SCHEMBL25565822

SCHEMBL25565822

Cc1ccc(-n2ccc(=O)[nH]c2=O)cc1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 3/20 0.56
DDB1 Q16531 1/20 0.56
HCAR1 Q9BXC0 1/20 0.54
ALDH1A1 P00352 6/20 0.49
HPGD P15428 1/20 0.49
GAA P10253 2/20 0.45
LMNA P02545 1/20 0.45
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
MAPT P10636 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ADRB1 P08588 1/20 0.41
ALKBH5 Q6P6C2 1/20 0.41
TSHR P16473 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
ATM Q13315 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP1 P29466 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23296161 0.84 CRBN (0.51) CRBNDDB1HCAR1ALDH1A1HPGD
SCHEMBL3340320 0.84 CRBN (0.51) CRBNDDB1HCAR1ALDH1A1HPGD
SCHEMBL848673 0.82 CRBN (0.53) CRBNDDB1HCAR1ALDH1A1HPGD
SCHEMBL25553210 0.82 CRBN (0.49) CRBNDDB1HCAR1ALDH1A1HPGD
SCHEMBL5325743 0.81 CRBN (0.66) CRBNDDB1HCAR1ALDH1A1HPGD
SCHEMBL11478341 0.79 CRBN (0.58) CRBNDDB1HCAR1ALDH1A1HPGD
SCHEMBL3340313 0.79 CRBN (0.46) CRBNDDB1HCAR1ALDH1A1HPGD
SCHEMBL23120610 0.77 CRBN (0.66) CRBNDDB1HCAR1ALDH1A1LMNA
SCHEMBL25551232 0.77 CRBN (0.44) CRBNDDB1HCAR1ALDH1A1MAPT
SCHEMBL14685529 0.76 CRBN (0.65) CRBNDDB1ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023096995-A1 COMPOSITIONS AND METHODS COMPRISING SUBSTITUTED N-(2-CHLORO-6-METHYLPHENYL)-2-((6-(6-MEMBERED HETEROCYCLOALKYL)-2-METHYLPYRIMIDIN-4-YL)AMINO)THIAZOLE-5-CARBOXAMIDE ANALOGUES ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC. (US) 2023-06-01 WO disclosed