SCHEMBL2552525

SCHEMBL2552525

O=c1[nH]c2ccc(O)cc2c2c(Cl)csc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 10/20 0.48
WEE1 P30291 11/20 0.45
CDK5 Q00535 4/20 0.45
DYRK1A Q13627 3/20 0.45
GSK3A P49840 3/20 0.45
GSK3B P49841 3/20 0.45
DAPK3 O43293 1/20 0.45
JAK2 O60674 1/20 0.45
PAK4 O96013 1/20 0.45
ABL1 P00519 1/20 0.45
LCK P06239 1/20 0.45
FYN P06241 1/20 0.45
PIM1 P11309 1/20 0.45
PRKACA P17612 1/20 0.45
CDK2 P24941 1/20 0.45
LTK P29376 1/20 0.45
KDR P35968 1/20 0.45
MAP2K2 P36507 1/20 0.45
SYK P43405 1/20 0.45
CSNK1A1 P48729 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2550135 0.99 CHEK1 (0.47) CHEK1WEE1CDK5DYRK1AGSK3A
SCHEMBL2564831 0.85 CHEK1 (0.47) CHEK1WEE1CDK5DYRK1AGSK3A
SCHEMBL2552481 0.83 CHEK1 (0.45) CHEK1WEE1CDK5DYRK1AGSK3A
Hydrochloric Acid SCHEMBL15092457 0.83 CHEK1 (0.45) CHEK1WEE1CDK5DYRK1AGSK3A
SCHEMBL2574942 0.81 WEE1 (0.53) CHEK1WEE1CDK2PRKCQMEN1
SCHEMBL2550354 0.81 CHEK1 (0.45) CHEK1WEE1CDK5DYRK1AGSK3A
SCHEMBL2551422 0.81 WEE1 (0.51) CHEK1WEE1CDK5DYRK1AGSK3A
SCHEMBL2550191 0.79 CHEK1 (0.42) CHEK1WEE1CDK5DYRK1AGSK3A
SCHEMBL2546633 0.77 NR1I2 (0.49) CHEK1WEE1CDK5DYRK1AGSK3A
SCHEMBL2549922 0.75 MAP2K7 (0.47) CHEK1WEE1CDK5DYRK1AGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552206-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-02-06 EP disclosed
WO-2011123419-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2011-10-06 WO disclosed