SCHEMBL255854

SCHEMBL255854

C[C@H](c1ccc(F)cc1)c1nc(Nc2cc[nH]n2)c2ccc(Br)cc2n1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2C8 P10632 3/20 0.42
CYP2C9 P11712 3/20 0.42
JAK1 P23458 3/20 0.42
TYK2 P29597 3/20 0.42
CYP2C19 P33261 3/20 0.42
JAK3 P52333 3/20 0.42
ADORA3 P0DMS8 2/20 0.42
CYP1A2 P05177 1/20 0.42
NTRK1 P04629 3/20 0.41
GRK6 P43250 6/20 0.40
AURKA O14965 3/20 0.36
AURKB Q96GD4 2/20 0.36
FBP1 P09467 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
EGFR P00533 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL720608 0.88 JAK2 (0.53) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL174916 0.88 JAK2 (0.53) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL720607 0.88 JAK2 (0.53) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL10224905 0.88 JAK2 (0.53) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL15434543 0.85 JAK2 (0.54) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL175039 0.76 JAK2 (0.54) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL175038 0.76 JAK2 (0.54) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL174692 0.76 JAK2 (0.54) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL10224881 0.76 JAK2 (0.54) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL13187150 0.75 JAK2 (0.64) JAK2CYP3A4CYP2C8CYP2C9JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012030918-A1 ADENOSINE A3 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2012-03-08 WO disclosed