SCHEMBL25540573

SCHEMBL25540573

CSc1ncc(C(F)(F)F)c(-c2cnn(C)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 5/20 0.46
RXFP1 Q9HBX9 1/20 0.39
CCNE1 P24864 7/20 0.39
CDK2 P24941 7/20 0.39
CDK1 P06493 4/20 0.39
CDK4 P11802 4/20 0.39
CCNB1 P14635 4/20 0.39
CCND1 P24385 4/20 0.39
CCND3 P30281 4/20 0.39
CDK6 Q00534 4/20 0.39
CCNT1 O60563 3/20 0.39
CDK7 P50613 3/20 0.39
CDK9 P50750 3/20 0.39
CCNH P51946 3/20 0.39
MNAT1 P51948 3/20 0.39
CCNE2 O96020 1/20 0.36
CLK2 P49760 1/20 0.36
PIK3CA P42336 1/20 0.35
NTRK1 P04629 1/20 0.35
KIT P10721 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30810412 0.82 CDK1 (0.51) LRRK2RXFP1CCNE1CDK2CDK1
SCHEMBL30837013 0.80 LRRK2 (0.47) LRRK2CCNE1CDK2CDK1CDK4
SCHEMBL27229135 0.80 LRRK2 (0.47) LRRK2CCNE1CDK2CDK1CDK4
SCHEMBL30291199 0.79 KDM5B (0.41) LRRK2RXFP1CCNE1CDK2CDK1
SCHEMBL30810528 0.77 CDK1 (0.54) RXFP1CCNE1CDK2CDK1CDK4
SCHEMBL14648923 0.77 RXFP1 (0.59) RXFP1NTRK1
SCHEMBL30291351 0.76 CCNE1 (0.43) RXFP1CCNE1CDK2CDK1CDK4
SCHEMBL30291251 0.76 CDK1 (0.41) RXFP1CCNE1CDK2CDK1CDK4
SCHEMBL21596308 0.75 PIK3CD (0.47) LRRK2
SCHEMBL30379895 0.75 PIK3CD (0.47) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091726-A1 INHIBITORS OF CYCLIN‑DEPENDENT KINASE 12 (CDK12) SYROS PHARMACEUTICALS, INC. (US) 2023-05-25 WO disclosed