SCHEMBL2556413

SCHEMBL2556413

CCNC(=O)Nc1cc2cccc(NC(=O)c3ccc[nH]3)c2cn1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.42
FGFR1 P11362 1/20 0.41
CDK8 P49336 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2559416 0.99 MAPK1 (0.42) MAPK1FGFR1CDK8
SCHEMBL2551801 0.85 NPC1 (0.50)
SCHEMBL2563512 0.85 MAPK1 (0.44) MAPK1
Hydrochloric Acid SCHEMBL2564290 0.84 MAPK1 (0.43) MAPK1
SCHEMBL2550944 0.78
SCHEMBL2551406 0.78 PIK3CA (0.49)
SCHEMBL14860044 0.77
Hydrochloric Acid SCHEMBL14860828 0.76
SCHEMBL2553090 0.76
SCHEMBL2552508 0.76 PIK3CA (0.53) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011121555-A1 ANTIBACTERIAL ISOQUINOLIN-3-YLUREA DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2011-10-06 WO claimed
WO-2011121555-A1 ANTIBACTERIAL ISOQUINOLIN-3-YLUREA DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2011-10-06 WO disclosed