SCHEMBL2550893

SCHEMBL2550893

NCc1ccc(-c2csc3c(=O)[nH]c4ccc(O)cc4c23)cc1

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NEK1 Q96PY6 9/20 0.51
WEE1 P30291 11/20 0.47
CHEK1 O14757 9/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2551422 0.89 WEE1 (0.51) WEE1CHEK1
SCHEMBL2574942 0.84 WEE1 (0.53) WEE1CHEK1
SCHEMBL2546633 0.82 NR1I2 (0.49) NEK1WEE1CHEK1
SCHEMBL2544993 0.77 TNKS (0.47)
SCHEMBL2564831 0.76 CHEK1 (0.47) WEE1CHEK1
Hydrochloric Acid SCHEMBL15092541 0.76 TNKS (0.46)
SCHEMBL14672729 0.75 NEK1 (0.57) NEK1WEE1CHEK1
SCHEMBL2550354 0.74 CHEK1 (0.45) WEE1CHEK1
SCHEMBL2546499 0.74 PARP1 (0.40) NEK1WEE1CHEK1
Hydrochloric Acid SCHEMBL15092457 0.74 CHEK1 (0.45) WEE1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552206-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-02-06 EP disclosed
WO-2011123419-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2011-10-06 WO disclosed