SCHEMBL255875

SCHEMBL255875

Cc1csc2nc(C(O)c3ccc(F)cc3)nc(Nc3cc[nH]n3)c12

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.45
CYP3A4 P08684 3/20 0.45
CYP2C8 P10632 3/20 0.45
CYP2C9 P11712 3/20 0.45
JAK1 P23458 3/20 0.45
TYK2 P29597 3/20 0.45
CYP2C19 P33261 3/20 0.45
JAK3 P52333 3/20 0.45
ADORA3 P0DMS8 2/20 0.45
CYP1A2 P05177 1/20 0.45
ESR1 P03372 1/20 0.34
PDE10A Q9Y233 1/20 0.34
TGM2 P21980 1/20 0.33
TGFBR1 P36897 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL175213 1.00 JAK2 (0.45) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL174850 0.85 JAK2 (0.63) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL173813 0.85 JAK2 (0.46) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL256527 0.85 JAK2 (0.46) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL10232408 0.81 JAK2 (0.50) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL174882 0.81 JAK2 (0.50) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL173921 0.78 AURKA (0.38) ADORA3ESR1TGM2TGFBR1
SCHEMBL255852 0.75 JAK2 (0.57) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL174255 0.75 JAK2 (0.57) JAK2CYP3A4CYP2C8CYP2C9JAK1
SCHEMBL174253 0.75 JAK2 (0.57) JAK2CYP3A4CYP2C8CYP2C9JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012030894-A1 THIENOPYRIDINE AND THIENOPYRIMIDINE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2012-03-08 WO disclosed