SCHEMBL2551982

SCHEMBL2551982

COc1cc2[nH]c(-c3ccccn3)nc2cc1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.58
RAB9A P51151 4/20 0.58
RUNX1 Q01196 1/20 0.58
CBFB Q13951 13/20 0.56
METAP2 P50579 4/20 0.56
METAP1 P53582 3/20 0.56
SMN1; SMN2 Q16637 3/20 0.55
KDM4E B2RXH2 2/20 0.55
PKM P14618 2/20 0.55
LMNA P02545 1/20 0.55
MAPT P10636 1/20 0.55
KMT2A Q03164 1/20 0.55
ALDH1A1 P00352 2/20 0.53
TP53 P04637 2/20 0.53
HPGD P15428 2/20 0.53
HSD17B10 Q99714 2/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
ALOX15 P16050 1/20 0.53
CYP2C19 P33261 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2551987 0.95 NPC1 (0.58) NPC1RAB9ARUNX1CBFBMETAP2
SCHEMBL179142 0.85 NPC1 (0.69) NPC1RAB9ARUNX1CBFBMETAP2
SCHEMBL1656372 0.83 GCK (0.63) NPC1RAB9ARUNX1CBFBMETAP2
SCHEMBL1657642 0.82 GCK (0.62) CBFBGCK
SCHEMBL14906668 0.81 CBFB (0.54) NPC1RAB9ARUNX1CBFBMETAP2
SCHEMBL17492287 0.81 CBFB (0.64) NPC1RAB9ARUNX1CBFBMETAP2
SCHEMBL1656346 0.80 GCK (0.71) CBFBCYP3A4CYP2C19GCK
SCHEMBL1657222 0.80 GCK (0.50) NPC1RAB9ARUNX1CBFBSMN1; SMN2
SCHEMBL15780004 0.79 CBFB (0.75) NPC1RAB9ARUNX1CBFBMETAP2
SCHEMBL179149 0.78 NPC1 (0.63) NPC1RAB9ARUNX1CBFBMETAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2556058-A1 RADIOPROTECTOR COMPOUNDS AND METHODS Peter MacCallum Cancer Institute (AU) 2013-02-13 EP disclosed
WO-2011123890-A1 RADIOPROTECTOR COMPOUNDS AND METHODS PETER MACCALLUM CANCER INSTITUTE (AU) 2011-10-13 WO disclosed