SCHEMBL25627

SCHEMBL25627

[CH]=CCC=C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21294346 0.82
SCHEMBL21294349 0.82
SCHEMBL28730964 0.79
SCHEMBL21294348 0.79
SCHEMBL21294351 0.79
SCHEMBL23546 0.71
SCHEMBL4665539 0.69
SCHEMBL4663538 0.69
SCHEMBL10458007 0.67
SCHEMBL18783524 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10666 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118136960-B Electrolyte and battery 深圳欣界能源科技有限公司 2024-07-16 CN claimed
CN-118136960-A Electrolyte and battery 深圳欣界能源科技有限公司 2024-06-04 CN claimed
EP-3753941-B1 PYRIMIDINE-FUSED CYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF SHANGHAI BLUERAY BIOPHARMA CO LTD (CN) 2024-05-01 EP claimed
WO-2023143312-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海艾力斯医药科技股份有限公司 2023-08-03 WO claimed
US-20210053989-A1 PYRIMIDINE-FUSED CYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF SHANGHAI BLUERAY BIOPHARMA CO., LTD. (CN) 2021-02-25 US claimed
EP-3753941-A1 PYRIMIDINE-FUSED CYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Shanghai Blueray Biopharma Co., Ltd. (CN) 2020-12-23 EP claimed
EP-3130594-B1 PHOSPHONATES OF ACETYLENIC BETULIN DERIVATIVES WITH ANTICANCER ACTIVITY, METHOD FOR THEIR PRODUCTION AND THEIR APPLICATION SLASKI UNIV MEDYCZNY W KATOWICACH (PL) 2020-11-11 EP claimed
CN-110128998-A A kind of allyl organic silicon potting adhesive and preparation method thereof 矽时代材料科技股份有限公司 2019-08-16 CN claimed
US-20080176858-A1 SELECTIVE ANTAGONISTS OF A2A ADENOSINE RECEPTORS ADENOSINE THERAPEUTICS, LLC (US) 2008-07-24 US claimed
EP-1054004-B1 NOVEL PYRIMIDINE-5-CARBOXAMIDE DERIVATIVES ASTELLAS PHARMA INC (JP) 2008-07-16 EP claimed
US-20070244134-A1 Selective antagonists of A2A adenosine receptors ADENOSINE THERAPEUTICS, LLC 2007-10-18 US claimed
US-7217702-B2 Selective antagonists of A2A adenosine receptors ADENOSINE THERAPEUTICS, LLC (US) 2007-05-15 US claimed
EP-1000070-B1 SILICON-CONTAINING CHAIN EXTENDERS AORTECH BIOMATERIALS PTY LTD (AU) 2003-09-10 EP claimed
EP-0984997-B1 SILICON-BASED POLYCARBONATES AORTECH BIOMATERIALS PTY LTD (AU) 2002-09-18 EP claimed
US-6420452-B1 POLYURETHANES WITH EXTENDERS AORTECH BIOMATERIALS PTY LTD (AU) 2002-07-16 US claimed
US-4710491-A N-glycosylated carboxylic acid derivatives as agents for combating rheumatic diseases TROPONWERKE GMBH & CO., KG (DE) 1987-12-01 US claimed
EP-0152630-A2 Organosiloxane polymers and compositions containing same curable upon exposure to gaseous oxygen UNION CARBIDE CORPORATION (US) 1985-08-28 EP claimed
WO-1985002854-A1 ORGANOSILOXANE POLYMERS AND COMPOSITIONS CONTAINING SAME CURABLE UPON EXPOSURE TO GASEOUS OXYGEN UNION CARBIDE CORPORATION (US) 1985-07-04 WO claimed
US-4526954-A Contains olefinically polyunsaturated radical containing 1,3- or 1,4-pentadienylene group bonded to silicon UNION CARBIDE CORPORATION (US) 1985-07-02 US claimed
US-12042479-B2 Use of topical formulations of cannabinoids in the treatment of epidermolysis bullosa and related connective tissue disorders INMED PHARMACEUTICALS INC. 2024-07-23 US disclosed
US-12042523-B2 Compositions and methods for managing or improving bone disorders, joint disorders, cartilage disorders, or a combination thereof UNIGEN, INC. (US) 2024-07-23 US disclosed
CN-118369335-A N1-modified pseudouridine and application thereof in mRNA synthesis 上海吉量医药工程有限公司 2024-07-19 CN disclosed
CN-118359666-A Tetravalent cisplatin prodrug, liposome and application thereof 杭州佰因泰医药科技有限公司 2024-07-19 CN disclosed
US-20240239751-A1 PROCESSES FOR PREPARING AG-10, ITS INTERMEDIATES, AND SALTS THEREOF BRIDGEBIO GENE THERAPY RESEARCH, INC. 2024-07-18 US disclosed
US-20240238427-A1 METHODS OF TREATING AN EYE DISORDER KODIAK SCIENCES INC. 2024-07-18 US disclosed
US-20240239755-A1 SUBSTITUTED PYRIDAZINONES, SALTS OR N-OXIDES THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2024-07-18 US disclosed
WO-2024151847-A1 IDENTIFICATION OF OTUD7B INHIBITOR 7BI AND ITS APPLICATION IN REDUCING GROWTH OF NSCLC AND LEUKEMIA CELLS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2024-07-18 WO disclosed
WO-2024152000-A1 DISRUPTABLE LINKER COMPOSITIONS, SWITCHABLE BISPECIFIC T CELL NANOENGAGER (SWITCH-BITE) COMPOSITIONS COMPRISING THE SAME, AND METHODS OF USE THEREOF THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2024-07-18 WO disclosed
WO-2024151489-A1 PHARMACEUTICAL PYRIDYL COMPOSITIONS AND METHODS FOR USE Unicycive Therapeutics Inc. (US) 2024-07-18 WO disclosed
US-20240238311-A1 AQUEOUS PHARMACEUTICAL FORMULATION OF HYDROCORTISONE SODIUM PHOSPHATE AND MONOTHIOGLYCEROL ANTARES PHARMA, INC. (US) 2024-07-18 US disclosed
US-20240238321-A1 MODIFIED OLIGOMERIC COMPOUNDS COMPRISING TRICYCLO-DNA NUCLEOSIDES AND USES THEREOF SYNTHENA AG (CH) 2024-07-18 US disclosed
US-20240239807-A1 SARS-COV2 MAIN PROTEASE INHIBITORS GILEAD SCIENCES, INC. 2024-07-18 US disclosed
US-20240238212-A1 LIPID COMPOUNDS AND LIPID NANOPARTICLE COMPOSITIONS Suzhou Abogen Biosciences Co., Ltd. (CN) 2024-07-18 US disclosed
US-20240238285-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2024-07-18 US disclosed
WO-2024150067-A2 ACYLOIN CONDENSATION REACTIONS, ENZYMES, AND PRODUCTS THEREOF MOJIA BIOTECH PTE. LTD. (SG) 2024-07-18 WO disclosed
US-20240239775-A1 FXR REGULATOR, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF BEIJING BEST PATHWAY MANAGEMENT CONSULTING CENTER (LIMITED PARTNERSHIP) (CN) 2024-07-18 US disclosed
US-20240238303-A1 LARGE-CONDUCTANCE POTASSIUM CHANNEL MODULATORS, COMPOSITIONS THEREOF, METHODS OF MANUFACTURING THEREOF, AND METHODS OF USE THEREOF ENALARE THERAPEUTICS INC (US) 2024-07-18 US disclosed
US-20240239762-A1 NOVEL HETEROCYCLIC COMPOUNDS FLORATEK PHARMA S A (CH) 2024-07-18 US disclosed
US-20240238438-A1 CD-90 Targeted Lipid Nanoparticles FRED HUTCHINSON CANCER CENTER 2024-07-18 US disclosed
US-20240239797-A1 AKT1 MODULATORS ALTEROME THERAPEUTICS, INC. 2024-07-18 US disclosed
CN-118136960-B Electrolyte and battery 深圳欣界能源科技有限公司 2024-07-16 CN disclosed
CN-118344348-A Heterocyclic substituted quinazoline and preparation method and application thereof 苏州泽璟生物制药股份有限公司 2024-07-16 CN disclosed
CN-113677665-B Substituted 2-heteroarylaminobenzenes and salts thereof, and their use as herbicides 拜耳公司 2024-07-16 CN disclosed
US-12036211-B2 Nicorandil derivatives Unicycive Therapeutics Inc. (US) 2024-07-16 US disclosed
CN-118339151-A Compound for inhibiting or degrading BRD9, composition and pharmaceutical application thereof 西藏海思科制药有限公司 2024-07-12 CN disclosed
CN-111447939-B Method for preparing conjugate 四川科伦博泰生物医药股份有限公司 2024-07-12 CN disclosed
CN-118324767-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-07-12 CN disclosed
CN-118324782-A Tricyclic compound for inhibiting HPK1 and medical application thereof 西藏海思科制药有限公司 2024-07-12 CN disclosed
CN-118339152-A Macrocyclic compounds having farnesyl transferase inhibitory activity 库拉肿瘤学公司 2024-07-12 CN disclosed
CN-118339168-A Fused ring heterocyclic derivative and application thereof in medicine 西藏海思科制药有限公司 2024-07-12 CN disclosed
US-20240228504-A1 SUBSTITUTED TRICYCLIC AMIDES, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2024-07-11 US disclosed
WO-2024148191-A1 MODULATORS OF TNF-α ACTIVITY FORWARD THERAPEUTICS, INC. (US) 2024-07-11 WO disclosed
US-20240226310-A1 Lipid Nanoparticle Therapeutics that Evade the Immune Response THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2024-07-11 US disclosed
US-20240228480-A1 PROCESSES FOR PREPARING PYRROLOPYRIDINE-ANILINE COMPOUNDS CURIA GLOBAL, INC. 2024-07-11 US disclosed
US-20240228499-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION (US) 2024-07-11 US disclosed
EP-4395550-A1 ADDITIVES FOR COLOR DRIFT REDUCTION IN COPPER-BASED ANTIMICROBIAL POLYMERIC FORMULATIONS Corning Incorporated (US) 2024-07-10 EP disclosed
EP-4395828-A1 BIFUNCTIONAL DEGRADERS COMPRISING A TEAD BINDER Novartis AG (CH) 2024-07-10 EP disclosed
CN-118317956-A Bis (hetero) aryl thioether oxadiazines as fungicidal compounds 拜耳公司 2024-07-09 CN disclosed
US-12030879-B2 Sulfonyl acetamides as NLRP3 inhibitors INFLAZOME LIMITED (IE) 2024-07-09 US disclosed
US-12030853-B2 MASP-2 inhibitors and methods of use OMEROS CORPORATION (US) 2024-07-09 US disclosed
CN-118317955-A N- (4-aminocyclohexyl) pyrimidine-4-carboxamide as CD38 inhibitor 塞里文斯股份有限公司 2024-07-09 CN disclosed
US-12029708-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2024-07-09 US disclosed
CN-112724349-B Polymer and use thereof 立邦涂料(中国)有限公司 2024-07-05 CN disclosed
CN-118302289-A Method for producing bioactive polymer filaments, and printing method using same 新加坡科技研究局 2024-07-05 CN disclosed
CN-116143757-B Multifunctional compound, composition and application of degradable BTK kinase 杭州和正医药有限公司 2024-07-05 CN disclosed
CN-118290446-A Compound for inhibiting and degrading c-MYC and medical application thereof 西藏海思科制药有限公司 2024-07-05 CN disclosed
US-20240218011-A1 GLUCOCORTICOID RECEPTOR AGONISTS AND CONJUGATES THEREOF FIREFLY BIO, INC. 2024-07-04 US disclosed
US-20240216346-A1 Substituted Chromenones, IRE1 Inhibitors, and Methods of Using Same THE WISTAR INST (US) 2024-07-04 US disclosed
US-20240218021-A1 CYCLIN INHIBITORS CIRCLE PHARMA, INC. 2024-07-04 US disclosed
US-20240216380-A1 BTK Inhibitors to Treat Solid Tumors Through Modulation of the Tumor Microenvironment ACERTA PHARMA BV (NL) 2024-07-04 US disclosed
US-20240216523-A1 Compositions and Methods for Targeting Lipid Nanoparticle Therapeutics to Stem Cells NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2024-07-04 US disclosed
WO-2024140653-A1 SELECTIVE CDK12/13 INHIBITOR AND APPLICATION THEREOF 南京圣和药业股份有限公司 2024-07-04 WO disclosed
WO-2024141052-A1 ESTROGEN-RECEPTOR MODULATOR AND USE THEREOF 江苏威凯尔医药科技有限公司 2024-07-04 WO disclosed
US-20240218399-A1 LIPID COMPOUNDS AND LIPID NANOPARTICLE COMPOSITIONS SUZHOU ABOGEN BIOSCIENCES CO LTD (CN) 2024-07-04 US disclosed
EP-4392409-A1 PYRAZINE COMPOUNDS AS IRREVERSIBLE INHIBITORS OF FLT3 Biomea Fusion, Inc. (US) 2024-07-03 EP disclosed
EP-4146348-B1 INHIBITORS OF NEK7 KINASE HALIA THERAPEUTICS INC (US) 2024-07-03 EP disclosed
EP-4013385-B1 IMPROVED LIPID NANOPARTICLES FOR DELIVERY OF NUCLEIC ACIDS ACUITAS THERAPEUTICS INC (CA) 2024-07-03 EP disclosed
EP-4394011-A2 MODIFICATION OF SURFACE PROPERTIES OF MICROFLUIDIC DEVICES Bio-Rad Laboratories, Inc. (US) 2024-07-03 EP disclosed
CN-118271316-A Cycloheptenyl-containing derivative, pharmaceutical composition and pharmaceutical application thereof 西藏海思科制药有限公司 2024-07-02 CN disclosed
CN-118271233-A Nilaparil manufacturing method 特沙诺有限公司 2024-07-02 CN disclosed
CN-118271284-A Estrogen receptor modulators and uses thereof 江苏威凯尔医药科技有限公司 2024-07-02 CN disclosed
CN-118284797-A Calibration assistance for optical imaging applications 斯特拉斯堡大学 2024-07-02 CN disclosed
US-12024595-B2 Polymer composition BASF SE (DE) 2024-07-02 US disclosed
US-12024731-B2 Methods and enzyme catalysts for the synthesis of non-canonical amino acids CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2024-07-02 US disclosed
CN-118271288-A Dual MAGL and FAAH inhibitors 灵北拉荷亚研究中心公司 2024-07-02 CN disclosed
CN-118284602-A Pyridine derivatives as sodium channel activators and uses thereof 泽农医药公司 2024-07-02 CN disclosed
CN-118284611-A Diazabicyclooctane derivatives useful as matrix metalloproteinase inhibitors VASA治疗有限责任公司 2024-07-02 CN disclosed
CN-118255746-A Selective CDK12/13 inhibitors and uses thereof 南京圣和药业股份有限公司 2024-06-28 CN disclosed
CN-118255780-A Compound for inhibiting and degrading c-MYC and medical application thereof 西藏海思科制药有限公司 2024-06-28 CN disclosed
WO-2024133610-A1 PROCCESSES FOR THE PREPARATION OF AN NLRP3 INHIBITOR F. HOFFMANN-LA ROCHE AG (CH) 2024-06-27 WO disclosed
US-20240209000-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE LLC 2024-06-27 US disclosed
WO-2024138052-A1 HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC. (US) 2024-06-27 WO disclosed
WO-2024134466-A1 SUBSTITUTED ARYLAMINE COMPOUNDS, SUBSTITUTED HETEROARYLAMINE COMPOUNDS, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2024-06-27 WO disclosed
US-20240208982-A1 PYRAZOLOPYRIMIDINONE COMPOUNDS Orphagen Pharmaceuticals, Inc. 2024-06-27 US disclosed
WO-2024137780-A1 PANK MODULATORS AND METHODS OF TREATMENT USING SAME YALE UNIVERSITY (US) 2024-06-27 WO disclosed
US-20240209076-A1 USE OF IL-6 ANTIBODIES AND VEGF TRAPS, AND FUSION CONSTRUCTS AND CONJUGATES THEREOF KODIAK SCIENCES INC. 2024-06-27 US disclosed
US-20240209214-A1 METHODS OF ATTACHING AZIDE COMPOUNDS TO SURFACES AND COMPOUNDS AND PRODUCTS THEREOF VANDERBILT UNIVERSITY 2024-06-27 US disclosed
WO-2024131843-A1 ANTIBODY-DRUG CONJUGATE, PREPARATION METHOD THEREFOR, AND USE THEREOF 苏州宜联生物医药有限公司 2024-06-27 WO disclosed
US-20240209011-A1 HETEROAROMATIC PHOSPHONIUM SALTS FOR TREATING CANCER FLORATEK PHARMA S A (CH) 2024-06-27 US disclosed
US-20240208975-A1 MACROCYCLIC HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC. 2024-06-27 US disclosed
US-20240208973-A1 TETRACYCLIC COMPOUNDS FOR TREATING BRAIN DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2024-06-27 US disclosed
EP-3356387-B1 ANTIMICROBIAL POLYMYXIN DERIVATIVE COMPOUNDS UNIV MONASH (AU) 2024-06-26 EP disclosed
EP-3908568-B1 LIPIDS FOR LIPID NANOPARTICLE DELIVERY OF ACTIVE AGENTS ACUITAS THERAPEUTICS INC (CA) 2024-06-26 EP disclosed
EP-4103160-B1 NANOPARTICLES ENCAPSULATING SMALL MOLECULES ETH ZUERICH (CH) 2024-06-26 EP disclosed
EP-4387977-A1 PHOSPHOLIPID COMPOUNDS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. (US) 2024-06-26 EP disclosed
EP-4387610-A1 TRICYCLIC SULTAMS AND SULFAMIDES AS ANTITUMOR AGENTS Peloton Therapeutics, Inc. (US) 2024-06-26 EP disclosed
EP-4388127-A1 METHODS AND COMPOSITIONS FOR IDENTIFYING METHYLATED CYTOSINES Illumina, Inc. (US) 2024-06-26 EP disclosed
CN-114502187-B Peptide amide composition and preparation thereof 西藏海思科制药有限公司 2024-06-25 CN disclosed
CN-118251216-A Method for biofilm disruption 尼尔利希尔有限公司 2024-06-25 CN disclosed
CN-115960109-B Preparation and application of condensed ring SHP2 phosphatase inhibitor 药雅科技(上海)有限公司 2024-06-25 CN disclosed
CN-118251389-A Pyridyl derivatives as sodium channel activators 泽农医药公司 2024-06-25 CN disclosed
US-12016856-B2 Compounds and methods for inhibiting NHE-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders ARDELYX, INC. (US) 2024-06-25 US disclosed
CN-118251393-A Novel substituted sulfonylurea compounds as inhibitors of interleukin-1 activity 唯久生物技术(苏州)有限公司 2024-06-25 CN disclosed
US-12016853-B2 Methods of treating RBP4 related diseases with triazolopyridines BELITE BIO, INC (KY) 2024-06-25 US disclosed
US-12021194-B2 Silicon-based energy storage devices with electrolyte containing a benzoyl peroxide based compound ENEVATE CORPORATION (US) 2024-06-25 US disclosed
US-12018011-B2 Macrocyclic compounds and compositions, and methods of preparing and using the same KURA ONCOLOGY, INC. (US) 2024-06-25 US disclosed
US-12018033-B2 Inhibitors of protein arginine deiminases FORWARD THERAPEUTICS, INC. (US) 2024-06-25 US disclosed
CN-114423739-B Improved enantioselective hydrogenation of 4-substituted 1, 2-dihydroquinolines in the presence of chiral iridium catalysts and additives 拜耳公司 2024-06-25 CN disclosed
CN-113395963-B Non-ATP/catalytic site p38 mitogen-activated protein kinase inhibitors 马里兰大学巴尔的摩分校 2024-06-25 CN disclosed
CN-118221656-A Compounds useful for the treatment of gastrointestinal disorders 阿德利克斯股份有限公司 2024-06-21 CN disclosed
CN-118221642-A Sulfonamide derivative and application thereof in medicine 西藏海思科制药有限公司 2024-06-21 CN disclosed
US-20240199596-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2024-06-20 US disclosed
US-20240199702-A1 CELL-PERMEABLE CYCLIC PEPTIDES AND USES THEREOF UNNATURAL PRODUCTS INC. 2024-06-20 US disclosed
US-20240199650-A1 PYRIMIDINE BASED MODULATORS AND USES THEREOF QUANTA THERAPEUTICS, INC. 2024-06-20 US disclosed
US-20240197742-A1 Therapeutic Combinations of a CD19 Inhibitor and a BTK Inhibitor ACERTA PHARMA BV (NL) 2024-06-20 US disclosed
US-20240199542-A1 SUBSTITUTED PYRROLIDIN-2-ONES, SALTS THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2024-06-20 US disclosed
WO-2024125603-A1 SHP2 INHIBITOR AND USE THEREOF 江苏威凯尔医药科技有限公司 2024-06-20 WO disclosed
WO-2024129763-A1 MODULATORS OF TNF-α ACTIVITY FORWARD THERAPEUTICS, INC. (US) 2024-06-20 WO disclosed
US-20240199699-A1 NICOTINIC ACETYLCHOLINE RECEPTOR PEPTIDE ANTAGONIST CONOTOXIN COMPOSITIONS AND RELATED METHODS GLO PHARMA, INC. 2024-06-20 US disclosed
US-20240197738-A1 COMPOUND 7AI IN TREATING EWING SARCOMA BY INHIBITING OTUD7A Atomwise Inc. 2024-06-20 US disclosed
US-20240197810-A1 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC. 2024-06-20 US disclosed
US-20240197694-A1 MODIFIED PROTEINS AND PROTEIN BINDERS CULLGEN (SHANGHAI), INC. (CN) 2024-06-20 US disclosed
WO-2024125639-A1 NOVEL GLUCOCORTICOID, METHOD FOR PREPARING SAME, AND USE THEREOF 津药生物科技(天津)有限公司 2024-06-20 WO disclosed
EP-4384506-A1 PROCESS FOR POLYAMIDE SYNTHESIS Design Therapeutics, Inc. (US) 2024-06-19 EP disclosed
EP-3562893-B1 MODIFICATION OF SURFACE PROPERTIES OF MICROFLUIDIC DEVICES BIO RAD LABORATORIES INC (US) 2024-06-19 EP disclosed
EP-4384522-A1 SELECTIVE KRAS INHIBITORS Erasca, Inc. (US) 2024-06-19 EP disclosed
EP-4384179-A1 COVALENT INHIBITORS OF MENIN-MLL INTERACTION FOR DIABETES MELLITUS Biomea Fusion, Inc. (US) 2024-06-19 EP disclosed
CN-118206558-A Compound capable of inhibiting and degrading AuroraA, pharmaceutical composition and pharmaceutical application thereof 西藏海思科制药有限公司 2024-06-18 CN disclosed
US-12012392-B2 Sulfonamide carboxamide compounds INFLAZOME LIMITED (IE) 2024-06-18 US disclosed
US-12015122-B2 Silicon-based energy storage devices with carboxylic ether, carboxylic acid based salt, or acrylate electrolyte containing electrolyte additives ENEVATE CORPORATION (US) 2024-06-18 US disclosed
CN-113318113-B Use of fibroblast growth factor receptor inhibitors 药捷安康(南京)科技股份有限公司 2024-06-18 CN disclosed
CN-118215472-A Lipid nanoparticles for oligonucleotide delivery 纪费亚斯公司 2024-06-18 CN disclosed
CN-110312730-B Cytotoxins and conjugates, uses thereof and methods of preparation 四川科伦博泰生物医药股份有限公司 2024-06-18 CN disclosed
CN-118215471-A Lipid nanoparticles for oligonucleotide delivery 纪费亚斯公司 2024-06-18 CN disclosed
CN-112638879-B Heteroaryl substituted sulfonamide compounds and their use as therapeutic agents 泽农医药公司 2024-06-18 CN disclosed
CN-118206550-A SHP2 inhibitor and application thereof 江苏威凯尔医药科技有限公司 2024-06-18 CN disclosed
CN-118201941-A CD73 compounds 吉利德科学公司 2024-06-14 CN disclosed
CN-118201612-A Compositions and methods for combination therapy for the treatment of lymphomas 上海睿跃生物科技有限公司 2024-06-14 CN disclosed
US-20240190865-A1 T-TYPE CALCIUM CHANNEL ANTAGONISTS AND USES THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2024-06-13 US disclosed
US-20240189304-A1 BET PROTEIN INHIBITORS AND USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-06-13 US disclosed
US-20240190839-A1 SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF INSILICO MEDICINE IP LIMITED (HK) 2024-06-13 US disclosed
US-20240190864-A1 Bruton's Tyrosine Kinase (BTK) INHIBITOR AND APPLICATION THEREOF YA THERAPEUTICS INC (CN) 2024-06-13 US disclosed
US-20240189445-A1 Targeted Therapeutic Lipid Nanoparticles and Methods of Use NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2024-06-13 US disclosed
US-20240190917-A1 PEPTIDES AND METHODS FOR REDUCING SKIN PIGMENTATION GLO PHARMA, INC. 2024-06-13 US disclosed
US-20240191035-A1 RING OPENING POLYMERIZATION OF CYCLIC SILOXANES CHT USA INC (US) 2024-06-13 US disclosed
WO-2024123791-A1 FORMULATIONS FOR DUAL VEGF/IL-6 INHIBITORS KODIAK SCIENCES INC. (US) 2024-06-13 WO disclosed
WO-2024124143-A2 HSC TARGETED LNP FOR DELIVERY OF PRO-APOPTOTIC MRNA AND METHODS OF USE THEREOF THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2024-06-13 WO disclosed
EP-4380566-A1 METHODS OF TREATING MIGRAINE WITH MNK INHIBITORS 4E Therapeutics, Inc. (US) 2024-06-12 EP disclosed
CN-114206463-B Lipid compounds and lipid nanoparticle compositions 苏州艾博生物科技有限公司 2024-06-11 CN disclosed
CN-118159536-A Substituted 1,2, 4-thiadiazolyl nicotinamide, salts or N-oxides thereof and their use as herbicidal active substances 拜耳公司 2024-06-07 CN disclosed
CN-118159300-A Antibody, drug conjugate and application thereof 苏州信诺维医药科技股份有限公司 2024-06-07 CN disclosed
CN-118159542-A Substituted 2, 3-dihydro [1,3] thiazolo [4,5-b ] pyridines, salts thereof and their use as herbicidal agents 拜耳公司 2024-06-07 CN disclosed
CN-118146224-A Nitrogen-containing tricyclic derivative and application thereof in medicine 西藏海思科制药有限公司 2024-06-07 CN disclosed
WO-2024119117-A1 MODIFIED 5' CAP FOR MRNA AND METHODS OF USE THEREOF PRIME MEDICINE, INC. (US) 2024-06-06 WO disclosed
WO-2024119099-A1 GALLIUM-SALOPHEN ANTIMICROBIAL COMPOUNDS AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2024-06-06 WO disclosed
US-20240180904-A1 Methods of Treating Chronic Lymphocytic Leukemia and Small Lymphocytic Leukemia Using a BTK Inhibitor ACERTA PHARMA BV (NL) 2024-06-06 US disclosed
US-20240182452-A1 6-PHENYL-4,5-DIHYDROPYRIDAZIN-3(2H)-ONE DERIVATIVES AS PDE3A AND PDE3B INHIBITORS FOR TREATING CANCER BAYER AKTIENGESELLSCHAFT (DE) 2024-06-06 US disclosed
US-20240182498-A1 DISILYLAMINE PRECURSORS AND RELATED METHODS ENTEGRIS INC (US) 2024-06-06 US disclosed
WO-2024114954-A1 CHLORIN K ANALOGUES SUITABLE FOR USE IN PHOTODYNAMIC THERAPY (PDT) RMW CHO GROUP LIMITED (CN) 2024-06-06 WO disclosed
WO-2024115525-A2 NOVEL COMPOUNDS RMW CHO GROUP LIMITED (CN) 2024-06-06 WO disclosed
WO-2024115524-A1 PORPHYRIN AND PHOSPHONIUM-PORPHYRIN BASED COMPOUNDS FOR PHOTODYNAMIC THERAPY AND DIAGNOSTICS RMW CHO GROUP LIMITED (CN) 2024-06-06 WO disclosed
WO-2024118840-A1 FUSED PYRIMIDINES AS MASP-2 INHIBITORS OMEROS CORPORATION (US) 2024-06-06 WO disclosed
WO-2024118571-A2 RING OPENING POLYMERIZATION OF CYCLIC SILOXANES CHT USA INC (US) 2024-06-06 WO disclosed
US-20240182467-A1 INHIBITORS OF RAF KINASES Pierre Fabre Médicament (FR) 2024-06-06 US disclosed
US-20240182464-A1 SELECTIVE BCL-XL PROTAC COMPOUNDS AND METHODS OF USE Les Laboratoirens Serviece (FR) 2024-06-06 US disclosed
US-20240182480-A1 5-HT2A AND/OR 5-HT2C RECEPTOR AGONISTS DIAMOND THERAPEUTICS INC. (CA) 2024-06-06 US disclosed
US-20240182476-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2024-06-06 US disclosed
US-20240182490-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2024-06-06 US disclosed
WO-2024114953-A1 PHYLLOCHLORIN ANALOGUES SUITABLE FOR USE IN PHOTODYNAMIC THERAPY (PDT) RMW CHO GROUP LIMITED (CN) 2024-06-06 WO disclosed
EP-3890737-B1 USP19 INHIBITORS FOR USE IN A METHOD OF TREATING OBESITY, INSULIN RESISTANCE AND TYPE II DIABETES ALMAC DISCOVERY LTD (GB) 2024-06-05 EP disclosed
EP-3570838-B1 SUBSTITUTED 3-DIALKYLAMINOMETHYL-PIPERIDIN-4-YL-BENZAMIDES AND METHODS OF MAKING AND USING SAME MEBIAS DISCOVERY INC (US) 2024-06-05 EP disclosed
EP-4376833-A1 COMPOSITIONS AND METHODS FOR TREATING LIPOMA PAIN Raziel Therapeutics Ltd. (IL) 2024-06-05 EP disclosed
US-11999733-B2 Diacylglycerol kinase modulating compounds GILEAD SCIENCES, INC. (US) 2024-06-04 US disclosed
US-11998539-B2 Substituted aminoquinolones as DGKalpha inhibitors for immune activation BAYER AKTIENGESELLSCHAFT (DE) 2024-06-04 US disclosed
CN-118136960-A Electrolyte and battery 深圳欣界能源科技有限公司 2024-06-04 CN disclosed
CN-118139860-A PARP-1 degrading agent and application thereof 西藏海思科制药有限公司 2024-06-04 CN disclosed
US-11999730-B1 AKT1 modulators ALTEROME THERAPEUTICS, INC. (US) 2024-06-04 US disclosed
CN-118126035-A Cycloalkyl or heterocycle substituted benzo or pyridopyridazine, and preparation method and application thereof 苏州泽璟生物制药股份有限公司 2024-06-04 CN disclosed
US-11999821-B2 Compound, a reaction product of said compound and production methods thereof AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2024-06-04 US disclosed
CN-114829368-B Method for sequencing by synthesis using a continuous labelling scheme 豪夫迈·罗氏有限公司 2024-06-04 CN disclosed
CN-118119275-A Additives for reducing color shift in copper-based antimicrobial polymer formulations 康宁公司 2024-05-31 CN disclosed
CN-118108711-A Glycollic acid oxidase inhibitor and application thereof in medicine 西藏海思科制药有限公司 2024-05-31 CN disclosed
CN-118119372-A Malodor-counteracting compositions, compositions and uses thereof 国际香料和香精公司 2024-05-31 CN disclosed
CN-113874341-B Process for preparing derivatives of 1, 1-dialkylethane-1, 2-diols useful as intermediates 科学与工业研究委员会 2024-05-31 CN disclosed
WO-2024112796-A1 MODULATORS OF TNF-α ACTIVITY FORWARD THERAPEUTICS, INC. (US) 2024-05-30 WO disclosed
WO-2024112611-A1 TARGETED PROTEIN MODIFICATION WEATHERWAX BIOTECHNOLOGIES CORPORATION (US) 2024-05-30 WO disclosed
WO-2024112882-A1 TARGETED DELIVERY OF GENE EDITING CONSTRUCTS AND METHODS OF USE THEREOF THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2024-05-30 WO disclosed
US-20240175023-A1 GALNAC COMPOSITIONS FOR IMPROVING SIRNA BIOAVAILABILITY EMPIRICO INC. 2024-05-30 US disclosed
US-20240174690-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER VANDERBILT UNIVERSITY 2024-05-30 US disclosed
US-20240174618-A1 SUBSTITUTED (2-HETEROARYLOXYPHENYL)SULFONATES, SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2024-05-30 US disclosed
WO-2024109798-A1 LIPID COMPOUND AND LIPID NANOPARTICLE COMPOSITION 苏州艾博生物科技有限公司 2024-05-30 WO disclosed
US-20240174699-A1 FUNCTIONALIZED ORGANOTIN PRECURSORS AND RELATED METHODS ENTEGRIS, INC. 2024-05-30 US disclosed
US-20240174667-A1 AKT1 MODULATORS ALTEROME THERAPEUTICS, INC. 2024-05-30 US disclosed
US-20240174715-A1 PEPTIDE LIBRARIES WITH NON-CANONICAL AMINO ACIDS INDI MOLECULAR, INC. 2024-05-30 US disclosed
US-20240174630-A1 SELECTIVE HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF HUMAN DISEASE SHUTTLE PARMACEUTICALS, LLC 2024-05-30 US disclosed
EP-4373823-A1 SYNTHESIS OF SUBSTITUTED TRICYCLIC AMIDES AND ANALOGUES THEREOF Arbutus Biopharma Corporation (CA) 2024-05-29 EP disclosed
CN-118084844-A PI3K alpha inhibitor and application thereof in medicine 西藏海思科制药有限公司 2024-05-28 CN disclosed
CN-118103372-A Heterocyclic compound capable of inhibiting IL-17A and application thereof 西藏海思科制药有限公司 2024-05-28 CN disclosed
CN-118084720-A Triarylmethane dye and application thereof in biological imaging and tumor photoacoustic imaging 华东理工大学 2024-05-28 CN disclosed
US-11993595-B2 Compounds MISSION THERAPEUTICS LIMITED (GB) 2024-05-28 US disclosed
CN-118076357-A Covalent inhibitors of Mennin-MLL interactions for diabetes 拜欧米富士恩公司 2024-05-24 CN disclosed
CN-115197221-B Dihydropyrazolopyrimidinone macrocyclic derivatives and their use 轩竹(北京)医药科技有限公司 2024-05-24 CN disclosed
CN-115279368-B Heteroaryl compounds 维瓦斯治疗公司 2024-05-24 CN disclosed
CN-118063537-A Prodrugs of directed lymphatics 莫纳什大学 2024-05-24 CN disclosed
CN-118076603-A CAMKK2 modulators as ligand-directed degradants 细胞基因公司 2024-05-24 CN disclosed
CN-118076612-A Sulfur-containing heteroaromatic tricyclic KRAS inhibitors 医睿世康药业研发公司 2024-05-24 CN disclosed
CN-118076354-A Methods of treating migraine with MNK inhibitors 4E治疗公司 2024-05-24 CN disclosed
CN-118063435-A Piperidine-2, 6-dione derivative and application thereof 西藏海思科制药有限公司 2024-05-24 CN disclosed
WO-2024105205-A1 ANTIBODY-DRUG CONJUGATES (A2DCS) WITH ENZYMATICALLY CLEAVABLE GROUPS BAYER AKTIENGESELLSCHAFT (DE) 2024-05-23 WO disclosed
WO-2024108090-A1 METHODS OF TREATING INFLAMMATORY CONDITIONS ATHIRA PHARMA, INC. (US) 2024-05-23 WO disclosed
WO-2024108131-A1 PHTHALAZINONE BASED MODULATORS FOR THE TREATMENT OF DISEASE SOLEY THERAPEUTICS, INC. (US) 2024-05-23 WO disclosed
WO-2024107565-A1 AKT1 MODULATORS ALTEROME THERAPEUTICS, INC. (US) 2024-05-23 WO disclosed
US-20240166625-A1 Substituted 4-Benzyl And 4-Benzoyl Piperidine Derivates CEPHALON LLC 2024-05-23 US disclosed
US-20240166641-A1 HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC. 2024-05-23 US disclosed
US-20240166661-A1 Spiropiperidine Derivatives CEPHALON LLC 2024-05-23 US disclosed
US-20240166658-A1 PORPHYRIN DERIVATIVES AND USES THEREOF UNIVERSITY OF TASMANIA (AU) 2024-05-23 US disclosed
WO-2024104956-A1 SUBSTITUTED CYCLOALKYLSULFANYLPHENYLURACILS AND THEIR SALTS, AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2024-05-23 WO disclosed
WO-2024104954-A1 SUBSTITUTED CYCLOALKYLOXYPHENYLURACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2024-05-23 WO disclosed
WO-2024104952-A1 SUBSTITUTED CYCLOPROPYLOXYPHENYLURACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2024-05-23 WO disclosed
EP-4370109-A1 SUBEROYLANILIDE HYDROXAMIC ACID (SAHA) DRUGS, CONJUGATES, AND NANOPARTICLES, AND METHODS OF USE THEREOF University of Maryland, Baltimore (US) 2024-05-22 EP disclosed
EP-4370506-A1 PYRAZINE COMPOUNDS AS INHIBITORS OF FLT3 Biomea Fusion, Inc. (US) 2024-05-22 EP disclosed
US-11990585-B2 Electrolyte formulations for optimal performance in Si-containing lithium ion batteries ENEVATE CORPORATION (US) 2024-05-21 US disclosed
US-11987597-B2 Modulators of TNF-α activity FORWARD THERAPEUTICS, INC. (US) 2024-05-21 US disclosed
US-11987560-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2024-05-21 US disclosed
CN-118056835-A Pyridazinones as PARP7 inhibitors 中山优理生物医药有限公司 2024-05-21 CN disclosed
CN-118047776-A Tricyclic compound, preparation method thereof, pharmaceutical composition containing tricyclic compound and application of tricyclic compound 上海优理惠生医药有限公司 2024-05-17 CN disclosed
CN-111566104-B Spiro aromatic ring compound and application thereof 上海奕拓医药科技有限责任公司 2024-05-17 CN disclosed
CN-115335050-B Compounds and compositions for treating skin disorders 卡玛瑞制药有限公司 2024-05-17 CN disclosed
CN-114514223-B Process for enantioselective hydrogenation of 4-substituted 1, 2-dihydroquinolines comprising using novel iridium catalysts 拜耳公司 2024-05-17 CN disclosed
CN-118055699-A Formulation for antimicrobial thermosetting coatings 康宁公司 2024-05-17 CN disclosed
WO-2024102621-A1 AKT1 MODULATORS ALTEROME THERAPEUTICS, INC. (US) 2024-05-16 WO disclosed
WO-2024103012-A1 POLYCYCLIC COMPOUNDS FOR USE IN NEURODEGENERATIVE CONDITIONS IMET INC. (US) 2024-05-16 WO disclosed
US-20240156791-A1 METHODS OF TREATING SPINAL CORD INJURY OR DAMAGE SPINOGENIX INC (US) 2024-05-16 US disclosed
US-20240158394-A1 NEK7 INHIBITORS Halia Therapeutics, Inc. 2024-05-16 US disclosed
US-20240158385-A1 NOVEL COMPOUNDS Cerevance, Inc. 2024-05-16 US disclosed
US-20240156808-A1 Compositions and methods to improve the therapeutic benefit of suboptimally chemical compounds and biological therapies including substituted camptothecins such as irinotecan and topotecan for the treatment of benign and neoplastic hyperproliferative disease conditions, infections, inflammatory and immunological diseases EDISON ONCOLOGY (US) 2024-05-16 US disclosed
US-20240156999-A1 MULTIMERIC CHELATOR COMPOUNDS FOR USE IN TARGETED RADIOTHERAPY BAYER AKTIENGESELLSCHAFT (DE) 2024-05-16 US disclosed
WO-2024100276-A2 SUBSTITUTED 1,3-DIOXOLAN-4-ONES AND 1,3-DIOXAN-4-ONES AS FRAGRANCE INGREDIENTS BASF SE (DE) 2024-05-16 WO disclosed
US-20240158410-A1 CAMPTOTHECIN COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2024-05-16 US disclosed
EP-4366829-A1 PHENYL ACETAMIDE BASED IL-17A MODULATORS AND USES THEREOF Dice Alpha, Inc. (US) 2024-05-15 EP disclosed
CN-118043322-A PARP inhibitors containing nitrogen heterocyclic derivatives and uses thereof 西藏海思科制药有限公司 2024-05-14 CN disclosed
CN-111212647-B Dihydro oxadiazinones 拜耳股份有限公司 2024-05-14 CN disclosed
CN-118043306-A Lipid compounds and lipid nanoparticle compositions 苏州艾博生物科技有限公司 2024-05-14 CN disclosed
US-11980614-B2 2024-05-14 US disclosed
US-11981667-B2 Sulfonamide carboxamide compounds INFLAZOME LIMITED (IE) 2024-05-14 US disclosed
CN-118043314-A Benzazepine heteroaromatic ring derivative and application thereof in medicine 西藏海思科制药有限公司 2024-05-14 CN disclosed
CN-114728910-B Pyrazole derivative for FGFR inhibitor and preparation method thereof 上海奕拓医药科技有限责任公司 2024-05-14 CN disclosed
CN-118043323-A Bicyclic derivative PARP inhibitors and uses thereof 西藏海思科制药有限公司 2024-05-14 CN disclosed
CN-115516044-B Fluorescent dimer compounds useful as probes for detection of endogenous receptors 斯特拉斯堡大学 2024-05-14 CN disclosed
CN-118005610-A PARP-1 degrading agent and application thereof 西藏海思科制药有限公司 2024-05-10 CN disclosed
WO-2024094875-A1 CHROMEN-4-ONE COMPOUNDS WITH ANTICANCER PROPERTIES Floratek Pharma SA (CH) 2024-05-10 WO disclosed
CN-118019737-A Beta-lactam derivatives for the treatment of diseases 英矽智能科技知识产权有限公司 2024-05-10 CN disclosed
CN-118019740-A Heteroaryl derivative PARP inhibitors and uses thereof 海思科医药集团股份有限公司 2024-05-10 CN disclosed
WO-2024095005-A1 DIARYL DIAZOLE AND DIARYL TRIAZOLE DERIVATIVES FOR USE IN TREATING A DISEASE ASSOCIATED WITH KCNK13 ACTIVITY Cerevance, Inc. (US) 2024-05-10 WO disclosed
WO-2024095003-A1 NICOTINAMIDE DERIVATIVES FOR USE IN TREATING DISORDERS ASSOCIATED WITH KCNK13 ACTIVITY Cerevance, Inc. (US) 2024-05-10 WO disclosed
WO-2024097632-A1 METHODS OF REDUCING MIRO1 OR PHOSPHORYLATED ALPHA-SYNUCLEIN ACUREX BIOSCIENCES CORPORATION (US) 2024-05-10 WO disclosed
CN-118019727-A Methods for preparing NLRP3 inhibitors 豪夫迈·罗氏有限公司 2024-05-10 CN disclosed
US-20240150291-A1 PROCESS FOR THE PREPARATION OF NLRP3 INHIBITORS HOFFMANN-LA ROCHE INC. (US) 2024-05-09 US disclosed
US-20240150315-A1 BETA-2 ADRENORECEPTOR MODULATORS AND METHODS OF USING SAME THOMAS JEFFERSON UNIVERSITY 2024-05-09 US disclosed
US-20240150653-A1 ETCHANT COMPOSITIONS AND RELATED METHODS ENTEGRIS, INC. 2024-05-09 US disclosed
US-20240150380-A1 SILANE PRECURSORS AND RELATED METHODS ENTEGRIS, INC. 2024-05-09 US disclosed
US-20240150320-A1 QUATERNARY INDAZOLE GLUCOCORTICOID RECEPTOR ANTAGONISTS SYGNATURE DISCOVERY LIMITED (GB) 2024-05-09 US disclosed
US-20240150306-A1 COMPOUNDS WITH CLEAVABLE DISULFIDE MOIETIES REINVIGORON THERATECH, INC. 2024-05-09 US disclosed
EP-4013756-B1 MLL1 INHIBITORS AND ANTI-CANCER AGENTS NOVARTIS AG (CH) 2024-05-08 EP disclosed
EP-3852766-B1 COMBINATION THERAPY FOR TREATING BLOOD CANCER SIGNALCHEM LIFESCIENCES CORP (CA) 2024-05-08 EP disclosed
EP-4362929-A1 METHODS OF TREATING OR PREVENTING CORONAVIRUS INFECTION WITH CANNABINOID ACIDS Oregon State University (US) 2024-05-08 EP disclosed
CN-113354811-B Oxazoline polymer with side chain containing amino and/or hydroxyl, preparation method and application thereof 华东理工大学 2024-05-07 CN disclosed
US-11978894-B2 Silicon anodes with water-soluble maleic anhydride-, and/or maleic acid-containing polymers/copolymers, derivatives, and/or combinations (with or without additives) as binders ENEVATE CORPORATION (US) 2024-05-07 US disclosed
US-11976219-B2 Photo-cleavable primer compositions and methods of use ORMCO CORPORATION (US) 2024-05-07 US disclosed
CN-117999073-A Use of nadolol to treat chronic obstructive pulmonary disease by blocking the inhibitor protein-2 pathway 慢性呼吸道治疗有限公司 2024-05-07 CN disclosed
CN-117959303-A PIM kinase inhibitors for the treatment of myeloproliferative neoplasms and cancer-related fibrosis 住友制药肿瘤公司 2024-05-03 CN disclosed
CN-114391008-B Lipid compounds and lipid nanoparticle compositions 苏州艾博生物科技有限公司 2024-05-03 CN disclosed
CN-117980306-A Compound, pharmaceutical composition containing same and application of compound 中山优理生物医药有限公司 2024-05-03 CN disclosed
US-20240141382-A1 GENE EDITING COMPONENTS, SYSTEMS, AND METHODS OF USE RENAGADE THERAPEUTICS MANAGEMENT INC., 2024-05-02 US disclosed
US-20240140953-A1 INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, INC. 2024-05-02 US disclosed
WO-2024092185-A1 ACYL SULFONAMIDE COMPOUNDS AS INHIBITORS OF POLYOMAVIRUS VIA NOVA THERAPEUTICS, INC. (US) 2024-05-02 WO disclosed
WO-2024088379-A1 TUMOR TREATMENT OR PREVENTION METHOD 香港科技大学 2024-05-02 WO disclosed
WO-2024088069-A1 PREPARATION FOR AROMATIC KRAS MUTANT PROTEIN INHIBITOR AND USE THEREOF 药雅科技(上海)有限公司 2024-05-02 WO disclosed
US-20240140940-A1 CARBOXYLIC ACID, ACYL SULFONAMIDE AND ACYL SULFAMIDE-DERIVATIZED BICYCLIC AZA-HETEROAROMATICS AS SELECTIVE MCL-1 INHIBITORS AND AS DUAL MCL-1/BCL-2 INHIBITORS UNIVERSITY OF MARYLAND, BALTIMORE 2024-05-02 US disclosed
WO-2024088377-A1 PYRIMIDOPYRROLE ANALOG 香港科技大学 2024-05-02 WO disclosed
EP-4359389-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2024-05-01 EP disclosed
EP-4359413-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2024-05-01 EP disclosed
EP-4359385-A2 PROCESS FOR THE PREPARATION OF NLRP3 INHIBITORS F. Hoffmann-La Roche AG (CH) 2024-05-01 EP disclosed
EP-3753941-B1 PYRIMIDINE-FUSED CYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF SHANGHAI BLUERAY BIOPHARMA CO LTD (CN) 2024-05-01 EP disclosed
EP-4359411-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2024-05-01 EP disclosed
US-11970506-B2 Bioactive molecule conjugate, preparation method and use thereof SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2024-04-30 US disclosed
US-RE49948-E1 Aryl ethers and uses thereof PELOTON THERAPEUTICS, INC. (US) 2024-04-30 US disclosed
US-11970497-B2 Tricyclic AKR1C3 dependent KARS inhibitors NOVARTIS AG (CH) 2024-04-30 US disclosed
US-11970552-B2 Nicotinic acetylcholine receptor peptide antagonist conotoxin compositions and related methods GLO PHARMA, INC. (US) 2024-04-30 US disclosed
US-11970731-B2 Enhancement of nucleic acid polymerization by aromatic compounds Roche Sequencing Solutions, Inc. (US) 2024-04-30 US disclosed
US-11969472-B2 Tropomyosin receptor kinase (TRK) degradation compounds and methods of use CULLGEN (SHANGHAI), INC. (CN) 2024-04-30 US disclosed
CN-117956990-A Compositions and methods for treating lipomatous pain 拉结尔治疗有限公司 2024-04-30 CN disclosed
CN-117957212-A IL-17A modulators based on phenylacetamide and uses thereof 戴斯阿尔法公司 2024-04-30 CN disclosed
CN-110769689-B Novel supercooling method for preserving biological samples 先时迈纳米生物科技股份有限公司 2024-04-26 CN disclosed
WO-2024086814-A2 CYCLIN INHIBITORS CIRCLE PHARMA, INC. (US) 2024-04-25 WO disclosed
WO-2024086614-A2 TARGETED LNP-MRNA WITH MINIMAL OFF-TARGET EXPRESSION AND METHODS OF USE THEREOF THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2024-04-25 WO disclosed
WO-2024086744-A2 COMPOSITIONS AND USES THEREOF SOLVE THERAPEUTICS, INC. (US) 2024-04-25 WO disclosed
US-20240131150-A1 NUCLEIC ACID VACCINES FOR CORONAVIRUS SUZHOU ABOGEN BIOSCIENCES CO LTD (CN) 2024-04-25 US disclosed
US-20240131181-A1 Therapeutic Targeting of Lipid Nanoparticles THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2024-04-25 US disclosed
WO-2024083172-A1 LIPID COMPOUND AND LIPID NANOPARTICLE COMPOSITION 苏州艾博生物科技有限公司 2024-04-25 WO disclosed
WO-2024083171-A1 LIPID COMPOUND AND LIPID NANOPARTICLE COMPOSITION 苏州艾博生物科技有限公司 2024-04-25 WO disclosed
US-20240132497-A1 AZABICYCLO AND DIAZEPINE DERIVATIVES ALCON INC. (CH) 2024-04-25 US disclosed
US-20240132484-A1 BROAD SPECTRUM ANTIVIRAL COMPOUNDS TARGETING THE SKI COMPLEX UNIVERSITY OF MARYLAND, BALTIMORE 2024-04-25 US disclosed
US-20240132461-A1 FLAVONE DEAZA SPERMIDINE ANALOGUES AND THEIR USE TREATING CANCER FLORATEK PHARMA S A (CH) 2024-04-25 US disclosed
WO-2024083671-A1 BROMINE- OR IODINE-PARA-SUBSTITUTED [(1,5-DIPHENYL-1H-1,2,4-TRIAZOL-3-YL)OXY]ACETIC ACID DERIVATIVES AND SALTS THEREOF, PROTECTION AGENTS COMPRISING THEM, FOR USEFUL PLANTS OR CROP PLANTS, METHODS FOR PRODUCING THEM AND USE THEREOF AS SAFENERS BAYER AKTIENGESELLSCHAFT (DE) 2024-04-25 WO disclosed
WO-2024084028-A1 PYRIDINE COMPOUNDS FOR COMBATTING DIHYDROOROTATE-DEHYDROGENASE INHIBITOR-RESISTANT PHYTOPATHOGENIC FUNGI BASF SE (DE) 2024-04-25 WO disclosed
US-20240130994-A1 IONIC LIQUID FORMULATIONS FOR TREATING DIABETES I2O THERAPEUTICS, INC. 2024-04-25 US disclosed
US-20240132493-A1 IMIDAZOPYRIDINE DERIVATIVES AS STING AGONISTS FULGENT GENETICS INC (US) 2024-04-25 US disclosed
US-20240130969-A1 LIPID NANOPARTICLES AND METHODS OF USE THEREOF RENAGADE THERAPEUTICS MANAGEMENT INC. 2024-04-25 US disclosed
US-20240131035-A1 AQUEOUS PHARMACEUTICAL FORMULATION OF HYDROCORTISONE SODIUM PHOSPHATE AND MONOTHIOGLYCEROL ANTARES PHARMA, INC. (US) 2024-04-25 US disclosed
WO-2024083670-A2 BROMINE- OR IODINE-PARA-SUBSTITUTED [(1,5-DIPHENYL-1H-1,2,4-TRIAZOL-3-YL)OXY]ACETIC ACID DERIVATIVES AND THEIR SALTS, AGENTS FOR PROTECTING USEFUL PLANTS OR CROP PLANTS COMPRISING THEM, METHODS FOR PRODUCING THEM AND THEIR USE AS SAFENERS BAYER AKTIENGESELLSCHAFT (DE) 2024-04-25 WO disclosed
WO-2024083024-A1 PREPARATION AND USE OF RET INHIBITOR 药雅科技(上海)有限公司 2024-04-25 WO disclosed
EP-4357020-A2 ASYMMETRIC PHASE TRANSFER CATALYSIS Merck Sharp & Dohme LLC (US) 2024-04-24 EP disclosed
US-11964052-B2 Lipid compounds and lipid nanoparticle compositions Suzhou Abogen Biosciences Co., Ltd. (CN) 2024-04-23 US disclosed
CN-114685487-B Pyrimidine heterocyclic compounds, preparation method and application 上海凌达生物医药有限公司 2024-04-19 CN disclosed
CN-117903016-A Fluorosulfonyl sulfonimide salt, preparation method and application thereof 中国科学院上海有机化学研究所 2024-04-19 CN disclosed
WO-2024079468-A1 COMPOUNDS FOR USE AS MEDICAMENTS CHARIOT INNOVATIONS LTD (GB) 2024-04-18 WO disclosed
WO-2024078906-A1 SUBSTITUTED N-PHENYLURACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2024-04-18 WO disclosed
WO-2024078263-A1 PREPARATION AND USE OF MACROCYCLIC HETEROCYCLIC COMPOUND AS EGFR INHIBITOR 药雅科技(上海)有限公司 2024-04-18 WO disclosed
US-20240122854-A1 NOVEL CARBONYL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS ACUITAS THERAPEUTICS INC (CA) 2024-04-18 US disclosed
US-20240124413-A1 COMPOUNDS AND COMPOSITIONS FOR USE IN TREATING SKIN DISORDERS KAMARI PHARMA LTD. (IL) 2024-04-18 US disclosed
US-20240124467-A1 FUSED PYRIMIDINE COMPOUNDS AS INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, INC. 2024-04-18 US disclosed
US-20240125773-A1 COMPOSITIONS AND METHODS FOR PREVENTING NON-SPECIFIC INTERACTIONS BETWEEN POLYMER DYES-ANTIBODY CONJUGATES BECKMAN COULTER, INC. 2024-04-18 US disclosed
WO-2024081789-A2 HISTONE DEMETHYLASE INHIBITORS FOR TREATING CANCERS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-04-18 WO disclosed
WO-2024081653-A2 METHODS OF LOWERING MIRO2 TO TREAT NEURODEGENERATIVE DISEASES ACUREX BIOSCIENCES CORPORATION (US) 2024-04-18 WO disclosed
WO-2024079252-A1 SOS1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2024-04-18 WO disclosed
US-20240124645-A1 COMPOSITION FOR REVERSIBLE POLYMERIZATION OF THIOESTER AND METHODS THEREOF UNIV COLORADO REGENTS (US) 2024-04-18 US disclosed
US-20240124503-A1 HETEROAROMATIC PHOSPHONIUM SALTS AND THEIR USE TREATING CANCER FLORATEK PHARMA S A (CH) 2024-04-18 US disclosed
EP-4351651-A1 LIPID NANOPARTICLES AND METHODS OF USE THEREOF Renagade Therapeutics Management Inc. (US) 2024-04-17 EP disclosed
EP-3893645-B1 SUBSTITUTED ARYLMETHYLUREAS AND HETEROARYLMETHYLUREAS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORP (CA) 2024-04-17 EP disclosed
EP-4353310-A2 FATTY LIVER DISEASE TREATMENT USING GLUCOCORTICOID AND MINERALOCORTICOID RECEPTOR ANTAGONISTS Corcept Therapeutics Incorporated (US) 2024-04-17 EP disclosed
EP-4353082-A1 HERBICIDAL COMPOSITIONS Bayer Aktiengesellschaft (DE) 2024-04-17 EP disclosed
EP-4352062-A2 5-HT2A AND/OR 5-HT2C RECEPTOR AGONISTS Diamond Therapeutics Inc. (CA) 2024-04-17 EP disclosed
EP-4351620-A1 CELL-PERMEABLE CYCLIC PEPTIDES AND USES THEREOF Unnatural Products Inc. (US) 2024-04-17 EP disclosed
EP-3737376-B1 SELECTIVE HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF HUMAN DISEASES SHUTTLE PHARMACEUTICALS INC (US) 2024-04-17 EP disclosed
CN-117897385-A Compound for degrading Bcl-2 family proteins and application of compound in medicine 西藏海思科制药有限公司 2024-04-16 CN disclosed
CN-113262175-B Skin care compositions and methods of use thereof 尤尼根公司 2024-04-16 CN disclosed
US-11958850-B2 Heteroaryl compounds for kinase inhibition TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2024-04-16 US disclosed
US-11961967-B2 Silicon-based energy storage devices with phosphorus containing electrolyte additives ENEVATE CORPORATION (US) 2024-04-16 US disclosed
US-11958854-B2 Substituted xanthines and methods of use thereof HYDRA BIOSCIENCES, LLC (US) 2024-04-16 US disclosed
US-11958833-B2 Compounds MISSION THERAPEUTICS LIMITED (GB) 2024-04-16 US disclosed
CN-117881795-A Methods and compositions for identifying methylated cytosines 因美纳有限公司 2024-04-12 CN disclosed
WO-2024077009-A1 FUNCTIONALIZED MACROMOLECULES AND SYSTEMS, METHODS OF SYNTHESIS, AND USES THEREOF SEER, INC. (US) 2024-04-11 WO disclosed
US-20240116877-A1 KIT KINASE INHIBITORS AND METHODS OF USE THEREOF DECIPHERA PHARMACEUTICALS, LLC 2024-04-11 US disclosed
US-20240117306-A1 METHOD OF INHIBITING TAU PHOSPHORYLATION CASSAVA SCIENCES, INC. (US) 2024-04-11 US disclosed
US-20240116946-A1 SARS-COV2 MAIN PROTEASE INHIBITORS GILEAD SCIENCES, INC. 2024-04-11 US disclosed
US-20240116928-A1 CD73 COMPOUNDS GILEAD SCIENCES, INC. 2024-04-11 US disclosed
WO-2024077057-A1 PHENYL OXY AMIDE KINASE INHIBITORS THE TRANSLATIONAL GENOMICS RESEARCH INSTITUTE (US) 2024-04-11 WO disclosed
US-20240116899-A1 BETA-LACTAM DERIVATIVES FOR THE TREATMENT OF DISEASES INSILICO MEDICINE IP LIMITED (HK) 2024-04-11 US disclosed
US-20240116949-A1 SPIRO AROMATIC RING COMPOUND AND USE THEREOF ETERN BIOPHARMA SHANGHAI CO LTD (CN) 2024-04-11 US disclosed
WO-2024074641-A1 METHOD FOR PREPARING AMIDES FROM ESTERS BASF SE (DE) 2024-04-11 WO disclosed
EP-3368556-B1 NOVEL POLYPEPTIDES WITH IMPROVED PROTEOLYTIC STABILITY, AND METHODS OF PREPARING AND USING SAME UNIV TUFTS (US) 2024-04-10 EP disclosed
EP-4347603-A1 SULFUR-CONTAINING HETEROAROMATIC TRICYCLIC KRAS INHIBITORS Erasca, Inc. (US) 2024-04-10 EP disclosed
EP-4349833-A1 PYRIDAZINONE COMPOUND AS PARP7 INHIBITOR Euregen Biopharma Co., Ltd. (CN) 2024-04-10 EP disclosed
EP-4349839-A2 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS Novartis AG (CH) 2024-04-10 EP disclosed
EP-4347607-A1 PENICILLIN-BINDING PROTEIN INHIBITORS Venatorx Pharmaceuticals, Inc. (US) 2024-04-10 EP disclosed
CN-117843567-A Diazaaryl ring substituted benzene derivatives, compositions and uses thereof 康迈迪森(北京)医药科技有限公司 2024-04-09 CN disclosed
CN-117838695-A PIM kinase inhibitors for the treatment of myeloproliferative neoplasms and cancer-related fibrosis 住友制药肿瘤公司 2024-04-09 CN disclosed
CN-117843566-A Polysubstituted benzene derivative, composition and use thereof 康迈迪森(北京)医药科技有限公司 2024-04-09 CN disclosed
CN-112638898-B Heteroaryl substituted sulfonamide compounds and their use as sodium channel inhibitors 泽农医药公司 2024-04-09 CN disclosed
US-11951100-B2 Formulations of RBP4 inhibitors and methods of use BELITE BIO, LLC (US) 2024-04-09 US disclosed
CN-117858881-A Phospholipid compounds and methods of making and using the same 吉利德科学公司 2024-04-09 CN disclosed
CN-115043841-B Preparation and application of heterocyclic compound serving as BTK inhibitor 药雅科技(上海)有限公司 2024-04-09 CN disclosed
CN-117836289-A Tropomyosin Receptor Kinase (TRK) degrading compounds and methods of use thereof 上海睿跃生物科技有限公司 2024-04-05 CN disclosed
CN-115181106-B Quinazoline KRAS G12D Preparation and application of mutant protein inhibitor 药雅科技(上海)有限公司 2024-04-05 CN disclosed
CN-117826534-A Method for forming semiconductor device 台湾积体电路制造股份有限公司 2024-04-05 CN disclosed
CN-117820305-A Heterocyclic substituted quinazoline and preparation method and application thereof 苏州泽璟生物制药股份有限公司 2024-04-05 CN disclosed
WO-2024073371-A1 AKT1 MODULATORS ALTEROME THERAPEUTICS, INC. (US) 2024-04-04 WO disclosed
WO-2024073426-A1 1,4-DIHYDROQUINAZOLINONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. (US) 2024-04-04 WO disclosed
WO-2024073410-A1 TERNARY SOLVENT ELECTROLYTES FOR HIGH VOLTAGE AND HIGH RATE LITHIUM BATTERIES SEPION TECHNOLOGIES, INC. (US) 2024-04-04 WO disclosed
WO-2024069448-A1 SUBSTITUTED 1-ARYLAMINOCARBONYL-1'-HETEROARYL COMPOUNDS, SUBSTITUTED 1-HETEROARYLAMINOCARBONYL-1'-HETEROARYL COMPOUNDS AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2024-04-04 WO disclosed
WO-2024067744-A1 HETEROCYCLIC SUBSTITUTED QUINAZOLINE, PREPARATION METHOD THEREFOR, AND USE THEREOF 苏州泽璟生物制药股份有限公司 2024-04-04 WO disclosed
WO-2024067401-A1 ULTRA-LONG-ACTING PLATFORM COMPRISING FC-ADVANCED FATTY ACID CHAIN 中美华世通生物医药科技(武汉)股份有限公司 2024-04-04 WO disclosed
US-20240108745-A1 BIOACTIVE SUBSTANCE CONJUGATE, PREPARATION METHOD THEREFOR AND USE THEREOF MEDILINK THERAPEUTICS (SUZHOU) CO., LTD. (CN) 2024-04-04 US disclosed
US-20240109927-A1 BIS (ARENE) METAL COMPLEXES AND RELATED METHODS ENTEGRIS, INC. 2024-04-04 US disclosed
US-20240109896-A1 FGFR KINASE INHIBITOR AND USE THEREOF YA THERAPEUTICS INC (CN) 2024-04-04 US disclosed
US-20240109913-A1 NEW SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2024-04-04 US disclosed
US-20240109891-A1 NOVEL SUBSTITUTED TRICYCLIC AZA-HETEROCYCLES AS SOS1 INHIBITORS VIVA STAR BIOSCIENCES (SUZHOU) CO., LTD. (CN) 2024-04-04 US disclosed
US-20240109887-A1 NOVEL SUBSTITUTED BICYCLIC AZA-HETEROCYCLES AS SOS1 INHIBITORS VIVA STAR BIOSCIENCES (SUZHOU) CO., LTD. (CN) 2024-04-04 US disclosed
WO-2024073610-A2 COMPOSITIONS AND USES THEREOF SOLVE THERAPEUTICS, INC. (US) 2024-04-04 WO disclosed
WO-2024073436-A2 COMPOSITIONS AND USES THEREOF SOLVE THERAPEUTICS, INC. (US) 2024-04-04 WO disclosed
WO-2024072908-A1 COMPOUNDS WITH CLEAVABLE DISULFIDE MOIETIES REINVIGORON THERATECH, INC. (US) 2024-04-04 WO disclosed
EP-3206692-B1 FATTY LIVER DISEASE TREATMENT USING GLUCOCORTICOID AND MINERALOCORTICOID RECEPTOR ANTAGONISTS CORCEPT THERAPEUTICS INC (US) 2024-04-03 EP disclosed
CN-117813288-A Arylamino derivative estrogen receptor modulator and use thereof 西藏海思科制药有限公司 2024-04-02 CN disclosed
US-11949072-B2 Silicon-based energy storage devices with electrolyte containing cyanate based compounds ENEVATE CORPORATION (US) 2024-04-02 US disclosed
US-11945785-B2 Pyrazine compounds as inhibitors of FLT3 BIOMEA FUSION, INC. (US) 2024-04-02 US disclosed
US-11945797-B2 1-cyano-pyrrolidine derivatives as dub inhibitors MISSION THERAPEUTICS LIMITED (GB) 2024-04-02 US disclosed
US-11945890-B2 Fluorinated PVC copolymer compositions for increased ultraviolet protection Mexichem Specialty Resins Inc. (US) 2024-04-02 US disclosed
US-11945812-B2 Annulated 2-amino-3-cyano thiophenes and derivatives for the treatment of cancer BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2024-04-02 US disclosed
CN-117800976-A Nitrogen-containing heterocyclic compound, preparation method and application 上海凌达生物医药有限公司 2024-04-02 CN disclosed
CN-117794929-A Selective BCL-XL PROTAC compounds and methods of use 法国施维雅药厂 2024-03-29 CN disclosed
CN-112469720-B Dual ATM and DNA-PK inhibitors for use in anti-tumor therapy 艾科思莱德制药公司 2024-03-29 CN disclosed
CN-114072207-B Bicyclic compounds 维瓦斯治疗公司 2024-03-29 CN disclosed
US-20240101544-A1 INHIBITORS OF QPCTL AND QPCT 858 THERAPEUTICS, INC. 2024-03-28 US disclosed
US-20240101535-A1 DIHYDROISOQUINOLINONE DERIVATIVE AND APPLICATION THEREOF ETERN BIOPHARMA (SHANGHAI) CO., LTD. (CN) 2024-03-28 US disclosed
WO-2024064701-A2 ADENOSINE ANALOGS FOR THE TREATMENT OF DISEASE BIOINTERVENE, INC. (US) 2024-03-28 WO disclosed
US-20240101531-A1 PYRIDINAMINE DERIVATIVES AND THEIR USE AS POTASSIUM CHANNEL MODULATORS XENON PHARMACEUTICALS INC. (CA) 2024-03-28 US disclosed
WO-2024064026-A1 AKT1 MODULATORS ALTEROME THERAPEUTICS, INC. (US) 2024-03-28 WO disclosed
US-20240100170-A1 CYCLIC-AMP RESPONSE ELEMENT BINDING PROTEIN (CBP) AND/OR ADENOVIRAL E1A BINDING PROTEIN OF 300 KDA (P300) DEGRADATION COMPOUNDS AND METHODS OF USE CULLGEN (SHANGHAI) , INC. (CN) 2024-03-28 US disclosed
US-20240101585-A1 HETEROAROMATIC PHOSPHONIUM SALTS AND THEIR USE TREATING CANCER FLORATEK PHARMA AG (CH) 2024-03-28 US disclosed
EP-3615510-B1 NOVEL CARBONYL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS ACUITAS THERAPEUTICS INC (CA) 2024-03-27 EP disclosed
EP-4340701-A1 BIOMARKERS FOR AGE-RELATED MACULAR DEGENERATION Belite Bio, LLC (US) 2024-03-27 EP disclosed
US-11942599-B2 Symmetrical or asymmetrical alkylsulfonyl imide or cyclic alkylene sulfonylimide salts as cathode additives, electrolyte additives, or SI anode additives for SI anode-based li-ion cells ENEVATE CORPORATION (US) 2024-03-26 US disclosed
US-11939335-B2 Substituted imidazo[1,2-a]quinazolines and imidazo [1,2-a]pyrido[4,3-e]pyrimidines as inhibitors of PARG 858 THERAPEUTICS, INC. (US) 2024-03-26 US disclosed
US-11939474-B2 Water soluble fluorescent or colored dyes and methods for their use Sony Group Corporation (JP) 2024-03-26 US disclosed
CN-117751106-A Novel triazole-pyridine substituted pyrrolidinyl and tetrahydro-2H-pyranylacetic acid compounds as LPA antagonists 唯久生物技术(苏州)有限公司 2024-03-22 CN disclosed
CN-117736178-A Dual MAGL and FAAH inhibitors 灵北拉荷亚研究中心公司 2024-03-22 CN disclosed
CN-117736207-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-03-22 CN disclosed
CN-115448923-B Pyrimidine-fused ring compound, preparation method and application thereof 上海青煜医药科技有限公司 2024-03-22 CN disclosed
CN-115362003-B Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-03-22 CN disclosed
US-20240092761-A1 QUINAZOLINE COMPOUNDS AND METHODS OF USE IAMBIC THERAPEUTICS, INC. 2024-03-21 US disclosed
US-20240092756-A1 METHODS AND COMPOSITION FOR KRAS MODIFICATIONS DUNAD THERAPEUTICS LTD. (GB) 2024-03-21 US disclosed
WO-2024056782-A1 SULFONE-SUBSTITUTED PYRIDO[3,4-D]PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF CANCER BAYER AKTIENGESELLSCHAFT (DE) 2024-03-21 WO disclosed
US-20240092788-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION (US) 2024-03-21 US disclosed
US-20240092810-A1 COMPOSITIONS FOR EXTREME ULTRAVIOLET LITHOGRAPHY AND RELATED METHODS ENTEGRIS, INC. 2024-03-21 US disclosed
US-20240092746-A1 OPIOID RECEPTOR MODULATORS EPIODYNE, INC. 2024-03-21 US disclosed
WO-2024059200-A1 NEK7 INHIBITORS Halia Therapeutics, Inc. (US) 2024-03-21 WO disclosed
WO-2024059085-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF INFLAMMATORY DISEASES INVEA THERAPEUTICS, INC. (US) 2024-03-21 WO disclosed
WO-2024059041-A1 BENZO-FUSED N-HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES, INC. (US) 2024-03-21 WO disclosed
EP-3641741-B1 MICROTUBULE POLYMERIZATION INHIBITOR PRODRUGS AND METHODS OF USING THE SAME UNIV MARYLAND (US) 2024-03-20 EP disclosed
EP-3609906-B1 NOVEL PEPTOID POLYMERS AND METHODS OF USE X THERMA INC (US) 2024-03-20 EP disclosed
US-11931347-B2 Method of screening for agents for differentiating stem cells MINERVA BIOTECHNOLOGIES CORPORATION (US) 2024-03-19 US disclosed
US-11932634-B2 Diacylglycerol kinase modulating compounds GILEAD SCIENCES, INC. (US) 2024-03-19 US disclosed
CN-117730082-A Synthesis of substituted tricyclic amides and analogs thereof 爱彼特生物制药公司 2024-03-19 CN disclosed
CN-117720517-A AR inhibitor, composition thereof and pharmaceutical application thereof 西藏海思科制药有限公司 2024-03-19 CN disclosed
CN-108137482-B Prodrugs of directed lymphatics 莫纳什大学 2024-03-15 CN disclosed
US-20240084074-A1 NOVEL PEPTOID POLYMERS AND METHODS OF USE X-THERMA, INC. (US) 2024-03-14 US disclosed
US-20240084308-A1 FIBROTIC TREATMENT MONASH UNIVERSITY (AU) 2024-03-14 US disclosed
US-20240084274-A1 GENE EDITING COMPONENTS, SYSTEMS, AND METHODS OF USE RENAGADE THERAPEUTICS MANAGEMENT INC. (US) 2024-03-14 US disclosed
US-20240083855-A1 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE SUMITOMO PHARMA AMERICA, INC. (US) 2024-03-14 US disclosed
US-20240084043-A1 METHODS OF TREATING AN EYE DISORDER KODIAK SCIENCES INC. 2024-03-14 US disclosed
WO-2024054387-A1 BIS (ARENE) METAL COMPLEXES AND RELATED METHODS ENTEGRIS, INC. (US) 2024-03-14 WO disclosed
US-20240083857-A1 2-Methyl-Quinazolines Bayer Pharma AG (DE) 2024-03-14 US disclosed
WO-2024054512-A1 AKT1 MODULATORS ALTEROME THERAPEUTICS, INC. (US) 2024-03-14 WO disclosed
US-20240084193-A1 METAL OXIDE, METAL BRONZE AND POLYOXOMETALATE AS CHARGE STORAGE MATERIALS IN ELECTROCHROMIC DEVICE Furcifer Inc. (US) 2024-03-14 US disclosed
EP-4335848-A2 DUAL MAGL AND FAAH INHIBITORS Lundbeck La Jolla Research Center, Inc. (US) 2024-03-13 EP disclosed
EP-4090655-B1 PROCESS FOR PREPARING CYCLIC CARBONATES WITH AN EXOCYCLIC VINYLIDENE GROUP BASF SE (DE) 2024-03-13 EP disclosed
CN-117693353-A Cell-permeable cyclic peptides and uses thereof 安奈彻产品股份有限公司 2024-03-12 CN disclosed
CN-116064598-B Nucleic acid vaccine for coronavirus 苏州艾博生物科技有限公司 2024-03-12 CN disclosed
US-11926600-B2 Sulfonylureas and sulfonylthioureas as NLRP3 inhibitors INFLAZOME LIMITED (IE) 2024-03-12 US disclosed
US-11926628-B2 Diacylglyercol kinase modulating compounds GILEAD SCIENCES, INC. (US) 2024-03-12 US disclosed
CN-117693511-A Penicillin binding protein inhibitors 维纳拓尔斯制药公司 2024-03-12 CN disclosed
CN-117659007-A Pyrazinone derivative and application thereof in medicine 西藏海思科制药有限公司 2024-03-08 CN disclosed
CN-110267944-B Compounds useful for the treatment of gastrointestinal disorders 阿德利克斯股份有限公司 2024-03-08 CN disclosed
US-20240076306-A1 MODULATORS OF TNF-ALPHA ACTIVITY FORWARD THERAPEUTICS, INC. 2024-03-07 US disclosed
US-20240076314-A1 PEPTIDE COMPOSITIONS AND METHODS FOR INHIBITING NICOTINIC ACETYLCHOLINE RECEPTOR ACTIVITY GLO PHARMA, INC. 2024-03-07 US disclosed
US-20240075163-A1 NOVEL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS ACUITAS THERAPEUTICS INC (CA) 2024-03-07 US disclosed
US-20240079653-A1 Electrolyte Formulations for Optimal Performance in Si-Containing Lithium Ion Batteries ENEVATE CORPORATION 2024-03-07 US disclosed
WO-2024049979-A2 NOVEL IONIZABLE LIPIDS AND LIPID NANOPARTICLES AND METHODS OF USING THE SAME SENDA BIOSCIENCES, INC. (US) 2024-03-07 WO disclosed
WO-2024049919-A1 COMPOSITIONS FOR EXTREME ULTRAVIOLET LITHOGRAPHY AND RELATED METHODS ENTEGRIS, INC. (US) 2024-03-07 WO disclosed
EP-4329816-A1 LIPID NANOPARTICLE THERAPEUTICS THAT EVADE THE IMMUNE RESPONSE The Trustees of the University of Pennsylvania (US) 2024-03-06 EP disclosed
EP-4330249-A1 NOVEL TRIAZOLE-PYRIDINE SUBSTITUTED PYRROLIDINYL AND TETRAHYDRO-2H-PYRANYL ACETIC ACID COMPOUNDS AS LPA ANTAGONISTS Viva Star Biosciences (Suzhou) Co., Ltd. (CN) 2024-03-06 EP disclosed
EP-4331669-A2 SELECTIVE P2X3 ANTAGONISTS FOR USE IN TREATING CHRONIC COUGH WITHOUT LOSS OF TASTE RESPONSE Bellus Health Inc. (CA) 2024-03-06 EP disclosed
EP-4330391-A1 COMPOSITIONS AND METHODS FOR TARGETING LIPID NANOPARTICLE THERAPEUTICS TO STEM CELLS The Trustees of the University of Pennsylvania (US) 2024-03-06 EP disclosed
EP-4329776-A1 CD-90 TARGETED LIPID NANOPARTICLES The Trustees of the University of Pennsylvania (US) 2024-03-06 EP disclosed
EP-4330234-A1 SUBSTITUTED PYRIDAZINONES, SALTS OR N-OXIDES THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES Bayer Aktiengesellschaft (DE) 2024-03-06 EP disclosed
EP-3615537-B1 6-6 FUSED BICYCLIC HETEROARYL COMPOUNDS AND THEIR USE AS LATS INHIBITORS NOVARTIS AG (CH) 2024-03-06 EP disclosed
EP-4330245-A1 NOVEL HETEROCYCLIC COMPOUNDS Floratek Pharma SA (CH) 2024-03-06 EP disclosed
EP-3512840-B1 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS TSENG YUFENG JANE (US) 2024-03-06 EP disclosed
EP-3691642-B1 [1,6]NAPHTHYRIDINE COMPOUNDS AND DERIVATIVES AS CDK8/CDK19 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2024-03-06 EP disclosed
US-11919869-B2 CD73 compounds GILEAD SCIENCES, INC. (US) 2024-03-05 US disclosed
US-11918951-B2 MOF compositions for selective separation of hydrocarbons RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2024-03-05 US disclosed
US-11923545-B2 Crown ethers as additives for silicon-based Li-ion batteries ENEVATE CORPORATION (US) 2024-03-05 US disclosed
US-11923506-B2 Silicon-based energy storage devices with ether containing electrolyte additives ENEVATE CORPORATION (US) 2024-03-05 US disclosed
US-11919972-B2 Peptide libraries with non-canonical amino acids REGENERON PHARMACEUTICALS, INC. (US) 2024-03-05 US disclosed
US-11919865-B2 Processes for preparing AG-10, its intermediates, and salts thereof Eidos Therapeutics, Inc. (US) 2024-03-05 US disclosed
CN-117651549-A Anti-angiogenic agents and related methods 新加坡科技研究局 2024-03-05 CN disclosed
CN-117651701-A Novel substituted bicyclic aza heterocycles as SOS1 inhibitors 唯久生物技术(苏州)有限公司 2024-03-05 CN disclosed
CN-117642397-A Modified proteins and protein binders 上海睿跃生物科技有限公司 2024-03-01 CN disclosed
CN-112739349-B Combination therapy for the treatment of hematological cancers 圣诺康生命科学公司 2024-03-01 CN disclosed
US-20240067625-A1 SMALL-MOLECULE MODULATORS OF THE ORPHAN NUCLEAR RECEPTOR TLX BAYLOR COLLEGE OF MEDICINE (US) 2024-02-29 US disclosed
US-20240066136-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS CULLGEN (SHANGHAI), INC. (CN) 2024-02-29 US disclosed
US-20240067623-A1 [(1-PHENYL-5-HETEROARYL-1H-PYRAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2024-02-29 US disclosed
WO-2024041976-A1 PROCESS FOR DISTILLATIVE RECOVERY OF 1,1,1,3,3,3-HEXAFLUORO-2-PROPANOL (HFIP) FROM MIXTURES WITH 4- SUBSTITUTED 1,2,3,4-TETRAHYDROQUINOLINES BAYER AKTIENGESELLSCHAFT (DE) 2024-02-29 WO disclosed
WO-2024044327-A1 DHNT MONOMERS AND POLYMER DYES WITH MODIFIED PHOTOPHYSICAL PROPERTIES BECKMAN COULTER, INC. (US) 2024-02-29 WO disclosed
US-20240067626-A1 INHIBITORS OF MET KINASE CELYN THERAPEUTICS, INC. 2024-02-29 US disclosed
WO-2024044728-A1 PEGYLATED LIPID COMPOUNDS AND METHODS OF USE THEREOF RENAGADE THERAPEUTICS MANAGEMENT INC. (US) 2024-02-29 WO disclosed
EP-3294811-B1 ULTRA BRIGHT DIMERIC OR POLYMERIC DYES SONY GROUP CORP (JP) 2024-02-28 EP disclosed
EP-3705480-B1 CLASS OF AMINO-SUBSTITUTED NITROGEN-CONTAINING FUSED RING COMPOUNDS, PREPARATION METHOD THEREFOR, AND USE THEREOF SHANGHAI RINGENE BIOPHARMA CO LTD (CN) 2024-02-28 EP disclosed
EP-4327877-A2 DUAL ATM AND DNA-PK INHIBITORS FOR USE IN ANTI-TUMOR THERAPY XRad Therapeutics, Inc. (US) 2024-02-28 EP disclosed
US-11912784-B2 Methods of treating an eye disorder KODIAK SCIENCES INC. (US) 2024-02-27 US disclosed
US-11912723-B2 KRAS modulators and uses thereof QUANTA THERAPEUTICS, INC. (US) 2024-02-27 US disclosed
US-11912708-B2 Macrocyclic heterocycles and uses thereof KUMQUAT BIOSCIENCES INC. (US) 2024-02-27 US disclosed
US-11911751-B2 Catalyst compositions for hydroformylation and methods of use thereof BOARD OF SUPERVISORS OF LOUISIANA STATE UNIVERSITY AND AGRICULTURAL AND MECHANICAL COLLEGE (US) 2024-02-27 US disclosed
US-11911392-B2 Non-catalytic substrate-selective p38α-specific MAPK inhibitors with endothelial-stabilizing and anti-inflammatory activity, and methods of use thereof UNIVERSITY OF MARYLAND, BALTIMORE (US) 2024-02-27 US disclosed
US-11911393-B2 Non-catalytic substrate-selective p38alpha-specific MAPK inhibitors with endothelial-stabilizing and anti-inflammatory activity, and methods of use thereof UNIVERSITY OF MARYLAND, BALTIMORE (US) 2024-02-27 US disclosed
CN-117597345-A Heterocyclic derivatives as CaMKK2 inhibitors 百时美施贵宝公司 2024-02-23 CN disclosed
CN-117597346-A NEK7 inhibitors 哈利亚治疗公司 2024-02-23 CN disclosed
WO-2024038356-A1 SYNTHESIS OF SUBSTITUTED 1-ARYL-1'-HETEROARYL COMPOUNDS AND SUBSTITUTED 1,1'-BIHETEROARYL COMPOUNDS, AND ANALOGUES THEREOF ARBUTUS BIOPHARMA CORPORATION (CA) 2024-02-22 WO disclosed
US-20240059671-A1 TYROSINE KINASE 2 (TYK2) DEGRADATION COMPOUNDS AND METHODS OF USE CULLGEN (SHANGHAI) , INC. (CN) 2024-02-22 US disclosed
WO-2024038357-A1 SYNTHESIS OF SUBSTITUTED TETRACYCLIC CARBOXYLIC ACIDS AND ANALOGUES THEREOF ARBUTUS BIOPHARMA CORPORATION (CA) 2024-02-22 WO disclosed
EP-4324825-A1 FXR REGULATOR, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF Beijing Best Pathway Management Consulting Center (Limited Partnership) (CN) 2024-02-21 EP disclosed
EP-4322962-A1 PHOSPHORUS DERIVATIVES AS NOVEL SOS1 INHIBITORS Bayer Aktiengesellschaft (DE) 2024-02-21 EP disclosed
EP-4323399-A1 METHODS OF TREATING AN EYE DISORDER Kodiak Sciences Inc. (US) 2024-02-21 EP disclosed
EP-3762365-B1 METHODS AND COMPOSITIONS OF ISOINDOLINE-1,3-DIONE AND ISOINDOLE PRODRUGS USEFUL FOR TREATING CANCER, ULCERATIVE COLITIS AND RELATED INFLAMMATORY DISEASES AMGEN EUROPE GMBH (CH) 2024-02-21 EP disclosed
EP-4323359-A2 TETRACYCLIC COMPOUNDS FOR TREATING BRAIN DISORDERS The Regents of the University of California (US) 2024-02-21 EP disclosed
CN-117580587-A Coronavirus nucleic acid vaccine based on sequences derived from SARS-CoV-2 Omikovia strain 苏州艾博生物科技有限公司 2024-02-20 CN disclosed
CN-114805361-B Amino substituted aromatic heterocyclic pyrazole compound, preparation method and application 上海凌达生物医药有限公司 2024-02-20 CN disclosed
CN-117580477-A Reducing viral infection 福克斯生物有限公司 2024-02-20 CN disclosed
US-11905291-B2 2024-02-20 US disclosed
US-11905444-B2 Quantum dots and processes for preparation thereof THE UNIVERSITY OF QUEENSLAND (AU) 2024-02-20 US disclosed
US-11905252-B2 Compounds INFLAZOME LIMITED (IE) 2024-02-20 US disclosed
CN-117567478-A Camptothecins compound and its preparation method and application 四川科伦博泰生物医药股份有限公司 2024-02-20 CN disclosed
US-20240050512-A1 REDUCTION OF VIRAL INFECTIONS PHOXBIO LIMITED (IE) 2024-02-15 US disclosed
WO-2024035339-A1 AN IMPROVED GALACTOSE OXIDASE ENZYME PANEL FOR OXIDATION OF SECONDARY ALCOHOLS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2024-02-15 WO disclosed
US-20240050437-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2024-02-15 US disclosed
US-20240050428-A1 COMPOUNDS AND METHODS OF TREATING CANCERS CULLGEN (SHANGHAI), INC. (CN) 2024-02-15 US disclosed
US-20240052092-A1 PHOTOACTIVE MACROMOLECULES AND USES THEREOF BECKMAN COULTER, INC. 2024-02-15 US disclosed
US-20240051896-A1 METHODS OF FORMING LOW SALT NITROGEN-BASED FERTILIZER Cynagra LLC 2024-02-15 US disclosed
US-20240050573-A1 LYMPH DIRECTING PRODRUGS MONASH UNIVERSITY (AU) 2024-02-15 US disclosed
US-20240051930-A1 HETEROAROMATIC SPERMIDINE ANALOGUES AND THEIR ANTICANCER ACTIVITY FLORATEK PHARMA S.A. (CH) 2024-02-15 US disclosed
EP-4320127-A1 NEK7 INHIBITORS Halia Therapeutics, Inc. (US) 2024-02-14 EP disclosed
EP-4320103-A1 PYRIMIDINE BASED RAS MODULATORS AND USES THEREOF Quanta Therapeutics, Inc. (US) 2024-02-14 EP disclosed
EP-4320105-A1 OPIOID RECEPTOR MODULATORS Epiodyne, Inc. (US) 2024-02-14 EP disclosed
CN-117551073-A Thienylaniline compounds for the treatment of dermatological disorders 恩福莱克逊治疗有限公司 2024-02-13 CN disclosed
CN-117561258-A Novel substituted tricyclic aza heterocycles as SOS1 inhibitors 唯久生物技术(苏州)有限公司 2024-02-13 CN disclosed
US-11897867-B2 6-phenyl-4,5-dihydropyridazin-3(2H)-one derivatives as PDE3A and PDE3B inhibitors for treating cancer BAYER AKTIENGESELLSCHAFT (DE) 2024-02-13 US disclosed
US-11901508-B2 Silicon-based energy storage devices with functionalized linear sulfonate ester derivative compound containing electrolyte additives ENEVATE CORPORATION (US) 2024-02-13 US disclosed
US-11897865-B2 ABHD12 inhibitors and methods of making and using same THE SCRIPPS RESEARCH INSTITUTE (US) 2024-02-13 US disclosed
CN-114656791-B Polymer-silica hybrid PDOT and methods of use thereof 华盛顿大学 2024-02-09 CN disclosed
US-20240047098-A1 POLYMER-SILICA HYBRID PDOTS AND METHODS OF USE THEREOF UNIVERSITY OF WASHINGTON (US) 2024-02-08 US disclosed
US-20240042010-A1 NUCLEIC ACID VACCINES FOR CORONAVIRUS SUZHOU ABOGEN BIOSCIENCES CO LTD (CN) 2024-02-08 US disclosed
US-20240042051-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE LES LABORATOIRES SERVIER (FR) 2024-02-08 US disclosed
US-20240043455-A1 WATER SOLUBLE FLUORSCENT OR COLORED DYES COMPRISING CONJUGATING GROUPS SONY GROUP CORP (JP) 2024-02-08 US disclosed
US-20240043382-A1 MODIFIED INDOLE ALKALOIDS FOR THERAPEUTIC USES COMPASS PATHFINDER LIMITED (GB) 2024-02-08 US disclosed
US-20240043387-A1 SUBSTITUTED 3-DIALKYLAMINOMETHYL-PIPERIDIN-4-YL-BENZAMIDES AND METHODS OF MAKING AND USING SAME MEBIAS DISCOVERY INC (US) 2024-02-08 US disclosed
US-20240041827-A1 COMPOSITIONS FOR THE TREATMENT OF FAT RELATED CONDITIONS AND DISORDERS RAZIEL THERAPEUTICS LTD. (IL) 2024-02-08 US disclosed
US-20240043427-A1 CD73 COMPOUNDS GILEAD SCIENCES, INC. 2024-02-08 US disclosed
US-20240043441-A1 INHIBITORS OF KRAS G12C ARAXES PHARMA LLC (US) 2024-02-08 US disclosed
US-20240043379-A1 PRODRUGS OF CYTOTOXIC ACTIVE AGENTS HAVING ENZYMATICALLY CLEAVABLE GROUPS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2024-02-08 US disclosed
WO-2024031089-A1 SARS-COV2 MAIN PROTEASE INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-08 WO disclosed
WO-2024027703-A1 PRMT5 INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 上海艾力斯医药科技股份有限公司 2024-02-08 WO disclosed
EP-4313100-A2 PEPTIDES AND METHODS FOR REDUCING SKIN PIGMENTATION GLO Pharma, Inc. (US) 2024-02-07 EP disclosed
EP-4315330-A1 HALOGENATED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC (US) 2024-02-07 EP disclosed
EP-4313968-A2 SUBSTITUTED 1-ARYL-1'-HETEROARYL COMPOUNDS, SUBSTITUTED 1,1'-BIHETEROARYL COMPOUNDS, AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2024-02-07 EP disclosed
EP-4313943-A1 SUBSTITUTED PYRROLIDIN-2-ONES, SALTS THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES Bayer Aktiengesellschaft (DE) 2024-02-07 EP disclosed
EP-4313988-A1 PYRAZOLOPYRIMIDINONE COMPOUNDS Orphagen Pharmaceuticals, Inc. (US) 2024-02-07 EP disclosed
CN-117510468-A Dual MAGL and FAAH inhibitors 灵北拉荷亚研究中心公司 2024-02-06 CN disclosed
US-11890275-B2 Therapeutic compounds CELGENE QUANTICEL RESEARCH, INC. 2024-02-06 US disclosed
US-11894519-B2 Silicon-based energy storage devices with linear carbonate containing electrolyte additives ENEVATE CORPORATION (US) 2024-02-06 US disclosed
US-11891404-B2 Substituted macrocyclic indole derivatives BAYER AKTIENGESELLSCHAFT (DE) 2024-02-06 US disclosed
CN-116478145-B ALK2 kinase inhibitors 杭州邦顺制药有限公司 2024-02-02 CN disclosed
CN-117500507-A Phosphorus derivatives as novel SOS1 inhibitors 拜耳公司 2024-02-02 CN disclosed
WO-2024023641-A1 METHODS OF TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITOR DOSING FIELD OF THE INVENTION NOVARTIS AG (CH) 2024-02-01 WO disclosed
WO-2024026500-A2 INHIBITORS OF PDE11A4 AND METHODS OF USING SAME UNIVERSITY OF MARYLAND, BALTIMORE (US) 2024-02-01 WO disclosed
US-20240034845-A1 POLYMER PARTICLES QUEENSLAND UNIVERSITY OF TECHNOLOGY (AU) 2024-02-01 US disclosed
WO-2024024963-A1 MODIFIED POLYISOCYANATE, COATING AND COATED METAL MATERIAL 関西ペイント株式会社 2024-02-01 WO disclosed
US-20240034731-A1 AZA-QUINAZOLINE COMPOUNDS AND METHODS OF USE IAMBIC THERAPEUTICS, INC. 2024-02-01 US disclosed
WO-2024022263-A1 LIPID COMPOUND AND LIPID NANOPARTICLE COMPOSITION 苏州艾博生物科技有限公司 2024-02-01 WO disclosed
CN-117479945-A Large conductance potassium channel modulators, compositions thereof, methods of making and methods of using the same 依那拉治疗股份有限公司 2024-01-30 CN disclosed
CN-117466868-A Dual MAGL and FAAH inhibitors 灵北拉荷亚研究中心公司 2024-01-30 CN disclosed
CN-117480155-A Diacylglycerol kinase modulating compounds 吉利德科学公司 2024-01-30 CN disclosed
US-11884645-B2 Sulfonyl acetamides as NLRP3 inhibitors INFLAZOME LIMITED (IE) 2024-01-30 US disclosed
US-11883381-B2 ASH1L inhibitors and methods of treatment therewith THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2024-01-30 US disclosed
US-11884648-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2024-01-30 US disclosed
US-11884666-B2 Azabicyclo and diazepine derivatives ALCON INC. (CH) 2024-01-30 US disclosed
US-11884673-B2 Modulators of ion channel receptors and uses thereof BIONOMICS LIMITED (AU) 2024-01-30 US disclosed
US-11883397-B2 Substituted pyrido[1,2-a]pyrrolo[1,2-d]pyrazines for treating viral infections GILEAD SCIENCES, INC. (US) 2024-01-30 US disclosed
US-11884680-B2 Bromodomain inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2024-01-30 US disclosed
US-11888114-B2 Silicon-based energy storage devices with fluorinated polymer containing electrolyte additives ENEVATE CORPORATION (US) 2024-01-30 US disclosed
CN-117460827-A Nucleic acid vaccine for rabies 苏州艾博生物科技有限公司 2024-01-26 CN disclosed
CN-117460518-A CD-90 targeted lipid nanoparticles 宾夕法尼亚大学理事会 2024-01-26 CN disclosed
WO-2024020164-A2 GLUCOCORTICOID RECEPTOR AGONISTS AND CONJUGATES THEREOF FIREFLY BIO, INC. (US) 2024-01-25 WO disclosed
WO-2024020419-A1 AZA-QUINAZOLINE COMPOUNDS AND METHODS OF USE IAMBIC THERAPEUTICS, INC. (US) 2024-01-25 WO disclosed
US-20240024403-A1 Compositions and Methods for Managing Weight UNIGEN, INC. (US) 2024-01-25 US disclosed
US-20240025868-A1 PHENOTHIAZINE COMPOUNDS FOR THE TREATMENT OF ALZHEIMER'S DISEASE AND OTHER AGE-RELATED AND NEUROLOGICAL DISEASES ICAHN SCHOOL MED MOUNT SINAI (US) 2024-01-25 US disclosed
US-20240025862-A1 SUBSTITUTED N-PHENYLURACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2024-01-25 US disclosed
WO-2024020380-A1 QUINAZOLINE COMPOUNDS AND METHODS OF USE IAMBIC THERAPEUTICS, INC. (US) 2024-01-25 WO disclosed
US-20240025851-A1 Modulators of BCL6 as Ligand Directed Degraders CELGENE CORPORATION (US) 2024-01-25 US disclosed
US-20240024870-A1 MODIFICATION OF SURFACE PROPERTIES OF MICROFLUIDIC DEVICES BIO RAD LABORATORIES INC (US) 2024-01-25 US disclosed
WO-2024019770-A1 METHODS OF MAKING IONIZABLE LIPIDS AND LIPID NANOPARTICLES FOR MRNA DELIVERY UNIVERSITY OF CINCINNATI (US) 2024-01-25 WO disclosed
US-20240025903-A1 Bicyclic Compounds and Uses Thereof for the Treatment of Diseases ATHIRA PHARMA, INC. (US) 2024-01-25 US disclosed
WO-2024020517-A1 3-(6-PYRIDIN-3-YL)-2-[4-(4-METHYL-4H-1,2,4-TRIAZOL-3-YL)PIPERIDIN-1-YL]BENZONITRILE DERIVATIVES AND SIMILAR COMPOUNDS AS QPCTL AND QPCT INHIBITORS FOR THE TREATMENT OF CANCER 858 THERAPEUTICS, INC. (US) 2024-01-25 WO disclosed
US-20240025913-A1 TERTIARY CARBOXAMIDE COMPOUNDS VIVACE THERAPEUTICS, INC. 2024-01-25 US disclosed
WO-2024018403-A1 SUBSTITUTED IMIDAZOAMIDE COMPOUNDS, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2024-01-25 WO disclosed
WO-2024018017-A1 CATIONIC CHROMENONES AND THEIR USE IN ONCOLOGY Floratek Pharma SA (CH) 2024-01-25 WO disclosed
WO-2024020346-A2 GENE EDITING COMPONENTS, SYSTEMS, AND METHODS OF USE RENAGADE THERAPEUTICS MANAGEMENT INC. (US) 2024-01-25 WO disclosed
EP-4308666-A1 MULTIFUNCTIONAL LIQUID CRYSTALLINE PHOTOREACTIVE POLYMERS FOR POLARIZATION HOLOGRAPHY META PLATFORMS TECHNOLOGIES, LLC (US) 2024-01-24 EP disclosed
EP-4308982-A1 RECORDING A LATENT HOLOGRAPHIC GRATING AND AMPLIFICATION OF ITS DYNAMIC RANGE META PLATFORMS TECHNOLOGIES, LLC (US) 2024-01-24 EP disclosed
EP-4308983-A1 SPATIALLY VARYING DYNAMIC RANGE IN HOLOGRAPHIC GRATINGS META PLATFORMS TECHNOLOGIES, LLC (US) 2024-01-24 EP disclosed
EP-4309002-A1 RECORDING A LATENT HOLOGRAPHIC GRATING AND AMPLIFICATION OF ITS DYNAMIC RANGE META PLATFORMS TECHNOLOGIES, LLC (US) 2024-01-24 EP disclosed
US-11878027-B2 Nicotinamide mononucleotide derivatives and their uses METRO INTERNATIONAL BIOTECH, LLC (US) 2024-01-23 US disclosed
US-11878982-B2 Spiropiperidine derivatives 89BIO LTD (IL) 2024-01-23 US disclosed
US-11879024-B1 Soft mold formulations for surface relief grating fabrication with imprinting lithography META PLATFORMS TECHNOLOGIES, LLC (US) 2024-01-23 US disclosed
US-11878985-B2 Substituted quinazolines as inhibitors of KRAS G12C ARAXES PHARMA LLC (US) 2024-01-23 US disclosed
US-11878966-B2 Substituted 4-benzyl and 4-benzoyl piperidine derivates 89BIO LTD (IL) 2024-01-23 US disclosed
CN-117440774-A Biomarkers of age-related macular degeneration 倍亮生物有限责任公司 2024-01-23 CN disclosed
CN-117430588-A Pyridazinone heterocyclic compound Myosin II inhibitor and application thereof 西藏海思科制药有限公司 2024-01-23 CN disclosed
CN-117425646-A Phosphono derivative, composition thereof and pharmaceutical application thereof 西藏海思科制药有限公司 2024-01-19 CN disclosed
CN-117425644-A Opioid receptor modulators 埃皮欧黛公司 2024-01-19 CN disclosed
CN-117425496-A Lipid nanoparticle therapy to evade immune responses 宾夕法尼亚大学理事会 2024-01-19 CN disclosed
CN-117417279-A Phenoxyacetic acid compound, isomer thereof, pharmaceutically acceptable salt or solvate thereof, pharmaceutical composition and medical application 中国人民解放军军事科学院军事医学研究院 2024-01-19 CN disclosed
CN-117417281-A Anti-inflammatory, anti-cancer and anti-angiogenic compounds, pharmaceutical compositions and methods of making and using the same 麦迪康制药公司 2024-01-19 CN disclosed
WO-2024015950-A1 METHODS AND COMPOSITIONS FOR PPO HERBICIDE TOLERANCE MONSANTO TECHNOLOGY LLC (US) 2024-01-18 WO disclosed
WO-2024012524-A1 ANTIBODY-DRUG CONJUGATE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 苏州宜联生物医药有限公司 2024-01-18 WO disclosed
WO-2024013015-A1 HERBICIDAL COMPOSITIONS BAYER AKTIENGESELLSCHAFT (DE) 2024-01-18 WO disclosed
WO-2024013193-A1 ALKOXYLATED ALKANOLS FOR ENHANCING THE ACTIVITY OF ANTIMICROBIAL AGENTS BASF SE (DE) 2024-01-18 WO disclosed
US-20240018149-A1 PROTEIN DEGRADATION COMPOUNDS AND METHODS OF USE ANHORN MEDICINES CO., LTD. (TW) 2024-01-18 US disclosed
US-20240016152-A1 ACTIVE COMPOUND COMBINATIONS BAYER AKTIENGESELLSCHAFT (DE) 2024-01-18 US disclosed
US-20240016786-A1 GLUCOSIDASE INHIBITORS FOR THE TREATMENT AND PREVENTION OF PULMONARY INFECTIONS COVIRIX Medical Pty Ltd (AU) 2024-01-18 US disclosed
WO-2024013016-A1 HERBICIDAL COMPOSITIONS BAYER AKTIENGESELLSCHAFT (DE) 2024-01-18 WO disclosed
US-20240018153-A1 BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF 2692372 ONTARIO, INC. (CA) 2024-01-18 US disclosed
WO-2024015949-A2 METHODS AND COMPOSITIONS FOR PPO HERBICIDE TOLERANCE MONSANTO TECHNOLOGY LLC (US) 2024-01-18 WO disclosed
US-20240016799-A1 ANTI-INFLAMMATORY, ANTI-CANCER, AND ANTI-ANGIOGENIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF MAKING AND USING THEREOF MEDICON PHARMACEUTICALS, INC. 2024-01-18 US disclosed
WO-2024013724-A1 ANTIBODY-DRUG CONJUGATES PHEON THERAPEUTICS LTD (GB) 2024-01-18 WO disclosed
WO-2024012523-A1 ANTIBODY-DRUG CONJUGATE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 苏州宜联生物医药有限公司 2024-01-18 WO disclosed
WO-2024013723-A1 ANTIBODY DRUG CONJUGATES THAT BIND CDCP1 AND USES THEREOF PHEON THERAPEUTICS LTD (GB) 2024-01-18 WO disclosed
EP-3384549-B1 SODIUM-ION ELECTROLYTE COMPOSITION UNIV DEAKIN (AU) 2024-01-17 EP disclosed
EP-4304717-A1 USE OF NADOLOL TO TREAT CHRONIC OBSTRUCTIVE PULMONARY DISEASE BY BLOCKAGE OF THE ARRESTIN-2 PATHWAY Chronic Airway Therapeutics Limited (AU) 2024-01-17 EP disclosed
EP-4304567-A1 TARGETED THERAPEUTIC LIPID NANOPARTICLES AND METHODS OF USE The Trustees of the University of Pennsylvania (US) 2024-01-17 EP disclosed
EP-4305030-A1 HETEROCYCLES AND USES THEREOF Kumquat Biosciences Inc. (US) 2024-01-17 EP disclosed
CN-117398474-A Bioactive conjugate, preparation method and application thereof 苏州宜联生物医药有限公司 2024-01-16 CN disclosed
CN-113816969-B Eptification control compound, antibody drug conjugate thereof and application thereof 联宁(苏州)生物制药有限公司 2024-01-16 CN disclosed
US-11872239-B2 Modified oligomeric compounds comprising tricyclo-DNA nucleosides and uses thereof SYNTHENA AG (CH) 2024-01-16 US disclosed
CN-117412959-A Substituted 1-aryl-1 '-heteroaryl compounds, substituted 1,1' -biaryl compounds, and methods of use thereof 爱彼特生物制药公司 2024-01-16 CN disclosed
US-11876180-B2 Silicon-based energy storage devices with metal sulfide containing electrolyte additives ENEVATE CORPORATION (US) 2024-01-16 US disclosed
US-11876179-B2 Silicon-based energy storage devices with electrolyte containing dimethoxyethane based compound ENEVATE CORPORATION (US) 2024-01-16 US disclosed
US-11873288-B2 Inhibitors for soluble epoxide hydrolase (sEH) and fatty acid amide hydrolase (FAAH) THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-01-16 US disclosed
CN-117396478-A Diacylglycerol kinase modulating compounds 吉利德科学公司 2024-01-12 CN disclosed
CN-117396604-A Compositions and methods for targeting lipid nanoparticle therapies to stem cells 宾夕法尼亚大学理事会 2024-01-12 CN disclosed
CN-117396480-A Pyrazolopyrimidinone compounds 奥弗恩制药公司 2024-01-12 CN disclosed
CN-117396194-A Targeted therapeutic lipid nanoparticles and methods of use 宾夕法尼亚大学理事会 2024-01-12 CN disclosed
CN-114106278-B Polyurethane/urea materials 联邦科学和工业研究组织 2024-01-12 CN disclosed
US-20240011976-A1 ADDITIVES FOR REDUCING NON-SPECIFIC INTERACTIONS BETWEEN FLUORESCENT POLYMER CONJUGATES AND CELLS IN A BIOLOGICAL SAMPLE BECKMAN COULTER, INC. 2024-01-11 US disclosed
EP-4301371-A1 SUBSTITUTED 3,6-DIHYDRO-2H-1,3,4-OXADIAZIN-2-ONES FOR THE TREATMENT OF SARCOMA Bayer Aktiengesellschaft (DE) 2024-01-10 EP disclosed
EP-4301759-A2 T-TYPE CALCIUM CHANNEL ANTAGONISTS AND USES THEREOF The Board of Trustees of the Leland Stanford Junior University (US) 2024-01-10 EP disclosed
EP-3813784-B1 PRC1 INHIBITORS AND PRC1 INHIBITORS FOR USE IN METHODS OF TREATMENT THEREWITH UNIV MICHIGAN REGENTS (US) 2024-01-10 EP disclosed
CN-117377664-A Small molecule modulators of orphan nuclear receptor TLX 贝勒医学院 2024-01-09 CN disclosed
US-11866431-B2 Bicyclic compounds VIVACE THERAPEUTICS, INC. (US) 2024-01-09 US disclosed
CN-117377671-A Diacylglycerol kinase modulating compounds 吉利德科学公司 2024-01-09 CN disclosed
CN-111454165-B Novel lipid and lipid nanoparticle formulations for delivery of nucleic acids 爱康泰生治疗公司 2024-01-05 CN disclosed
CN-115919859-B Pharmaceutical composition of heteroaryl derivative and application of pharmaceutical composition in medicine 四川海思科制药有限公司 2024-01-05 CN disclosed
US-20240002611-A1 MULTIFUNCTIONAL RESINS FOR 3D PRINTED MATERIALS AND METHODS OF MAKING SAME META PLATFORMS TECHNOLOGIES, LLC (US) 2024-01-04 US disclosed
WO-2024006391-A1 MENIN-MLL INHIBITORS AND COMPOSITIONS FOR PROLIFERATION OF BETA CELLS BIOMEA FUSION, INC. (US) 2024-01-04 WO disclosed
WO-2024003749-A1 COMPOUNDS AND METHODS FOR DEGRADING CASEIN KINASE 1 ALPHA PIN THERAPEUTICS, INC. (KR) 2024-01-04 WO disclosed
WO-2024007016-A2 NOVEL FLUORESCENT DYES AND POLYMERS FROM DIHYDROPHENANTHRENE DERIVATIVES BECKMAN COULTER, INC. (US) 2024-01-04 WO disclosed
WO-2024006929-A1 CD73 COMPOUNDS GILEAD SCIENCES, INC. (US) 2024-01-04 WO disclosed
EP-4297746-A2 COMPOSITIONS AND METHODS TO IMPROVE THE THERAPEUTIC BENEFIT OF SUBOPTIMALLY ADMINISTERED COMPOUNDS AND THERAPIES FOR THE TREATMENT OF DISEASES Edison Oncology (US) 2024-01-03 EP disclosed
EP-3684368-B1 SELECTIVE P2X3 ANTAGONISTS FOR USE IN TREATING CHRONIC COUGH WITHOUT LOSS OF TASTE RESPONSE BELLUS HEALTH COUGH INC (CA) 2024-01-03 EP disclosed
EP-4298101-A1 PORPHYRIN DERIVATIVES AND USES THEREOF University Of Tasmania (AU) 2024-01-03 EP disclosed
US-11857555-B2 Aqueous pharmaceutical formulation of hydrocortisone sodium phosphate and monothioglycerol ANTARES PHARMA, INC. (US) 2024-01-02 US disclosed
US-11859130-B2 Metal oxide, metal bronze and polyoxometalate as charge storage materials in electrochromic device Furcifer Inc. (US) 2024-01-02 US disclosed
CN-111050765-B Spiro compounds and methods of making and using the same H.隆德贝克有限公司 2024-01-02 CN disclosed
US-11858925-B2 GAS41 inhibitors and methods of use thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2024-01-02 US disclosed
CN-112105355-B ABHD12 inhibitors and methods of making and using the same 斯克利普斯研究所 2024-01-02 CN disclosed
CN-115626927-B Tropomyosin Receptor Kinase (TRK) degrading compounds and methods of use 上海睿跃生物科技有限公司 2024-01-02 CN disclosed
CN-117337289-A Tetracyclic compounds for the treatment of brain disorders 加利福尼亚大学董事会 2024-01-02 CN disclosed
CN-113527299-B Nitrogen-containing condensed ring compound, preparation method and application 上海凌达生物医药有限公司 2023-12-29 CN disclosed
CN-114907350-B Nitrogen-containing condensed ring compound, preparation method and application 上海凌达生物医药有限公司 2023-12-29 CN disclosed
US-20230416269-A1 TOPICAL PHOSPHOINOSITIDE 3-KINASE INHIBITORS COA THERAPEUTICS, INC. 2023-12-28 US disclosed
US-20230416245-A1 ADENOSINE ANALOGS FOR THE TREATMENT OF DISEASE BIOINTERVENE, INC. 2023-12-28 US disclosed
US-20230414624-A1 METHODS OF TREATING NEUROLOGICAL VENTILATORY INSUFFICIENCY ENALARE THERAPEUTICS INC (US) 2023-12-28 US disclosed
US-20230416468-A1 BIOACTIVE POLYETHYLENE COPOLYMER, POLYETHYLENE MACROMOLECULE AND RELATED METHODS THEREOF MITSUI CHEMICALS, INC. (JP) 2023-12-28 US disclosed
US-20230416229-A1 [(1,5-DIHETEROARYL-1H-1,2,4-TRIAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2023-12-28 US disclosed
US-20230416259-A1 INHIBITORS OF NEK7 KINASE HALIA THERAPEUTICS INC (US) 2023-12-28 US disclosed
US-20230416452-A1 MULTICOLORED ELECTROCHROMIC POLYMER COMPOSITIONS AND METHODS OF MAKING AND USING THE SAME LANNRAY ADVANCED MATERIALS CO. LTD (CN) 2023-12-28 US disclosed
US-20230416286-A1 INHIBITORS OF MEK KINASE MOSAICA MEDICINES, INC. 2023-12-28 US disclosed
WO-2023250141-A2 METHODS OF TREATING NEUROLOGICAL VENTILATORY INSUFFICIENCY ENALARE THERAPEUTICS INC. (US) 2023-12-28 WO disclosed
WO-2023250427-A2 FORMULATIONS FOR MODULATING MYC EXPRESSION FLAGSHIP PIONEERING INNOVATIONS V, INC. (US) 2023-12-28 WO disclosed
WO-2023250429-A2 COMBINATION THERAPIES COMPRISING MYC MODULATION FLAGSHIP PIONEERING INNOVATIONS V, INC. (US) 2023-12-28 WO disclosed
CN-117295727-A Pyridazinones as PARP7 inhibitors 中山优理生物医药有限公司 2023-12-26 CN disclosed
CN-117263950-A Pyridazine compound, pharmaceutical composition and application thereof 上海优理惠生医药有限公司 2023-12-22 CN disclosed
CN-115073469-B Preparation and application of pyrrolopyrimidine compound as kinase inhibitor 药雅科技(上海)有限公司 2023-12-22 CN disclosed
CN-114057749-B Preparation method and application of irreversible alkyne heterocyclic compound FGFR inhibitor 药雅科技(上海)有限公司 2023-12-22 CN disclosed
CN-115073468-B Preparation and application of imidazopyrazines BTK inhibitor 药雅科技(上海)有限公司 2023-12-22 CN disclosed
CN-117279644-A Substituted 3, 6-dihydro-2H-1, 3, 4-oxadiazin-2-ones for the treatment of sarcomas 拜耳股份有限公司 2023-12-22 CN disclosed
CN-117263959-A Preparation and application of aromatic KRAS mutant protein inhibitor 药雅科技(上海)有限公司 2023-12-22 CN disclosed
CN-117263999-A Camptothecin prodrugs and pharmaceutical compositions thereof 天津和美奥康医药科技有限公司 2023-12-22 CN disclosed
CN-115028633-B Preparation and application of pyrrolopyrimidine compound 药雅科技(上海)有限公司 2023-12-22 CN disclosed
CN-117279913-A Heterocyclic compounds and their use 金橘生物科技公司 2023-12-22 CN disclosed
US-20230413432-A1 SELF-HEALABLE, RECYCLABLE, AND RECONFIGURABLE WEARABLE ELECTRONICS DEVICE NATIONAL SCIENCE FOUNDATION 2023-12-21 US disclosed
US-20230404984-A1 FORMULATIONS OF RBP4 INHIBITORS AND METHODS OF USE Belite Bio (HK) Limited (HK) 2023-12-21 US disclosed
US-20230405015-A1 SUBSTITUTED 3,6-DIHYDRO-2H-1,3,4-OXADIAZIN-2-ONES FOR THE TREATMENT OF SARCOMA BAYER AKTIENGESELLSCHAFT (DE) 2023-12-21 US disclosed
EP-4292655-A2 HEXADECAHYDRO-1H-CYCLOPENTA[A]PHENANTHRENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION Taro Pharmaceuticals Inc. (CA) 2023-12-20 EP disclosed
CN-111757884-B Substituted macrocyclic indole derivatives 拜耳股份公司 2023-12-19 CN disclosed
US-11845761-B2 Tricyclic pyridones and pyrimidones ERASCA, INC. (US) 2023-12-19 US disclosed
US-11845723-B2 Diacylglycerol kinase modulating compounds GILEAD SCIENCES, INC. (US) 2023-12-19 US disclosed
US-11848419-B2 Metal amide bases as electrolyte additives for Si anode-based Li-ion batteries ENEVATE CORPORATION (US) 2023-12-19 US disclosed
US-11845753-B2 Inhibitors of menin-mll interaction BIOMEA FUSION, INC. (US) 2023-12-19 US disclosed
US-11848418-B2 Single lithium-ion conductive polymer electrolytes for Si anode-based lithium-ion batteries ENEVATE CORPORATION (US) 2023-12-19 US disclosed
CN-117229300-A Preparation and application of EGFR inhibitor 药雅科技(上海)有限公司 2023-12-15 CN disclosed
CN-117229262-A Preparation and application of polyaromatic ring EGFR inhibitor 药雅科技(上海)有限公司 2023-12-15 CN disclosed
CN-117229292-A Preparation and application of RET inhibitor 药雅科技(上海)有限公司 2023-12-15 CN disclosed
CN-117229263-A Compound for inhibiting or degrading Bcl6 and application of compound in medicine 四川海思科制药有限公司 2023-12-15 CN disclosed
CN-117229289-A Preparation and application of EGFR inhibitor with macrocyclic structure 药雅科技(上海)有限公司 2023-12-15 CN disclosed
CN-117229261-A Preparation and application of EGFR inhibitor 药雅科技(上海)有限公司 2023-12-15 CN disclosed
CN-117224593-A Compositions and methods for managing or improving bone disorders, cartilage disorders, or both 尤尼根公司 2023-12-15 CN disclosed
US-20230399565-A1 POLYMER DYES AND USES THEREOF BECKMAN COULTER, INC. 2023-12-14 US disclosed
US-20230399314-A1 CD73 INHIBITOR AND USE THEREOF Wuhan Humanwell Innovative Drug Research and Development Center Limited Company (CN) 2023-12-14 US disclosed
US-20230397604-A1 [(1-PHENYL-5-(HETEROARYL)-1H-1,2,4-TRIAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS BAYER AKTIENGELLSCHAFT (DE) 2023-12-14 US disclosed
US-20230399312-A1 SUBSTITUTED PYRIMIDINES AND METHODS OF USE THERAVANCE BIOPHARMA R&D IP LLC (US) 2023-12-14 US disclosed
US-20230398224-A1 TARGETED PLASMA PROTEIN DEGRADATION NOVARTIS AG (CH) 2023-12-14 US disclosed
US-20230399457-A1 Bioactive Synthetic Copolymer, Bioactive Macromolecule and Related Methods Thereof AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2023-12-14 US disclosed
WO-2023240253-A2 MODULATORS OF TNF-ALPHA ACTIVITY FORWARD THERAPEUTICS, INC. (US) 2023-12-14 WO disclosed
EP-4288418-A1 SUBSTITUTED (2-HETEROARYLOXYPHENYL)SULFONATES, SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS Bayer Aktiengesellschaft (DE) 2023-12-13 EP disclosed
EP-4288422-A1 HETEROAROMATIC SPERMIDINE ANALOGUES AND THEIR ANTICANCER ACTIVITY Floratek Pharma SA (CH) 2023-12-13 EP disclosed
EP-4288433-A1 NOVEL COMPOUNDS Cerevance, Inc. (US) 2023-12-13 EP disclosed
EP-4288421-A1 FLAVONE DEAZA SPERMIDINE ANALOGUES AND THEIR USE TREATING CANCER Floratek Pharma SA (CH) 2023-12-13 EP disclosed
EP-3612532-B1 VMAT2 INHIBITOR COMPOUNDS AND COMPOSITIONS THEREOF NEUROCRINE BIOSCIENCES INC (US) 2023-12-13 EP disclosed
EP-4289425-A2 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS Tseng, Yufeng, Jane (US) 2023-12-13 EP disclosed
EP-4288423-A1 COMBINATION OF DUAL ATM AND DNA-PK INHIBITORS AND IMMUNOTHERAPEUTIC AGENTS FOR USE IN CANCER THERAPY XRad Therapeutics, Inc. (US) 2023-12-13 EP disclosed
EP-4288434-A1 SELECTIVE BCL-XL PROTAC COMPOUNDS AND METHODS OF USE Les Laboratoires Servier (FR) 2023-12-13 EP disclosed
EP-4289851-A1 CAMPTOTHECIN COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2023-12-13 EP disclosed
US-11840543-B2 Compounds and uses THE UNIVERSITY OF QUEENSLAND (AU) 2023-12-12 US disclosed
CN-117222409-A Methods of treating spinal cord injury or damage 斯皮诺吉尼克斯公司 2023-12-12 CN disclosed
CN-117222642-A Analogues for the treatment of disease 英矽智能科技知识产权有限公司 2023-12-12 CN disclosed
CN-117222625-A Substituted pyridazinones, salts or N-oxides thereof and their use as herbicidal agents 拜耳公司 2023-12-12 CN disclosed
CN-117222641-A Analogues for the treatment of disease 英矽智能科技知识产权有限公司 2023-12-12 CN disclosed
CN-117202895-A Lipid compounds and lipid nanoparticle compositions 苏州艾博生物科技有限公司 2023-12-08 CN disclosed
WO-2023235880-A1 CD38 MODULATORS AND USES THEREOF AEOVIAN PHARMACEUTICALS, INC. (US) 2023-12-07 WO disclosed
WO-2023235618-A1 FUSED PYRIMIDINE COMPOUNDS AS INHIBITORS OF MENIN BIOMEA FUSION, INC. (US) 2023-12-07 WO disclosed
WO-2023235321-A1 CO-MONOMERS FOR POLYMERIZATION OF DECONSTRUCTABLE THERMOSETS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-12-07 WO disclosed
WO-2023232048-A1 CAMPTOTHECIN PRODRUG AND PHARMACEUTICAL COMPOSITION THEREOF 天津和美奥康医药科技有限公司 2023-12-07 WO disclosed
WO-2023231988-A1 PREPARATION METHOD FOR DRUG LINKER CONJUGATE AND INTERMEDIATE THEREOF 苏州宜联生物医药有限公司 2023-12-07 WO disclosed
US-20230390354-A1 CYTOTOXIC AND ANTI-MITOTIC COMPOUNDS, AND METHODS OF USING THE SAME ZYMEWORKS BC INC. (CA) 2023-12-07 US disclosed
US-20230389542-A1 USE OF [(1,5-DIPHENYL-1H-PYRAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AND THEIR SALTS AND COMPOSITIONS CONTAINING THEM, FOR REDUCING PHYTOTOXIC EFFECTS OF AGROCHEMICALS, IN PARTICULAR OF HERBICIDES, IN USEFUL PLANTS AND CROP PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2023-12-07 US disclosed
US-20230391723-A1 1,4-Substituted Piperidine Derivatives CEPHALON LLC 2023-12-07 US disclosed
US-20230391765-A1 HETEROBIFUNCTIONAL COMPOUNDS AS DEGRADERS OF ENL ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI 2023-12-07 US disclosed
US-20230391790-A1 INDENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION TARO PHARMACEUTICALS INC. (CA) 2023-12-07 US disclosed
US-20230391784-A1 IRREVERSIBLE INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, INC. 2023-12-07 US disclosed
US-20230391815-A1 EFFICIENT AND SCALABLE SYNTHESES OF NICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, MODIFIED DERIVATIVES THEREOF, PHOSPHORYLATED ANALOGS THEREOF, ADENYLYL DINUCLEOTIDE CONJUGATES THEREOF, AND NOVEL CRYSTALLINE FORMS THEREOF THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2023-12-07 US disclosed
WO-2023235753-A2 ALDH2 INHIBITORS AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-12-07 WO disclosed
EP-4284517-A1 HETEROAROMATIC PHOSPHONIUM SALTS FOR TREATING CANCER Floratek Pharma SA (CH) 2023-12-06 EP disclosed
EP-4284515-A1 HETEROAROMATIC PHOSPHONIUM SALTS AND THEIR USE TREATING CANCER Floratek Pharma SA (CH) 2023-12-06 EP disclosed
EP-4286381-A2 TREATMENT OF MERKEL CELLL CARCINOMA Celgene Quanticel Research, Inc. (US) 2023-12-06 EP disclosed
EP-4284514-A1 HETEROAROMATIC PHOSPHONIUM SALTS AND THEIR USE TREATING CANCER Floratek Pharma SA (CH) 2023-12-06 EP disclosed
EP-3496721-B1 TREATMENT OF MERKEL CELLL CARCINOMA CELGENE QUANTICEL RES INC (US) 2023-12-06 EP disclosed
US-11837711-B2 Silicon-based energy storage devices with anhydride containing electrolyte additives ENEVATE CORPORATION (US) 2023-12-05 US disclosed
CN-110143999-B Cytotoxic and antimitotic compounds and methods of use thereof 酵活英属哥伦比亚省公司 2023-12-05 CN disclosed
US-11834551-B2 Photoactive macromolecules and uses thereof BECKMAN COULTER, INC. (US) 2023-12-05 US disclosed
US-11834440-B2 Beta-lactam derivatives for the treatment of diseases INSILICO MEDICINE IP LIMITED (HK) 2023-12-05 US disclosed
US-11834466-B2 Benzoxaborole compounds and formulations thereof 5METIS, INC. (US) 2023-12-05 US disclosed
US-11834663-B2 Fibrotic treatment MONASH UNIVERSITY (AU) 2023-12-05 US disclosed
CN-117164657-A Prodrugs of directed lymphatics 莫纳什大学 2023-12-05 CN disclosed
US-11833210-B2 ASH1L inhibitors and methods of treatment therewith THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2023-12-05 US disclosed
US-11834433-B2 Compounds INFLAZOME LIMITED (IE) 2023-12-05 US disclosed
US-11834434-B2 Substituted 2-heteroaryloxypyridines and salts thereof and their use as herbicidal agents BAYER AKTIENGESELLSCHAFT (DE) 2023-12-05 US disclosed
US-11833137-B2 Substituted chromenones, IRE1 inhibitors, and methods of using same THE WISTAR INSTITUTE (US) 2023-12-05 US disclosed
CN-117164661-A Peptide compound, preparation method thereof, pharmaceutical composition containing peptide compound and application of pharmaceutical composition 上海优理惠生医药有限公司 2023-12-05 CN disclosed
CN-117143177-A Preparation method of drug connector conjugate and intermediate thereof 苏州宜联生物医药有限公司 2023-12-01 CN disclosed
CN-114524810-B Pyrimidine heterocyclic compounds, preparation method and application 上海凌达生物医药有限公司 2023-12-01 CN disclosed
CN-117143079-A Spiro aromatic ring compound and application thereof 上海奕拓医药科技有限责任公司 2023-12-01 CN disclosed
CN-113563323-B Benzothiazolyl biaryl compound, preparation method and application 上海凌达生物医药有限公司 2023-12-01 CN disclosed
CN-117157285-A Pharmaceutical compounds as ubiquitin-specific protease 19 (USP 19) inhibitors 阿尔麦克探索有限公司 2023-12-01 CN disclosed
CN-117143178-A Preparation method of drug connector conjugate and intermediate thereof 苏州宜联生物医药有限公司 2023-12-01 CN disclosed
US-20230381329-A1 Zwitterion Polymer-Drug Conjugates UNIV UTAH RES FOUND (US) 2023-11-30 US disclosed
WO-2023230472-A1 INHIBITORS OF MOLLUSCUM CONTAGIOSUM INFECTION AND METHODS USING THE SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2023-11-30 WO disclosed
US-20230383038-A1 CO-MONOMERS FOR POLYMERIZATION OF DECONSTRUCTABLE THERMOSETS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2023-11-30 US disclosed
US-20230382983-A1 COMPLEMENT FACTOR D ANTAGONIST ANTIBODIES AND CONJUGATES THEREOF KODIAK SCIENCES INC. 2023-11-30 US disclosed
US-20230382874-A1 [(5-PHENYL-1-HETEROARYL-1H-TRIAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2023-11-30 US disclosed
WO-2023230190-A1 PYRIMIDINE BASED MODULATORS AND USES THEREOF QUANTA THERAPEUTICS, INC. (US) 2023-11-30 WO disclosed
WO-2023227867-A1 HETEROBICYCLIC AMIDES AS INHIBITORS OF CD38 Cerevance, Inc. (US) 2023-11-30 WO disclosed
US-20230382940-A1 ANTIVIRAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. 2023-11-30 US disclosed
EP-3735404-B1 ASK1 INHIBITOR COMPOUNDS AND USES THEREOF SEAL ROCK THERAPEUTICS INC (US) 2023-11-29 EP disclosed
EP-4281069-A1 PROCESSES FOR PREPARING PYRROLOPYRIDINE-ANILINE COMPOUNDS NFlection Therapeutics, Inc. (US) 2023-11-29 EP disclosed
US-11827661-B2 Water soluble fluorescent or colored dyes comprising conjugating groups Sony Group Corporation (JP) 2023-11-28 US disclosed
CN-117136056-A Process for preparing pyrrolopyridine-anilines 恩福莱克逊治疗有限公司 2023-11-28 CN disclosed
CN-115028634-B Acetylenic pyrazino heterocycle FGFR inhibitor and preparation method and application thereof 药雅科技(上海)有限公司 2023-11-28 CN disclosed
CN-117136076-A MCL-1 inhibitor antibody drug conjugates and methods of use 诺华股份有限公司 2023-11-28 CN disclosed
CN-111902399-B Enantioselective hydrogenation of 4-substituted 1, 2-dihydroquinolines in the presence of chiral iridium catalysts 拜耳公司 2023-11-28 CN disclosed
CN-117120415-A Modified indole alkaloids for therapeutic use 指南针探路者有限公司 2023-11-24 CN disclosed
CN-114853723-B Preparation and application of indole compound BTK inhibitor 药雅科技(上海)有限公司 2023-11-24 CN disclosed
US-20230374036-A1 KRAS G12D MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2023-11-23 US disclosed
WO-2023225005-A1 FLT3 COMBINATION THERAPY FOR CANCER AND COMPOSITIONS THEREFOR BIOMEA FUSION, INC. (US) 2023-11-23 WO disclosed
WO-2023225336-A1 MET BCL-XL INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE THEREOF NOVARTIS AG (CH) 2023-11-23 WO disclosed
WO-2023223097-A1 ANTIBODY DRUG CONJUGATES NOVARTIS AG (CH) 2023-11-23 WO disclosed
US-20230374042-A1 KRAS MODULATORS AND USES THEREOF QUANTA THERAPEUTICS, INC. 2023-11-23 US disclosed
US-20230374022-A1 INHIBITORS OF PARG 858 THERAPEUTICS, INC. 2023-11-23 US disclosed
WO-2023221975-A1 ANTIBODY-DRUG CONJUGATE CONTAINING PROTEIN DEGRADATION AGENT BIOACTIVE COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF 苏州宜联生物医药有限公司 2023-11-23 WO disclosed
WO-2023224998-A1 INHIBITORS OF PARG 858 THERAPEUTICS, INC. (US) 2023-11-23 WO disclosed
WO-2023225359-A1 ANTIBODY-DRUG CONJUGATES OF ANTINEOPLASTIC COMPOUNDS AND METHODS OF USE THEREOF NOVARTIS AG (CH) 2023-11-23 WO disclosed
US-20230372337-A1 Combination Therapy Comprising an AXL Inhibitor BERGENBIO ASA (NO) 2023-11-23 US disclosed
US-20230374015-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR KINASES KINNATE BIOPHARMA INC. 2023-11-23 US disclosed
US-20230373832-A1 MICROBIAL REMEDIATION OF HALOGENATED COMPOUNDS VIA CHAIN ELONGATION AND DEHALOGENATION NATIONAL SCIENCE FOUNDATION 2023-11-23 US disclosed
WO-2023225664-A1 LACTAM SUBSTITUTED IMIDAZOPYRIDAZINE IL-17A MODULATORS AND USES THEREOF DICE ALPHA, INC. (US) 2023-11-23 WO disclosed
US-20230372537-A1 LIPID NANOPARTICLE FORMULATIONS ACUITAS THERAPEUTICS INC (CA) 2023-11-23 US disclosed
WO-2023225001-A1 NAPHTHYRIDINE BASED ENPP1 MODULATORS AND USES THEREOF Vir Biotechnology, Inc. (US) 2023-11-23 WO disclosed
EP-3586835-B1 PHARMACEUTICAL COMPOSITIONS COMPRISING ARYL ETHERS PELOTON THERAPEUTICS INC (US) 2023-11-22 EP disclosed
EP-3988631-B1 POLYMER-SILICA HYBRID PDOTS UNIV WASHINGTON (US) 2023-11-22 EP disclosed
US-11820728-B2 Carbonyl lipids and lipid nanoparticle formulations for delivery of nucleic acids Acuitas Therapeutics, Inc. (CA) 2023-11-21 US disclosed
US-11823809-B2 Polymer-silica hybrid pdots and methods of use thereof UNIVERSITY OF WASHINGTON (US) 2023-11-21 US disclosed
US-11819531-B2 Multifunctional zwitterionic polymer conjugates KODIAK SCIENCES INC. (US) 2023-11-21 US disclosed
CN-111132974-B Sulfonamide carboxamide compounds 英夫拉索姆有限公司 2023-11-21 CN disclosed
CN-117088931-A Prodrugs of directed lymphatics 莫纳什大学 2023-11-21 CN disclosed
CN-112218873-B Metallocene synthesis process 埃克森美孚化学专利公司 2023-11-21 CN disclosed
CN-117069785-A Lipid compounds and lipid nanoparticle compositions 中生复诺健生物科技(上海)有限公司 2023-11-17 CN disclosed
CN-117083274-A Fused ring heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2023-11-17 CN disclosed
CN-117069682-A Phenoxyacetic acid compound, pharmaceutical composition and medical application thereof 中国人民解放军军事科学院军事医学研究院 2023-11-17 CN disclosed
CN-117083291-A Coronavirus nucleic acid vaccine based on sequences derived from SARS-CoV-2Delta strain 苏州艾博生物科技有限公司 2023-11-17 CN disclosed
US-20230364082-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CONTINEUM THERAPEUTICS, INC. 2023-11-16 US disclosed
US-20230365577-A1 Photodynamic Therapy and Diagnosis RMW CHO GROUP LIMITED (HK) 2023-11-16 US disclosed
WO-2023220741-A1 ALPHA 4 BETA 7 INTEGRIN MODULATORS AND USES THEREOF DICE MOLECULES SV, INC. (US) 2023-11-16 WO disclosed
US-20230364074-A1 Compounds and Compositions for Disrupting Programmed Ribosomal Frameshifting NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-11-16 US disclosed
WO-2023216956-A1 CAMPTOTHECIN COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2023-11-16 WO disclosed
US-20230364097-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS INFINITY PHARMACEUTICALS, INC. (US) 2023-11-16 US disclosed
EP-4276126-A1 POLYURETHANE/UREA MATERIALS Commonwealth Scientific and Industrial Research Organisation (AU) 2023-11-15 EP disclosed
CN-117050058-A Fused heterocyclic compound, composition thereof and pharmaceutical application thereof 四川海思科制药有限公司 2023-11-14 CN disclosed
US-11814384-B2 Inhibtors of Raf kinases KINNATE BIOPHARMA INC. (US) 2023-11-14 US disclosed
US-11814380-B2 Benzylamino substituted pyridopyrimidinones and derivatives as SOS1 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-11-14 US disclosed
US-11813304-B2 Compounds and methods for inhibiting phosphate transport ARDELYX, INC. (US) 2023-11-14 US disclosed
CN-113061132-B Condensed ring lactam compound, preparation method and application 上海凌达生物医药有限公司 2023-11-14 CN disclosed
CN-112262142-B Benzenesulfonamide compounds and their use as therapeutic agents 泽农医药公司 2023-11-14 CN disclosed
US-11817578-B2 Silicon-based energy storage devices with silyl amine compounds or derivatives of silyl amine containing electrolyte additives ENEVATE CORPORATION (US) 2023-11-14 US disclosed
US-11814795-B2 Coating for recyclable paper JL DARLING LLC (US) 2023-11-14 US disclosed
CN-110582480-B Therapeutic compounds and methods 塔斯马尼亚大学 2023-11-10 CN disclosed
CN-117043862-A Halogenated monomers and polymers for volume Bragg gratings 元平台技术有限公司 2023-11-10 CN disclosed
CN-117043343-A Nucleic acid vaccine for mutant coronaviruses 苏州艾博生物科技有限公司 2023-11-10 CN disclosed
CN-117043140-A Substituted pyrrolidin-2-ones, salts thereof and their use as herbicidal active substances 拜耳公司 2023-11-10 CN disclosed
CN-117043143-A Substituted 2- (heteroaryloxyphenyl) sulfonates, salts thereof and their use as herbicides 拜耳公司 2023-11-10 CN disclosed
CN-117042780-A In vivo targeting of T cells for mRNA therapeutic agents 宾夕法尼亚大学理事会 2023-11-10 CN disclosed
WO-2023215377-A1 METHODS OF TREATING NEUROINFLAMMATORY CONDITIONS ATHIRA PHARMA, INC. (US) 2023-11-09 WO disclosed
WO-2023215709-A1 EFFICIENT METHOD OF SYNTHESIZING LINEAR OLIGOMERS AND APPLICATION TO FRONTAL RING-OPENING METATHESIS POLYMERIZATION THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-11-09 WO disclosed
US-20230357239-A1 PYRIDO[2,3-D]PYRIMIDIN-4-AMINES AS SOS1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2023-11-09 US disclosed
US-20230357490-A1 EFFICIENT METHOD OF SYNTHESIZING LINEAR OLIGOMERS AND APPLICATION TO FRONTAL RING-OPENING METATHESIS POLYMERIZATION THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-11-09 US disclosed
WO-2023215710-A1 EVERGREEN UPCYCLING PROCESS FOR THERMOSETS AND THERMOPLASTICS WITH DECONSTRUCTABLE AND UPGRADABLE MONOMERS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2023-11-09 WO disclosed
US-20230357259-A1 BIOACTIVE CONJUGATE, PREPARATION METHOD THEREFOR AND USE THEREOF SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2023-11-09 US disclosed
US-20230357459-A1 MECHANICALLY STIMULATED MECHANOPHORES, POLYMERS THEREOF, METHODS OF PREPARATION THEREOF, AND SYSTEMS THEREOF FOR CONTROLLED EMISSION OF SMALL MOLECULES THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2023-11-09 US disclosed
US-20230355584-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF LIPID-RELATED DISORDERS RAZIEL THERAPEUTICS LTD. (IL) 2023-11-09 US disclosed
WO-2023215376-A1 METHODS OF TREATING NEUROPATHIES ATHIRA PHARMA, INC. (US) 2023-11-09 WO disclosed
EP-3401314-B1 COVALENT INHIBITORS OF KRAS G12C ARAXES PHARMA LLC (US) 2023-11-08 EP disclosed
EP-4273147-A1 SUBSTITUTED SPIROLACTAMS, SALTS THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES Bayer Aktiengesellschaft (DE) 2023-11-08 EP disclosed
CN-117003658-A Lipid Nanoparticle Compositions 苏州艾博生物科技有限公司 2023-11-07 CN disclosed
US-11807646-B2 4-hydroxypiperidine derivatives and their use as inhibitors of ubiquitin specific protease 19 (USP19) ALMAC DISCOVERY LIMITED (GB) 2023-11-07 US disclosed
US-11807621-B2 Compounds and compositions for use in treating skin disorders KAMARI PHARMA LTD. (IL) 2023-11-07 US disclosed
CN-117015711-A Compositions and methods for preventing non-specific interactions between polymer dye-antibody conjugates 贝克曼库尔特有限公司 2023-11-07 CN disclosed
CN-117015534-A Combination of dual ATM and DNA-PK inhibitors for cancer therapy and immunotherapeutic agents 艾科思莱德制药公司 2023-11-07 CN disclosed
CN-117015745-A Recording a latent holographic grating and magnifying its dynamic range 元平台技术有限公司 2023-11-07 CN disclosed
CN-111655666-B Anti-inflammatory, anti-cancer and anti-angiogenic compounds, pharmaceutical compositions and methods of making and using the same 麦迪康制药公司 2023-11-07 CN disclosed
US-11807641-B2 MASP-2 inhibitors and methods of use OMEROS CORPORATION (US) 2023-11-07 US disclosed
CN-116997827-A Spatially varying dynamic range in holographic gratings 元平台技术有限公司 2023-11-03 CN disclosed
CN-110312533-B Prodrugs of cytotoxic active agents having enzymatically cleavable groups 拜耳公司 2023-11-03 CN disclosed
CN-116987509-A Liquid crystal compound, composition and application thereof 北京燕化集联光电技术有限公司 2023-11-03 CN disclosed
CN-116997797-A Additives for reducing non-specific interactions between fluorescent polymer conjugates and cells in biological samples 贝克曼库尔特有限公司 2023-11-03 CN disclosed
US-20230348852-A1 METHODS AND COMPOSITIONS FOR OCULAR CELL THERAPY NOVARTIS AG (CH) 2023-11-02 US disclosed
WO-2023212147-A1 HETEROCYCLIC COMPOUNDS AS MODULATORS OF BCL6 AS LIGAND DIRECTED DEGRADERS CELGENE CORPORATION (US) 2023-11-02 WO disclosed
WO-2023212612-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS QIAN SHAWN (US) 2023-11-02 WO disclosed
US-20230348674-A1 HYDROGELS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2023-11-02 US disclosed
US-20230348689-A1 EVERGREEN UPCYCLING PROCESS FOR THERMOSETS AND THERMOPLASTICS WITH DECONSTRUCTABLE AND UPGRADABLE MONOMERS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2023-11-02 US disclosed
WO-2023212548-A1 TRICYCLIC PYRIDONES AND PYRIMIDONES ERASCA, INC. (US) 2023-11-02 WO disclosed
US-20230348362-A1 LIPID COMPOUNDS AND LIPID NANOPARTICLE COMPOSITIONS Suzhou Abogen Biosciences Co., Ltd. (CN) 2023-11-02 US disclosed
US-20230348419-A1 BIAMINOQUINOLINES AND NANOFORMULATIONS FOR CANCER TREATMENT THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2023-11-02 US disclosed
US-20230348392-A1 PYRIDINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2023-11-02 US disclosed
US-20230346927-A1 COMBINATION of ATR KINASE INHIBITORS and PD-1/PD-L1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2023-11-02 US disclosed
WO-2023209368-A1 NITROGEN COMPRISING HETEROCYCLIC DERIVATIVES FOR THE TREATMENT OF DISORDERS ASSOCIATED WITH GPR55 RECEPTOR Cerevance, Inc. (US) 2023-11-02 WO disclosed
WO-2023211977-A1 TRYPTANTHRIN DERIVATIVES AND USES THEREOF VISCIENT BIO, INC. (US) 2023-11-02 WO disclosed
US-20230348475-A1 IMIDAZOPYRIDAZINE AND IMIDAZOPYRAZINE COMPOUNDS AS INHIBITORS OF CDK7 TRANSLATIONAL GENOMICS RES INST (US) 2023-11-02 US disclosed
WO-2023212549-A1 TRICYCLIC PYRIDONES AND PYRIMIDONES ERASCA, INC. (US) 2023-11-02 WO disclosed
EP-4267561-A1 SMALL-MOLECULE MODULATORS OF THE ORPHAN NUCLEAR RECEPTOR TLX Baylor College of Medicine (US) 2023-11-01 EP disclosed
CN-112707893-B 1-cyanopyrrolidine compounds as USP30 inhibitors 特殊治疗有限公司 2023-10-31 CN disclosed
CN-111801314-B ASK1 inhibitor compounds and uses thereof 西尔洛克治疗公司 2023-10-31 CN disclosed
CN-116969921-A Compound for inhibiting or degrading HPK1 kinase and application thereof in medicine 四川海思科制药有限公司 2023-10-31 CN disclosed
CN-116981665-A Novel compounds 思瑞万斯公司 2023-10-31 CN disclosed
CN-116981968-A Recording latent holographic grating and amplification of dynamic range thereof 元平台技术有限公司 2023-10-31 CN disclosed
CN-116948657-A Liquid crystal compound, composition and application thereof 北京燕化集联光电技术有限公司 2023-10-27 CN disclosed
CN-114805359-B Preparation method and application of acetylenic heterocyclic compound FGFR inhibitor 药雅科技(上海)有限公司 2023-10-27 CN disclosed
CN-116947877-A Benzimidazole derivative and application thereof in medicine 四川海思科制药有限公司 2023-10-27 CN disclosed
WO-2023204822-A1 PHENYL PHOSPHINE OXIDE COMPOUNDS AND METHODS OF USE THEREOF VIVACE THERAPEUTICS, INC. (US) 2023-10-26 WO disclosed
WO-2023202582-A1 GPCR REGULATOR AND USE THEREOF 北京昌平实验室 2023-10-26 WO disclosed
WO-2023205701-A1 MACROCYCLIC HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC. (US) 2023-10-26 WO disclosed
US-20230339867-A1 PYRAZINE COMPOUNDS AS INHIBITORS OF FLT3 BIOMEA FUSION, INC. 2023-10-26 US disclosed
WO-2023205719-A1 KRAS G12D MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2023-10-26 WO disclosed
US-20230339878-A1 SLC26A3 INHIBITORS AND USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2023-10-26 US disclosed
US-20230338565-A1 ANTIBODY DRUG CONJUGATE, PREPARATION METHOD THEREFOR AND USE THEREOF SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2023-10-26 US disclosed
WO-2023205116-A1 PYRIDINE DERIVATIVES FOR TREATING PSYCHIATRIC DISORDERS GILGAMESH PHARMACEUTICALS, INC. (US) 2023-10-26 WO disclosed
US-20230339952-A1 MACROCYCLIC HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC. 2023-10-26 US disclosed
US-20230339981-A1 KRAS G12D MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2023-10-26 US disclosed
EP-4265616-A1 SPIROCYCLIC COMPOUND AS KRAS-G12C INHIBITOR Shanghai Euregen Biopharma Co., Ltd. (CN) 2023-10-25 EP disclosed
EP-4263504-A1 MODIFIED INDOLE ALKALOIDS FOR THERAPEUTIC USES COMPASS Pathfinder Limited (GB) 2023-10-25 EP disclosed
EP-3659591-B1 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC (US) 2023-10-25 EP disclosed
EP-3601216-B1 SUBSTITUTED DIHYDROINDENE-4-CARBOXAMIDES AND ANALOGS THEREOF, AND METHODS USING SAME FOR THE TREATMENT OF HEPATITIS B VIRUS INFECTION ARBUTUS BIOPHARMA CORP (CA) 2023-10-25 EP disclosed
EP-4013500-B1 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS NOVARTIS AG (CH) 2023-10-25 EP disclosed
EP-3041830-B1 POLYMER-FLAVONOID CONJUGATES AND HYDROGELS FOR BIOMEDICAL APPLICATIONS AGENCY SCIENCE TECH & RES (SG) 2023-10-25 EP disclosed
EP-4263542-A1 FUSED PYRIMIDINE COMPOUNDS AS INHIBITORS OF MENIN-MLL INTERACTION Biomea Fusion, Inc. (US) 2023-10-25 EP disclosed
CN-116940679-A Oligomeric compounds for dystrophin rescue in DMD patients by skipping of exon-51 SQY治疗公司 2023-10-24 CN disclosed
CN-116925070-A Substituted aza-fused ring compounds and medical uses thereof 扬子江药业集团有限公司 2023-10-24 CN disclosed
US-11795136-B2 Methods for the treatment of diabetic retinopathy and other ophthalmic diseases ACUCELA INC. (US) 2023-10-24 US disclosed
CN-115368381-B Preparation and application of heterocyclic inhibitor 药雅科技(上海)有限公司 2023-10-24 CN disclosed
CN-116940685-A Coronavirus multivalent nucleic acid vaccine based on sequences derived from SARS-CoV-2Beta and Delta strains 苏州艾博生物科技有限公司 2023-10-24 CN disclosed
CN-116903695-A Cyclic peptide compound, preparation method thereof, pharmaceutical composition containing cyclic peptide compound and application of cyclic peptide compound 上海优理惠生医药有限公司 2023-10-20 CN disclosed
CN-116903563-A GPCR modulators and uses thereof 北京昌平实验室 2023-10-20 CN disclosed
CN-116917440-A Multifunctional liquid crystal photoreactive polymers for polarization holography 元平台技术有限公司 2023-10-20 CN disclosed
CN-116903609-A Compound, pharmaceutical composition containing same and application of compound 上海优理惠生医药有限公司 2023-10-20 CN disclosed
CN-116903610-A Heterocyclic condensed pyridines, pharmaceutical compositions and uses thereof 上海优理惠生医药有限公司 2023-10-20 CN disclosed
CN-114591334-B Dihydropyrazolopyrimidinone derivatives 山东轩竹医药科技有限公司 2023-10-20 CN disclosed
CN-116903696-A Peptide compound, preparation method thereof, pharmaceutical composition containing peptide compound and application of pharmaceutical composition 上海优理惠生医药有限公司 2023-10-20 CN disclosed
CN-116903611-A Phthalazinone compound, preparation method thereof, pharmaceutical composition containing phthalazinone compound and application of pharmaceutical composition 上海优理惠生医药有限公司 2023-10-20 CN disclosed
CN-116917289-A T-type calcium channel antagonists and uses thereof 小利兰·斯坦福大学董事会 2023-10-20 CN disclosed
WO-2023200766-A1 METHODS, COMPOSITIONS AND SYSTEMS FOR EVALUATION OF VISUAL FUNCTION BELITE BIO, INC (US) 2023-10-19 WO disclosed
US-20230331655-A1 HYDROXYNORKETAMINE COMPOUNDS AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-10-19 US disclosed
WO-2023198114-A1 ALK2 KINASE INHIBITOR 杭州邦顺制药有限公司 2023-10-19 WO disclosed
US-20230331719-A1 Pyrazolopyridine Compounds and Methods of Inhibiting IRE1 Using Same OPTIKIRA LLC (US) 2023-10-19 US disclosed
EP-4261211-A1 DIHYDROISOQUINOLINONE DERIVATIVE AND APPLICATION THEREOF Etern Biopharma (Shanghai) Co., Ltd. (CN) 2023-10-18 EP disclosed
EP-4259105-A1 IN VIVO TARGETING OF CD4+ -T CELLS FOR MRNA THERAPEUTICS The Trustees of the University of Pennsylvania (US) 2023-10-18 EP disclosed
US-11787783-B2 Heparanase inhibitors and use thereof Beta Therapeutics Pty Ltd (AU) 2023-10-17 US disclosed
US-11787780-B2 Quaternary indazole glucocorticoid receptor antagonists CORCEPT THERAPEUTICS INCORPORATED (US) 2023-10-17 US disclosed
US-11786519-B2 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases ABBVIE INC. (US) 2023-10-17 US disclosed
US-11786602-B2 ASH1L degraders and methods of treatment therewith THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2023-10-17 US disclosed
CN-116888127-A Tri-fused ring HPK1 inhibitor and application thereof 轩竹生物科技股份有限公司 2023-10-13 CN disclosed
US-20230323031-A1 POLYMER COMPRISING A PLURALITY OF ACTIVE AMINE GROUPS, RELATED POLYMERS AND RELATED METHODS THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2023-10-12 US disclosed
US-20230322672-A1 COMPOUNDS AND FORMULATIONS FOR TREATING OPHTHALMIC DISEASES VIEWPOINT THERAPEUTICS, INC. 2023-10-12 US disclosed
US-20230322711-A1 MACROCYCLIC COMPOUNDS AND COMPOSITIONS, AND METHODS OF PREPARING AND USING THE SAME WUXI APPTEC (HONG KONG) LIMITED (CN) 2023-10-12 US disclosed
US-20230321050-A1 Heterocyclic Compounds and Uses Thereof MILLENNIUM PHARMACEUTICALS, INC. 2023-10-12 US disclosed
EP-4257154-A1 BIOACTIVE SUBSTANCE CONJUGATE, PREPARATION METHOD THEREFOR AND USE THEREOF Medilink Therapeutics (Suzhou) Co., Ltd. (CN) 2023-10-11 EP disclosed
EP-3784671-B1 DUAL ATM AND DNA-PK INHIBITORS FOR USE IN ANTI-TUMOR THERAPY XRAD THERAPEUTICS INC (US) 2023-10-11 EP disclosed
EP-4257591-A2 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Celgene Quanticel Research, Inc. (US) 2023-10-11 EP disclosed
US-11780862-B2 Inhibitors of MEK kinase KINNATE BIOPHARMA INC. (US) 2023-10-10 US disclosed
US-RE49687-E1 Thienopyrimidine and thienopyridine compounds and methods of use thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2023-10-10 US disclosed
US-11780850-B2 Purification of rapamycin derivatives using temperature induced phase separation BIOSENSORS INTERNATIONAL GROUP, LTD. (BM) 2023-10-10 US disclosed
US-11780819-B2 Aromatic substituted alkane-core monomers and polymers thereof for volume Bragg gratings META PLATFORMS TECHNOLOGIES, LLC (US) 2023-10-10 US disclosed
CN-116850163-A Methods for treating diabetic retinopathy and other ophthalmic diseases 奥克塞拉有限公司 2023-10-10 CN disclosed
CN-116854709-A Reversible inhibitors of Bruton's tyrosine kinase and application thereof 药雅科技(上海)有限公司 2023-10-10 CN disclosed
CN-116867372-A [ (5-phenyl-1-heteroaryl-1H-pyrazol-3-yl) oxy ] acetic acid derivatives as safeners for protecting useful plants and crop plants 拜耳公司 2023-10-10 CN disclosed
US-20230312481-A1 SUBSTITUTED (PHTHALAZIN-1-YLMETHYL)UREAS, SUBSTITUTED N-(PHTHALAZIN-1-YLMETHYL)AMIDES, AND ANALOGUES THEREOF ARBUTUS BIOPHARMA CORP (CA) 2023-10-05 US disclosed
US-20230310398-A1 NICORANDIL DERIVATIVES Unicycive Therapeutics Inc. 2023-10-05 US disclosed
US-20230310440-A1 RESPIRATORY STIMULANT NASAL FORMULATIONS ENALARE THERAPEUTICS INC. 2023-10-05 US disclosed
US-20230312564-A1 AROMATIC RING-LACTAM COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI RINGENE BIOPHARMA CO., LTD. (CN) 2023-10-05 US disclosed
US-20230313245-A1 Engineered Enzymes and Method for the Synthesis of Diverse Tyrosine Analogs CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2023-10-05 US disclosed
US-20230312557-A1 P2X3 MODULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.3) LIMITED (GB) 2023-10-05 US disclosed
US-20230312498-A1 NON-ATP/CATALYTIC SITE p38 MITOGEN ACTIVATED PROTEIN KINASE INHIBITORS UNIVERSITY OF MARYLAND, BALTIMORE 2023-10-05 US disclosed
US-20230312713-A1 In vivo targeting of T cells for mRNA therapeutics THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2023-10-05 US disclosed
WO-2023190111-A1 RAFT POLYMERIZATION REACTION SOLUTION AND RAFT POLYMERIZATION REACTION SOLUTION PRODUCTION METHOD テクノUMG株式会社 2023-10-05 WO disclosed
WO-2023187670-A1 DIAZABICYCLOOCTANE DERIVATIVES USEFUL AS MATRIX METALLOPROTEINASE INHIBITORS VASA THERAPEUTICS SPOLKA Z OGRANICZONA ODPOWIEDZIALNOSCIA (PL) 2023-10-05 WO disclosed
WO-2023186842-A1 SYNTHESIS OF ISOMERICALLY PURE POLYOL-BASED PHOSPHORAMIDITES F. HOFFMANN-LA ROCHE AG (CH) 2023-10-05 WO disclosed
WO-2023192602-A2 RESPIRATORY STIMULANT NASAL FORMULATIONS ENALARE THERAPEUTICS INC. (US) 2023-10-05 WO disclosed
EP-4251627-A1 PHOTODYNAMIC THERAPY AND DIAGNOSIS RMW Cho Group Limited (CN) 2023-10-04 EP disclosed
EP-4251209-A1 BCL-XL INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE THEREOF Novartis AG (CH) 2023-10-04 EP disclosed
EP-4251208-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE Novartis AG (CH) 2023-10-04 EP disclosed
EP-3774836-B1 HEXADECAHYDRO-1H-CYCLOPENTA[A]PHENANTHRENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION TARO PHARMACEUTICALS INC (CA) 2023-10-04 EP disclosed
EP-4250991-A1 REDUCTION OF VIRAL INFECTIONS Phoxbio Limited (IE) 2023-10-04 EP disclosed
CN-111557942-B Fatty liver disease treatment using glucocorticoid and mineralocorticoid receptor antagonists 科赛普特治疗学股份有限公司 2023-10-03 CN disclosed
US-11773096-B2 Small-molecule PI5P4K alpha/beta inhibitors and methods of treatment using same YALE UNIVERSITY (US) 2023-10-03 US disclosed
US-11773058-B2 Sulfonamide carboxamide compounds INFLAZOME LIMITED (IE) 2023-10-03 US disclosed
CN-116836184-A Preparation and application of Wee1 kinase inhibitor 药雅科技(上海)有限公司 2023-10-03 CN disclosed
US-11773108-B2 Indene derivatives useful in treating pain and inflammation TARO PHARMACEUTICALS INC. (CA) 2023-10-03 US disclosed
US-11773214-B2 Multicolored electrochromic polymer compositions and methods of making and using the same Furcifer Inc. (US) 2023-10-03 US disclosed
US-11773114-B2 Protective groups and methods for protecting benzoxaboroles or oxaboroles SAINT JOSEPH'S UNIVERSITY (US) 2023-10-03 US disclosed
US-11773070-B2 Dihydrooxadiazinones BAYER AKTIENGESELLSCHAFT (DE) 2023-10-03 US disclosed
US-11771696-B2 Methods of treating chronic lymphocytic leukemia and small lymphocytic leukemia using a BTK inhibitor ACERTA PHARMA B.V. (NL) 2023-10-03 US disclosed
CN-116829197-A Polychelator compounds for targeted radiation therapy 拜耳股份有限公司 2023-09-29 CN disclosed
CN-109414596-B ASH1L inhibitors and methods of treatment therewith 密歇根大学董事会 2023-09-29 CN disclosed
CN-116813647-A Nitrogen-containing condensed ring STING regulator compound, preparation method and application 上海凌达生物医药有限公司 2023-09-29 CN disclosed
CN-116829561-A Camptothecins compound and its preparation method and application 四川科伦博泰生物医药股份有限公司 2023-09-29 CN disclosed
CN-116829578-A Polynucleotides encoding interleukin-12 (IL-12) and compositions and methods related thereto 苏州艾博生物科技有限公司 2023-09-29 CN disclosed
CN-116829570-A WEE1 degrading compounds 北京星奇原生物科技有限公司 2023-09-29 CN disclosed
US-20230303739-A1 FLUORINATED PVC COPOLYMER COMPOSITIONS FOR INCREASED ULTRAVIOLET PROTECTION Mexichem Specialty Resins Inc. 2023-09-28 US disclosed
US-20230301948-A1 REDUCTION OF VIRAL INFECTIONS PHOXBIO LIMITED (IE) 2023-09-28 US disclosed
WO-2023183807-A1 AQUEOUS PHARMACEUTICAL FORMULATION OF HYDROCORTISONE SODIUM PHOSPHATE AND MONOTHIOGLYCEROL ANTARES PHARMA, INC. (US) 2023-09-28 WO disclosed
US-20230302016-A1 AQUEOUS PHARMACEUTICAL FORMULATION OF HYDROCORTISONE SODIUM PHOSPHATE AND MONOTHIOGLYCEROL ANTARES PHARMA, INC. (US) 2023-09-28 US disclosed
US-20230303586-A1 INHIBITORS OF KRAS G12C ARAXES PHARMA LLC (US) 2023-09-28 US disclosed
US-20230303549-A1 SUBSTITUTED HETEROARYLOXYPYRIDINES, THE SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2023-09-28 US disclosed
US-20230303566-A1 INHIBITORS OF RAF KINASES Pierre Fabre Médicament (FR) 2023-09-28 US disclosed
WO-2023183755-A1 TRICYCLIC PYRIMIDONES ERASCA, INC. (US) 2023-09-28 WO disclosed
WO-2023183616-A1 NOVEL IONIZABLE LIPIDS AND LIPID NANOPARTICLES AND METHODS OF USING THE SAME SENDA BIOSCIENCES, INC. (US) 2023-09-28 WO disclosed
EP-4249519-A1 FLUORINATED PVC COPOLYMER COMPOSITIONS FOR INCREASED ULTRAVIOLET PROTECTION Mexichem Specialty Resins Inc. (US) 2023-09-27 EP disclosed
EP-4247794-A2 BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF 2692372 Ontario, Inc. (CA) 2023-09-27 EP disclosed
EP-4247787-A2 METHODS AND COMPOSITION FOR KRAS MODIFICATIONS 2692372 Ontario, Inc. (CA) 2023-09-27 EP disclosed
EP-3546454-B1 BENZOHETEROCYCLYL ALKYLAMINE COMPOUND AND USE THEREOF UNIV EAST CHINA SCIENCE & TECH (CN) 2023-09-27 EP disclosed
CN-116804020-A Nitrogen-containing heterocyclic organic compound and application thereof in OLED device 北京燕化集联光电技术有限公司 2023-09-26 CN disclosed
US-11767295-B2 Isoindole derivative TIANJIN HEMAY PHARMACEUTICAL CO., LTD. (CN) 2023-09-26 US disclosed
CN-112011002-B Method of controlled radical polymerization and apparatus for controlled radical polymerization 立邦工业涂料(上海)有限公司 2023-09-26 CN disclosed
CN-114853739-B Acetylenic pyrazine FGFR inhibitor and preparation method and application thereof 药雅科技(上海)有限公司 2023-09-22 CN disclosed
CN-116785342-A Compositions and methods for managing or improving bone disorders, cartilage disorders, or both 尤尼根公司 2023-09-22 CN disclosed
CN-113185740-B Method for improving antibacterial activity and biocompatibility of substrate surface 华东理工大学 2023-09-22 CN disclosed
CN-116789677-A Organic electroluminescent compound and application thereof 北京燕化集联光电技术有限公司 2023-09-22 CN disclosed
US-20230295115-A1 SUBSTITUTED ISOQUINOLINYLMETHYL AMIDES, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORP (CA) 2023-09-21 US disclosed
WO-2023175536-A1 LIPID MONOMERS FOR THERAPEUTIC DELIVERY OF RNA JANSSEN BIOTECH, INC. (US) 2023-09-21 WO disclosed
US-20230295135-A1 CERTAIN CHEMICAL COMPOSITIONS AND METHODS OF USE THEREOF ALGEN BIOTECHNOLOGIES, INC. 2023-09-21 US disclosed
US-20230295075-A1 LIPIDS FOR USE IN LIPID NANOPARTICLE FORMULATIONS Acuitas Therapeutics, Inc. (CA) 2023-09-21 US disclosed
US-20230293524-A1 OTIC FORMULATIONS FOR DRUG-INDUCED OTOTOXICITY SPIRAL THERAPEUTICS INC. 2023-09-21 US disclosed
US-20230295138-A1 HETEROCYCLYL PYRIDINES AS NOVEL FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-09-21 US disclosed
US-20230292741-A1 NOVEL SUPERCOOLING METHODS FOR PRESERVATION OF BIOLOGICAL SAMPLES X-THERMA, INC. (US) 2023-09-21 US disclosed
US-20230295201-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. 2023-09-21 US disclosed
WO-2023178144-A2 GALNAC COMPOSITIONS FOR IMPROVING SIRNA BIOAVAILABILITY EMPIRICO INC. (US) 2023-09-21 WO disclosed
WO-2023175615-A1 ARTS MIMETIC COMPONDS AND COMBINATIONS THEREOF FOR TREATING HIGH-RISK NEUROBLASTOMA CARMEL-HAIFA UNIVERSITY ECONOMIC CORPORATION LTD. (IL) 2023-09-21 WO disclosed
US-20230295106-A1 ERGOLINE-LIKE COMPOUNDS FOR PROMOTING NEURAL PLASTICITY DELIX THERAPEUTICS, INC. 2023-09-21 US disclosed
US-20230295630-A1 GALNAC COMPOSITIONS FOR IMPROVING SIRNA BIOAVAILABILITY EMPIRICO INC. 2023-09-21 US disclosed
EP-4244625-A1 ADDITIVES FOR REDUCING NON-SPECIFIC INTERACTIONS BETWEEN FLUORESCENT POLYMER CONJUGATES AND CELLS IN A BIOLOGICAL SAMPLE Beckman Coulter, Inc. (US) 2023-09-20 EP disclosed
EP-3159344-B1 AMINO PYRANOID RING DERIVATIVE AND COMPOSITION AND USE THEREOF SICHUAN HAISCO PHARMACEUTICAL CO LTD (CN) 2023-09-20 EP disclosed
EP-4244203-A1 SUBSTITUTED PROPANE-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC (US) 2023-09-20 EP disclosed
EP-4244204-A1 SUBSTITUTED MONO- AND POLY-PHENYL-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC (US) 2023-09-20 EP disclosed
CN-116783188-A Dihydro-isoquinolone derivative and application thereof 上海奕拓医药科技有限责任公司 2023-09-19 CN disclosed
US-11760752-B2 Carboxylic acid, acyl sulfonamide and acyl sulfamide-derivatized bicyclic aza-heteroaromatics as selective Mcl-1 inhibitors and as dual Mcl-1/Bcl-2 inhibitors UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-09-19 US disclosed
US-11759780-B2 Modification of surface properties of microfluidic devices BIO-RAD LABORATORIES, INC. (US) 2023-09-19 US disclosed
CN-116751156-A Substituted 3-dialkylaminomethyl-piperidin-4-yl-benzamides and methods of making and using the same 梅比斯发现公司 2023-09-15 CN disclosed
CN-116761635-A BCL-XL inhibitor antibody drug conjugates and methods of use thereof 诺华股份有限公司 2023-09-15 CN disclosed
CN-116751200-A Tricyclic compounds containing substituted pyridones and methods of using the same 爱彼特生物制药公司 2023-09-15 CN disclosed
CN-111138412-B Spiro aromatic ring compound and application thereof 上海奕拓医药科技有限责任公司 2023-09-15 CN disclosed
CN-114075196-B Aromatic ring lactam compound, preparation method and application thereof 上海凌达生物医药有限公司 2023-09-15 CN disclosed
CN-116761510-A Use of [ (1, 5-diphenyl-1H-pyrazol-3-yl) oxy ] acetic acid derivatives and salts thereof and compositions containing them for reducing the phytotoxic effect of agrochemicals, in particular herbicides, on useful plants and crops 拜耳公司 2023-09-15 CN disclosed
CN-114751903-B Nitrogen-containing fused heterocycle SHP2 inhibitor compound, preparation method and application 上海凌达生物医药有限公司 2023-09-15 CN disclosed
US-20230286902-A1 LIPID NANOPARTICLE COMPOSITION Suzhou Abogen Biosciences Co., Ltd. (CN) 2023-09-14 US disclosed
WO-2023278691-A9 METHODS OF TREATING OR PREVENTING CORONAVIRUS INFECTION WITH CANNABINOID ACIDS OREGON STATE UNIVERSITY (US) 2023-09-14 WO disclosed
US-20230285378-A1 Anti-Viral Compounds ABBVIE INC. (US) 2023-09-14 US disclosed
WO-2023168484-A1 \"COMPOUNDS AND METHODS\ DemAgtech Pty Ltd (AU) 2023-09-14 WO disclosed
WO-2023170160-A1 POLYMERIC IMIDAZOLIUM COMPOUNDS FOR ENHANCING THE ACTIVITY OF ANTIMICROBIAL AGENTS BASF SE (DE) 2023-09-14 WO disclosed
US-20230286917-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2023-09-14 US disclosed
US-20230286934-A1 Use of Multi-Kinase Inhibitors to Treat RNA Virus Infections ICAHN SCHOOL MED MOUNT SINAI (US) 2023-09-14 US disclosed
WO-2023169438-A1 NITROGEN-CONTAINING HETEROCYCLIC CELL CYCLE INHIBITOR COMPOUNDS AS WELL AS PREPARATION METHOD THEREFOR AND USE THEREOF 上海凌达生物医药有限公司 2023-09-14 WO disclosed
WO-2023170142-A1 PRINTABLE SUBSTRATES WITH BARRIER PROPERTIES KNOWFORT HOLDING B.V. (NL) 2023-09-14 WO disclosed
US-20230286983-A1 PYRIDINE-1,5-DIONES EXHIBITING MNK INHIBITION AND THEIR METHOD OF USE NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-09-14 US disclosed
EP-4240723-A1 USE OF [(1,5-DIPHENYL-1H-PYRAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AND THEIR SALTS AND COMPOSITIONS CONTAINING THEM, FOR REDUCING PHYTOTOXIC EFFECTS OF AGROCHEMICALS, IN PARTICULAR OF HERBICIDES, IN USEFUL PLANTS AND CROP PLANTS Bayer Aktiengesellschaft (DE) 2023-09-13 EP disclosed
EP-4242255-A1 PRINTABLE SUBSTRATES WITH BARRIER PROPERTIES Knowfort Holding B.V. (NL) 2023-09-13 EP disclosed
EP-4240727-A1 [(5-PHENYL-5-HETEROARYL-1H-PYRAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS Bayer Aktiengesellschaft (DE) 2023-09-13 EP disclosed
EP-3774735-B1 ENANTIOSELECTIVE HYDROGENATION OF 4-SUBSTITUTED 1,2-DIHYDROQUINOLINES IN PRESENCE OF A CHIRAL IRIDIUM CATALYST BAYER AG (DE) 2023-09-13 EP disclosed
EP-4240355-A1 INHIBITING AN IMMUNE RESPONSE MEDIATED BY ONE OR MORE OF TLR2, RAGE, CCR5, CXCR4 AND CD4 Cassava Sciences, Inc. (US) 2023-09-13 EP disclosed
EP-4240725-A1 [(1-PHENYL-5-HETEROARYL-1H-PYRAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS Bayer Aktiengesellschaft (DE) 2023-09-13 EP disclosed
EP-4240726-A1 [(1-PHENYL-5-(HETEROARYL)-1H-1,2,4-TRIAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS Bayer Aktiengesellschaft (DE) 2023-09-13 EP disclosed
EP-4241541-A1 SELF-HEALABLE, RECYCLABLE, AND RECONFIGURABLE WEARABLE ELECTRONICS DEVICE The Regents of the University of Colorado, a body corporate (US) 2023-09-13 EP disclosed
EP-3661517-B1 DIHYDROOXADIAZINONES BAYER AG (DE) 2023-09-13 EP disclosed
EP-4242204-A1 CD73 INHIBITOR AND USE THEREOF Wuhan Humanwell Innovative Drug Research and Development Center Limited Company (CN) 2023-09-13 EP disclosed
EP-4240728-A1 [(5-PHENYL-1-HETEROARYL-1H-TRIAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS Bayer Aktiengesellschaft (DE) 2023-09-13 EP disclosed
EP-4240731-A1 [(1,5-DIHETEROARYL-1H-1,2,4-TRIAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS Bayer Aktiengesellschaft (DE) 2023-09-13 EP disclosed
CN-116745285-A [ (1-phenyl-5- (heteroaryl) -1H-1,2, 4-triazol-3-yl) oxy ] acetic acid derivatives as safeners for protecting useful plants and crop plants 拜耳公司 2023-09-12 CN disclosed
US-11752146-B2 Anti-inflammatory, anti-cancer, and anti-angiogenic compounds, pharmaceutical compositions, and methods of making and using thereof MEDICON PHARMACEUTICALS, INC. (US) 2023-09-12 US disclosed
CN-116730920-A AG-10 preparation method, intermediate and salt thereof 文涵治疗有限公司 2023-09-12 CN disclosed
CN-116730921-A AG-10 preparation method, intermediate and salt thereof 文涵治疗有限公司 2023-09-12 CN disclosed
CN-116745268-A Benzenesulfonamide derivatives and uses thereof 2692372安大略公司 2023-09-12 CN disclosed
US-11752149-B2 Muscarinic acetylcholine M1 receptor antagonists Pipeline Therapeutics, Inc. (US) 2023-09-12 US disclosed
CN-116745264-A Methods and compositions for KRAS modification 2692372安大略公司 2023-09-12 CN disclosed
US-11753395-B2 Inhibitors of MET kinase KINNATE BIOPHARMA INC. (US) 2023-09-12 US disclosed
CN-111542324-B Cytotoxic agent and conjugate thereof, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-09-12 CN disclosed
CN-116724043-A Photodynamic therapy and diagnosis RMW曹氏集团有限公司 2023-09-08 CN disclosed
CN-116715668-A Nitrogen-containing heterocyclic cell cycle inhibitor compound, preparation method and application 上海凌达生物医药有限公司 2023-09-08 CN disclosed
US-20230276788-A1 COMPOSITIONS AND METHODS FOR REDUCING ICE CRYSTAL FORMATION X-THERMA, INC. 2023-09-07 US disclosed
WO-2023168291-A1 COVALENT MODIFIERS OF AKT1 AND USES THEREOF TERREMOTO BIOSCIENCES, INC. (US) 2023-09-07 WO disclosed
US-20230277652-A1 NUCLEIC ACID VACCINES FOR CORONAVIRUS SUZHOU ABOGEN BIOSCIENCES CO LTD (CN) 2023-09-07 US disclosed
WO-2023168203-A1 INHIBITORS OF MEK KINASE KINNATE BIOPHARMA INC. (US) 2023-09-07 WO disclosed
WO-2023168254-A1 ANTIVIRAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. (US) 2023-09-07 WO disclosed
WO-2023166507-A1 APOPTOSIS RELATED PROTEIN IN THE TGF-BETA SIGNALING PATHWAY (ARTS) AND ARTS MIMETIC SMALL MOLECULE COMPOUNDS FOR UPREGULATING P53 LEVEL CARMEL-HAIFA UNIVERSITY ECONOMIC CORPORATION LTD. (IL) 2023-09-07 WO disclosed
US-20230277616-A9 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC. 2023-09-07 US disclosed
US-20230278994-A1 HETEROCYCLYL PYRIMIDINES AND TRIAZINES AS NOVEL FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-09-07 US disclosed
US-20230279033-A1 INHIBITORS OF MEK KINASE MOSAICA MEDICINES, INC. 2023-09-07 US disclosed
US-20230279026-A1 NOVEL BICYCLIC SUBSTITUTED SULFONYLUREA COMPOUNDS AS INHIBITORS OF INTERLEUKIN-1 ACTIVITY VIVA STAR BIOSCIENCES (SUZHOU) CO., LTD. (CN) 2023-09-07 US disclosed
WO-2023165958-A1 SUBSTITUTED 1,2,4-THIADIAZOLYL ISONICOTINAMIDES, SALTS OR N-OXIDES THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2023-09-07 WO disclosed
WO-2023166488-A1 BROAD SPECTRUM AMINOGLYCOSIDES AND USES THEREOF REVAGENIX, INC. (US) 2023-09-07 WO disclosed
EP-4238972-A1 SUBSTITUTED 1,2,4-THIADIAZOLYL PICOLINAMIDES, SALTS OR N-OXIDES THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES Bayer AG (DE) 2023-09-06 EP disclosed
EP-4238973-A1 SUBSTITUTED 1,2,4-THIADIAZOLYL ISONICOTINAMIDES, SALTS OR N-OXIDES THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES Bayer AG (DE) 2023-09-06 EP disclosed
EP-3436445-B1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2023-09-06 EP disclosed
EP-4236944-A1 BICYCLIC COMPOUNDS AND USES THEREOF FOR THE TREATMENT OF DISEASES Athira Pharma, Inc. (US) 2023-09-06 EP disclosed
EP-3316890-B1 NOVEL BREATHING CONTROL MODULATING COMPOUNDS, AND METHODS OF MAKING AND USING SAME NEURAD LTD (IL) 2023-09-06 EP disclosed
EP-4237423-A1 SUBSTITUTED 1H-PYRAZOLO[4,3-C]PYRIDINES AND DERIVATIVES AS EGFR INHIBITORS Boehringer Ingelheim International GmbH (DE) 2023-09-06 EP disclosed
EP-3475387-B1 PHOTOCHROMIC WATER HARVESTING PLATFORM WARNER BABCOCK INST FOR GREEN CHEMISTRY LLC (US) 2023-09-06 EP disclosed
CN-116693411-A Novel carbonyl lipid and lipid nanoparticle formulations for delivery of nucleic acids 爱康泰生治疗公司 2023-09-05 CN disclosed
CN-116709916-A [ (1-phenyl-5-heteroaryl-1H-pyrazol-3-yl) oxy ] acetic acid derivatives as safeners for protecting useful plants and crop plants 拜耳公司 2023-09-05 CN disclosed
CN-116710457-A Spirocyclic compounds as KRAS-G12C inhibitors 上海优理惠生医药有限公司 2023-09-05 CN disclosed
US-11749839-B2 Silicon-based energy storage devices with electrolyte containing sulfonate or carboxylate salt based compounds ENEVATE CORPORATION (US) 2023-09-05 US disclosed
US-11746095-B2 Inhibtors of RAF kinases KINNATE BIOPHARMA INC. (US) 2023-09-05 US disclosed
CN-116693542-A Tetrahydroquinoline compound containing spiro structure and preparation method thereof 云南农业大学 2023-09-05 CN disclosed
US-11746123-B2 Efficient and scalable syntheses of nicotinoyl ribosides and reduced nicotinoyl ribosides, modified derivatives thereof, phosphorylated analogs thereof, adenylyl dinucleotide conjugates thereof, and novel crystalline forms thereof THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2023-09-05 US disclosed
US-11745147-B2 Curable poly(RTIL)-based mixed-matrix membranes and methods using same THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2023-09-05 US disclosed
CN-116685316-A Compositions and methods for treating lipid-related disorders 拉结尔治疗有限公司 2023-09-01 CN disclosed
CN-116675674-A Novel substituted benzimidazole derivatives as inhibitors of D-amino acid oxidase (DAAO) 宇凤·简·曾 2023-09-01 CN disclosed
WO-2023163971-A1 METHODS OF TREATING COVID-RELATED DISORDERS ATHIRA PHARMA, INC. (US) 2023-08-31 WO disclosed
US-20230270700-A1 PHARMACOLOGY OF VISUAL CYCLE MODULATORS ACUCELA INC. 2023-08-31 US disclosed
WO-2023161940-A1 APOPTOSIS RELATED PROTEIN IN THE TGF-BETA SIGNALING PATHWAY (ARTS) MIMETIC COMPOUNDS, COMPOSITIONS, METHODS AND USES THEREOF IN INDUCTION OF APOPTOSIS CARMEL-HAIFA UNIVERSITY ECONOMIC CORPORATION LTD. (IL) 2023-08-31 WO disclosed
WO-2023164057-A1 DI-CYCLOPROPYL BASED IL-17A MODULATORS AND USES THEREOF DICE ALPHA, INC. (US) 2023-08-31 WO disclosed
US-20230275230-A1 AQUEOUS BASED POLYMERS FOR SILICON ANODES ENEVATE CORPORATION 2023-08-31 US disclosed
WO-2023161172-A1 SUBSTITUTED N-BENZOIC ACID URACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2023-08-31 WO disclosed
EP-3699184-B1 TRIPTOLIDE DERIVATIVE AND PREPARATION METHOD THEREFOR AND USE THEREOF CINKATE PHARMACEUTICAL INTERMEDIATES CO LTD (CN) 2023-08-30 EP disclosed
EP-3151919-B1 CARBON MONOXIDE-RELEASING MOLECULES FOR THERAPEUTIC APPLICATIONS AND METHODS OF MAKING AND USING THEREOF UNIV GEORGIA STATE RES FOUND (US) 2023-08-30 EP disclosed
EP-4233865-A2 ARYL-ANILINE AND HETEROARYL-ANILINE COMPOUNDS FOR TREATMENT OF SKIN CANCERS NFlection Therapeutics, Inc. (US) 2023-08-30 EP disclosed
EP-4233871-A2 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL Eli Lilly and Company (US) 2023-08-30 EP disclosed
EP-4233834-A2 ARYL-ANILINE AND HETEROARYL-ANILINE COMPOUNDS FOR TREATMENT OF BIRTHMARKS NFlection Therapeutics, Inc. (US) 2023-08-30 EP disclosed
CN-106715456-B Prodrugs of directed lymphatics 莫纳什大学 2023-08-29 CN disclosed
US-11742519-B2 Silicon-based energy storage devices with electrolyte additive compounds ENEVATE CORPORATION (US) 2023-08-29 US disclosed
US-11738087-B2 Lymph directing prodrugs MONASH UNIVERSITY (AU) 2023-08-29 US disclosed
CN-116669727-A Triazole-pyridinyl substituted azacyclohexylacetic acid compounds as LPA receptor antagonists 唯久生物有限公司 2023-08-29 CN disclosed
CN-116670267-A Tetravalent mRNA vaccine for influenza virus 苏州艾博生物科技有限公司 2023-08-29 CN disclosed
CN-116670928-A Self-healing, recyclable and reconfigurable wearable electronic device 科罗拉多大学评议会公司 2023-08-29 CN disclosed
US-11739077-B2 Small molecule inhibitors of ubiquitin specific protease 1 (USP1) and uses thereof INSILICO MEDICINE IP LIMITED (HK) 2023-08-29 US disclosed
US-11739223-B2 Surface primer compositions and methods of use ENVISTA (US) 2023-08-29 US disclosed
CN-111448226-B Polymerization process 埃克森美孚化学专利公司 2023-08-25 CN disclosed
CN-116640140-A Polycyclic-carbamoyl pyridone compounds and pharmaceutical uses thereof 吉利德科学公司 2023-08-25 CN disclosed
CN-116640157-A METTL3 inhibitor and composition thereof and application of METTL3 inhibitor and composition thereof in medicine 海思科医药集团股份有限公司 2023-08-25 CN disclosed
CN-111526877-B Compounds and compositions for IRE1 inhibition 奥普提卡拉公司 2023-08-25 CN disclosed
CN-116648472-A Bioactive synthetic copolymers, bioactive macromolecules and related methods 新加坡科技研究局 2023-08-25 CN disclosed
CN-116648471-A Bioactive polyethylene copolymers, polyethylene macromolecules and related methods 新加坡科技研究局 2023-08-25 CN disclosed
WO-2023158824-A1 NOVEL BICYCLIC SUBSTITUTED SULFONYLUREA COMPOUNDS AS INHIBITORS OF INTERLEUKIN- 1 ACTIVITY VIVA STAR BIOSCIENCES (SUZHOU) CO., LTD. (CN) 2023-08-24 WO disclosed
WO-2023155808-A1 CONJUGATE OF ANTIBODY-ERIBULIN OR DERIVATIVE THEREOF, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 苏州宜联生物医药有限公司 2023-08-24 WO disclosed
US-20230265173-A1 SULFONAMIDE-CONTAINING LINKAGE SYSTEMS FOR DRUG CONJUGATES ZYMEWORKS BC INC. (CA) 2023-08-24 US disclosed
US-20230263790-A1 HISTONE DEACETYLASE INHIBITORS FOR IMMUNOMODULATION IN TUMOR MICROENVIRONMENT Great Novel Therapeutics Biotech & Medicals Corporation (TW) 2023-08-24 US disclosed
EP-4228601-A1 IN VIVO TARGETING OF FIBROSIS BY ANTI-CD5-TARGETED FAP-CAR T MRNA-LNP The Trustees of the University of Pennsylvania (US) 2023-08-23 EP disclosed
EP-3370518-B1 COMPOSITIONS AND METHODS FOR REDUCING ICE CRYSTAL FORMATION X THERMA INC (US) 2023-08-23 EP disclosed
EP-4230620-A1 SUBSTITUTED N-AMINO-N-BENZOIC ACID URACILS, THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS Bayer Aktiengesellschaft (DE) 2023-08-23 EP disclosed
EP-4228602-A1 IN VIVO TARGETING OF T CELLS FOR MRNA THERAPEUTICS The Trustees of the University of Pennsylvania (US) 2023-08-23 EP disclosed
EP-4229045-A1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER The Broad Institute Inc. (US) 2023-08-23 EP disclosed
EP-4230621-A1 SUBSTITUTED N-BENZOIC ACID URACILS, THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS Bayer AG (DE) 2023-08-23 EP disclosed
CN-115043832-B FGFR inhibitor acetylenic heterocyclic compound and preparation method and application thereof 药雅科技(上海)有限公司 2023-08-22 CN disclosed
CN-113816990-B Modified amino acids and their use in ADCs 联宁(苏州)生物制药有限公司 2023-08-22 CN disclosed
CN-114957242-B Preparation and application of pyrido heterocyclic compounds as kinase inhibitors 药雅科技(上海)有限公司 2023-08-22 CN disclosed
CN-115141176-B Acetylenic indole FGFR inhibitor and preparation method and application thereof 药雅科技(上海)有限公司 2023-08-22 CN disclosed
CN-113939544-B non-core-shell polymer particles 悉尼大学 2023-08-22 CN disclosed
CN-114957241-B Preparation and Application of Heterocyclic Compounds as Kinase Inhibitors 药雅科技(上海)有限公司 2023-08-22 CN disclosed
US-11731954-B2 Histone demethylase inhibitors CELGENE QUANTICEL RES INC (US) 2023-08-22 US disclosed
CN-116635023-A Ionic liquid preparation for treating diabetes I2O治疗公司 2023-08-22 CN disclosed
CN-114853752-B Preparation and application of BTK inhibitor pyrido heterocyclic compound 药雅科技(上海)有限公司 2023-08-22 CN disclosed
US-11732259-B2 Peptide oligonucleotide conjugates SAREPTA THERAPEUTICS, INC. (US) 2023-08-22 US disclosed
CN-116615468-A Polymer particles 昆士兰科技大学 2023-08-18 CN disclosed
CN-116615428-A Tricyclic pyridones and pyrimidinones 医睿世康药业研发公司 2023-08-18 CN disclosed
CN-116615472-A Polymer conjugated lipid compounds and lipid nanoparticle compositions 苏州艾博生物科技有限公司 2023-08-18 CN disclosed
US-20230257380-A1 TROPOMYOSIN RECEPTOR KINASE (TRK) DEGRADATION COMPOUNDS AND METHODS OF USE CULLGEN (SHANGHAI), INC. (CN) 2023-08-17 US disclosed
US-20230257428-A1 METHODS OF TREATMENT USING CHLOROTOXIN CONJUGATES Blaze Bioscience, Inc. 2023-08-17 US disclosed
WO-2023154822-A2 METHODS OF PURIFYING A PRODUCT KODIAK SCIENCES INC. (US) 2023-08-17 WO disclosed
US-20230255945-A1 FORMULATIONS OF PYRROLOPYRIDINE-ANILINE COMPOUNDS NFLECTION THERAPEUTICS, INC. 2023-08-17 US disclosed
US-20230257374-A1 NOVEL KRAS G12C PROTEIN INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF INNOVENT BIOLOGICS (SUZHOU) CO., LTD. (CN) 2023-08-17 US disclosed
WO-2023154766-A1 KRAS MODULATORS AND USES THEREOF QUANTA THERAPEUTICS, INC. (US) 2023-08-17 WO disclosed
EP-3253752-B1 [9,10-DIMETHOXY-3-(2-METHYLPROPYL)-1H,2H,3H,4H,6H,7H,11BH-PYRIDO-[2,1-A]ISOQUINOLIN-2-YL]METHANOL AND COMPOUNDS, COMPOSITIONS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES INC (US) 2023-08-16 EP disclosed
EP-4225915-A1 OLIGOMERIC COMPOUND FOR DYSTROPHIN RESCUE IN DMD PATIENTS THROUGHOUT SKIPPING OF EXON-51 SQY Therapeutics (FR) 2023-08-16 EP disclosed
EP-4225811-A1 POLYMER PARTICLES Queensland University Of Technology (AU) 2023-08-16 EP disclosed
EP-3959202-B1 ACYL SULFONAMIDES FOR TREATING CANCER BAYER AG (DE) 2023-08-16 EP disclosed
CN-111410659-B PDE9 inhibitors and uses thereof 药捷安康(南京)科技股份有限公司 2023-08-15 CN disclosed
CN-111909083-B Inhibitors of histone demethylase 赛尔基因昆蒂赛尔研究公司 2023-08-15 CN disclosed
CN-116601152-A Pyrrolopyridine-anilines for the treatment of cognitive dysfunction 恩福莱克逊治疗有限公司 2023-08-15 CN disclosed
US-11723944-B2 Botulinum neurotoxin-specific capture agents, compositions, and methods of using and making INDI MOLECULAR, INC. (US) 2023-08-15 US disclosed
CN-116570594-A Selective p38α -specific MAPK inhibitors 马里兰大学巴尔的摩分校 2023-08-11 CN disclosed
CN-116583509-A Compounds and methods for treating cancer 上海睿跃生物科技有限公司 2023-08-11 CN disclosed
CN-116574104-A Biaryl benzylamine compound, preparation method and application 如东凌达生物医药科技有限公司 2023-08-11 CN disclosed
CN-116574105-A Quinoline derivatives having indoleamine-2, 3-dioxygenase inhibitory activity 深圳微芯生物科技股份有限公司 2023-08-11 CN disclosed
WO-2023150663-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS RETUNE PHARMA INC. (US) 2023-08-10 WO disclosed
WO-2023150681-A1 INHIBITORS OF RAF KINASES KINNATE BIOPHARMA INC. (US) 2023-08-10 WO disclosed
US-20230248736-A1 SELECTIVE P2X3 MODULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.3) LIMITED (GB) 2023-08-10 US disclosed
US-20230250536-A1 MODIFICATION OF METALLIC SURFACES WITH PHOSPHONIC ACIDS BIOLOGICAL DYNAMICS, INC. 2023-08-10 US disclosed
US-20230250104-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELLTAXIS LLC (US) 2023-08-10 US disclosed
US-20230248752-A1 PRODRUGS OF ALOX-15 INHIBITORS AND METHODS OF USING THE SAME EMPIRICO INC. 2023-08-10 US disclosed
US-20230250133-A1 METHODS OF PURIFYING A PRODUCT KODIAK SCIENCES GMBH (CH) 2023-08-10 US disclosed
US-20230248835-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR THE TREATMENT OF FIBROTIC DISEASES AND CANCER PURDUE RESEARCH FOUNDATION 2023-08-10 US disclosed
US-20230250169-A1 AXL Inhibitors for Antiviral Therapy BERGENBIO ASA (NO) 2023-08-10 US disclosed
EP-3966202-B1 THIANTHRENE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS FACEBOOK TECH LLC (US) 2023-08-09 EP disclosed
US-11718609-B2 Heparanase inhibitors and use thereof Beta Therapeutics Pty Ltd (AU) 2023-08-08 US disclosed
CN-116568669-A Substituted mono-and poly-benzene nuclear monomers and polymers thereof for volume Bragg gratings 元平台技术有限公司 2023-08-08 CN disclosed
CN-116554461-A Use of polymers to promote endothelialization of interventional/implant materials 华东理工大学 2023-08-08 CN disclosed
CN-116549598-A Polypeptide polymer or polypeptide mimic and application thereof in treating tumors 华东理工大学 2023-08-08 CN disclosed
US-11718580-B2 Fluorene derivatized monomers and polymers for volume Bragg gratings META PLATFORMS TECHNOLOGIES, LLC (US) 2023-08-08 US disclosed
CN-116568136-A [ (5-phenyl-1-heteroaryl-1H-triazol-3-yl) oxy ] acetic acid derivatives as safeners for protecting useful plants and crop plants 拜耳公司 2023-08-08 CN disclosed
CN-116568301-A Bicyclic compounds for treating diseases and uses thereof 雅斯娜制药公司 2023-08-08 CN disclosed
US-11718620-B2 Method for treating a cancer mediated by abnormality of multi-kinases TRANSTHERA SCIENCES (NANJING), INC. (CN) 2023-08-08 US disclosed
CN-116554147-A Pyrazole derivative, composition and pharmaceutical application thereof 四川海思科制药有限公司 2023-08-08 CN disclosed
CN-116554166-A Pyridazinopyridone compound, pharmaceutical composition and application thereof 上海优理惠生医药有限公司 2023-08-08 CN disclosed
US-11721809-B2 Silicate and organosilicon containing additives for silicon-based Li ion batteries ENEVATE CORPORATION (US) 2023-08-08 US disclosed
US-11718595-B2 Non-ATP/catalytic site p38 Mitogen Activated Protein Kinase inhibitors UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-08-08 US disclosed
CN-116547281-A Isoxazolidines as RIPK1 inhibitors and uses thereof 赛诺菲 2023-08-04 CN disclosed
CN-116546991-A mRNA therapeutic agent versus CD4 + In vivo targeting of T cells 宾夕法尼亚大学理事会 2023-08-04 CN disclosed
US-20230242514-A1 BICYCLIC INDAZOLE GLUCOCORTICOID RECEPTOR ANTAGONISTS CORCEPT THERAPEUTICS INCORPORATED 2023-08-03 US disclosed
US-20230241034-A1 MICROTUBULE POLYMERIZATION INHIBITOR PRODRUGS AND METHODS OF USING THE SAME UNIV MARYLAND (US) 2023-08-03 US disclosed
WO-2023147372-A1 INHIBITORS OF CDK4/6 KINASE KINNATE BIOPHARMA INC. (US) 2023-08-03 WO disclosed
WO-2023143147-A1 PYRIDAZOPYRIDONE COMPOUNDS, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 上海优理惠生医药有限公司 2023-08-03 WO disclosed
US-20230242538-A1 PanK Modulators and Methods Using Same UNIV YALE (US) 2023-08-03 US disclosed
WO-2023143263-A1 ANTIBODY AGAINST HER3, CONJUGATE AND USE THEREOF 苏州宜联生物医药有限公司 2023-08-03 WO disclosed
WO-2023147312-A1 AMPK AGONISTS AND METHODS OF USE THEREOF EVVIA THERAPEUTICS, INC. (US) 2023-08-03 WO disclosed
WO-2023143210-A1 PHTHALAZINONE COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION CONTAINING PHTHALAZINONE COMPOUNDS AND USES THEREOF 上海优理惠生医药有限公司 2023-08-03 WO disclosed
US-20230242551-A1 ISOTOPE-SUBSTITUTED SPIRO AROMATIC RING COMPOUND AND APPLICATION THEREOF ETERN BIOPHARMA (SHANGHAI) CO., LTD. (CN) 2023-08-03 US disclosed
WO-2023146831-A1 NOVEL EXCITATORY AMINO ACID GLUTAMATE TRANSPORT MODULATORS AND METHODS USING THE SAME DREXEL UNIVERSITY (US) 2023-08-03 WO disclosed
WO-2023146512-A1 COMPOUNDS AND METHODS OF USE THEREOF VIVACE THERAPEUTICS, INC. (US) 2023-08-03 WO disclosed
WO-2023143312-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海艾力斯医药科技股份有限公司 2023-08-03 WO disclosed
WO-2023146513-A1 COMPOUNDS AND METHODS OF USE THEREOF VIVACE THERAPEUTICS, INC. (US) 2023-08-03 WO disclosed
WO-2023146511-A1 COMPOUNDS AND METHODS OF USE THEREOF VIVACE THERAPEUTICS, INC. (US) 2023-08-03 WO disclosed
EP-3898612-B1 SUBSTITUTED PYRIDINYLOXYBENZENES, THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS BAYER AG (DE) 2023-08-02 EP disclosed
EP-4216952-A1 TREATMENT OF COGNITIVE DYSFUNCTION WITH PYRROLOPYRIDINE-ANILINE COMPOUNDS NFlection Therapeutics, Inc. (US) 2023-08-02 EP disclosed
EP-4219460-A1 TRANSGLUTAMINASE 2 (TG2) INHIBITORS Sitari Pharma, Inc. (US) 2023-08-02 EP disclosed
EP-4219493-A1 BENZYLAMINO SUBSTITUTED PYRIDOPYRIMIDINONES AND DERIVATIVES AS SOS1 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2023-08-02 EP disclosed
US-11712481-B2 Lipid nanoparticle formulations Acuitas Therapeutics, Inc. (CA) 2023-08-01 US disclosed
CN-112262145-B 2-aminopyrimidine derivative and preparation method and application thereof 上海奕拓医药科技有限责任公司 2023-08-01 CN disclosed
CN-114853740-B Preparation method and application of acetylenic pyrimidine compound as FGFR inhibitor 药雅科技(上海)有限公司 2023-08-01 CN disclosed
US-11713321-B2 Inhibitors of NEK7 kinase Halia Therapeutics, Inc. (US) 2023-08-01 US disclosed
CN-107216312-B Compound with mutant IDH inhibitory activity, preparation method and application thereof 上海海和药物研究开发股份有限公司 2023-08-01 CN disclosed
CN-116528674-A [ (1, 5-bis (heteroaryl) -1H-1,2, 4-triazol-3-yl) oxy ] acetic acid derivatives as safeners for protecting useful plants and crop plants 拜耳公司 2023-08-01 CN disclosed
CN-116529248-A Benzene ring derivative, composition and pharmaceutical application thereof 四川海思科制药有限公司 2023-08-01 CN disclosed
CN-116496318-A Heterocyclic derivative, composition and pharmaceutical application thereof 四川海思科制药有限公司 2023-07-28 CN disclosed
CN-116507333-A Cyclic AMP response element binding protein (CBP) and/or 300KDA adenovirus E1A binding protein (P300) degrading compounds and methods of use 上海睿跃生物科技有限公司 2023-07-28 CN disclosed
CN-116507618-A Spiro compound, pharmaceutical composition containing spiro compound and application of spiro compound 上海优理惠生医药有限公司 2023-07-28 CN disclosed
WO-2023141364-A1 SILYL-LIPID N-ACYL L-HOMOSERINE LACTONES AS QUORUM SENSING MOLECULES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-07-27 WO disclosed
US-20230233706-A1 In vivo targeting of CD4+-T cells for mRNA therapeutics THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2023-07-27 US disclosed
US-20230234945-A1 AZABICYCLYL-SUBSTITUTED HETEROCYCLES AS FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-07-27 US disclosed
US-20230233468-A1 LIPID COMPOUNDS AND LIPID NANOPARTICLE COMPOSITIONS Suzhou Abogen Biosciences Co., Ltd. (CN) 2023-07-27 US disclosed
EP-4213835-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF LIPID-RELATED DISORDERS Raziel Therapeutics Ltd. (IL) 2023-07-26 EP disclosed
EP-4213827-A1 AQUEOUS PHARMACEUTICAL FORMULATION OF HYDROCORTISONE SODIUM PHOSPHATE AND MONOTHIOGLYCEROL Antares Pharma, Inc. (US) 2023-07-26 EP disclosed
EP-4065564-B1 [ (1,5-DIPHENYL-1H-1,2,4-TRIAZOL-3-YL) OXY ] ACETIC ACID DERIVATIVES AND SALTS THEREOF, USEFUL OR CULTIVATING AGENTS CONTAINING THEM, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS SAFENERS BAYER AG (DE) 2023-07-26 EP disclosed
EP-4214204-A1 PYRIDO[2,3-D]PYRIMIDIN-4-AMINES AS SOS1 INHIBITORS Bayer Aktiengesellschaft (DE) 2023-07-26 EP disclosed
CN-116478145-A ALK2 kinase inhibitors 杭州邦顺制药有限公司 2023-07-25 CN disclosed
CN-116473965-A Pyrazole MAGL inhibitors H.隆德贝克有限公司 2023-07-25 CN disclosed
CN-116490501-A Tyrosine kinase 2 (TYK 2) degrading compounds and methods of use 上海睿跃生物科技有限公司 2023-07-25 CN disclosed
US-11710854-B2 Functional epoxides in catalyst-based electrolyte compositions for Li-ion batteries ENEVATE CORPORATION (US) 2023-07-25 US disclosed
CN-116462679-A Pyrazolopyrimidine derivative and application thereof in medicine 四川海思科制药有限公司 2023-07-21 CN disclosed
CN-116472275-A Lipid compounds and lipid nanoparticle compositions 苏州艾博生物科技有限公司 2023-07-21 CN disclosed
CN-116472292-A Modified proteins and protein degrading agents 上海睿跃生物科技有限公司 2023-07-21 CN disclosed
CN-110381940-B AG-10 preparation method, intermediate and salt thereof 文涵治疗有限公司 2023-07-21 CN disclosed
CN-110092750-B Pentafluoro sulfanyl substituted amide compound, preparation method and application thereof in medicine 北京诺诚健华医药科技有限公司 2023-07-21 CN disclosed
US-20230227458-A1 IRREVERSIBLE INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, INC. 2023-07-20 US disclosed
US-20230227470-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER VANDERBILT UNIVERSITY 2023-07-20 US disclosed
US-20230227476-A1 GALLIUM-SALOPHEN ANTIMICROBIAL COMPOUNDS AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-07-20 US disclosed
WO-2023134374-A1 PYRIMIDO-HETEROCYCLIC COMPOUND, PREPARATION METHOD, AND USE 如东凌达生物医药科技有限公司 2023-07-20 WO disclosed
EP-4212510-A1 NOVEL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS Acuitas Therapeutics Inc. (CA) 2023-07-19 EP disclosed
CN-116444497-A Pyridazinone compound, preparation and application thereof 如东凌达生物医药科技有限公司 2023-07-18 CN disclosed
US-11702388-B2 1,4-substituted piperidine derivatives 89BIO LTD (IL) 2023-07-18 US disclosed
CN-116457356-A A3 adenosine receptor agonists for use in medicine 生物干预公司 2023-07-18 CN disclosed
US-11702427-B2 Substituted 2-pyridone tricyclic compounds, analogues thereof, and methods using same ARBUTUS BIOPHARMA CORPORATION (CA) 2023-07-18 US disclosed
US-11701345-B2 Car activator agents for cyclophosphamide-based treatments of cancer UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-07-18 US disclosed
US-11701377-B2 Methods for treating cancers by prodrugs of clofarabine BoYen Therapeutics, Inc. (TW) 2023-07-18 US disclosed
CN-116457336-A Substituted propane nuclear monomer for volume Bragg grating and polymer thereof 元平台技术有限公司 2023-07-18 CN disclosed
US-11702421-B2 Substituted pyridines as irreversible inhibitors of menin-MLL interaction BIOMEA FUSION, LLC (US) 2023-07-18 US disclosed
CN-116425796-A Pyrimidine heterocyclic compounds, preparation method and application 如东凌达生物医药科技有限公司 2023-07-14 CN disclosed
CN-116438183-A Thienopyrimidine compound, pharmaceutical composition containing thienopyrimidine compound and application of thienopyrimidine compound 上海优理惠生医药有限公司 2023-07-14 CN disclosed
WO-2023131254-A1 PSEUDOURIDINE MODIFIED AT N1 POSITION AND USE THEREOF IN MRNA SYNTHESIS 上海吉量医药工程有限公司 2023-07-13 WO disclosed
US-20230219937-A1 ISOXAZOLIDINES AS RIPK1 INHIBITORS AND USE THEREOF SANOFI (FR) 2023-07-13 US disclosed
US-20230219929-A1 INHIBITORS OF MET KINASE CELYN THERAPEUTICS, INC. 2023-07-13 US disclosed
US-20230218597-A1 SUBSTITUTED PYRIDINES AND METHODS OF USE THERAVANCE BIOPHARMA R&D IP LLC (US) 2023-07-13 US disclosed
US-20230219897-A1 PYRAZOLE MAGL INHIBITORS H. LUNDBECK A/S (DK) 2023-07-13 US disclosed
US-20230218549-A1 ALKOXY COMPOUNDS FOR DISEASE TREATMENT ACUCELA INC. 2023-07-13 US disclosed
WO-2023133507-A1 ESTRADIOL PRODRUGS AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-07-13 WO disclosed
US-20230218621-A1 FATTY LIVER DISEASE TREATMENT USING GLUCOCORTICOID AND MINERALOCORTICOID RECEPTOR ANTAGONISTS CORCEPT THERAPEUTICS, INC. (US) 2023-07-13 US disclosed
US-20230219994-A1 MODIFIED NUCLEOSIDE AND SYNTHESIS METHOD THEREFOR Stemirna Therapeutics Co., Ltd. (CN) 2023-07-13 US disclosed
EP-3675847-B1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME H LUNDBECK AS (DK) 2023-07-12 EP disclosed
EP-4208160-A1 IONIC LIQUID FORMULATIONS FOR TREATING DIABETES I2O Therapeutics, Inc. (US) 2023-07-12 EP disclosed
CN-111511781-B Catalyst system and polymerization process using the same 埃克森美孚化学专利公司 2023-07-11 CN disclosed
CN-116419754-A Glucosidase inhibitors for the treatment and prevention of pulmonary infections 科威里克斯医疗有限公司 2023-07-11 CN disclosed
US-11697713-B2 Chromophoric polymer dots with narrow-band emission UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2023-07-11 US disclosed
WO-2023129502-A1 RESPIRATORY STIMULANT PARENTERAL FORMULATIONS ENALARE THERAPEUTICS INC. (US) 2023-07-06 WO disclosed
WO-2023129667-A1 PYRAZINE COMPOUNDS AS INHIBITORS OF FLT3 BIOMEA FUSION, INC. (US) 2023-07-06 WO disclosed
US-20230210857-A1 RESPIRATORY STIMULANT PARENTERAL FORMULATIONS ENALARE THERAPEUTICS INC. 2023-07-06 US disclosed
US-20230212183-A9 INHIBITORS OF KRAS G12C ARAXES PHARMA LLC (US) 2023-07-06 US disclosed
US-20230212164-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-07-06 US disclosed
US-20230212199-A1 PHOSPHOLIPID COMPOUNDS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. 2023-07-06 US disclosed
US-20230211000-A1 TISSUE-HOMING PEPTIDE CONJUGATES AND METHODS OF USE THEREOF Blaze Bioscience, Inc. 2023-07-06 US disclosed
US-20230210853-A1 TARGETED NEK7 INHIBITION FOR MODULATION OF THE NLRP3 INFLAMMASOME Halia Therapeutics, Inc. 2023-07-06 US disclosed
EP-4206199-A1 AROMATIC RING-LACTAM COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Ringene BioPharma Co., Ltd. (CN) 2023-07-05 EP disclosed
EP-3966195-B1 FLUORENE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS FACEBOOK TECH LLC (US) 2023-07-05 EP disclosed
EP-4203954-A1 GLUCOSIDASE INHIBITORS FOR THE TREATMENT AND PREVENTION OF PULMONARY INFECTIONS Covirix Medical Pty Ltd (AU) 2023-07-05 EP disclosed
EP-3541820-B1 MAGL INHIBITORS H LUNDBECK AS (DK) 2023-07-05 EP disclosed
EP-4204414-A1 COMPOUNDS AND FORMULATIONS FOR TREATING OPHTHALMIC DISEASES Viewpoint Therapeutics, Inc. (US) 2023-07-05 EP disclosed
EP-3474835-B1 NON-CATALYTIC SUBSTRATE-SELECTIVE P38 -SPECIFIC MAPK INHIBITORS WITH ENDOTHELIAL-STABILIZING AND ANTI-INFLAMMATORY ACTIVITY, AND METHODS OF USE THEREOF UNIV MARYLAND (US) 2023-07-05 EP disclosed
CN-116375742-A Azaaromatic ring derivative, composition and pharmaceutical application thereof 海思科医药集团股份有限公司 2023-07-04 CN disclosed
US-11690911-B2 Combination of ATR kinase inhibitors and PD-1/PD-L1 inhibitors BAYER AKTIENGESELLSCHAFT (DE) 2023-07-04 US disclosed
CN-110114071-B Tricyclic compounds containing substituted pyridones and methods of using the same 爱彼特生物制药公司 2023-07-04 CN disclosed
US-11691975-B2 MAGL inhibitors H. LUNDBECKA/S (DK) 2023-07-04 US disclosed
CN-110392571-B Substituted 3-dialkylaminomethyl-piperidin-4-yl-benzamides and methods of making and using the same 梅比斯发现公司 2023-07-04 CN disclosed
US-11690921-B2 Delivery of target specific nucleases SANGAMO THERAPEUTICS, INC. (US) 2023-07-04 US disclosed
CN-116354957-A CDK9 inhibitors and uses thereof 药捷安康(南京)科技股份有限公司 2023-06-30 CN disclosed
CN-111592534-B New compounds 特殊治疗有限公司 2023-06-30 CN disclosed
CN-116367835-A Aqueous pharmaceutical formulations of hydrocortisone sodium phosphate and monothioglycerol 安塔雷斯药品公司 2023-06-30 CN disclosed
US-20230201295-A1 Compositions and Methods for Managing or Improving Bone Disorders, Joint Disorders, Cartilage Disorders, or a Combination Thereof UNIGEN, INC. (US) 2023-06-29 US disclosed
US-20230203077-A1 NOVEL PRECATALYST SCAFFOLDS FOR CROSS-COUPLING REACTIONS, AND METHODS OF MAKING AND USING SAME NATIONAL SCIENCE FOUNDATION 2023-06-29 US disclosed
WO-2023115167-A1 COMPOUNDS Psylo Pty Ltd (AU) 2023-06-29 WO disclosed
WO-2023116779-A1 DIALKYNE COMPOUND AND USE THEREOF 上海艾力斯医药科技股份有限公司 2023-06-29 WO disclosed
WO-2023116707-A1 PREPARATION FOR THIOPHENE DERIVATIVE 赣州和美药业有限公司 2023-06-29 WO disclosed
US-20230203538-A1 In vivo targeting of Fibrosis by anti-CD5-targeted FAP-CAR T mRNA-LNP THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2023-06-29 US disclosed
US-20230203007-A1 PYRIDINYLACETAMIDE DERIVATIVES AS SODIUM CHANNEL ACTIVATORS X-CHEM GLOBAL HQ 2023-06-29 US disclosed
US-20230203089-A1 HEXADECAHYDRO-1H-CYCLOPENTA[A]PHENANTHRENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION TARO PHARMACEUTICALS INC. (CA) 2023-06-29 US disclosed
US-20230203018-A1 COVALENT INHIBITORS OF KRAS ARAXES PHARMA LLC (US) 2023-06-29 US disclosed
US-20230203045-A1 INHIBITORS OF NEK7 KINASE Halia Therapeutics, Inc. 2023-06-29 US disclosed
WO-2023115165-A1 COMPOUNDS Psylo Pty Ltd (AU) 2023-06-29 WO disclosed
WO-2023116763-A1 PYRIDAZINE COMPOUND, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF 上海优理惠生医药有限公司 2023-06-29 WO disclosed
WO-2023116804-A1 LIPID COMPOUND AND LIPID NANOPARTICLE COMPOSITION 苏州艾博生物科技有限公司 2023-06-29 WO disclosed
WO-2023122600-A1 PIPERAZINE INDAZOLE GLUCOCORTICOID RECEPTOR ANTAGONISTS CORCEPT THERAPEUTICS INCORPORATED (US) 2023-06-29 WO disclosed
US-20230201186-A1 SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION BAYER AKTIENGESELLSCHAFT (DE) 2023-06-29 US disclosed
US-20230201211-A1 NON-CATALYTIC SUBSTRATE-SELECTIVE p38alpha-SPECIFIC MAPK INHIBITORS WITH ENDOTHELIAL-STABILIZING AND ANTI-INFLAMMATORY ACTIVITY, AND METHODS OF USE THEREOF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2023-06-29 US disclosed
US-20230203063-A1 TRICYCLIC PYRIDONES AND PYRIMIDONES ERASCA, INC. 2023-06-29 US disclosed
EP-4200282-A1 SUBSTITUTED N-PHENYLURACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES Bayer Aktiengesellschaft (DE) 2023-06-28 EP disclosed
CN-110799492-B Novel carbonyl lipid and lipid nanoparticle formulations for delivery of nucleic acids 爱康泰生治疗公司 2023-06-27 CN disclosed
US-11685748-B2 Spiro aromatic ring compound and application thereof ETERN BIOPHARMA (SHANGHAI) CO., LTD. (CN) 2023-06-27 US disclosed
US-11685714-B2 Prodrugs of cytotoxic active agents having enzymatically cleavable groups BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2023-06-27 US disclosed
US-11685801-B2 Derivatizable monomers and polymers, and methods for making and using same RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2023-06-27 US disclosed
CN-116332960-A Pyridazine compound, pharmaceutical composition and application thereof 上海优理惠生医药有限公司 2023-06-27 CN disclosed
CN-116332954-A Preparation of thiophene derivatives 赣州和美药业股份有限公司 2023-06-27 CN disclosed
CN-116332830-A Lipid compounds and lipid nanoparticle compositions 苏州艾博生物科技有限公司 2023-06-27 CN disclosed
CN-116348638-A Modification of metal surfaces by phosphonic acids 生物动力学公司 2023-06-27 CN disclosed
CN-116348451-A ENPP1 modulators and uses thereof 维艾尔生物科技有限公司 2023-06-27 CN disclosed
CN-116323623-A Pyrido [2,3-d ] pyrimidin-4-amines as SOS1 inhibitors 拜耳公司 2023-06-23 CN disclosed
CN-116323627-A Lipid compounds and lipid nanoparticle compositions 苏州艾博生物科技有限公司 2023-06-23 CN disclosed
CN-116323570-A Compounds and methods for treating diseases 上海睿跃生物科技有限公司 2023-06-23 CN disclosed
US-20230190751-A1 6-6 Fused Bicyclic Heteroaryl Compounds and their Use as LATS Inhibitors NOVARTIS INSTITUTE FOR FUNTIONAL GENOMICS, INC., DBA GENOMICS INSTITUTE OF THE NOVARTIS RESEARCH FOUNDATION 2023-06-22 US disclosed
WO-2023114943-A2 LIPIDS FOR USE IN LIPID NANOPARTICLE FORMULATIONS Acuitas Therapeutics, Inc. (CA) 2023-06-22 WO disclosed
US-20230192700-A1 PYRAZOLOPYRAZINES ACTING ON CANCERS VIA INHIBITION OF CDK12 BAYER AKTIENGESELLSCHAFT (DE) 2023-06-22 US disclosed
US-20230192666-A1 PIPERAZINE INDAZOLE GLUCOCORTICOID RECEPTOR ANTAGONISTS CORCEPT THERAPEUTICS INCORPORATED 2023-06-22 US disclosed
WO-2023114710-A1 FUSED BENZOISOXAZOLYL COMPOUNDS AS KAT6A INHIBITORS AURIGENE ONCOLOGY LIMITED (IN) 2023-06-22 WO disclosed
US-20230192760-A1 SYSTEMS AND METHODS FOR TYROSINASE-MEDIATED SITE-SPECIFIC PROTEIN CONJUGATION GENENTECH, INC. 2023-06-22 US disclosed
US-20230192617-A1 AZABICYCLIC(THIO)AMIDES AS FUNGICIDAL COMPOUNDS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2023-06-22 US disclosed
WO-2023114428-A1 HETEROCYCLE DERIVATIVES FOR THE TREATMENT OF DISEASE Vir Biotechnology, Inc. (US) 2023-06-22 WO disclosed
WO-2023109959-A1 CDK9 INHIBITOR AND USE THEREOF 药捷安康(南京)科技股份有限公司 2023-06-22 WO disclosed
WO-2023115060-A1 PSYCHOPLASTOGENS FOR TREATING HEARING-RELATED DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-06-22 WO disclosed
US-20230190852-A1 COMPOSITIONS AND METHODS FOR JOINT HEALTH UNIGEN, INC. (US) 2023-06-22 US disclosed
WO-2023114809-A1 INHIBITORS OF MET KINASE KINNATE BIOPHARMA INC. (US) 2023-06-22 WO disclosed
US-20230192667-A1 BETA-LACTAM DERIVATIVES FOR THE TREATMENT OF DISEASES INSILICO MEDICINE IP LIMITED (HK) 2023-06-22 US disclosed
WO-2023114733-A1 KRAS MODULATORS AND USES THEREOF QUANTA THERAPEUTICS, INC. (US) 2023-06-22 WO disclosed
WO-2023114456-A1 USES OF BICYCLIC COMPOUNDS FOR THE TREATMENT OF DISEASES ATHIRA PHARMA, INC. (US) 2023-06-22 WO disclosed
WO-2023114472-A1 HETEROCYCLIC COMPOUNDS AS 5HT2A BIASED AGONISTS ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2023-06-22 WO disclosed
EP-3735409-B1 ENHANCEMENT OF NUCLEIC ACID POLYMERIZATION BY AROMATIC COMPOUNDS STRATOS GENOMICS INC (US) 2023-06-21 EP disclosed
EP-3271370-B1 NICOTINIC ACID RIBOSIDE OR NICOTINAMIDE RIBOSIDE COMPOSITIONS, REDUCED DERIVATIVES THEREOF, AND THE USE THEREOF CHROMADEX INC (US) 2023-06-21 EP disclosed
EP-4196219-A1 A3 ADENOSINE RECEPTOR AGONISTS FOR USE IN MEDICINE Biointervene, Inc. (US) 2023-06-21 EP disclosed
EP-3615502-B1 THERAPEUTIC COMPOUNDS AND METHODS UNIV TASMANIA (AU) 2023-06-21 EP disclosed
EP-4196220-A1 TRIAZOLE-PYRIDINYL SUBSTITUTED AZACYCLOHEXYL ACETIC ACID COMPOUNDS AS LPA RECEPTOR ANTAGONISTS Viva Star Biosciences Limited (HK) 2023-06-21 EP disclosed
EP-4198024-A1 PYRAZOLE MAGL INHIBITORS H. Lundbeck A/S (DK) 2023-06-21 EP disclosed
CN-110950842-B Quinoline derivatives having indoleamine-2, 3-dioxygenase inhibitory activity 深圳微芯生物科技股份有限公司 2023-06-20 CN disclosed
CN-116262753-A Novel PIM kinase inhibitors 杭州邦顺制药有限公司 2023-06-16 CN disclosed
US-20230180756-A1 TRIAZINE AND PYRIMIDINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2023-06-15 US disclosed
US-20230183210-A1 SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF INSILICO MEDICINE IP LIMITED (HK) 2023-06-15 US disclosed
US-20230180758-A1 SUBSTITUTED PYRROLINE-2-ONES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2023-06-15 US disclosed
WO-2023107863-A1 HETEROCYCLIC COMPOUNDS AS KIT KINASE INHIBITORS DECIPHERA PHARMACEUTICALS, LLC (US) 2023-06-15 WO disclosed
WO-2023102600-A1 SYNTHESIS OF AMPHIPHILIC BLOCK COPOLYMERS AND POLYMERIC NANOFIBERS PRODUCED THEREFROM NEWSOUTH INNOVATIONS PTY LIMITED (AU) 2023-06-15 WO disclosed
US-20230183188-A1 ENPP1 MODULATORS AND USES THEREOF Vir Biotechnology, Inc. 2023-06-15 US disclosed
WO-2023107870-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR KINASES KINNATE BIOPHARMA INC. (US) 2023-06-15 WO disclosed
US-20230183189-A1 CD73 COMPOUNDS GILEAD SCIENCES, INC. 2023-06-15 US disclosed
EP-4192431-A1 FORMULATIONS OF PHOSPHOINOSITIDE 3-KINASE INHIBITORS Venthera, Inc. (US) 2023-06-14 EP disclosed
EP-3884935-B1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX INC (US) 2023-06-14 EP disclosed
EP-4192462-A1 PYRAZOLOPYRIDINE COMPOUNDS AND METHODS OF INHIBITING IRE1 USING SAME Optikira LLC (US) 2023-06-14 EP disclosed
CN-116253717-A Pyridazine derivative and application thereof in medicine 海思科医药集团股份有限公司 2023-06-13 CN disclosed
CN-116261561-A Certain chemical compositions and methods of use thereof 奧基生物技术有限公司 2023-06-13 CN disclosed
US-11673879-B2 Substituted pyrimidines and methods of use THERAVANCE BIOPHARMA R&D IP, LLC (US) 2023-06-13 US disclosed
US-11674964-B2 Encoded chromophoric polymer particles and methods of use thereof UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2023-06-13 US disclosed
CN-110678177-B Pyrazole MAGL inhibitors H.隆德贝克有限公司 2023-06-13 CN disclosed
US-11672788-B2 Histone deacetylase inhibitors for immunomodulation in tumor microenvironment Great Novel Therapeutics Biotech & Medicals Corporation (TW) 2023-06-13 US disclosed
US-20230174526-A1 BENZOTHIAZOLYL BIARYL COMPOUND, AND PREPARATION METHOD AND USE SHANGHAI RINGENE THERAPEUTICS CO. LTD (CN) 2023-06-08 US disclosed
US-20230172886-A1 (S)-2-AMINO-6-((3-AMINOPROPYL)AMINO)HEXANOIC ACID (APL) FOR USE IN THE TREATMENT OF NON-ALCOHOLIC STEATOHEPATITIS (NASH), LIVER INFLAMMATION, HEPATOCELLULAR BALLOONING, LIVER FIBROSIS AND STEATOSIS TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2023-06-08 US disclosed
US-20230174535-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR KINASES KINNATE BIOPHARMA INC. 2023-06-08 US disclosed
WO-2023099612-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-06-08 WO disclosed
WO-2023102378-A1 MACROCYCLIC COMPOUNDS HAVING FARNESYLTRANSFERASE INHIBITORY ACTIVITY KURA ONCOLOGY, INC. (US) 2023-06-08 WO disclosed
WO-2023099623-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-06-08 WO disclosed
WO-2023099620-A1 KRAS DEGRADING COMPOUNDS COMPRISING ANNULATED 2-AMINO-3-CYANO THIOPHENES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-06-08 WO disclosed
US-20230174506-A1 (DI)AMINATION OF ACTIVATED ALLENE COMPOUNDS, DERIVATIVES THEREOF, AND METHODS FOR SYNTHESIS OF THE SAME PURDUE RESEARCH FOUNDATION 2023-06-08 US disclosed
US-20230178803-A1 Silicon-Based Energy Storage Devices With Electrolyte Containing Sulfonate or Carboxylate Salt Based Compounds ENEVATE CORPORATION 2023-06-08 US disclosed
US-20230173081-A1 FACTOR VIII ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC. 2023-06-08 US disclosed
US-20230174480-A1 FLUOROGENIC DIMER COMPOUND, USEFUL AS A PROBE FOR DETECTION OF ENDOGENOUS RECEPTORS UNIVERSITE DE STRASBOURG (FR) 2023-06-08 US disclosed
WO-2023099624-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-06-08 WO disclosed
WO-2023099445-A1 BIS(HETERO)ARYL THIOETHER OXADIAZINES AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2023-06-08 WO disclosed
US-20230174477-A1 METHODS FOR SYNTHESIS OF THE TRICYCLIC PROSTAGLANDIN D2 METABOLITE METHYL ESTER PURDUE RESEARCH FOUNDATION 2023-06-08 US disclosed
EP-3445359-B1 USE OF NICOTINIC ACID RIBOSIDE OR NICOTINAMIDE RIBOSITE DERIVATIVES, AND REDUCED DERIVATIVES THEREOF, AS NAD+INCREASING PRECURSORS CHROMADEX INC (US) 2023-06-07 EP disclosed
EP-3717525-B1 CATALYST SYSTEMS AND POLYMERIZATION PROCESSES FOR USING THE SAME EXXONMOBIL CHEMICAL PATENTS INC (US) 2023-06-07 EP disclosed
CN-111511465-B Method for producing organic silicon dioxide material and use thereof 埃克森美孚科技工程公司 2023-06-06 CN disclosed
CN-116217581-A Methods and compositions for inhibiting interactions of multiple endocrine oncostatin proteins with MLL proteins 库拉肿瘤学公司 2023-06-06 CN disclosed
US-11667669-B2 Epoxy-(meth)acrylate monomers and polymers and methods of making and using the same ROWAN UNIVERSITY (US) 2023-06-06 US disclosed
US-11667634-B2 Inhibitors of RAF kinases KINNATE BIOPHARMA INC. (US) 2023-06-06 US disclosed
US-11666588-B2 Prodrugs of ALOX-15 inhibitors and methods of using the same EMPIRICO INC. (US) 2023-06-06 US disclosed
CN-116199685-A HER2 degradation agent and application thereof 四川海思科制药有限公司 2023-06-02 CN disclosed
US-20230165252-A1 ACTIVE COMPOUND COMBINATIONS BAYER AKTIENGESELLSCHAFT (DE) 2023-06-01 US disclosed
WO-2023094679-A1 PHOTODYNAMIC THERAPY AND DIAGNOSIS RMW CHO GROUP LIMITED (CN) 2023-06-01 WO disclosed
WO-2023096845-A1 ANTIMICROBIAL POLYMER COMPOSITIONS, ANTIMICROBIAL POLYMER ARTICLES, AND METHODS OF MAKING THE SAME CORNING INCORPORATED (US) 2023-06-01 WO disclosed
WO-2023092195-A1 ANALOGUES OF MDMA FOR MODULATING SERT, DAT, AND / OR NET ACTIVITY THE UNIVERSITY OF WESTERN AUSTRALIA (AU) 2023-06-01 WO disclosed
WO-2023039240-A9 IRREVERSIBLE INHIBITORS OF KRas BIOMEA FUSION, INC. (US) 2023-06-01 WO disclosed
WO-2023094680-A1 PHOTODYNAMIC THERAPY AND DIAGNOSIS RMW CHO GROUP LIMITED (CN) 2023-06-01 WO disclosed
US-20230165857-A1 AXL KINASE INHIBITORS AND USE OF THE SAME SUMITOMO PHARMA ONCOLOGY, INC. 2023-06-01 US disclosed
WO-2023096935-A1 FORMULATIONS OF PYRROLOPYRIDINE-ANILINE COMPOUNDS NFLECTION THERAPEUTICS, INC. (US) 2023-06-01 WO disclosed
WO-2023094677-A1 PHOTODYNAMIC THERAPY AND DIAGNOSIS RMW CHO GROUP LIMITED (CN) 2023-06-01 WO disclosed
US-20230167106-A1 SERINE THREONINE KINASE (AKT) DEGRADATION / DISRUPTION COMPOUNDS AND METHODS OF USE ICAHN SCHOOL MED MOUNT SINAI (US) 2023-06-01 US disclosed
WO-2023094594-A1 SUBSTITUTED DIHYDROPYRANOPYRIDINES, SALTS OR N-OXIDES THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2023-06-01 WO disclosed
WO-2023097020-A1 HETEROBIFUNCTIONAL COMPOUNDS AS HPK1 DEGRADERS ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2023-06-01 WO disclosed
US-20230167088-A1 1-PYRAZINYLPYRAZOLYL-3-OXYALKYL ACIDS AND THEIR DERIVATIVES, AND THEIR USE FOR CONTROL OF UNDESIRED PLANT GROWTH BAYER AKTIENGESELLSCHAFT (DE) 2023-06-01 US disclosed
WO-2023097221-A1 TABLET FORMULATIONS OF RBP4 INHIBITORS AND METHODS OF USE BELITE BIO, INC (US) 2023-06-01 WO disclosed
CN-116194448-A Compounds and formulations for the treatment of ophthalmic diseases 视点医疗股份有限公司 2023-05-30 CN disclosed
US-11661421-B2 Indolizine compounds, preparation method and use thereof HAIHE BIOPHARMA CO., LTD. (CN) 2023-05-30 US disclosed
CN-116178360-A PRMT5 inhibitors and uses thereof 四川海思科制药有限公司 2023-05-30 CN disclosed
US-11661429-B2 Topical phosphoinositide 3-kinase inhibitors VENTHERA, INC. (US) 2023-05-30 US disclosed
US-11660301-B2 Combination of ATR kinase inhibitors with PARP inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2023-05-30 US disclosed
US-11661580-B2 Method of inhibiting tau phosphorylation CASSAVA SCIENCES, INC. (US) 2023-05-30 US disclosed
US-11661418-B2 MASP-2 inhibitors and methods of use OMEROS CORPORATION (US) 2023-05-30 US disclosed
US-11661403-B2 Oxadiazole compounds VIVACE THERAPEUTICS, INC. (US) 2023-05-30 US disclosed
CN-116194112-A Pyridine-1, 5-diones exhibiting MNK inhibition and methods of use thereof 4E治疗公司 2023-05-30 CN disclosed
CN-114573566-B Selective ROCK2 kinase inhibitors 杭州邦顺制药有限公司 2023-05-30 CN disclosed
CN-116194463-A Cyclic peptide compounds and methods of use 李丰桥 2023-05-30 CN disclosed
CN-111527090-B Pyrazolo-pyrrolo-pyrimidine-dione derivatives as P2X3 inhibitors 拜耳公司 2023-05-26 CN disclosed
US-20230159544-A1 AZEPINO-INDOLES FOR THE TREATMENT OF NEUROLOGICAL AND PSYCHIATRIC DISORDERS TERRAN BIOSCIENCES INC (US) 2023-05-25 US disclosed
WO-2023091707-A1 BICYCLIC INHIBITORS OF JAK AND METHODS OF USE THERAVANCE BIOPHARMA R&D IP, LLC (US) 2023-05-25 WO disclosed
US-20230158469-A1 DEVICES AND METHODS FOR SYNTHESIS Twist Bioscience Corporation 2023-05-25 US disclosed
WO-2023091606-A1 PYRIDAZINONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. (US) 2023-05-25 WO disclosed
US-20230159563-A1 TRICYCLIC PYRIDONES AND PYRIMIDONES ERASCA, INC. 2023-05-25 US disclosed
WO-2023092133-A1 STEREOSELECTIVE COVALENT LIGANDS FOR ONCOGENIC AND IMMUNOLOGICAL PROTEINS THE SCRIPPS RESEARCH INSTITUTE (US) 2023-05-25 WO disclosed
WO-2023091490-A1 NOVEL IONIZABLE LIPIDS AND LIPID NANOPARTICLES AND METHODS OF USING THE SAME SENDA BIOSCIENCES, INC. (US) 2023-05-25 WO disclosed
US-20230159456-A1 N-SUBSTITUTED INDOLES TERRAN BIOSCIENCES INC (US) 2023-05-25 US disclosed
US-20230158053-A1 NICOTINAMIDE MONONUCLEOTIDE DERIVATIVES AND THEIR USES METROBIOTECH, LLC 2023-05-25 US disclosed
US-20230159569-A1 DUAL HDAC6/PROTEASOME INHIBITORS, AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-05-25 US disclosed
US-20230158146-A1 HSP70 Inhibitors and Methods of Using Same THE WISTAR INST (US) 2023-05-25 US disclosed
EP-4183853-A1 PHOTOACTIVE MACROMOLECULES AND USES THEREOF Beckman Coulter, Inc. (US) 2023-05-24 EP disclosed
US-11655217-B2 Pyrazole MAGL inhibitors H. LUNDBECK A/S (DK) 2023-05-23 US disclosed
CN-116157388-A Carbocyclic amide derivative and application thereof in medicine 四川海思科制药有限公司 2023-05-23 CN disclosed
CN-116143766-A CDK2 degrading agent and application thereof 四川海思科制药有限公司 2023-05-23 CN disclosed
CN-116143744-A Aromatic ester compound and application thereof 陈艳莉 2023-05-23 CN disclosed
CN-114206827-B Lipid nanoparticle compositions 苏州艾博生物科技有限公司 2023-05-23 CN disclosed
CN-110139644-B Compositions and methods for treating insulin resistance 坦普尔大学 2023-05-23 CN disclosed
CN-109640970-B Selective p38α -specific MAPK inhibitors 马里兰大学巴尔的摩分校 2023-05-23 CN disclosed
CN-116157397-A Heterocyclylpyridines as novel fungicides 拜耳公司 2023-05-23 CN disclosed
CN-116143805-A Nitrogen-containing heterocyclic biaryl compounds, preparation method and application 上海凌达生物医药有限公司 2023-05-23 CN disclosed
CN-116143777-A Heterocyclic compound capable of inhibiting IL-17A and application thereof 四川海思科制药有限公司 2023-05-23 CN disclosed
CN-116143806-A Nitrogen-containing heterocyclic compound, preparation method and application 上海凌达生物医药有限公司 2023-05-23 CN disclosed
US-11654143-B2 Therapeutic combinations of a BTK inhibitor, a PI3K inhibitor, a JAK-2 inhibitor, and/or a BCL-2 inhibitor ACERTA PHARMA B.V. (NL) 2023-05-23 US disclosed
WO-2023086520-A2 ENGINEERED ENZYMES AND METHOD FOR THE SYNTHESIS OF DIVERSE TYROSINE ANALOGS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2023-05-19 WO disclosed
WO-2023086417-A1 COMPOUNDS AND METHODS OF USE THEREOF ALGEN BIOTECHNOLOGIES, INC. (US) 2023-05-19 WO disclosed
WO-2023084206-A1 N-(4-AMINOCYCLOHEXYL)PYRIMIDINE-4-CARBOXAMIDE DERIVATIVES AS CD38 INHIBITORS CEREVANCE LTD (GB) 2023-05-19 WO disclosed
WO-2023086341-A1 INHIBITORS OF KRAS BIOMEA FUSION, INC. (US) 2023-05-19 WO disclosed
WO-2023086638-A1 ENPP1 MODULATORS AND USES THEREOF Vir Biotechnology, Inc. (US) 2023-05-19 WO disclosed
WO-2023086830-A1 INTRASPINAL DELIVERY OF THERAPEUTIC AGENTS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2023-05-19 WO disclosed
CN-111587256-B Catalyst system and polymerization process using the same 埃克森美孚化学专利公司 2023-05-19 CN disclosed
US-20230150972-A1 PYRIDINYL DERIVATIVES AS SODIUM CHANNEL ACTIVATORS XENON PHARMACEUTICALS INC. (CA) 2023-05-18 US disclosed
US-20230151025-A1 SUBSTITUTED THIAZOLOPYRIDINES, SALTS THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES BAYER AG (DE) 2023-05-18 US disclosed
US-20230149397-A1 Combination Therapy with AXL Inhibitor and Immune Checkpoint Modulator or Oncolytic Virus BERGENBIO ASA (NO) 2023-05-18 US disclosed
US-20230151018-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES FORWARD THERAPEUTICS, INC. 2023-05-18 US disclosed
US-20230151100-A1 Method of Selecting Patients for Treatment with a Combination of an AXL Inhibitor and an Immune Checkpoint Modulator BERGENBIO ASA (NO) 2023-05-18 US disclosed
EP-4179133-A1 MODIFICATION OF METALLIC SURFACES WITH PHOSPHONIC ACIDS Biological Dynamics, Inc. (US) 2023-05-17 EP disclosed
EP-4178574-A2 COMPOUNDS, COMPOSITIONS, AND METHODS FOR THE TREATMENT OF FIBROTIC DISEASES AND CANCER Purdue Research Foundation (US) 2023-05-17 EP disclosed
EP-4178571-A1 GAS41 INHIBITORS AND METHODS OF USE THEREOF The Regents Of The University Of Michigan (US) 2023-05-17 EP disclosed
CN-109996790-B Piperazine carbamates and methods of making and using the same H.隆德贝克有限公司 2023-05-16 CN disclosed
US-11652239-B2 Silicon-based energy storage devices with electrolyte containing dihydrofuranone based compound ENEVATE CORPORATION (US) 2023-05-16 US disclosed
US-11648324-B2 Lipids and lipid nanoparticle formulations for delivery of nucleic acids Acuitas Therapeutics, Inc. (CA) 2023-05-16 US disclosed
US-11649237-B2 Substituted imidazo[1,5-a]pyrazines for IRE1 inhibition OPTIKIRA LLC (US) 2023-05-16 US disclosed
CN-111542315-B Benzosulfonyl compounds 维瓦斯治疗公司 2023-05-12 CN disclosed
CN-116113406-A GAS41 inhibitors and methods of use thereof 密歇根大学董事会 2023-05-12 CN disclosed
US-20230142139-A1 CATALYST COMPOSITIONS FOR HYDROFORMYLATION AND METHODS OF USE THEREOF BOARD OF SUPERVISORS OF LOUISIANA STATE UNIVERSITY AND AGRICULTURAL AND MECHANICAL COLLEGE 2023-05-11 US disclosed
US-20230147053-A1 FUSED N-HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC (US) 2023-05-11 US disclosed
US-20230144095-A1 PYRIDINE DERIVATIVES AND THEIR USE AS SODIUM CHANNEL ACTIVATORS X-CHEM GLOBAL HQ 2023-05-11 US disclosed
US-20230148194-A1 SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION BAYER AKTIENGESELLSCHAFT (DE) 2023-05-11 US disclosed
WO-2023081185-A1 METHODS OF TREATING RESPIRATORY DEPRESSION MODULATED BY A NON-OPIOID AGENT ENALARE THERAPEUTICS INC. (US) 2023-05-11 WO disclosed
US-20230140941-A1 NON-ATP/CATALYTIC SITE P38 MITOGEN ACTIVATED PROTEIN KINASE INHIBITORS THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2023-05-11 US disclosed
WO-2023078915-A1 BIS(HETERO)ARYL THIOETHER (THIO)AMIDES AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2023-05-11 WO disclosed
US-20230143612-A1 SUBSTITUTED 1,1'-BIPHENYL COMPOUNDS AND METHODS USING SAME ARBUTUS BIOPHARMA CORP (US) 2023-05-11 US disclosed
WO-2023078946-A1 LIPID NANOPARTICLES FOR OLIGONUCLEOTIDE DELIVERY ZIPHIUS VACCINES NV (BE) 2023-05-11 WO disclosed
US-20230146903-A1 CXCR5 Antagonists and Methods of Treating Diseases or Disorders Using Same YALE UNIVERSITY 2023-05-11 US disclosed
WO-2023078954-A1 LIPID NANOPARTICLES FOR OLIGONUCLEOTIDE DELIVERY ZIPHIUS VACCINES NV (BE) 2023-05-11 WO disclosed
WO-2023081312-A1 SMALL MOLECULE INDUCERS OF AUTOPHAGY Vir Biotechnology, Inc. (US) 2023-05-11 WO disclosed
US-20230148152-A1 METHOD OF SYNTHESIZING SINGLE-STRANDED NUCLEOTIDE SEQUENCE, BLOCKED NUCLEOSIDE TRIPHOSPHATES AND RELATED METHODS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2023-05-11 US disclosed
WO-2023078426-A1 COMPOUND, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND USE THEREOF 上海优理惠生医药有限公司 2023-05-11 WO disclosed
WO-2023078950-A1 LIPID NANOPARTICLES FOR OLIGONUCLEOTIDE DELIVERY ZIPHIUS VACCINES NV (BE) 2023-05-11 WO disclosed
EP-3851469-B1 POLYURETHANE/UREA MATERIALS COMMW SCIENT IND RES ORG (AU) 2023-05-10 EP disclosed
EP-4175503-A1 REDUCTION OF VIRAL INFECTIONS Phoxbio Limited (IE) 2023-05-10 EP disclosed
CN-112390904-B Polyethylene containing polar functional groups and preparation method thereof 中国科学院上海有机化学研究所 2023-05-09 CN disclosed
CN-116096707-A Inhibitors of fibroblast growth factor receptor kinase 金耐特生物制药公司 2023-05-09 CN disclosed
US-11646449-B2 Cyclodextrin-based compounds and their derivatives for silicon-based li-ion batteries ENEVATE CORPORATION (US) 2023-05-09 US disclosed
CN-116075303-A Method of selecting patients treated with a combination of an AXL inhibitor and an immune checkpoint modulator 卑尔根生物股份公司 2023-05-05 CN disclosed
CN-116059390-A Prodrugs of cytotoxic actives with enzymatically cleavable groups 拜耳制药股份公司 2023-05-05 CN disclosed
CN-112778336-B Nitrogen-containing condensed ring STING regulator compound, preparation method and application 上海凌达生物医药有限公司 2023-05-05 CN disclosed
CN-116063639-A Multiblock copolymers and uses thereof 广州立邦涂料有限公司 2023-05-05 CN disclosed
CN-116075513-A Inhibitors of NEK7 kinase 哈利亚治疗公司 2023-05-05 CN disclosed
CN-116064598-A Nucleic acid vaccine for coronavirus 苏州艾博生物科技有限公司 2023-05-05 CN disclosed
WO-2023077146-A1 CANNABIGEROL FOR TREATMENT OF SEIZURES AND EPILEPSY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-05-04 WO disclosed
US-20230134760-A1 CAR AND NRF2 DUAL ACTIVATOR AGENTS FOR CYCLOPHOSPHAMIDE-BASED AND DOXORUBICIN-BASED TREATMENTS OF CANCER NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-05-04 US disclosed
WO-2023077125-A2 AZEPINO-INDOLES FOR THE TREATMENT OF NEUROLOGICAL AND PSYCHIATRIC DISORDERS TERRAN BIOSCIENCES, INC. (US) 2023-05-04 WO disclosed
WO-2023077127-A2 N-SUBSTITUTED INDOLES TERRAN BIOSCIENCES, INC. (US) 2023-05-04 WO disclosed
WO-2023076687-A1 DEVICES AND METHODS FOR SYNTHESIS Twist Bioscience Corporation (US) 2023-05-04 WO disclosed
WO-2023073423-A1 ERGOLINE-DERIVED AGONISTS OF THE 5-HT2A RECEPTOR DIAMOND THERAPEUTICS INC. (CA) 2023-05-04 WO disclosed
WO-2023077030-A1 CD73 COMPOUNDS GILEAD SCIENCES, INC. (US) 2023-05-04 WO disclosed
US-20230140606-A1 METHODS OF TREATING RESPIRATORY DEPRESSION MODULATED BY A NON-OPIOID AGENT ENALARE THERAPEUTICS INC. 2023-05-04 US disclosed
EP-4172272-A1 HYDROGELS Commonwealth Scientific and Industrial Research Organisation (AU) 2023-05-03 EP disclosed
EP-4171565-A2 PYRIDINE-1,5-DIONES EXHIBITNG MNK INHIBITION AND THEIR METHOD OF USE 4E Therapeutics, Inc. (US) 2023-05-03 EP disclosed
EP-3590932-B1 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE SUMITOMO PHARMA ONCOLOGY INC (US) 2023-05-03 EP disclosed
EP-3511319-B1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2023-05-03 EP disclosed
EP-4172153-A1 SUBSTITUTED HETEROARYLOXYPYRIDINES, THE SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS Bayer Aktiengesellschaft (DE) 2023-05-03 EP disclosed
CN-116057056-A Azabicyclo-substituted heterocyclic compounds as fungicides 拜耳公司 2023-05-02 CN disclosed
CN-110678456-B Pyrazole MAGL inhibitors H.隆德贝克有限公司 2023-05-02 CN disclosed
CN-111032034-B Spiro compounds and methods of making and using the same H.隆德贝克有限公司 2023-05-02 CN disclosed
CN-116057045-A Fibroblast growth factor receptor kinase inhibitors 金耐特生物制药公司 2023-05-02 CN disclosed
US-11639329-B2 Lipids for use in lipid nanoparticle formulations Acuitas Therapeutics, Inc. (CA) 2023-05-02 US disclosed
US-11639351-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. 2023-05-02 US disclosed
US-11639333-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC (US) 2023-05-02 US disclosed
US-11639346-B2 Quinazoline derivatives as modulators of mutant KRAS, HRAS or NRAS ARAXES PHARMA LLC (US) 2023-05-02 US disclosed
US-11639332-B2 Methods and compositions of isoindoline-1,3-dione and isoindole prodrugs useful for treating cancer, ulcerative colitis and related inflammatory diseases Amgen (Europe) GmbH (CH) 2023-05-02 US disclosed
CN-113929729-B Veratramine compound, preparation method and application thereof 上海医药工业研究院有限公司 2023-04-28 CN disclosed
CN-116033904-A Histone deacetylase inhibitor for tumor microenvironment immunomodulation 华上生技医药股份有限公司 2023-04-28 CN disclosed
US-20230131260-A1 SUBSTITUTED THIOPHENYL URACILS, SALTS THEREOF AND THE USE THEREOF AS HERBICIDAL AGENTS SYNGENTA CROP PROTECTION AG (CH) 2023-04-27 US disclosed
WO-2023070053-A1 INHIBITORS OF RAF KINASES KINNATE BIOPHARMA INC. (US) 2023-04-27 WO disclosed
US-20230128972-A1 Anat Inhibitors and Methods of Use Thereof Atomwise Inc. 2023-04-27 US disclosed
US-20230127931-A1 SINGLE LITHIUM-ION CONDUCTIVE POLYMER ELECTROLYTES FOR SI ANODE-BASED LITHIUM-ION BATTERIES ENEVATE CORPORATION 2023-04-27 US disclosed
US-20230126893-A1 [(1,4,5-TRISUBSTITUTED-1H-PYRAZOL-3-YL)SULFANYL]ACETIC ACID DERIVATIVES, SALTS THEREOF, AND USE THEREOF AS ACTIVE HERBICIDAL INGREDIENTS BAYER AKTIENGESELLSCHAFT (DE) 2023-04-27 US disclosed
WO-2023070114-A2 REVERSIBLE LYSINE COVALENT MODIFIERS OF EGFR AND USES THEREOF TERREMOTO BIOSCIENCES, INC. (US) 2023-04-27 WO disclosed
WO-2023069727-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF HYPERPROLIFERATIVE, INFLAMMATORY, AND IMMUNOLOGICAL DISEASES, AND INFECTIONS EDISON ONCOLOGY (US) 2023-04-27 WO disclosed
WO-2023069548-A1 MALODOR-COUNTERACTING COMPOUNDS, COMPOSITIONS, AND USES THEREOF INTERNATIONAL FLAVORS AND FRAGRANCES INC. (US) 2023-04-27 WO disclosed
EP-3675858-B1 IMIDAZO[1,5-A]PYRAZINE COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION OPTIKIRA LLC (US) 2023-04-26 EP disclosed
EP-4167740-A1 ACTIVE COMPOUND COMBINATIONS Bayer Aktiengesellschaft (DE) 2023-04-26 EP disclosed
EP-4168402-A1 QUATERNARY INDAZOLE GLUCOCORTICOID RECEPTOR ANTAGONISTS Corcept Therapeutics Incorporated (US) 2023-04-26 EP disclosed
US-11634528-B2 Latent imaging for volume Bragg gratings META PLATFORMS TECHNOLOGIES, LLC (US) 2023-04-25 US disclosed
CN-110573511-B 6-6 fused bicyclic heteroaryl compounds and their use as LATS inhibitors 诺华股份有限公司 2023-04-25 CN disclosed
US-11633490-B2 2023-04-25 US disclosed
US-11634396-B2 Opioid receptor modulators EPIODYNE, INC. (US) 2023-04-25 US disclosed
CN-115996923-A Nitrile derivative as dipeptidyl peptidase 1 inhibitor and application thereof 四川海思科制药有限公司 2023-04-21 CN disclosed
CN-115996638-A Substituted N-phenyluracils and salts thereof and their use as herbicidal agents 拜耳股份有限公司 2023-04-21 CN disclosed
CN-115996919-A Substituted heteroaryloxy pyridines, salts thereof and their use as herbicides 拜耳公司 2023-04-21 CN disclosed
US-20230117519-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2023-04-20 US disclosed
US-20230117034-A1 PYRAZOLOTRIAZINES BAYER AKTIENGESELLSCHAFT (DE) 2023-04-20 US disclosed
US-20230117791-A1 SUBSTITUTED 1,2,3,4,5,6-HEXAHYDROAZEPINO[4,5-b]INDOLES FOR TREATING BRAIN DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2023-04-20 US disclosed
US-20230121768-A1 MLL1 INHIBITORS AND ANTI-CANCER AGENTS CHINA NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH CO., LTD. (CN) 2023-04-20 US disclosed
US-20230120115-A1 COVALENT INHIBITORS OF MENIN-MLL INTERACTION FOR DIABETES MELLITUS BIOMEA FUSION, INC. 2023-04-20 US disclosed
US-20230121031-A1 MASKED FLUOROGENIC COMPOUNDS AND METHODS OF USING THE SAME RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2023-04-20 US disclosed
US-20230118233-A1 PRC1 INHIBITORS AND METHODS OF TREATMENT THEREWITH NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-04-20 US disclosed
US-20230121952-A1 COMPOUNDS INFLAZOME LIMITED (IE) 2023-04-20 US disclosed
US-20230123534-A1 LIPIDS FOR LIPID NANOPARTICLE DELIVERY OF ACTIVE AGENTS ACUITAS THERAPEUTICS INC (CA) 2023-04-20 US disclosed
US-20230119934-A1 NETWORK POLYMERS AND METHODS OF MAKING AND USING SAME UNIV COLORADO REGENTS (US) 2023-04-20 US disclosed
WO-2023064152-A1 TRICYCLIC SULFAMIDES AND SULTAMS MERCK SHARP & DOHME LLC (US) 2023-04-20 WO disclosed
WO-2023064058-A1 TRICYCLIC SULTAMS AND SULFAMIDES AS ANTITUMOR AGENTS PELOTON THERAPEUTICS INC. (US) 2023-04-20 WO disclosed
WO-2023062492-A1 DIAZABICYCLOOCTANE DERIVATIVES USEFUL AS MATRIX METALLOPROTEINASE INHIBITORS VASA THERAPEUTICS SPÓŁKA Z OGRANICZONĄ ODPOWIEDZIALNOŚCIĄ (PL) 2023-04-20 WO disclosed
EP-4165038-A1 AZABICYCLYL-SUBSTITUTED HETEROCYCLES AS FUNGICIDES Bayer Aktiengesellschaft (DE) 2023-04-19 EP disclosed
EP-4166549-A1 ISOTOPE-SUBSTITUTED SPIRO AROMATIC RING COMPOUND AND APPLICATION THEREOF Etern Biopharma (Shanghai) Co., Ltd. (CN) 2023-04-19 EP disclosed
US-11629230-B1 Ternary orthogonal photopolymers META PLATFORMS TECHNOLOGIES, LLC (US) 2023-04-18 US disclosed
US-11629137-B2 Methods of manufacturing of niraparib TESARO, INC. (US) 2023-04-18 US disclosed
CN-115960098-A Preparation method and application of nitrogen-containing fused ring compounds 上海凌达生物医药有限公司 2023-04-14 CN disclosed
CN-115960109-A Preparation and application of fused-ring SHP2 phosphatase inhibitor 药雅科技(上海)有限公司 2023-04-14 CN disclosed
CN-114096550-B Modified nucleosides and methods of synthesis thereof 斯微(上海)生物科技股份有限公司 2023-04-14 CN disclosed
US-20230112489-A1 COMPOSITIONS AND METHODS OF MAKING EXPANDED HEMATOPOIETIC STEM CELLS USING DERIVATIVES OF FLUORENE TRANSFUSION HEALTH LLC 2023-04-13 US disclosed
US-20230116632-A1 ANALOGS FOR THE TREATMENT OF DISEASE Insilico Medicine Hong Kong Limited (CN) 2023-04-13 US disclosed
US-20230116253-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2023-04-13 US disclosed
US-20230115836-A1 ANALOGS FOR THE TREATMENT OF DISEASE Insilico Medicine Hong Kong Limited (CN) 2023-04-13 US disclosed
US-20230114728-A1 PENICILLIN-BINDING PROTEIN INHIBITORS VenatoRx Pharmaceuticals, Inc. 2023-04-13 US disclosed
US-20230111793-A1 ANTIMALARIAL COMPOSITIONS AND USES THEREOF SCRIPPS RESEARCH INST (US) 2023-04-13 US disclosed
US-20230115890-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH LINEAR CARBONATE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2023-04-13 US disclosed
US-20230112086-A1 PHOTO-CLEAVABLE PRIMER COMPOSITIONS AND METHODS OF USE ORMCO CORPORATION 2023-04-13 US disclosed
US-20230112244-A1 SUBSTITUTED MACROCYCLIC INDOLE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2023-04-13 US disclosed
EP-4162950-A1 NUCLEIC ACID VACCINES FOR CORONAVIRUS Suzhou Abogen Biosciences Co., Ltd. (CN) 2023-04-12 EP disclosed
EP-4161916-A1 SUBSTITUTED ISOQUINOLINYLMETHYL AMIDES, ANALOGUES THEREOF, AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2023-04-12 EP disclosed
EP-4161379-A1 GALLIUM-SALOPHEN ANTIMICROBIAL COMPOUNDS AND METHODS OF USE THEREOF University of Maryland, Baltimore (US) 2023-04-12 EP disclosed
EP-4161905-A1 SUBSTITUTED (PHTHALAZIN-1-YLMETHYL)UREAS, SUBSTITUTED N-(PHTHALAZIN-1-YLMETHYL)AMIDES, AND ANALOGUES THEREOF Arbutus Biopharma Corporation (CA) 2023-04-12 EP disclosed
EP-4161656-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR KINASES Kinnate Biopharma Inc. (US) 2023-04-12 EP disclosed
EP-4161933-A1 INHIBITORS OF NEK7 KINASE Halia Therapeutics, Inc. (US) 2023-04-12 EP disclosed
EP-4161914-A1 HETEROCYCLYL PYRIDINES AS NOVEL FUNGICIDES Bayer Aktiengesellschaft (DE) 2023-04-12 EP disclosed
EP-4161657-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR KINASES Kinnate Biopharma Inc. (US) 2023-04-12 EP disclosed
EP-4161906-A1 HETEROCYCLYL PYRIMIDINES AND TRIAZINES AS NOVEL FUNGICIDES Bayer Aktiengesellschaft (DE) 2023-04-12 EP disclosed
EP-4161922-A1 USE OF MULTI-KINASE INHIBITORS TO TREAT RNA VIRUS INFECTIONS Icahn School of Medicine at Mount Sinai (US) 2023-04-12 EP disclosed
US-11622960-B2 Microtubule polymerization inhibitor prodrugs and methods of using the same UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-04-11 US disclosed
US-11623922-B2 Compounds INFLAZOME LIMITED (IE) 2023-04-11 US disclosed
CN-115955916-A Active compound combinations 拜耳公司 2023-04-11 CN disclosed
CN-111303152-B Polycyclic-carbamoylpyridone compounds and their pharmaceutical use 吉利德科学公司 2023-04-11 CN disclosed
CN-115943143-A 1-pyrazinylpyrazolyl-3-oxyalkyl acids and derivatives thereof and their use for controlling undesired vegetation 拜耳公司 2023-04-07 CN disclosed
CN-111848573-B Benzothiophene amide compound and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-04-07 CN disclosed
US-20230108157-A1 FORMULATIONS OF (S)-3-(1-(9H-PURIN-6-YLAMINO)ETHYL)-8-CHLORO-2-PHENYLISOQUINOLIN-1(2H)-ONE INTELLIKINE LLC 2023-04-06 US disclosed
US-20230107642-A1 TRICYCLIC PYRIDONES AND PYRIMIDONES ERASCA, INC. 2023-04-06 US disclosed
US-20230103958-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ELECTROLYTE CONTAINING A BENZOYL PEROXIDE BASED COMPOUND ENEVATE CORPORATION 2023-04-06 US disclosed
WO-2023056460-A1 WATER-SOLUBLE TETRAHYDROPYRENE BASED FLUORESCENT POLYMERS BECKMAN COULTER, INC. (US) 2023-04-06 WO disclosed
US-20230106583-A1 HETEROARYL COMPOUNDS VIVACE THERAPEUTICS, INC. 2023-04-06 US disclosed
WO-2023055702-A1 MAIN PROTEASE (M PRO) INHIBITORS AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2023-04-06 WO disclosed
WO-2023056264-A1 NOVEL SUBSTITUTED SULFONYLUREA COMPOUNDS AS INHIBITORS OF INTERLEUKIN-1 ACTIVITY VIVA STAR BIOSCIENCES (SUZHOU) CO., LTD. (CN) 2023-04-06 WO disclosed
WO-2023052363-A1 NOVEL TETRAHYDROQUINOLINES AND PROTEOLYSIS TARGETING CHIMERA (PROTACS) COMPRISING THEM AS DEGRADERS OF SMARCA BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-04-06 WO disclosed
US-20230106032-A1 IMIDAZOTRIAZINES ACTING ON CANCER VIA INHIBITION OF CDK12 BAYER AKTIENGESELLSCHAFT (DE) 2023-04-06 US disclosed
US-20230108463-A1 PHOSPHORUS-CONTAINING COMPOUNDS AS ADDITIVES FOR SILICON-BASED LI ION BATTERIES ENEVATE CORPORATION 2023-04-06 US disclosed
US-20230108906-A1 SUBSTITUTED BICYCLIC AND TRICYCLIC UREAS AND AMIDES, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2023-04-06 US disclosed
EP-3755694-B1 NEW BENZIMIDAZOLE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2023-04-05 EP disclosed
EP-4157836-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER Boehringer Ingelheim International GmbH (DE) 2023-04-05 EP disclosed
EP-4157837-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER Boehringer Ingelheim International GmbH (DE) 2023-04-05 EP disclosed
EP-4157835-A1 ISOXAZOLIDINES AS RIPK1 INHIBITORS AND USE THEREOF SANOFI (FR) 2023-04-05 EP disclosed
EP-4157851-A1 SUBSTITUTED PYRROLINE-2-ONES AND THEIR USE AS HERBICIDES Bayer Aktiengesellschaft (DE) 2023-04-05 EP disclosed
EP-4156936-A1 ACTIVE COMPOUND COMBINATIONS Bayer Aktiengesellschaft (DE) 2023-04-05 EP disclosed
CN-115916342-A Compounds, compositions and methods for treating fibrotic diseases and cancer 普渡研究基金会 2023-04-04 CN disclosed
CN-115915941-A Pyridine (thio) amides as fungicidal compounds 拜耳公司 2023-04-04 CN disclosed
CN-115916344-A AXL inhibitors for antiviral therapy 卑尔根生物股份公司 2023-04-04 CN disclosed
US-11617777-B2 Cytotoxic and anti-mitotic compounds, and methods of using the same ZYMEWORKS BC INC. 2023-04-04 US disclosed
CN-109311789-B Process for preparing 2, 3-unsaturated alcohols 巴斯夫欧洲公司 2023-04-04 CN disclosed
CN-115916747-A Fused heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2023-04-04 CN disclosed
US-20230099165-A1 AQUEOUS PHARMACEUTICAL FORMULATION OF HYDROCORTISONE SODIUM PHOSPHATE AND MONOTHIOGLYCEROL ANTARES PHARMA, INC. (US) 2023-03-30 US disclosed
US-20230101934-A1 CYCLODEXTRIN-BASED COMPOUNDS AND THEIR DERIVATIVES FOR SILICON-BASED LI-ION BATTERIES ENEVATE CORPORATION 2023-03-30 US disclosed
US-20230096870-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. 2023-03-30 US disclosed
US-20230094796-A1 PROCESS FOR PREPARING CYCLIC CARBONATES WITH AN EXOCYCLIC VINYLIDENE GROUP BASF SE (DE) 2023-03-30 US disclosed
US-20230096965-A1 SILICATE AND ORGANOSILICON CONTAINING ADDITIVES FOR SILICON-BASED LI ION BATTERIES ENEVATE CORPORATION 2023-03-30 US disclosed
US-20230102829-A1 Heteroaryl Compounds For Kinase Inhibition ARIAD PHARMACEUTICALS, INC. 2023-03-30 US disclosed
WO-2023049919-A1 INHIBITORS OF MOLLUSCUM CONTAGIOSUM INFECTION AND METHODS USING THE SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2023-03-30 WO disclosed
WO-2023046729-A1 CALIBRATION AID FOR OPTICAL IMAGING APPLICATIONS UNIVERSITE DE STRASBOURG (FR) 2023-03-30 WO disclosed
US-20230103027-A1 SURFACE PRIMER COMPOSITIONS AND METHODS OF USE ENVISTA (US) 2023-03-30 US disclosed
US-20230097090-A1 IMPROVED LIPID NANOPARTICLES FOR DELIVERY OF NUCLEIC ACIDS Acuitas Therapeutics, Inc. (CA) 2023-03-30 US disclosed
US-20230095171-A1 ORGANIC ACID ADDITIVES FOR SILICON-BASED LI ION BATTERIES ENEVATE CORPORATION 2023-03-30 US disclosed
US-20230099618-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH CYCLIC CARBONATE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2023-03-30 US disclosed
US-20230096187-A1 Compounds, Compositions, and Methods for Coloring Edible Materials THE PENN STATE RESEARCH FOUNDATION 2023-03-30 US disclosed
US-20230094087-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH PHOSPHAZENE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2023-03-30 US disclosed
EP-4155293-A1 PRC1 INHIBITORS AND METHODS OF TREATMENT THEREWITH The Regents of The University of Michigan (US) 2023-03-29 EP disclosed
EP-4155694-A1 CALIBRATION AID FOR OPTICAL IMAGING APPLICATIONS Université de Strasbourg (FR) 2023-03-29 EP disclosed
EP-4153566-A1 AZABICYCLIC(THIO)AMIDES AS FUNGICIDAL COMPOUNDS Bayer CropScience Aktiengesellschaft (DE) 2023-03-29 EP disclosed
CN-111655693-B Inhibition of transient receptor potential A1 ion channels 伊莱利利公司 2023-03-28 CN disclosed
US-11613542-B2 Sulfonylureas and sulfonylthioureas as NLRP3 inhibitors INFLAZOME LIMITED (IE) 2023-03-28 US disclosed
CN-110090308-B Method for preparing conjugate 四川科伦博泰生物医药股份有限公司 2023-03-24 CN disclosed
CN-110770236-B VMAT2 inhibitor compounds and compositions thereof 纽罗克里生物科学有限公司 2023-03-24 CN disclosed
CN-115843272-A Inhibitors of NEK7 kinase 哈利亚治疗公司 2023-03-24 CN disclosed
US-20230091510-A1 ANTIBODY DRUG CONJUGATES HAVING LINKERS COMPRISING HYDROPHILIC GROUPS NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2023-03-23 US disclosed
US-20230089484-A1 COMPOSITIONS FOR THE TREATMENT OF ANGIOLIPOMA RAZIEL THERAPEUTICS LTD. (IL) 2023-03-23 US disclosed
US-20230087744-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES INC (US) 2023-03-23 US disclosed
US-20230089921-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CONTINEUM THERAPEUTICS, INC. 2023-03-23 US disclosed
US-20230093099-A1 COMPOUNDS AND METHODS OF TREATING CANCERS CULLGEN (SHANGHAI), INC. (CN) 2023-03-23 US disclosed
US-20230092679-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2023-03-23 US disclosed
US-20230091115-A1 CROSSLINKABLE POLYSILOXANE COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2023-03-23 US disclosed
EP-4151235-A1 ANTIBODY DRUG CONJUGATE, PREPARATION METHOD THEREFOR AND USE THEREOF Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2023-03-22 EP disclosed
EP-4150009-A1 FLUOROGENIC DIMER COMPOUND, USEFUL AS A PROBE FOR DETECTION OF ENDOGENOUS RECEPTORS Université de Strasbourg (FR) 2023-03-22 EP disclosed
EP-4149927-A1 ENPP1 MODULATORS AND USES THEREOF VIR Biotechnology, Inc. (US) 2023-03-22 EP disclosed
EP-4149941-A1 CERTAIN CHEMICAL COMPOSITIONS AND METHODS OF USE THEREOF Algen Biotechnologies, Inc. (US) 2023-03-22 EP disclosed
EP-4149945-A1 SUBSTITUTED TRICYCLIC AMIDES, ANALOGUES THEREOF, AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2023-03-22 EP disclosed
EP-4149929-A1 TRIAZINE AND PYRIMIDINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS Bayer Aktiengesellschaft (DE) 2023-03-22 EP disclosed
CN-111448223-B Polyethylene compositions and articles made therefrom 埃克森美孚化学专利公司 2023-03-21 CN disclosed
US-11608414-B2 Peptoid polymers and methods of use X-THERMA, INC. (US) 2023-03-21 US disclosed
CN-110878048-B Anilines as psychotropic disorders 中国科学院上海药物研究所 2023-03-17 CN disclosed
US-20230081720-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2023-03-16 US disclosed
WO-2023036706-A1 SUBSTITUTED THIAZOLOPYRIDINES, SALTS THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2023-03-16 WO disclosed
US-20230078839-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR KINASES KHORA SPV 1, LLC 2023-03-16 US disclosed
US-20230083973-A1 SUBSTITUTED CYCLOPROPYL-2,2'-BIPYRIMIDINYL COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2023-03-16 US disclosed
US-20230080270-A1 NANOPARTICLES ENCAPSULATING SMALL MOLECULES ETH ZURICH (CH) 2023-03-16 US disclosed
WO-2023039240-A1 IRREVERSIBLE INHIBITORS OF KRas BIOMEA FUSION, INC. (US) 2023-03-16 WO disclosed
US-20230081390-A1 INHIBITORS OF RAF KINASES Pierre Fabre Médicament (FR) 2023-03-16 US disclosed
EP-4146168-A1 USE OF IL-6 ANTIBODIES AND VEGF TRAPS, AND FUSION CONSTRUCTS AND CONJUGATES THEREOF Kodiak Sciences Inc. (US) 2023-03-15 EP disclosed
EP-4146665-A1 SYSTEMS AND METHODS FOR TYROSINASE-MEDIATED SITE-SPECIFIC PROTEIN CONJUGATION GENENTECH, INC. (US) 2023-03-15 EP disclosed
EP-4146628-A1 PYRIDINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS Bayer Aktiengesellschaft (DE) 2023-03-15 EP disclosed
EP-4146348-A1 INHIBITORS OF NEK7 KINASE Halia Therapeutics, Inc. (US) 2023-03-15 EP disclosed
CN-115803320-A Heterocyclyl pyrimidines and triazines as novel fungicides 拜耳公司 2023-03-14 CN disclosed
US-11603381-B2 Precatalyst scaffolds for cross-coupling reactions, and methods of making and using same YALE UNIVERSITY (US) 2023-03-14 US disclosed
US-11605813-B2 Silicon-based energy storage devices with functional terthiophene compound or thiophene oligomer compound containing electrolyte additives ENEVATE CORPORATION (US) 2023-03-14 US disclosed
CN-115803317-A Azabicyclo (thio) amides as fungicidal compounds 拜耳作物科学股份公司 2023-03-14 CN disclosed
CN-112390832-B Metal complex, intermediate, preparation method and application thereof 中国科学院上海有机化学研究所 2023-03-14 CN disclosed
CN-110234635-B Novel substituted benzimidazole derivatives as D-amino oxidase (DAAO) inhibitors 宇凤·简·曾 2023-03-10 CN disclosed
WO-2023033723-A2 A MEMBRANE AND A METHOD OF MAKING THE SAME AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2023-03-09 WO disclosed
WO-2023034262-A1 FORMULATIONS FOR ANTIMICROBIAL THERMOSET COATINGS CORNING INCORPORATED (US) 2023-03-09 WO disclosed
WO-2023034393-A1 ADDITIVES FOR COLOR DRIFT REDUCTION IN COPPER-BASED ANTIMICROBIAL POLYMERIC FORMULATIONS CORNING INCORPORATED (US) 2023-03-09 WO disclosed
WO-2023031801-A1 BIFUNCTIONAL DEGRADERS COMPRISING A TEAD BINDER NOVARTIS AG (CH) 2023-03-09 WO disclosed
US-20230073334-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES TAKEDA PHARMACEUTICALS CO (JP) 2023-03-09 US disclosed
US-20230072421-A1 TARGETED RADIOPHARMACEUTICALS FOR THE DIAGNOSIS AND TREATMENT OF PROSTATE CANCER BAYER AS (NO) 2023-03-09 US disclosed
US-20230073777-A1 CYCLIC-AMP RESPONSE ELEMENT BINDING PROTEIN (CBP) AND/OR ADENOVIRAL E1A BINDING PROTEIN OF 300 KDA (P300) DEGRADATION COMPOUNDS AND METHODS OF USE CULLGEN (SHANGHAI), INC. (CN) 2023-03-09 US disclosed
US-20230070613-A1 PROTEIN TYROSINE KINASE 6 (PTK6) DEGRADATION / DISRUPTION COMPOUNDS AND METHODS OF USE ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI 2023-03-09 US disclosed
US-20230074545-A1 TREATMENT OF CANCER WITH CDK12/13 INHIBITORS KINNATE BIOPHARMA INC. 2023-03-09 US disclosed
EP-4143194-A1 CD73 INHIBITING 2,4-DIOXOPYRIMIDINE COMPOUNDS GILEAD SCIENCES, INC. (US) 2023-03-08 EP disclosed
EP-4144732-A1 BENZOTHIAZOLYL BIARYL COMPOUND, AND PREPARATION METHOD AND USE Shanghai Ringene BioPharma Co., Ltd. (CN) 2023-03-08 EP disclosed
EP-4142879-A1 METHODS AND COMPOSITIONS FOR OCULAR CELL THERAPY Novartis AG (CH) 2023-03-08 EP disclosed
EP-3867263-B1 PROTEOLYSIS TARGETING CHIMERA (PROTACS) AS DEGRADERS OF SMARCA2 AND/OR SMARCA4 BOEHRINGER INGELHEIM INT (DE) 2023-03-08 EP disclosed
EP-4143181-A1 1-PYRAZINYLPYRAZOLYL-3-OXYALKYL ACIDS AND THEIR DERIVATIVES, AND THEIR USE FOR CONTROL OF UNDESIRED PLANT GROWTH Bayer Aktiengesellschaft (DE) 2023-03-08 EP disclosed
CN-115746227-A Fluorine-containing block copolymer and use thereof 广州立邦涂料有限公司 2023-03-07 CN disclosed
CN-115747223-A Nucleic acid compositions of anti-coronavirus antibodies 中国人民解放军军事科学院军事医学研究院 2023-03-07 CN disclosed
US-11596615-B2 Compositions and methods for treatment of insulin resistance Temple University—Of the Commonwealth System of Higher Education (US) 2023-03-07 US disclosed
CN-115724920-A Nucleic acid vaccine for coronavirus and influenza virus 中国人民解放军军事科学院军事医学研究院 2023-03-03 CN disclosed
WO-2023027966-A1 PYRAZINE COMPOUNDS AS IRREVERSIBLE INHIBITORS OF FLT3 BIOMEA FUSION, INC. (US) 2023-03-02 WO disclosed
US-20230062100-A1 SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION BAYER AKTIENGESELLSCHAFT (DE) 2023-03-02 US disclosed
US-20230066946-A1 1,5-DIPHENYLPYRAZOLYL-3-OXYALKYL ACIDS AND 1-PHENYL-5-THIENYLPYRAZOLYL-3-OXYALKYL ACIDS AND THE USE THEREOF FOR CONTROL OF UNWANTED PLANT GROWTH BAYER AKTIENGESELLSCHAFT (DE) 2023-03-02 US disclosed
US-20230064576-A1 HETEROCYCLYL PYRIDAZINE AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2023-03-02 US disclosed
US-20230061438-A1 METHODS OF SEQUENCING BY SYNTHESIS USING A CONSECUTIVE LABELING SCHEME Roche Sequencing Solutions, Inc. 2023-03-02 US disclosed
US-20230064809-A1 SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION BAYER AKTIENGESELLSCHAFT (DE) 2023-03-02 US disclosed
US-20230061429-A1 BICYCLIC COMPOUNDS VIVACE THERAPEUTICS, INC. 2023-03-02 US disclosed
EP-4138812-A1 (S)-2-AMINO-6-((3-AMINOPROPYL)AMINO)HEXANOIC ACID (APL) FOR USE IN THE TREATMENT OF NON-ALCOHOLIC STEATOHEPATITIS (NASH), LIVER INFLAMMATION, HEPATOCELLULAR BALLOONING, LIVER FIBROSIS AND STEATOSIS Temple University - Of The Commonwealth System of Higher Education (US) 2023-03-01 EP disclosed
EP-4138823-A1 METHOD OF SELECTING PATIENTS FOR TREATMENT WITH A COMBINATION OF AN AXL INHIBITOR AND AN IMMUNE CHECKPOINT MODULATOR BerGenBio ASA (NO) 2023-03-01 EP disclosed
CN-109311813-B Palladium-catalyzed meta-C-H functionalized universal ligands 斯克利普斯研究院 2023-02-28 CN disclosed
US-11591355-B2 CD73 inhibitors and uses thereof PELOTON THERAPEUTICS INC. (US) 2023-02-28 US disclosed
US-11590135-B2 Fatty liver disease treatment using glucocorticoid and mineralocorticoid receptor antagonists CORCEPT THERAPEUTICS, INC. (US) 2023-02-28 US disclosed
US-11591333-B2 Substituted pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors CINAKATE PHARM TECH (SHANGHAI) CO., LTD. (CN) 2023-02-28 US disclosed
US-11591304-B2 SLC26A3 inhibitors and use thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-02-28 US disclosed
US-11591322-B2 Certain chemical compositions and methods of use thereof ALGEN BIOTECHNOLOGIES, INC. (US) 2023-02-28 US disclosed
US-11590235-B2 Factor VIII zwitterionic polymer conjugates KODIAK SCIENCES INC. (US) 2023-02-28 US disclosed
US-11594733-B1 Aqueous-based solid polymer suspensions in a polymer solution as a binder for Si dominant anodes ENEVATE CORPORATION (US) 2023-02-28 US disclosed
US-11590116-B2 Substituted pyridines and methods of use THERAVANCE BIOPHARMA R&D IP, LLC (US) 2023-02-28 US disclosed
CN-115715202-A Antibody drug conjugate, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-02-24 CN disclosed
US-20230054449-A1 PYRIDAZINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2023-02-23 US disclosed
US-20230053437-A1 LIPID COMPOUNDS AND LIPID NANOPARTICLE COMPOSITIONS Suzhou Abogen Biosciences Co., Ltd. (CN) 2023-02-23 US disclosed
WO-2023023500-A1 METHODS AND COMPOSITIONS FOR IDENTIFYING METHYLATED CYTOSINES ILLUMINA, INC. (US) 2023-02-23 WO disclosed
WO-2023023527-A1 PHOSPHOLIPID COMPOUNDS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. (US) 2023-02-23 WO disclosed
US-20230057177-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS CULLGEN (SHANGHAI), INC. (CN) 2023-02-23 US disclosed
US-20230055961-A1 PENTAFLUOROBENZENESULFONAMIDE DERIVATIVES AND USES THEREOF DUNAD THERAPEUTICS LTD. (GB) 2023-02-23 US disclosed
US-20230060004-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2023-02-23 US disclosed
EP-3529254-B1 PRODRUGS OF CLOFARABINE WU LAURENCE I (TW) 2023-02-22 EP disclosed
EP-3652111-B1 ELECTROCHROMIC POLYMER THIN FILMS HAVING REDUCED SELF-BLEACHING BEHAVIOR AND ENHANCED CYCLING STABILITY FURCIFER INC (US) 2023-02-22 EP disclosed
CN-115707710-A Sample derivatization reagent and application thereof in detecting optical isomer 中国科学院上海有机化学研究所 2023-02-21 CN disclosed
US-11584790-B2 Complement factor D antagonist antibodies and conjugates thereof KODIAK SCIENCES INC. (US) 2023-02-21 US disclosed
US-11584733-B2 Selective histone deacetylase inhibitors for the treatment of human disease SHUTTLE PHARMACEUTICALS, INC. (US) 2023-02-21 US disclosed
CN-115707708-A Wee1 kinase inhibitors 轩竹生物科技股份有限公司 2023-02-21 CN disclosed
CN-113616656-B Heterocyclic compounds for the treatment of PI 3K-gamma mediated disorders 无限药品股份有限公司 2023-02-17 CN disclosed
WO-2023018825-A1 COVALENT INHIBITORS OF MENIN-MLL INTERACTION FOR DIABETES MELLITUS BIOMEA FUSION, INC. (US) 2023-02-16 WO disclosed
WO-2023018699-A1 SELECTIVE KRAS INHIBITORS ERASCA, INC. (US) 2023-02-16 WO disclosed
WO-2023019163-A1 METHODS AND COMPOSITIONS FOR EDMAN-LIKE REACTIONS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-02-16 WO disclosed
US-20230052191-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2023-02-16 US disclosed
US-20230046340-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2023-02-16 US disclosed
US-20230046569-A1 NSD FAMILY INHIBITORS AND METHODS OF TREATMENT THEREWITH THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2023-02-16 US disclosed
US-20230047816-A1 PFKFB3 INHIBITORS AND THEIR USES GERO PTE. LTD. (SG) 2023-02-16 US disclosed
EP-4132947-A2 PEPTIDE COMPOSITIONS AND METHODS FOR INHIBITING NICOTINIC ACETYLCHOLINE RECEPTOR ACTIVITY GLO Pharma, Inc. (US) 2023-02-15 EP disclosed
EP-4132652-A1 AXL INHIBITORS FOR ANTIVIRAL THERAPY BerGenBio ASA (NO) 2023-02-15 EP disclosed
EP-4132938-A1 SUBSTITUTED THIAZOLOPYRIDINES, SALTS THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES Bayer Aktiengesellschaft (DE) 2023-02-15 EP disclosed
EP-3728254-B1 BENZYLAMINO SUBSTITUTED PYRIDOPYRIMIDINONES AND DERIVATIVES AS SOS1 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2023-02-15 EP disclosed
EP-4134364-A2 BROMODOMAIN INHIBITORS Celgene Quanticel Research, Inc. (US) 2023-02-15 EP disclosed
CN-115702161-A Peptide compositions and methods for inhibiting nicotinic acetylcholine receptor activity 格罗制药公司 2023-02-14 CN disclosed
CN-110526912-B Heteroaryl compounds for kinase inhibition 武田药品工业株式会社 2023-02-14 CN disclosed
CN-115702157-A Substituted pyrrolin-2-ones and their use as herbicides 拜耳公司 2023-02-14 CN disclosed
US-20230039244-A1 2-BETA-NAPHTHYL-ACETIC ACID ANALOGS AS AKR1C3 INHIBITORS AND METHODS OF USING SAME UNIV PENNSYLVANIA (US) 2023-02-09 US disclosed
WO-2023014793-A1 PROCESS FOR POLYAMIDE SYNTHESIS Design Therapeutics, Inc. (US) 2023-02-09 WO disclosed
US-20230044488-A1 AMINE COMPOUND, REACTIVE COALESCING AGENT, COATING COMPOSITION, COATING LAYER AND RELATED METHODS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2023-02-09 US disclosed
WO-2023014943-A1 METHODS OF TREATING MIGRAINE WITH MNK INHIBITORS 4E THERAPEUTICS, INC. (US) 2023-02-09 WO disclosed
US-20230037660-A1 METHODS OF TREATING VASCULAR LESIONS AND MALFORMATIONS Blaze Bioscience, Inc. 2023-02-09 US disclosed
US-20230040259-A1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES, LLC (US) 2023-02-09 US disclosed
US-20230039341-A1 ANTIBODY DRUG CONJUGATES (ADCS) AND ANTIBODY PRODRUG CONJUGATES (APDCS) WITH ENZYMATICALLY CLEAVABLE GROUPS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2023-02-09 US disclosed
US-20230044323-A1 COMPOSITIONS AND METHODS FOR POTENTIATING IMMUNE ACTIVITY KUMQUAT BIOSCIENCES INC. 2023-02-09 US disclosed
US-20230045421-A1 SUBSTITUTED ARYLMETHYLUREAS AND HETEROARYLMETHYLUREAS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORP (CA) 2023-02-09 US disclosed
US-20230039553-A1 CD73 COMPOUNDS GILEAD SCIENCES, INC. 2023-02-09 US disclosed
EP-4126824-A1 SUBSTITUTED PYRIMIDINES AND METHODS OF USE Theravance Biopharma R&D IP, LLC (US) 2023-02-08 EP disclosed
EP-4125908-A1 COMBINATION THERAPY COMPRISING AN AXL INHIBITOR BerGenBio ASA (NO) 2023-02-08 EP disclosed
US-11572353-B2 Alkynyl-substituted heterocyclic compound, preparation method therefor and medical use thereof BEIJING INNOCARE PHARMA TECH CO., LTD. (CN) 2023-02-07 US disclosed
US-11572344-B2 Cyanoaryl-aniline compounds for treatment of dermal disorders NFLECTION THERAPEUTICS, INC. (US) 2023-02-07 US disclosed
CN-111344316-B Polyethylene compositions and articles made therefrom 埃克森美孚化学专利公司 2023-02-03 CN disclosed
CN-115697986-A Isotopically substituted spiroaromatic ring compounds and their use 上海奕拓医药科技有限责任公司 2023-02-03 CN disclosed
CN-115697059-A Active compound combinations 拜耳公司 2023-02-03 CN disclosed
CN-115698009-A CD73 inhibiting 2,4-dioxopyrimidine compounds 吉利德科学公司 2023-02-03 CN disclosed
CN-115698021-A Substituted thiazolopyridines, salts thereof and their use as herbicidal active substances 拜耳公司 2023-02-03 CN disclosed
CN-115697989-A Tropomyosin Receptor Kinase (TRK) degrading compounds and methods of use 上海睿跃生物科技有限公司 2023-02-03 CN disclosed
US-20230032612-A1 QUATERNARY INDAZOLE GLUCOCORTICOID RECEPTOR ANTAGONISTS CORCEPT THERAPEUTICS INCORPORATED 2023-02-02 US disclosed
US-20230037255-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LTD (IE) 2023-02-02 US disclosed
US-20230031776-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC. (US) 2023-02-02 US disclosed
WO-2023009629-A1 ISOFORM SPECIFIC AGONISTS TARGETING AKT KINASE THOMAS JEFFERSON UNIVERSITY (US) 2023-02-02 WO disclosed
WO-2023007247-A1 COMPOSITIONS AND METHODS FOR TREATING LIPOMA PAIN RAZIEL THERAPEUTICS LTD. (IL) 2023-02-02 WO disclosed
WO-2022086937-A9 HETEROBIFUNCTIONAL COMPOUNDS AS DEGRADERS OF ENL ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2023-02-02 WO disclosed
CN-115667504-A Methods and compositions for ocular cell therapy 诺华股份有限公司 2023-01-31 CN disclosed
US-11566002-B2 Substituted tetrahydrocyclopenta[C]pyrroles, substituted dihydropyrrolizines, analogues thereof, and methods using same ARBUTUS BIOPHARMA CORPORATION (CA) 2023-01-31 US disclosed
US-11564388-B2 Supercooling methods for preservation of biological samples X-THERMA, INC. (US) 2023-01-31 US disclosed
CN-115667238-A Five-membered ring derivative and application thereof in medicine 四川海思科制药有限公司 2023-01-31 CN disclosed
CN-110294742-B Fused ring ASK1 inhibitor and application thereof 山东轩竹医药科技有限公司 2023-01-31 CN disclosed
US-11569530-B2 Silicon-based energy storage devices with functional thiophene compounds or derivatives of thiophene containing electrolyte additives ENEVATE CORPORATION (US) 2023-01-31 US disclosed
WO-2023002323-A1 SYNTHESIS OF SUBSTITUTED TRICYCLIC AMIDES AND ANALOGUES THEREOF ARBUTUS BIOPHARMA CORPORATION (CA) 2023-01-26 WO disclosed
US-20230027219-A1 Skin Care Compositions and Methods of Use Thereof UNIGEN, INC. (US) 2023-01-26 US disclosed
US-20230022524-A1 HETEROBIFUNCTIONAL COMPOUNDS AS DEGRADERS OF HPK1 ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI 2023-01-26 US disclosed
US-20230029385-A1 2-METHYL-AZA-QUINAZOLINES BAYER AG (DE) 2023-01-26 US disclosed
US-20230029191-A1 PRELITHIATION OF FREE-STANDING SILICON DOMINANT ANODE BATTERIES ENEVATE CORPORATION 2023-01-26 US disclosed
US-20230022235-A1 DUAL ANDROGEN RECEPTOR/AKR1C3 INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-01-26 US disclosed
EP-3630744-B1 PYRAZOLE MAGL INHIBITORS H LUNDBECK AS (DK) 2023-01-25 EP disclosed
EP-4122929-A1 NOVEL COMPOUNDS Mission Therapeutics Limited (GB) 2023-01-25 EP disclosed
EP-4122935-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE Gilead Sciences, Inc. (US) 2023-01-25 EP disclosed
US-11560422-B2 Sulfonamide-containing linkage systems for drug conjugates ZYMEWORKS INC. 2023-01-24 US disclosed
US-11559580-B1 Tissue-homing peptide conjugates and methods of use thereof Blaze Bioscience, Inc. (US) 2023-01-24 US disclosed
CN-115626927-A Tropomyosin Receptor Kinase (TRK) degrading compounds and methods of use 上海睿跃生物科技有限公司 2023-01-20 CN disclosed
US-20230019280-A1 SUBSTITUTED ISOINDOLONYL 2,2'-BIPYRIMIDINYL COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2023-01-19 US disclosed
WO-2023287984-A1 SUBEROYLANILIDE HYDROXAMIC ACID (SAHA) DRUGS, CONJUGATES, AND NANOPARTICLES, AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2023-01-19 WO disclosed
US-20230013227-A1 ARYL-ANILINE AND HETEROARYL-ANILINE COMPOUNDS FOR TREATMENT OF BIRTHMARKS NFLECTION THERAPEUTICS, INC. 2023-01-19 US disclosed
US-20230018615-A1 STEROIDS AND METHODS OF MANUFACTURE TRUSTEES OF DARTMOUTH COLLEGE 2023-01-19 US disclosed
US-20230017200-A1 DIHYDROOXADIAZINONES BAYER AKTIENGESELLSCHAFT (DE) 2023-01-19 US disclosed
US-20230018423-A1 BENZIMIDAZOLE DERIVATIVES FOR TREATMENT AND/OR PREVENTION OF DISEASES AND DISORDERS MEDIATED BY NLRP3 YODA THERAPEUTICS INC. (TW) 2023-01-19 US disclosed
US-20230019342-A1 PHOSPHORYLATED AKT-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING CALIFORNIA INSTITUTE OF TECHNOLOGY 2023-01-19 US disclosed
US-11554153-B2 Compositions and methods for managing or improving bone disorders, joint disorders, cartilage disorders, or a combination thereof UNIGEN, INC. (US) 2023-01-17 US disclosed
US-11555010-B2 Diamide antimicrobial agents BROWN UNIVERSITY (US) 2023-01-17 US disclosed
CN-115605462-A Triazine and pyrimidine (thio) amides as fungicidal compounds 拜耳公司(DE) 2023-01-13 CN disclosed
WO-2023283453-A1 PHENYL ACETAMIDE BASED IL-17A MODULATORS AND USES THEREOF DICE ALPHA, INC. (US) 2023-01-12 WO disclosed
EP-4114837-A1 PYRAZOLOPYRAZINES ACTING ON CANCERS VIA INHIBITION OF CDK12 Bayer Aktiengesellschaft (DE) 2023-01-11 EP disclosed
EP-4114528-A1 IMIDAZOTRIAZINES ACTING ON CANCER VIA INHIBITION OF CDK12 Bayer Aktiengesellschaft (DE) 2023-01-11 EP disclosed
US-11547697-B2 Heterocyclic compounds and uses thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2023-01-10 US disclosed
US-11552334-B1 Nitrogen-containing compounds as additives for silicon-based Li-ion batteries ENEVATE CORPORATION (US) 2023-01-10 US disclosed
US-11548901-B2 Substituted 1,4-methanopyrido[1′,2′:4,5]pyrazino[1,2-a]pyrimidines for treating viral infections GILEAD SCIENCES, INC. (US) 2023-01-10 US disclosed
US-11548892-B1 Transglutaminase 2 (TG2) inhibitors SITARI PHARMA, INC. (US) 2023-01-10 US disclosed
CN-111349128-B Flavonol derivative and preparation method and application thereof 上海医药工业研究院 2023-01-06 CN disclosed
US-20230002388-A1 PIPERIDINYL-METHYL-PURINEAMINES AS NSD2 INHIBITORS AND ANTI-CANCER AGENTS CHINA NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH CO., LTD. (CN) 2023-01-05 US disclosed
US-20230001008-A1 COMPOSITIONS AND METHODS FOR TARGETING CELLULAR MOLECULES KUMQUAT BIOSCIENCES INC. 2023-01-05 US disclosed
US-20230006252-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH FUNCTIONALIZED LINEAR SULFONATE ESTER DERIVATIVE COMPOUND CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2023-01-05 US disclosed
US-20230002366-A1 INDENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION TARO PHARMACEUTICALS INC. (CA) 2023-01-05 US disclosed
WO-2023278691-A1 METHODS OF TREATING OR PREVENTING CORONAVIRUS INFECTION WITH CANNABINOID ACIDS OREGON STATE UNIVERSITY (US) 2023-01-05 WO disclosed
WO-2023274257-A1 IMIDAZOLE COMPOUND, AND INTERMEDIATE AND APPLICATION THEREOF 诸葛国琴 2023-01-05 WO disclosed
EP-4112602-A1 ENANTIOSELECTIVE HYDROGENATION OF 4-SUBSTITUTED 1,2-DIHYDROQUINOLINES IN PRESENCE OF A CHIRAL IRIDIUM CATALYST Bayer Aktiengesellschaft (DE) 2023-01-04 EP disclosed
US-11543584-B2 Inorganic matrix nanoimprint lithographs and methods of making thereof with reduced carbon META PLATFORMS TECHNOLOGIES, LLC (US) 2023-01-03 US disclosed
US-11542291-B2 Compounds, compositions, and methods for coloring edible materials THE PENN STATE RESEARCH FOUNDATION (US) 2023-01-03 US disclosed
US-11541059-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2023-01-03 US disclosed
US-11542248-B2 Methods and compositions for inhibiting the interaction of menin with MLL proteins KURA ONCOLOGY, INC. (US) 2023-01-03 US disclosed
US-11542225-B2 Lipids for use in lipid nanoparticle formulations Acuitas Therapeutics, Inc. (CA) 2023-01-03 US disclosed
US-11542255-B2 Sulfonylureas and sulfonylthioureas as NLRP3 inhibitors INFLAZOME LIMITED (IE) 2023-01-03 US disclosed
CN-115557898-A Imidazole compound, intermediate and application thereof 诸葛国琴 2023-01-03 CN disclosed
CN-115551864-A Substituted tricyclic amides, analogs thereof, and methods of using the same 爱彼特生物制药公司 2022-12-30 CN disclosed
CN-109843379-B Substituted ureas and methods of making and using the same 梅比斯发现公司 2022-12-30 CN disclosed
CN-115551875-A Systems and methods for tyrosinase-mediated site-specific protein conjugation 基因泰克公司 2022-12-30 CN disclosed
WO-2022271658-A1 TRICYCLIC KRAS INHIBITORS ERASCA, INC. (US) 2022-12-29 WO disclosed
WO-2022271659-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2022-12-29 WO disclosed
WO-2022271677-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2022-12-29 WO disclosed
WO-2022271650-A1 DIACYLGLYERCOL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2022-12-29 WO disclosed
WO-2022268935-A2 NOVEL PROCESS F. HOFFMANN-LA ROCHE AG (CH) 2022-12-29 WO disclosed
WO-2022268520-A1 USE OF SUBSTITUTED PYRROLIDINONES OR THEIR SALTS FOR INCREASING STRESS TOLERANCE OF PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2022-12-29 WO disclosed
US-20220409707-A1 DEVICES AND METHODS FOR MODULATING ADMA IN BLOOD THE TRUSTEES OF INDIANA UNIVERSITY 2022-12-29 US disclosed
US-20220411448-A1 CHROMENE-4-ONE DERIVATIVES AS BRAIN-DERIVED NEUROTROPHIC FACTOR (BDNF) MIMETICS Floratek Pharma SA (CH) 2022-12-29 US disclosed
EP-4106877-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2022-12-28 EP disclosed
EP-4108240-A2 BENZIMIDAZOLE DERIVATIVES FOR TREATMENT AND/OR PREVENTION OF DISEASES AND DISORDERS MEDIATED BY NLRP3 Yoda Pharmaceuticals Inc. (KY) 2022-12-28 EP disclosed
EP-4107153-A1 COMPOUNDS Inflazome Limited (IE) 2022-12-28 EP disclosed
EP-3889237-B1 PHOTOACTIVE MACROMOLECULES AND USES THEREOF BECKMAN COULTER INC (US) 2022-12-28 EP disclosed
US-11535616-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC (US) 2022-12-27 US disclosed
US-11534440-B2 Combination therapy with Axl inhibitor and immune checkpoint modulator or oncolytic virus BERGENBIO ASA (NO) 2022-12-27 US disclosed
US-11539077-B2 Electrolyte additives containing one, two, or more triple-bonded moieties for silicon anode-based li-ion batteries ENEVATE CORPORATION (US) 2022-12-27 US disclosed
US-11535713-B2 Network polymers and methods of making and using same THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2022-12-27 US disclosed
CN-115516044-A Fluorescent dimeric compounds useful as probes for the detection of endogenous receptors 斯特拉斯堡大学 2022-12-23 CN disclosed
CN-115504962-A Benzimidazole derivatives for the treatment and/or prevention of diseases and disorders mediated by NLRP3 思捷优达股份有限公司 2022-12-23 CN disclosed
US-20220401335-A1 SILK HAIR CARE COMPOSITIONS EVOLVED BY NATURE, INC. (US) 2022-12-22 US disclosed
US-20220402889-A1 NOVEL HETEROCYCLIC COMPOUNDS Floratek Pharma SA (CH) 2022-12-22 US disclosed
WO-2022265974-A1 AMINOHETEROCYCLE-SUBSTITUTED TRICYCLIC KRAS INHIBITORS ERASCA, INC. (US) 2022-12-22 WO disclosed
WO-2022266491-A1 PROTEOLYSIS TARGETING CHIMERAS AND POLYPHARMACOLOGICAL AGENTS TARGETING BCL-2, AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2022-12-22 WO disclosed
WO-2022265913-A1 COPOLYMERS AND ELECTROCHEMICAL SYSTEMS AND METHODS FOR THE REMEDIATION OF ORGANIC POLLUTANTS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2022-12-22 WO disclosed
WO-2022266206-A1 KRAS INHIBITOR CONJUGATES ERASCA, INC. (US) 2022-12-22 WO disclosed
WO-2022266167-A1 AMIDE AND UREA-CONTAINING TRICYCLIC KRAS INHIBITORS ERASCA, INC. (US) 2022-12-22 WO disclosed
WO-2022266069-A1 TRICYCLIC KRAS G12D INHIBITORS ERASCA, INC. (US) 2022-12-22 WO disclosed
EP-4103564-A1 P2X3 MODULATORS Bellus Health Cough Inc. (CA) 2022-12-21 EP disclosed
EP-4103160-A1 NANOPARTICLES ENCAPSULATING SMALL MOLECULES ETH Zurich (CH) 2022-12-21 EP disclosed
CN-115490709-A KRASG12D inhibitor and application thereof in medicine 四川海思科制药有限公司 2022-12-20 CN disclosed
US-11530199-B2 Analogs for the treatment of disease INSILICO MEDICINE IP LIMITED (HK) 2022-12-20 US disclosed
US-11530197-B2 Analogs for the treatment of disease INSILICO MEDICINE IP LIMITED (HK) 2022-12-20 US disclosed
US-11529356-B2 2-(morpholin-4-yl)-1,7-naphthyridines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2022-12-20 US disclosed
US-11530200-B2 Compounds INFLAZOME LIMITED (IE) 2022-12-20 US disclosed
CN-115477640-A Pyridazinones as PARP7 inhibitors 由理生物医药(上海)有限公司 2022-12-16 CN disclosed
US-20220396556-A1 Lipid and Lipid Nanoparticle Formulation for Drug Delivery THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2022-12-15 US disclosed
US-20220396554-A1 DIHYDROOXADIAZINONES BAYER AKTIENGESELLSCHAFT (DE) 2022-12-15 US disclosed
US-20220396549-A1 SMALL MOLECULE INHIBITORS OF THE MCL-1 ONCOPROTEIN AND USES THEROF UNIV MARYLAND (US) 2022-12-15 US disclosed
WO-2022261220-A1 PROTEOLYSIS TARGETING CHIMERAS AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2022-12-15 WO disclosed
WO-2022261210-A1 KRAS MODULATORS AND USES THEREOF QUANTA THERAPEUTICS, INC. (US) 2022-12-15 WO disclosed
EP-4100381-A1 SUBSTITUTED 1,1'-BIPHENYL COMPOUNDS AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2022-12-14 EP disclosed
EP-3746432-B1 4-HYDROXYPIPERIDINE DERIVATIVES AND THEIR USE AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 19 (USP19) ALMAC DISCOVERY LTD (GB) 2022-12-14 EP disclosed
US-11524932-B2 Lipids for use in lipid nanoparticle formulations Acuitas Therapeutics, Inc. (CA) 2022-12-13 US disclosed
US-11525123-B2 Diverse carbene transferase enzyme catalysts derived from a P450 enzyme CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-12-13 US disclosed
US-11524943-B1 Benzocarbonyl compounds VIVACE THERAPEUTICS, INC. (US) 2022-12-13 US disclosed
CN-107474024-B Glutaminase inhibitor and composition and application thereof 北京赛林泰医药技术有限公司 2022-12-13 CN disclosed
CN-115448923-A Pyrimido-cyclic compounds, process for their preparation and their use 青煜医药研发(上海)有限公司 2022-12-09 CN disclosed
CN-115461049-A (S) -2-amino-6- ((3-aminopropyl) amino) hexanoic Acid (APL) for the treatment of non-alcoholic steatohepatitis (NASH), liver inflammation, hepatocellular ballooning, liver fibrosis and steatosis 坦普尔大学 2022-12-09 CN disclosed
US-20220393174-A1 CROWN ETHERS AS ADDITIVES FOR SILICON-BASED LI-ION BATTERIES ENEVATE CORPORATION 2022-12-08 US disclosed
US-20220389031-A1 MACROCYCLIC SULFONYLAMIDE DERIVATIVES USEFUL AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2022-12-08 US disclosed
US-20220388990-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASES KINNATE BIOPHARMA INC. 2022-12-08 US disclosed
US-20220388971-A1 [(1,5-DIPHENYL-1H-1,2,4-TRIAZOL-3-YL)OXY]ACETIC ACID DERIVATIVES AND SALTS THEREOF, CROP PROTECTION COMPOSITIONS COMPRISING THEM, METHODS FOR PRODUCING THEM AND USE THEREOF AS SAFENERS BAYER AKTIENGESELLSCHAFT (DE) 2022-12-08 US disclosed
US-20220387608-A1 ADRENOMEDULLIN-ANALOGUES FOR LONG-TERM STABILIZATION AND THEIR USE BAYER AKTIENGESELLSCHAFT (DE) 2022-12-08 US disclosed
WO-2022256459-A1 KRAS MODULATORS AND USES THEREOF QUANTA THERAPEUTICS, INC. (US) 2022-12-08 WO disclosed
US-20220387400-A1 FORMULATIONS OF RBP4 INHIBITORS AND METHODS OF USE Belite Bio (HK) Limited (HK) 2022-12-08 US disclosed
WO-2022253101-A1 PYRIDAZINONE COMPOUND AS PARP7 INHIBITOR 上海优理惠生医药有限公司 2022-12-08 WO disclosed
EP-3368507-B1 NOVEL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS ACUITAS THERAPEUTICS INC (CA) 2022-12-07 EP disclosed
EP-4096653-A1 COMPOSITIONS FOR THE TREATMENT OF ANGIOLIPOMA Raziel Therapeutics Ltd. (IL) 2022-12-07 EP disclosed
EP-4096661-A1 COMPOUNDS AND COMPOSITIONS FOR USE IN TREATING SKIN DISORDERS Kamari Pharma Ltd. (IL) 2022-12-07 EP disclosed
EP-4096415-A1 WATER RESISTANT MATERIALS FOR FOOD-SAFE USES JL Darling LLC (US) 2022-12-07 EP disclosed
EP-4097087-A1 [(1,4,5-TRISUBSTITUTED-1H-PYRAZOL-3-YL)SULFANYL]ACETIC ACID DERIVATIVES, SALTS THEREOF, AND USE THEREOF AS HERBICIDAL INGREDIENTS Bayer Aktiengesellschaft (DE) 2022-12-07 EP disclosed
CN-115443269-A Substituted pyrimidines and methods of use 施万生物制药研发IP有限责任公司 2022-12-06 CN disclosed
CN-115433190-A Preparation method and application of irreversible heterocyclic compound FGFR inhibitor 药雅科技(上海)有限公司 2022-12-06 CN disclosed
US-11518739-B2 Sulfonamide carboxamide compounds INFLAZOME LIMITED (IE) 2022-12-06 US disclosed
US-11522223-B2 Silicon-based energy storage devices with phosphazene containing electrolyte additives ENEVATE CORPORATION (US) 2022-12-06 US disclosed
US-11518840-B2 Dynamic covalent thermoset nanocomposites and uses thereof THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2022-12-06 US disclosed
US-11518768-B2 Artificial metalloenzymes containing noble metal-porphyrins THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-12-06 US disclosed
CN-111471059-B PDE9 inhibitors and uses thereof 药捷安康(南京)科技股份有限公司 2022-12-02 CN disclosed
US-20220380371-A1 MLL1 INHIBITORS AND ANTI-CANCER AGENTS CHINA NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH CO., LTD. (CN) 2022-12-01 US disclosed
EP-3080100-B1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2022-11-30 EP disclosed
CN-115413279-A P2X3 modulators 贝卢斯医疗咳嗽病公司 2022-11-29 CN disclosed
US-11512066-B2 Sulfonyl piperidine derivatives and their use for treating prokineticin mediated diseases TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2022-11-29 US disclosed
CN-115413275-A Substituted 1,1 , -biphenyl compounds and methods of use thereof 爱彼特生物制药公司 2022-11-29 CN disclosed
CN-110945001-B FMS-like tyrosine kinase inhibitors 硕英生医股份有限公司 2022-11-25 CN disclosed
EP-4090655-A1 PROCESS FOR PREPARING CYCLIC CARBONATES WITH AN EXOCYCLIC VINYLIDENE GROUP BASF SE (DE) 2022-11-23 EP disclosed
CN-115379831-A Nanoparticles encapsulating small molecules 苏黎世联邦理工学院 2022-11-22 CN disclosed
CN-115368381-A Preparation and application of heterocyclic inhibitor 药雅科技(上海)有限公司 2022-11-22 CN disclosed
CN-113710661-B Compounds and methods for treating cancer 上海睿跃生物科技有限公司 2022-11-22 CN disclosed
CN-115362003-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2022-11-18 CN disclosed
CN-113861195-B Multi-condensed-ring EGFR inhibitor as well as preparation method and application thereof 上海和誉生物医药科技有限公司 2022-11-18 CN disclosed
CN-115362152-A Compound (I) 英夫拉索姆有限公司 2022-11-18 CN disclosed
WO-2022200540-A9 HETERO BENZYL AMINES AND THEIR USE TREATING CENTRAL NERVOUS SYSTEM DISORDERS Floratek Pharma SA (CH) 2022-11-17 WO disclosed
US-11498930-B2 Pyrimidine-fused cyclic compound, preparation method therefor and application thereof Blueray Therapeutics (Shanghai) Co., Ltd (CN) 2022-11-15 US disclosed
CN-109790160-B Pyrido five-membered aromatic ring compound, preparation method and application thereof 上海海和药物研究开发股份有限公司 2022-11-15 CN disclosed
CN-115340552-A Heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2022-11-15 CN disclosed
CN-115340561-A Preparation and application of SHP2 phosphatase fused ring inhibitor 药雅科技(上海)有限公司 2022-11-15 CN disclosed
CN-115340559-A Preparation and application of SHP2 phosphatase heterocyclic inhibitor 药雅科技(上海)有限公司 2022-11-15 CN disclosed
CN-115335081-A Targeted plasma protein degradation 诺华股份有限公司 2022-11-11 CN disclosed
CN-115335047-A Composition for treating vascular lipoma 拉结尔治疗有限公司 2022-11-11 CN disclosed
CN-115335050-A Compounds and compositions for treating skin conditions 卡玛瑞制药有限公司 2022-11-11 CN disclosed
WO-2022234339-A2 5-HT2A AND/OR 5-HT2C RECEPTOR AGONISTS DIAMOND THERAPEUTICS INC. (CA) 2022-11-10 WO disclosed
CN-115304623-A Pyrimido-cyclic derivative and application thereof in medicine 四川海思科制药有限公司 2022-11-08 CN disclosed
CN-111196816-B Seven-membered ring compound and application thereof in preventing and treating diabetes and metabolic syndrome 中国科学院上海药物研究所 2022-11-04 CN disclosed
WO-2022232552-A1 LIPID NANOPARTICLE THERAPEUTICS THAT EVADE THE IMMUNE RESPONSE THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2022-11-03 WO disclosed
WO-2022232514-A1 COMPOSITIONS AND METHODS FOR TARGETING LIPID NANOPARTICLE THERAPEUTICS TO STEM CELLS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2022-11-03 WO disclosed
CN-115279368-A Heteroaryl compounds 维瓦斯治疗公司 2022-11-01 CN disclosed
CN-115260214-A Condensed ring KRASG12DPreparation and application of mutant protein inhibitor 药雅科技(上海)有限公司 2022-11-01 CN disclosed
CN-115279417-A Bioactive substance conjugate and preparation method and application thereof 苏州宜联生物医药有限公司 2022-11-01 CN disclosed
CN-115252762-A Growth factor binding application of macromolecular compound 华东理工大学 2022-11-01 CN disclosed
CN-111278872-B Polyethylene compositions and articles made therefrom 埃克森美孚化学专利公司 2022-10-28 CN disclosed
US-11478451-B1 Macrocyclic chlorine substituted indole derivatives BAYER AKTIENGESELLSCHAFT (DE) 2022-10-25 US disclosed
CN-110317212-B Synthesis of polycyclic carbamoylpyridone compounds 吉利德科学公司 2022-10-21 CN disclosed
CN-115215823-A FXR (FXR) regulator and preparation method, pharmaceutical composition and application thereof 青岛睿吉医疗技术有限公司 2022-10-21 CN disclosed
CN-115215868-A Preparation method and application of heterocyclic compound FGFR inhibitor 药雅科技(上海)有限公司 2022-10-21 CN disclosed
WO-2022218440-A1 FXR REGULATOR, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF 青岛睿吉医疗技术有限公司 2022-10-20 WO disclosed
WO-2022221395-A1 METHODS OF TREATING AN EYE DISORDER KODIAK SCIENCES INC. (US) 2022-10-20 WO disclosed
US-20220332721-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CONTINEUM THERAPEUTICS, INC. 2022-10-20 US disclosed
CN-111465626-B Polyethylene compositions and films made therefrom 埃克森美孚化学专利公司 2022-10-18 CN disclosed
CN-115210225-A Substituted aminoquinolones as immuno-activated DGKALPHA inhibitors 拜耳公司 2022-10-18 CN disclosed
US-11472799-B2 Serine threonine kinase (AKT) degradation / disruption compounds and methods of use ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2022-10-18 US disclosed
CN-115197221-A Dihydropyrazolopyrimidinone macrocyclic derivatives and application thereof 轩竹生物科技股份有限公司 2022-10-18 CN disclosed
US-11472766-B2 Lipid nanoparticle composition Suzhou Abogen Biosciences Co., Ltd. (CN) 2022-10-18 US disclosed
CN-110551105-B Substituted triazoles useful as AXL inhibitors 里格尔制药公司 2022-10-18 CN disclosed
CN-115181106-A Quinazoline KRAS G12D Preparation and application of mutant protein inhibitor 药雅科技(上海)有限公司 2022-10-14 CN disclosed
WO-2022216386-A2 T-TYPE CALCIUM CHANNEL ANTAGONISTS AND USES THEREOF THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2022-10-13 WO disclosed
US-20220324866-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2022-10-13 US disclosed
US-20220323378-A1 Pharmaceutical Compositions and Methods for Treating Mental Health Disorders and Promoting Neural Plasticity JOSEPH SHAWN (US) 2022-10-13 US disclosed
CN-115175735-A Antiviral compounds 吉利德科学公司 2022-10-11 CN disclosed
CN-115175899-A Treatment of cancer using CDK12/13 inhibitors 金耐特生物制药公司 2022-10-11 CN disclosed
US-20220315706-A1 PHOTOPOLYMERIZABLE THERMOPLASTICS AND METHODS OF MAKING AND USING SAME UNIV COLORADO REGENTS (US) 2022-10-06 US disclosed
US-20220315895-A1 METHODS OF MAKING OLIGOPOTENT AND UNIPOTENT PRECURSORS IMMUNEBRIDGE LLC 2022-10-06 US disclosed
WO-2022212326-A1 NEK7 INHIBITORS Halia Therapeutics, Inc. (US) 2022-10-06 WO disclosed
EP-4066834-A1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF PI3K-GAMMA MEDIATED DISORDERS Infinity Pharmaceuticals, Inc. (US) 2022-10-05 EP disclosed
EP-4065552-A1 ANTHRAQUINONE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS Facebook Technologies, LLC (US) 2022-10-05 EP disclosed
EP-4067355-A1 SPIRO-CONDENSED PYRROLIDINE DERIVATIVES AS DEUBIQUITYLATING ENZYME (DUB) INHIBITORS Mission Therapeutics Limited (GB) 2022-10-05 EP disclosed
EP-4065551-A1 AROMATIC SUBSTITUTED METHANE-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS Facebook Technologies, LLC (US) 2022-10-05 EP disclosed
EP-4065570-A1 SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION Bayer Aktiengesellschaft (DE) 2022-10-05 EP disclosed
CN-110156770-B Aminopyridine derivatives as inhibitors of TAM family kinases 圣诺康生命科学公司 2022-10-04 CN disclosed
CN-115141176-A Alkyne-indole FGFR inhibitor and preparation method and application thereof 药雅科技(上海)有限公司 2022-10-04 CN disclosed
CN-109568323-B Antibacterial composition and use thereof 吉林四环制药有限公司 2022-09-30 CN disclosed
CN-115135152-A 1, 5-diphenylpyrazolyl-3-oxyalkyl acids and 1-phenyl-5-thienylpyrazolyl-3-oxyalkyl acids and their use for controlling undesired vegetation 拜耳公司 2022-09-30 CN disclosed
WO-2022200208-A1 SUBSTITUTED PYRROLIDIN-2-ONES, SALTS THEREOF AND THEIR USE AS HERBICIDALLY ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2022-09-29 WO disclosed
WO-2022204301-A1 ELECTROCHEMICAL POLYNUCLEOTIDE SYNTHESIS Twist Bioscience Corporation (US) 2022-09-29 WO disclosed
WO-2022204481-A1 PYRAZOLOPYRIMIDINONE COMPOUNDS Orphagen Pharmaceuticals, Inc. (US) 2022-09-29 WO disclosed
CN-115112898-A IL-17F-specific capture agents, compositions, and methods of use and manufacture 加州理工学院 2022-09-27 CN disclosed
CN-115108988-A Synthesis and use of polyfunctional diaziridines binders for elastomer bonding 元平台技术有限公司 2022-09-27 CN disclosed
US-11453790-B2 Photo-cleavable primer compositions and methods of use ENVISTA (US) 2022-09-27 US disclosed
CN-115103907-A Compositions and methods for enhancing immune activity 金橘生物科技公司 2022-09-23 CN disclosed
CN-115103709-A MASP-2 inhibitors and methods of use 奥默罗斯公司 2022-09-23 CN disclosed
US-20220298420-A1 MULTIFUNCTIONAL LIQUID CRYSTALLINE PHOTOREACTIVE POLYMERS FOR POLARIZATION HOLOGRAPHY META PLATFORMS TECHNOLOGIES, LLC 2022-09-22 US disclosed
US-20220298102-A1 BICYCLIC COMPOUNDS VIVACE THERAPEUTICS, INC. 2022-09-22 US disclosed
US-20220299938-A1 SPATIALLY VARYING DYNAMIC RANGE IN HOLOGRAPHIC GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2022-09-22 US disclosed
CN-115073468-A Preparation and application of imidazopyrazine BTK inhibitor 药雅科技(上海)有限公司 2022-09-20 CN disclosed
CN-115068574-A Compositions and methods for joint health 尤妮金公司 2022-09-20 CN disclosed
CN-115073469-A Preparation and application of pyrrolopyrimidine compound as kinase inhibitor 药雅科技(上海)有限公司 2022-09-20 CN disclosed
CN-115087486-A Substituted bicyclic and tricyclic ureas and amides, analogs thereof, and methods of use thereof 爱彼特生物制药公司 2022-09-20 CN disclosed
CN-115073451-A KRAS G12D Preparation and application of mutant protein inhibitor 药雅科技(上海)有限公司 2022-09-20 CN disclosed
CN-115073450-A KRAS G12C Preparation and application of mutant protein inhibitor 药雅科技(上海)有限公司 2022-09-20 CN disclosed
US-11447504-B2 Macrocyclic chlorine substituted indole derivatives BAYER AKTIENGESELLSCHAFT (DE) 2022-09-20 US disclosed
CN-115066241-A Compositions for treating solid tumors 拉结尔治疗有限公司 2022-09-16 CN disclosed
CN-115066457-A Crosslinkable polysiloxanes 联邦科学和工业研究组织 2022-09-16 CN disclosed
US-20220294016-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ETHER CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2022-09-15 US disclosed
WO-2022192598-A1 HETEROCYCLES AND USES THEREOF KUMQUAT BIOSCIENCES INC. (US) 2022-09-15 WO disclosed
US-20220289708-A1 SUBSTITUTED N-PHENYL URACILS, SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2022-09-15 US disclosed
CN-115043841-A Preparation and application of heterocyclic compound as BTK inhibitor 药雅科技(上海)有限公司 2022-09-13 CN disclosed
US-11440923-B2 Substituted macrocyclic indole derivatives BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2022-09-13 US disclosed
CN-115052604-A MASP-2 inhibitors and methods of use 奥默罗斯公司 2022-09-13 CN disclosed
CN-115052862-A MASP-2 inhibitors and methods of use 奥默罗斯公司 2022-09-13 CN disclosed
CN-115043832-A FGFR inhibitor alkyne-substituted heterocyclic compound and preparation method and application thereof 药雅科技(上海)有限公司 2022-09-13 CN disclosed
WO-2022184748-A1 SUBSTITUTED 3,6-DIHYDRO-2H-1,3,4-OXADIAZIN-2-ONES FOR THE TREATMENT OF SARCOMA BAYER AKTIENGESELLSCHAFT (DE) 2022-09-09 WO disclosed
CN-111658653-B Use of phosphodiesterase inhibitors 药捷安康(南京)科技股份有限公司 2022-09-09 CN disclosed
CN-115028634-A Alkynylpyrazine heterocyclic FGFR inhibitor and preparation method and application thereof 药雅科技(上海)有限公司 2022-09-09 CN disclosed
CN-115028633-A Preparation and application of pyrrolopyrimidine compounds 药雅科技(上海)有限公司 2022-09-09 CN disclosed
US-11433065-B2 Certain chemical entities, compositions and methods INTELLIKINE LLC (US) 2022-09-06 US disclosed
CN-115023418-A Bis-aminoquinoline and nanoformulation for cancer treatment 加利福尼亚大学董事会 2022-09-06 CN disclosed
CN-115023427-A Pyrazolotriazines 拜耳公司 2022-09-06 CN disclosed
CN-115003656-A [ (1,4, 5-trisubstituted-1H-pyrazol-3-yl) sulfanyl ] acetic acid derivatives and salts thereof, and their use as active herbicidal agents 拜耳公司 2022-09-02 CN disclosed
CN-109311822-B Histone demethylase inhibitors 赛尔基因昆蒂赛尔研究公司 2022-09-02 CN disclosed
CN-115003665-A Substituted aminoquinolones as immunoactive DGK alpha inhibitors 拜耳公司 2022-09-02 CN disclosed
US-20220274954-A1 SUBSTITUTED N-PHENYL-N-AMINOUARCILS AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2022-09-01 US disclosed
CN-114957242-A Preparation and application of pyrido-heterocyclic compound as kinase inhibitor 药雅科技(上海)有限公司 2022-08-30 CN disclosed
CN-114957241-A Preparation and application of heterocyclic compound as kinase inhibitor 药雅科技(上海)有限公司 2022-08-30 CN disclosed
CN-114957150-A Cyclic anhydride monomer and preparation method and application thereof 华东理工大学 2022-08-30 CN disclosed
US-11431029-B2 Silicon-based energy storage devices with functionalized linear sulfonate ester derivative compound containing electrolyte additives ENEVATE CORPORATION (US) 2022-08-30 US disclosed
CN-114949267-A Drug conjugates and uses thereof 米度(南京)生物技术有限公司 2022-08-30 CN disclosed
CN-108473483-B Compounds for medical use 奥斯维尔医疗私人有限公司 2022-08-30 CN disclosed
CN-114981255-A Method for preparing cyclic carbonate with exocyclic vinylidene 巴斯夫欧洲公司 2022-08-30 CN disclosed
CN-114981270-A MLL1 inhibitors and anticancer agents 诺华公司 2022-08-30 CN disclosed
US-11431027-B1 Single lithium-ion conductive polymer electrolytes for Si anode-based lithium-ion batteries ENEVATE CORPORATION (US) 2022-08-30 US disclosed
CN-109790112-B Cyanopyrrolidine derivatives having activity as USP30 inhibitors 特殊治疗有限公司 2022-08-26 CN disclosed
US-20220267303-A1 Compounds and Methods for Treating or Preventing Bacterial Infections BAYLOR COLLEGE OF MEDICINE 2022-08-25 US disclosed
EP-4045505-A1 2-METHYL-AZA-QUINAZOLINES Bayer Aktiengesellschaft (DE) 2022-08-24 EP disclosed
US-11420962-B2 Indene derivatives useful in treating pain and inflammation TARO PHARMACEUTICALS INC. (CA) 2022-08-23 US disclosed
US-11420970-B1 Piperidinyl-methyl-purineamines as NSD2 inhibitors and anti-cancer agents NOVARTIS AG (CH) 2022-08-23 US disclosed
CN-109790146-B Pharmaceutical compounds 阿尔麦克探索有限公司 2022-08-23 CN disclosed
CN-109563045-B Pd (II) -catalysed enantioselective beta-methylene C (sp) 3 ) -H bond activation 斯克里普斯研究学院 2022-08-23 CN disclosed
CN-114929705-A MLL1 inhibitor and anticancer agent 诺华公司 2022-08-19 CN disclosed
CN-114917361-A Antibody Drug Conjugates (ADC) and antibody prodrug conjugates (APDC) with enzyme cleavable groups 拜耳医药股份有限公司 2022-08-19 CN disclosed
WO-2022170971-A1 BIOACTIVE SUBSTANCE CONJUGATE, PREPARATION METHOD THEREFOR AND USE THEREOF 苏州宜联生物医药有限公司 2022-08-18 WO disclosed
CN-114907350-A Nitrogen-containing condensed ring compounds, preparation method and application 上海凌达生物医药有限公司 2022-08-16 CN disclosed
CN-114901253-A Improved lipid nanoparticles for delivery of nucleic acids 爱康泰生治疗公司 2022-08-12 CN disclosed
WO-2022167696-A1 FLAVONE DEAZA SPERMIDINE ANALOGUES AND THEIR USE TREATING CANCER Floratek Pharma SA (CH) 2022-08-11 WO disclosed
US-11407737-B2 Inhibitors of RAF kinases KINNATE BIOPHARMA INC. (US) 2022-08-09 US disclosed
CN-114853723-A Preparation and application of indole compound BTK inhibitor 药雅科技(上海)有限公司 2022-08-05 CN disclosed
CN-114853739-A Alkynyl pyrazine FGFR inhibitor and preparation method and application thereof 药雅科技(上海)有限公司 2022-08-05 CN disclosed
CN-114853752-A Preparation and application of BTK inhibitor pyridine heterocyclic compound 药雅科技(上海)有限公司 2022-08-05 CN disclosed
CN-114853740-A Preparation method and application of alkyne pyrimidine compound as FGFR inhibitor 药雅科技(上海)有限公司 2022-08-05 CN disclosed
WO-2022162025-A1 HETEROAROMATIC PHOSPHONIUM SALTS AND THEIR USE TREATING CANCER FLORATEK PHARMA AG (CH) 2022-08-04 WO disclosed
US-20220242823-A1 AGENTS FOR DIFFERENTIATING STEM CELLS AND TREATING CANCER MINERVA BIOTECHNOLOGIES CORPORATION 2022-08-04 US disclosed
EP-4034528-A1 PROCESS COMPRISING THE USE OF NEW IRIDIUM CATALYSTS FOR ENANTIOSELECTIVE HYDROGENATION OF 4-SUBSTITUTED 1,2-DIHYDROQUINOLINES Bayer Aktiengesellschaft (DE) 2022-08-03 EP disclosed
CN-107108527-B Ataxia telangiectasia and Rad 3-Associated (ATR) protein kinase inhibitors 阿特林制药有限责任公司 2022-08-02 CN disclosed
CN-114845711-A Inhibitors of RAF kinase 金耐特生物制药公司 2022-08-02 CN disclosed
CN-114845721-A Otic formulations for drug-induced ototoxicity 奥德纳米有限公司 2022-08-02 CN disclosed
CN-112384508-B Tricyclic ASK1 inhibitor and application thereof 山东轩竹医药科技有限公司 2022-08-02 CN disclosed
CN-114805359-A Preparation method and application of alkynyl heterocyclic compound FGFR inhibitor 药雅科技(上海)有限公司 2022-07-29 CN disclosed
CN-114805361-A Amino-substituted aromatic heterocyclic pyrazole compounds, preparation method and application 上海凌达生物医药有限公司 2022-07-29 CN disclosed
CN-114828836-A Lipid and lipid nanoparticle formulations for drug delivery 宾夕法尼亚大学理事会 2022-07-29 CN disclosed
CN-114829368-A Method for sequencing by synthesis using a sequential labelling scheme 豪夫迈·罗氏有限公司 2022-07-29 CN disclosed
CN-114828837-A Lipid nanoparticles for CAR mRNA delivery and formulations thereof 宾夕法尼亚大学理事会 2022-07-29 CN disclosed
US-20220233525-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2022-07-28 US disclosed
EP-3207128-B1 BUTYRYLCHOLINESTERASE ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC (US) 2022-07-27 EP disclosed
US-11398641-B2 Silicon-based energy storage devices with silicon containing electrolyte additives ENEVATE CORPORATION (US) 2022-07-26 US disclosed
CN-113004788-B Surface finishing composition 3M中国有限公司 2022-07-26 CN disclosed
CN-114786731-A Methods of treating ocular disorders 科达制药股份有限公司 2022-07-22 CN disclosed
US-20220226461-A1 Nucleoside-modified RNA for Inducing an Adaptive Immune Response THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2022-07-21 US disclosed
US-20220229065-A1 SENSORS AND METHODS FOR RAPID MICROBIAL DETECTION BAMBU VAULT LLC (US) 2022-07-21 US disclosed
US-20220226279-A1 ACYL SULFONAMIDES FOR TREATING CANCER THE BROAD INSTITUTE, INC. 2022-07-21 US disclosed
EP-4029510-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS Kodiak Sciences Inc. (US) 2022-07-20 EP disclosed
EP-3615513-B1 METHODS OF MANUFACTURING OF NIRAPARIB TESARO INC (US) 2022-07-20 EP disclosed
CN-108341774-B Substituted quinolinone inhibitors 首药控股(北京)股份有限公司 2022-07-19 CN disclosed
US-11390584-B2 1-cyano-pyrrolidine compounds as USP30 inhibitors MISSION THERAPEUTICS LIMITED (GB) 2022-07-19 US disclosed
US-11390618-B2 Inhibitors of cyclin-dependent kinases KINNATE BIOPHARMA INC. (US) 2022-07-19 US disclosed
US-11389444-B2 Methods of treating metabolic diseases with fused bicyclic pyrazoles BELITE BIO, INC (KY) 2022-07-19 US disclosed
US-11389445-B2 Pentafluorosulfanyl-substituted amide derivatives, preparation methods thereof and medical uses thereof BEIJING INNOCARE PHARMA TECH CO., LTD. (CN) 2022-07-19 US disclosed
CN-114751903-A Nitrogen-containing fused heterocyclic SHP2 inhibitor compound, preparation method and application 上海凌达生物医药有限公司 2022-07-15 CN disclosed
US-20220218816-A1 NUCLEIC ACID VACCINES FOR CORONAVIRUS Suzhou Abogen Biosciences Co., Ltd. (CN) 2022-07-14 US disclosed
EP-4025565-A1 NLRP3 INHIBITORS Inflazome Limited (IE) 2022-07-13 EP disclosed
EP-4025564-A1 NITRIFICATION INHIBITORS The University of Melbourne (AU) 2022-07-13 EP disclosed
EP-4026832-A1 PIPERIDINE DERIVATIVES AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 7 Almac Discovery Limited (GB) 2022-07-13 EP disclosed
EP-3612546-B1 MODIFIED OLIGOMERIC COMPOUNDS COMPRISING TRICYCLO-DNA NUCLEOSIDES AND USES THEREOF SYNTHENA AG (CH) 2022-07-13 EP disclosed
CN-109535155-B Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases 艾伯维公司 2022-07-12 CN disclosed
CN-111087612-B Phosphorus-containing flame-retardant nylon and preparation method and application thereof 今创景新材料科技(上海)有限公司 2022-07-12 CN disclosed
US-11384049-B2 2022-07-12 US disclosed
US-11384085-B2 Modulators of ion channel receptors and uses thereof BIONOMICS LIMITED (AU) 2022-07-12 US disclosed
US-11385221-B2 Alzheimer's disease assay in a living patient PAIN THERAPEUTICS, INC. (US) 2022-07-12 US disclosed
CN-111087796-B Phosphorus-containing copolymerized nylon and preparation method and application thereof 今创景新材料科技(上海)有限公司 2022-07-12 CN disclosed
CN-114728910-A Pyrazole derivatives for FGFR inhibitor and preparation method thereof 上海奕拓医药科技有限责任公司 2022-07-08 CN disclosed
CN-114728915-A [ (1, 5-diphenyl-1H-1, 2, 4-triazol-3-yl) oxy ] acetic acid derivatives and salts thereof, crop protection compositions comprising the same, method for the production thereof and use thereof as safeners 拜耳公司 2022-07-08 CN disclosed
CN-109415623-B Photosensitive macromolecules and uses thereof 拜克门寇尔特公司 2022-07-08 CN disclosed
CN-114728888-A Aromatic substituted ethane-core monomers and polymers thereof for volume bragg gratings 脸谱科技有限责任公司 2022-07-08 CN disclosed
CN-114728889-A Aromatic substituted alkane-nuclear monomers and polymers thereof for volume bragg gratings 脸谱科技有限责任公司 2022-07-08 CN disclosed
CN-110723748-B Metal oxides, metal bronzes and polyoxometallates as charge storage materials in electrochromic devices 菲尔齐费尔公司 2022-07-08 CN disclosed
CN-114728941-A Substituted 1, 5-naphthyridines or quinolines as ALK5 inhibitors 施万生物制药研发IP有限责任公司 2022-07-08 CN disclosed
CN-114728076-A MCL-1 inhibitor antibody-drug conjugates and methods of use 诺华股份有限公司 2022-07-08 CN disclosed
CN-114728077-A MCL-1 inhibitor antibody-drug conjugates and methods of use 诺华股份有限公司 2022-07-08 CN disclosed
CN-114728992-A Method for producing phosphate compound 斯泰拉化工公司 2022-07-08 CN disclosed
CN-114728993-A Thiophosphate and phosphine sulfide derivative monomer and polymer for volume Bragg grating 脸谱科技有限责任公司 2022-07-08 CN disclosed
CN-114728893-A Aromatic substituted methane-core monomers and polymers thereof for volume bragg gratings 脸谱科技有限责任公司 2022-07-08 CN disclosed
CN-114728894-A Anthraquinone derivative monomer and polymer for volume Bragg grating 脸谱科技有限责任公司 2022-07-08 CN disclosed
CN-114729044-A Muscarinic acetylcholine M1Receptor antagonists 帕珀莱恩医疗公司 2022-07-08 CN disclosed
CN-108026142-B Ligands for orphan nuclear receptor Nur77 and uses thereof 艾凯奇(厦门)生物科技有限公司 2022-07-08 CN disclosed
CN-114727975-A Antiandrogen receptor/AKR 1C3 inhibitors 加利福尼亚大学董事会 2022-07-08 CN disclosed
US-20220213260-A1 PHOTOACTIVE MACROMOLECULES AND USES THEREOF BECKMAN COULTER, INC. 2022-07-07 US disclosed
US-20220211664-A1 LYMPH DIRECTING PRODRUGS MONASH UNIVERSITY (AU) 2022-07-07 US disclosed
WO-2022147189-A1 VARENICLINE PRODRUGS ANTARES PHARMA, INC. (US) 2022-07-07 WO disclosed
WO-2022147180-A1 HIGH REFRACTIVE INDEX OVERCOAT FORMULATION AND METHOD OF USE WITH INKJET PRINTING META PLATFORMS TECHNOLOGIES, LLC (US) 2022-07-07 WO disclosed
EP-3608325-B1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES INC (US) 2022-07-06 EP disclosed
EP-4023639-A1 PYRAZOLE DERIVATIVE FOR FGFR INHIBITOR AND PREPARATION METHOD THEREFOR Etern Biopharma (Shanghai) Co., Ltd. (CN) 2022-07-06 EP disclosed
EP-3527573-B9 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES INC (US) 2022-07-06 EP disclosed
EP-3710449-B1 MACROCYCLIC FLUORINE SUBSTITUTED INDOLE DERIVATIVES AS MCL-1 INHIBITORS, FOR USE IN THE TREATMENT OF CANCER BROAD INST INC (US) 2022-07-06 EP disclosed
EP-3280262-B1 SYNERGISTIC BENZOXABOROLE-CONTAINING ANTI-FUNGICIDAL COMPOSITION PENN STATE RES FOUND (US) 2022-07-06 EP disclosed
CN-114703144-A 6-6 fused bicyclic heteroaryl compounds and their use as LATS inhibitors 诺华股份有限公司 2022-07-05 CN disclosed
US-11377441-B2 Covalent inhibitors of KRAS ARAXES PHARMA LLC (US) 2022-07-05 US disclosed
US-11377431-B2 Inhibitors of RAF kinases KINNATE BIOPHARMA INC. (US) 2022-07-05 US disclosed
CN-114685487-A Pyrimidine heterocyclic compound, preparation method and application 上海凌达生物医药有限公司 2022-07-01 CN disclosed
CN-114685502-A Spirocyclic compounds as KRAS-G12C inhibitors 由理生物医药(上海)有限公司 2022-07-01 CN disclosed
WO-2022133544-A1 CBD CANNABINOIDS AND CBD CANNABINOID ANALOGUES Botanix Pharmaceuticals Limited (AU) 2022-06-30 WO disclosed
WO-2022140643-A1 SMALL-MOLECULE MODULATORS OF THE ORPHAN NUCLEAR RECEPTOR TLX BAYLOR COLLEGE OF MEDICINE (US) 2022-06-30 WO disclosed
US-20220204790-A1 HIGH REFRACTIVE INDEX OVERCOAT FORMULATION AND METHOD OF USE WITH INKJET PRINTING META PLATFORMS TECHNOLOGIES, LLC 2022-06-30 US disclosed
US-20220209227-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH FLUORINATED CYCLIC COMPOUND CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORP (US) 2022-06-30 US disclosed
US-20220205165-A1 CHEMICALLY LINKED SILK FIBROIN COATINGS AND METHODS OF MAKING AND USING THEREOF EVOLVED BY NATURE, INC. (US) 2022-06-30 US disclosed
US-20220204486-A1 THIENYL-ANILINE COMPOUNDS FOR TREATMENT OF DERMAL DISORDERS NFLECTION THERAPEUTICS, INC. 2022-06-30 US disclosed
EP-4019516-A1 ASYMMETRIC PHASE TRANSFER CATALYSIS Merck Sharp & Dohme Corp. (US) 2022-06-29 EP disclosed
EP-4017843-A1 BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF 2692372 Ontario, Inc. (CA) 2022-06-29 EP disclosed
EP-3265453-B1 NEW PYRIDINONES AND ISOQUINOLINONES AS INHIBITORS OF THE BROMODOMAIN BRD9 BOEHRINGER INGELHEIM INT (DE) 2022-06-29 EP disclosed
EP-3517535-B1 ALKYNYL-SUBSTITUTED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF BEIJING INNOCARE PHARMA TECH CO LTD (CN) 2022-06-29 EP disclosed
US-11370775-B2 Substituted benzimidazole derivatives as D-amino acid oxidase (DAAO) inhibitors Tseng, Yufeng Jane (US) 2022-06-28 US disclosed
US-11371994-B2 Phosphorylated Akt-specific capture agents, compositions, and methods of using and making CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-06-28 US disclosed
US-11370784-B2 Cyano-substituted heterocycles with activity as inhibitors of USP30 MISSION THERAPEUTICS LIMITED (GB) 2022-06-28 US disclosed
US-11370776-B2 Sulfonylureas and sulfonylthioureas as NLRP3 inhibitors INFLAZOME LIMITED (IE) 2022-06-28 US disclosed
CN-109476680-B Organic magnesium phosphide, process for producing the same, complex thereof, process for producing the same, and process for producing organic phosphorus compound using the same 北兴化学工业株式会社 2022-06-28 CN disclosed
CN-111763217-B Thieno-nitrogen heterocyclic compounds, preparation method and application 上海凌达生物医药有限公司 2022-06-28 CN disclosed
CN-114656791-A Polymer-silica hybrid PDOT and methods of use thereof 华盛顿大学 2022-06-24 CN disclosed
CN-108290927-B IL-17F-specific capture agents, compositions, and methods of use and manufacture 加州理工学院 2022-06-24 CN disclosed
US-20220194945-A1 Imidazolopyridine Compounds For IRE1 Inhibition Optikira, LLC 2022-06-23 US disclosed
WO-2022133314-A1 MODIFIED INDOLE ALKALOIDS FOR THERAPEUTIC USES NEW ATLAS BIOTECHNOLOGIES, INC. (US) 2022-06-23 WO disclosed
WO-2022133280-A1 COMPOSITION FOR REVERSIBLE POLYMERIZATION OF THIOESTER AND METHODS THEREOF THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2022-06-23 WO disclosed
WO-2022133345-A1 TRICYCLIC PYRIDONES AND PYRIMIDONES ERASCA, INC. (US) 2022-06-23 WO disclosed
US-20220192984-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING OTIC THERAPEUTIC AGENTS AND RELATED METHODS Frequency Therapeutics, Inc. 2022-06-23 US disclosed
WO-2022133064-A1 FUSED PYRIMIDINE COMPOUNDS AS INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, INC. (US) 2022-06-23 WO disclosed
US-20220194923-A1 NOVEL SULFONAMIDEUREA COMPOUNDS INFLAZOME LIMITED (IE) 2022-06-23 US disclosed
EP-4013755-A1 PIPERIDINYL-METHYL-PURINEAMINES AS NSD2 INHIBITORS AND ANTI-CANCER AGENTS Novartis AG (CH) 2022-06-22 EP disclosed
EP-4013762-A1 MACROCYCLIC SULFONYLAMIDE DERIVATIVES USEFUL AS NLRP3 INHIBITORS Inflazome Limited (IE) 2022-06-22 EP disclosed
EP-4013756-A1 MLL1 INHIBITORS AND ANTI-CANCER AGENTS Novartis AG (CH) 2022-06-22 EP disclosed
EP-4013761-A1 MACROCYCLIC SULFONYLUREA DERIVATIVES USEFUL AS NLRP3 INHIBITORS Inflazome Limited (IE) 2022-06-22 EP disclosed
EP-4013500-A1 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS Novartis AG (CH) 2022-06-22 EP disclosed
EP-3652235-B1 ELECTROCHROMIC POLYMER AND SYNTHESIS AND USES THEREOF FURCIFER INC (US) 2022-06-22 EP disclosed
CN-109071446-B Organic reaction in aqueous solution in the presence of hydroxyalkyl (alkyl) cellulose or alkylcellulose 艾伯维德国有限责任两合公司 2022-06-21 CN disclosed
US-11365220-B2 Methods of making anti-GP41 antibody-specific capture agents CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-06-21 US disclosed
US-11365219-B2 Cyclic peptides as protein targeting agents CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-06-21 US disclosed
CN-110229157-B Pyrimido five-membered heteroaromatic compound, preparation method and application thereof 上海海和药物研究开发股份有限公司 2022-06-21 CN disclosed
CN-110437230-B Tertiary amine compound, diphosphine ligand, intermediate and preparation method thereof 中国科学院上海有机化学研究所 2022-06-21 CN disclosed
CN-109843873-B Alkyne heterocyclic compound, preparation method and application thereof in medicine and pharmacology 北京诺诚健华医药科技有限公司 2022-06-17 CN disclosed
US-20220185808-A1 ACYLAMINOPYRROLO-PYRIDONE COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI RINGENE BIOPHARMA CO., LTD. (CN) 2022-06-16 US disclosed
US-20220185846-A1 METHODS FOR SYNTHESIZING BETA-HOMOAMINO ACIDS PROTAGONIST THERAPEUTICS, INC. 2022-06-16 US disclosed
US-20220183998-A1 USE OF 8,9- DIHYDROCANNABIDIOL COMPOUNDS UNIV CALIFORNIA (US) 2022-06-16 US disclosed
EP-3837301-B1 POLYMER COMPOSITION BASF SE (DE) 2022-06-15 EP disclosed
EP-4011876-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2022-06-15 EP disclosed
CN-114621222-A 6-6 fused bicyclic heteroaryl compounds and their use as LATS inhibitors 诺华股份有限公司 2022-06-14 CN disclosed
US-11357856-B2 Lipids for delivery of active agents Acuitas Therapeutics, Inc. (CA) 2022-06-14 US disclosed
US-11357770-B2 Method of treating immunoglobulin light chain amyloidosis Alterity Therapeutics Limited (AU) 2022-06-14 US disclosed
US-11358959-B2 Benzothiophene and benzothiazole compounds and methods of use thereof ARAXES PHARMA LLC (US) 2022-06-14 US disclosed
US-11358958-B2 2022-06-14 US disclosed
CN-110177822-B Synthesis of polycarbonate siloxane diol 奥特克国际公开有限公司 2022-06-14 CN disclosed
US-11357781-B2 Non-catalytic substrate-selective, p38α-specific MAPK inhibitors with endothelial-stabilizing and anti-inflammatory activity, and methods of use thereof UNIVERSITY OF MARYLAND, BALTIMORE (US) 2022-06-14 US disclosed
CN-114616227-A Nitrification inhibitors 墨尔本大学 2022-06-10 CN disclosed
US-20220177451-A1 1-CYANO-PYRROLIDINE DERIVATIVES AS DUB INHIBITORS MISSION THERAPEUTICS LIMITED (GB) 2022-06-09 US disclosed
US-20220177659-A1 NON-CORE SHELL POLYMER PARTICLES THE UNIVERSITY OF SYDNEY (AU) 2022-06-09 US disclosed
WO-2022120207-A1 BROAD SPECTRUM ANTIVIRAL COMPOUNDS TARGETING THE SKI COMPLEX UNIVERSITY OF MARYLAND, BALTIMORE (US) 2022-06-09 WO disclosed
EP-4007578-A1 SUBSTITUTED CYCLOPROPYL-2,2'-BIPYRIMIDINYL COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME Arbutus Biopharma, Inc. (US) 2022-06-08 EP disclosed
US-11352554-B2 Photochromic water harvesting platform WARNER BABCOCK INSTITUTE FOR GREEN CHEMISTRY, LLC (US) 2022-06-07 US disclosed
US-11352339-B2 1-cyano-pyrrolidine derivatives as DUB inhibitors MISSION THERAPEUTICS LIMITED (GB) 2022-06-07 US disclosed
US-11352512-B2 Surface primer compositions and methods of use ENVISTA (US) 2022-06-07 US disclosed
US-11352367-B2 Indene derivatives useful in treating pain and inflammation TARO PHARMACEUTICALS INC. (CA) 2022-06-07 US disclosed
CN-109790148-B Cyano-substituted heterocycles having USP30 inhibitor activity 特殊治疗有限公司 2022-06-07 CN disclosed
CN-114591334-A Dihydropyrazolopyrimidinone derivatives 山东轩竹医药科技有限公司 2022-06-07 CN disclosed
CN-114599408-A Devices and methods for modulating ADMA in blood 印地安纳大学理事会 2022-06-07 CN disclosed
CN-114569552-A Anti-malarial compositions and uses thereof 斯克利普斯研究院 2022-06-03 CN disclosed
CN-114573566-A Selective ROCK2 kinase inhibitors 杭州邦顺制药有限公司 2022-06-03 CN disclosed
CN-110156786-B Pyrimido-cyclic compounds, process for their preparation and their use 青煜医药研发(上海)有限公司 2022-06-03 CN disclosed
CN-114585622-A Piperidinyl-methyl-purinamines as NSD2 inhibitors and anticancer agents 诺华股份有限公司 2022-06-03 CN disclosed
WO-2022112430-A1 REDUCTION OF VIRAL INFECTIONS PHOXBIO LIMITED (IE) 2022-06-02 WO disclosed
US-20220169618-A1 SUBSTITUTED 2-HETEROARYLAMINOBENZENES AND THE SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2022-06-02 US disclosed
WO-2022115451-A1 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE NOVARTIS AG (CH) 2022-06-02 WO disclosed
WO-2022115477-A1 BCL-XL INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE THEREOF NOVARTIS AG (CH) 2022-06-02 WO disclosed
WO-2022112537-A1 PHOTODYNAMIC THERAPY AND DIAGNOSIS RMW CHO GROUP LIMITED (CN) 2022-06-02 WO disclosed
US-20220169627-A1 IRREVERSIBLE INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, LLC 2022-06-02 US disclosed
US-20220170053-A1 HIGH GRAVITY, FED-BATCH IONIC LIQUID BASED PROCESS FOR DECONSTRUCTING BIOMASS UNITED STATES DEPARTMENT OF ENERGY 2022-06-02 US disclosed
EP-4003981-A1 SUBSTITUTED N-PHENYL URACILS, SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS Bayer Aktiengesellschaft (DE) 2022-06-01 EP disclosed
EP-4006030-A2 METHODS AND COMPOSITIONS FOR INHIBITING THE INTERACTION OF MENIN WITH MLL PROTEINS Kura Oncology, Inc. (US) 2022-06-01 EP disclosed
EP-4003345-A1 DUAL ATM AND DNA-PK INHIBITORS FOR USE IN ANTI-TUMOR THERAPY XRad Therapeutics, Inc. (US) 2022-06-01 EP disclosed
EP-4003975-A1 SUBSTITUTED N-PHENYL-N-AMINOUARCILS AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL AGENTS Bayer Aktiengesellschaft (DE) 2022-06-01 EP disclosed
EP-4003959-A1 TARGETED RADIOPHARMACEUTICALS FOR THE DIAGNOSIS AND TREATMENT OF PROSTATE CANCER Bayer AS (NO) 2022-06-01 EP disclosed
CN-112204025-B Compounds for the treatment of pain, compositions comprising the same and methods of using the same 瑟赛治疗公司 2022-05-31 CN disclosed
US-11349153-B2 Silicon-based energy storage devices with ether containing electrolyte additives ENEVATE CORPORATION (US) 2022-05-31 US disclosed
CN-114560893-A Planar chiral metallocene compound, and synthesis method and application thereof 中国科学院上海有机化学研究所 2022-05-31 CN disclosed
US-11345720-B2 Efficient and scalable syntheses of nicotinoyl ribosides and reduced nicotinoyl ribosides, modified derivatives thereof, phosphorylated analogs thereof, adenylyl dinucleotide conjugates thereof, and novel crystalline forms thereof THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2022-05-31 US disclosed
US-11344559-B2 PI3KGAMMA inhibitors THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-05-31 US disclosed
US-11345681-B1 Inhibitors of fibroblast growth factor receptor kinases KINNATE BIOPHARMA INC. (US) 2022-05-31 US disclosed
CN-114555609-A Macrocyclic sulfonamide derivatives useful as NLRP3 inhibitors 英夫拉索姆有限公司 2022-05-27 CN disclosed
CN-110325531-B Benzenesulfonamides and their use as therapeutic agents 泽农医药公司 2022-05-27 CN disclosed
WO-2022106902-A2 BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF 2692372 ONTARIO, INC. (CA) 2022-05-27 WO disclosed
WO-2022106897-A2 METHODS AND COMPOSITION FOR KRAS MODIFICATIONS 2692372 ONTARIO, INC. (CA) 2022-05-27 WO disclosed
US-20220160696-A1 USES OF PHOSPHODIESTERASE INHIBITORS TRANSTHERA SCIENCES (NANJING), INC. (CN) 2022-05-26 US disclosed
US-20220162193-A1 PYRAZOLESULFONAMIDES AS ANTITUMOR AGENTS PELOTON THERAPEUTICS, INC. (US) 2022-05-26 US disclosed
US-20220160724-A1 SELECTIVE P2X3 MODULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.3) LIMITED (GB) 2022-05-26 US disclosed
EP-3999061-A1 HETEROCYCLIC COMPOUNDS AS MODULATORS OF BETA-CATENIN / TCF4 INTERACTION Agency for Science, Technology and Research (SG) 2022-05-25 EP disclosed
EP-3999498-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASES Kinnate Biopharma Inc. (US) 2022-05-25 EP disclosed
EP-3423454-B1 SPIRO-CONDENSED PYRROLIDINE DERIVATIVES AS DEUBIQUITYLATING ENZYMES (DUB) INHIBITORS MISSION THERAPEUTICS LTD (GB) 2022-05-25 EP disclosed
EP-4000610-A1 PHARMACOLOGY OF VISUAL CYCLE MODULATORS Acucela Inc. (US) 2022-05-25 EP disclosed
US-11342588-B2 Silicon-based energy storage devices with electrolyte containing dihydrofuranone based compound ENEVATE CORPORATION (US) 2022-05-24 US disclosed
CN-114524810-A Pyrimidine heterocyclic compound, preparation method and application 上海凌达生物医药有限公司 2022-05-24 CN disclosed
CN-114516883-A Thienopyrimidine compound, and pharmaceutical composition and application thereof 苏州优理生物医药科技有限公司 2022-05-20 CN disclosed
CN-114516873-A Spiro compound, pharmaceutical composition containing same and application thereof 苏州优理生物医药科技有限公司 2022-05-20 CN disclosed
US-20220153895-A1 SUBSTITUTED PROPANE-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2022-05-19 US disclosed
US-20220153686-A1 LIPID NANOPARTICLE COMPOSITION Suzhou Abogen Biosciences Co., Ltd. (CN) 2022-05-19 US disclosed
WO-2022104113-A1 SUBSTITUTED MONO- AND POLY-PHENYL-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS FACEBOOK TECHNOLOGIES, LLC (US) 2022-05-19 WO disclosed
WO-2022104137-A1 SUBSTITUTED PROPANE-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS FACEBOOK TECHNOLOGIES, LLC (US) 2022-05-19 WO disclosed
WO-2022104070-A2 PHENOTHIAZINE COMPOUNDS FOR THE TREATMENT OF ALZHEIMER'S DISEASE AND OTHER AGE-RELATED AND NEUROLOGICAL DISEASES ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2022-05-19 WO disclosed
WO-2022104147-A1 ADDITIVES FOR REDUCING NON-SPECIFIC INTERACTIONS BETWEEN FLUORESCENT POLYMER CONJUGATES AND CELLS IN A BIOLOGICAL SAMPLE BECKMAN COULTER, INC. (US) 2022-05-19 WO disclosed
US-20220153731-A1 Compounds for Pain Treatment, Compositions Comprising Same, and Methods of Using Same ACADIA PHARM INC (US) 2022-05-19 US disclosed
US-20220153734-A1 Pyrazolopyridine Compounds For IRE1 Inhibition Optikira, LLC 2022-05-19 US disclosed
US-20220153693-A1 SUBSTITUTED MONO- AND POLY-PHENYL-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2022-05-19 US disclosed
US-20220153706-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2022-05-19 US disclosed
EP-3996714-A1 FORMULATIONS OF RBP4 INHIBITORS AND METHODS OF USE Belite Bio, LLC (US) 2022-05-18 EP disclosed
CN-114514322-A Method for producing oligoenergetic and monoenergetic precursors 投资健康有限责任公司 2022-05-17 CN disclosed
CN-114507190-A Deuterated 1, 4-benzodiazepine-2, 5-diketone compound and application thereof 宁波康柏睿格医药科技有限公司 2022-05-17 CN disclosed
US-11332453-B2 MAGL inhibitors H. LUNDBECK A/S (DK) 2022-05-17 US disclosed
US-11332476-B2 Fms-like tyrosine kinase inhibitors 3SM BIOTRON INC. (TW) 2022-05-17 US disclosed
CN-114514223-A Process comprising enantioselective hydrogenation of 4-substituted 1, 2-dihydroquinolines using a novel iridium catalyst 拜耳公司 2022-05-17 CN disclosed
US-11332485-B2 Penicillin-binding protein inhibitors VenatoRx Pharmaceuticals, Inc. (US) 2022-05-17 US disclosed
CN-114478568-A Thienopyrimidine compound, pharmaceutical composition containing thienopyrimidine compound and application of thienopyrimidine compound 苏州优理生物医药科技有限公司 2022-05-13 CN disclosed
CN-114478409-A Histone demethylase inhibitors 赛尔基因昆蒂赛尔研究公司 2022-05-13 CN disclosed
CN-109721620-B HPK1 inhibitors and uses thereof 药捷安康(南京)科技股份有限公司 2022-05-13 CN disclosed
CN-114478585-A Nitrogen-containing fused heterocyclic compound and preparation method and application thereof 上海青煜医药科技有限公司 2022-05-13 CN disclosed
CN-111885914-B Compositions and methods for producing expanded hematopoietic stem cells using fluorene derivatives 投资健康有限责任公司 2022-05-13 CN disclosed
CN-114502533-A Benzenesulfonamide derivatives and use thereof 2692372安大略公司 2022-05-13 CN disclosed
WO-2022096446-A1 [(1-PHENYL-5-(HETEROARYL)-1H-1,2,4-TRIAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2022-05-12 WO disclosed
US-20220144819-A1 NAPHTHYRIDINONE-ANILINE COMPOUNDS FOR TREATMENT OF DERMAL DISORDERS NFLECTION THERAPEUTICS, INC. 2022-05-12 US disclosed
US-20220144815-A1 1,3,4-OXADIAZOLES AND THEIR DERIVATIVES AS NEW ANTIFUNGAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2022-05-12 US disclosed
US-20220144845-A1 SUBSTITUTED PYRROLO[1,2-a]QUINOXALIN-4(5H)-ONES AS CX3CR1 ANTAGONISTS UNIV DREXEL (US) 2022-05-12 US disclosed
US-20220142995-A1 DUAL ATM AND DNA-PK INHIBITORS FOR USE IN ANTI-TUMOR THERAPY XRAD HOLDING CAYMAN LIMITED (KY) 2022-05-12 US disclosed
US-20220145171-A1 QUANTUM DOTS AND PROCESSES FOR PREPARATION THEREOF THE UNIVERSITY OF QUEENSLAND (AU) 2022-05-12 US disclosed
WO-2022098892-A1 SELF-HEALABLE, RECYCLABLE, AND RECONFIGURABLE WEARABLE ELECTRONICS DEVICE THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2022-05-12 WO disclosed
WO-2022098700-A1 INHIBITING AN IMMUNE RESPONSE MEDIATED BY ONE OR MORE OF TLR2, RAGE, CCR5, CXCR4 AND CD4 CASSAVA SCIENCES, INC. (US) 2022-05-12 WO disclosed
WO-2022096448-A1 [(5-PHENYL-5-HETEROARYL-1H-PYRAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2022-05-12 WO disclosed
WO-2022096442-A1 [(5-PHENYL-1-HETEROARYL-1H-TRIAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2022-05-12 WO disclosed
WO-2022096445-A1 [(1-PHENYL-5-HETEROARYL-1H-PYRAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2022-05-12 WO disclosed
WO-2022096449-A1 [(1,5-DIHETEROARYL-1H-1,2,4-TRIAZOL-3-YL)OXY] ACETIC ACID DERIVATIVES AS SAFENERS FOR THE PROTECTION OF USEFUL PLANTS AND CROP PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2022-05-12 WO disclosed
EP-3661917-B1 6-((3-TRIFLUOROMETHYL)PHENYL)-4,5-DIHYDROPYRIDAZIN-3(2H)-ONE DERIVATIVES AS PDE3A AND PDE3B INHIBITORS FOR TREATING CANCER BAYER AG (DE) 2022-05-11 EP disclosed
EP-3994262-A1 ENHANCEMENT OF NUCLEIC ACID POLYMERIZATION BY AROMATIC COMPOUNDS Stratos Genomics Inc. (US) 2022-05-11 EP disclosed
EP-3995611-A1 HIGH THROUGHPUT METHOD FOR CONSTRUCTING AND SCREENING COMPOUND LIBRARY AND REACTION DEVICE Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CN) 2022-05-11 EP disclosed
EP-3102207-B1 2,4,5-TRI-SUBSTITUTED AZOLE-BASED CASEIN KINASE 1 INHIBITORS AS INDUCERS FOR CARDIOMYOGENESIS AGENCY SCIENCE TECH & RES (SG) 2022-05-11 EP disclosed
EP-3179992-B1 THERAPEUTIC COMBINATIONS OF A BTK INHIBITOR, A PD-1 INHIBITOR AND/OR A PD-L1 INHIBITOR ACERTA PHARMA BV (NL) 2022-05-11 EP disclosed
US-11325902-B2 Benzenesulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2022-05-10 US disclosed
US-11324729-B2 NSD family inhibitors and methods of treatment therewith THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2022-05-10 US disclosed
US-11325111-B2 Catalysts and methods of making the same EXXONMOBIL RESEARCH & ENGINEERING COMPANY (US) 2022-05-10 US disclosed
CN-109384790-B Fibroblast growth factor receptor inhibitors and uses thereof 药捷安康(南京)科技股份有限公司 2022-05-10 CN disclosed
CN-108101826-B Indole-substituted alkylamine compound and application thereof 华东理工大学 2022-05-10 CN disclosed
CN-114437039-A CD73 inhibitor and application thereof 武汉人福创新药物研发中心有限公司 2022-05-06 CN disclosed
WO-2022094400-A1 BICYCLIC COMPOUNDS AND USES THEREOF FOR THE TREATMENT OF DISEASES ATHIRA PHARMA, INC. (US) 2022-05-05 WO disclosed
US-20220135612-A1 MODIFIED NUCLEOSIDE AND SYNTHETIC METHODS THEREOF Stemirna Therapeutics Co., Ltd. (CN) 2022-05-05 US disclosed
US-20220140392-A1 FUNCTIONAL EPOXIDES IN CATALYST-BASED ELECTROLYTE COMPOSITIONS FOR LI-ION BATTERIES ENEVATE CORPORATION 2022-05-05 US disclosed
US-20220133734-A1 SUBSTITUTED 1H-PYRAZOLO[4,3-C]PYRIDINES AND DERIVATIVES AS EGFR INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-05-05 US disclosed
US-20220135563-A1 MAGL INHIBITORS H. LUNDBECK A/S (DK) 2022-05-05 US disclosed
WO-2022090481-A1 SUBSTITUTED 1H-PYRAZOLO[4,3-C]PYRIDINES AND DERIVATIVES AS EGFR INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-05-05 WO disclosed
EP-3433246-B1 1-CYANO-PYRROLIDINE DERIVATIVES AS DBU INHIBITORS MISSION THERAPEUTICS LTD (GB) 2022-05-04 EP disclosed
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-05-03 US disclosed
US-11318129-B2 Compounds and methods for inhibiting NHE-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders ARDELYX, INC. (US) 2022-05-03 US disclosed
US-11319287-B2 Cyanopyrrolidines as dub inhibitors for the treatment of cancer MISSION THERAPEUTICS LIMITED (GB) 2022-05-03 US disclosed
US-11319324-B2 Pyrazolo-pyrrolo-pyrimidine-dione derivatives as P2X3 inhibitors BAYER AKTIENGESELLSCHAFT (DE) 2022-05-03 US disclosed
US-11319302-B2 PRC1 inhibitors and methods of treatment therewith THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2022-05-03 US disclosed
US-11319344-B2 Non-membrane disruptive P53 activating stapled peptides AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2022-05-03 US disclosed
US-11319290-B2 Substituted 3-dialkylaminomethyl-piperidin-4-yl-benzamides and methods of making and using same MEBIAS DISCOVERY, INC. (US) 2022-05-03 US disclosed
CN-114423463-A Heterobifunctional compounds as HPK1 degradants 西奈山伊坎医学院 2022-04-29 CN disclosed
CN-114423739-A Improved enantioselective hydrogenation of 4-substituted 1, 2-dihydroquinolines in the presence of chiral iridium catalysts and additives 拜耳公司 2022-04-29 CN disclosed
CN-114404588-A Compounds and methods for inhibiting phosphate transport 阿德利克斯公司 2022-04-29 CN disclosed
US-20220127613-A1 Functionally-Modified Oligonucleotides And Subunits Thereof SAREPTA THERAPEUTICS INC (US) 2022-04-28 US disclosed
US-20220125771-A1 SUBSTITUTED POLYCYCLIC CARBOXYLIC ACIDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2022-04-28 US disclosed
US-20220131148-A1 BORON-CONTAINING CHEMICALS AS CATHODE ADDITIVES, SI ANODE ADDITIVES, ELECTROLYTE ADDITIVES OR SEPARATOR MODIFIERS FOR LI-ION BATTERIES ENEVATE CORPORATION 2022-04-28 US disclosed
US-20220126270-A1 CAPTURE OF FLUORINATED CARBON COMPOUNDS THE UNIVERSITY OF QUEENSLAND (AU) 2022-04-28 US disclosed
US-20220131195-A1 ELECTROLYTE ADDITIVES CONTAINING ONE, TWO, OR MORE TRIPLE-BONDED MOIETIES FOR SILICON ANODE-BASED LI-ION BATTERIES ENEVATE CORPORATION 2022-04-28 US disclosed
US-20220131194-A1 METAL AMIDE BASES AS ELECTROLYTE ADDITIVES FOR SI ANODE-BASED LI-ION BATTERIES ENEVATE CORPORATION 2022-04-28 US disclosed
US-20220127271-A1 NITROGEN-CONTAINING FUSED HETEROCYCLIC SHP2 INHIBITOR COMPOUND, PREPARATION METHOD, AND USE SHANGHAI RINGENE BIOPHARMA CO., LTD. (CN) 2022-04-28 US disclosed
US-20220131193-A1 SYMMETRICAL OR ASYMMETRICAL ALKYLSULFONYL IMIDE OR CYCLIC ALKYLENE SULFONYLIMIDE SALTS AS CATHODE ADDITIVES, ELECTROLYTE ADDITIVES, OR SI ANODE ADDITIVES FOR SI ANODE-BASED LI-ION CELLS ENEVATE CORPORATION 2022-04-28 US disclosed
WO-2022087008-A1 TERTIARY CARBOXAMIDE COMPOUNDS VIVACE THERAPEUTICS, INC. (US) 2022-04-28 WO disclosed
WO-2022087456-A1 NEW COMPOUNDS FOR THE TREATMENT OF ALZHEIMER'S DISEASE ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2022-04-28 WO disclosed
WO-2022086937-A1 HETEROBIFUNCTIONAL COMPOUNDS AS DEGRADERS OF ENL ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2022-04-28 WO disclosed
EP-3986408-A1 ANTICANCER COMBINATION THERAPY Boehringer Ingelheim International GmbH (DE) 2022-04-27 EP disclosed
EP-3986874-A1 BENZYLPHENYL HYDROXYISOXAZOLINES AND ANALOGUES AS NEW ANTIFUNGAL AGENTS Bayer Aktiengesellschaft (DE) 2022-04-27 EP disclosed
EP-3986875-A1 PHENOXYPHENYL HYDROXYISOXAZOLINES AND ANALOGUES AS NEW ANTIFUNGAL AGENTS Bayer Aktiengesellschaft (DE) 2022-04-27 EP disclosed
EP-3986564-A1 NEW MACROCYCLIC COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS Boehringer Ingelheim International GmbH (DE) 2022-04-27 EP disclosed
EP-3988120-A1 NHE3-BINDING COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT Ardelyx, Inc. (US) 2022-04-27 EP disclosed
EP-3988631-A1 POLYMER-SILICA HYBRID PDOTS University of Washington (US) 2022-04-27 EP disclosed
EP-3458459-B1 MACROCYCLIC INDOLE DERIVATIVES BAYER AG (DE) 2022-04-27 EP disclosed
EP-3986918-A1 ADRENOMEDULLIN-ANALOGUES FOR LONG-TERM STABILIZATION AND THEIR USE Bayer Aktiengesellschaft (DE) 2022-04-27 EP disclosed
US-11311512-B2 Lymph directing prodrugs MONASH UNIVERSITY (AU) 2022-04-26 US disclosed
US-11311520-B2 Substituted dihydroimidazopyridinediones as MKNK1 and MKNK2 inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2022-04-26 US disclosed
US-11312718-B2 Formulations of (S)-3-(1-(9H-purin-6-ylamino)ethyl)-8-chloro-2-phenylisoquinolin-1(2H)-one INFINITY PHARMACEUTICALS, INC. (US) 2022-04-26 US disclosed
US-11312668-B2 Organic reactions carried out in aqueous solution in the presence of a hydroxyalkyl(alkyl)cellulose or an alkylcellulose ABBVIE INC. (US) 2022-04-26 US disclosed
CN-109803963-B Cyano-substituted heterocycles having USP30 inhibitor activity 特殊治疗有限公司 2022-04-26 CN disclosed
CN-114395065-A Spray-dried olefin polymerization catalyst composition and polymerization process using the same 埃克森美孚化学专利公司 2022-04-26 CN disclosed
CN-114401956-A Substituted N-phenyluracils, their salts and their use as herbicides 拜耳公司 2022-04-26 CN disclosed
CN-114401971-A Macrocyclic sulfonylurea derivatives as NLRP3 inhibitors 英夫拉索姆有限公司 2022-04-26 CN disclosed
CN-109689652-B Fused heterocyclic derivative, preparation method and medical application thereof 北京诺诚健华医药科技有限公司 2022-04-26 CN disclosed
CN-109313954-B Polymer-silica hybrid PDOT and methods of use thereof 华盛顿大学 2022-04-26 CN disclosed
CN-114401955-A Inhibitors of cyclin dependent kinases 金耐特生物制药公司 2022-04-26 CN disclosed
CN-114394983-A Synthesis of polycyclic carbamoylpyridone compounds 吉利德科学公司 2022-04-26 CN disclosed
CN-108473502-B 4, 6-dihydropyrrolo [3,4-C ] pyrazole-5 (1H) -carbonitrile derivatives for the treatment of cancer 特殊治疗有限公司 2022-04-26 CN disclosed
CN-114390920-A Chemically linked silk fibroin coatings and methods of making and using the same 自然进化公司 2022-04-22 CN disclosed
CN-114391008-A Lipid compounds and lipid nanoparticle compositions 苏州艾博生物科技有限公司 2022-04-22 CN disclosed
WO-2022081702-A1 IN VIVO TARGETING OF CD4+-T CELLS FOR MRNA THERAPEUTICS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2022-04-21 WO disclosed
WO-2022081842-A1 SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER THE BROAD INSTITUTE, INC. (US) 2022-04-21 WO disclosed
WO-2022081699-A1 IN VIVO TARGETING OF T CELLS FOR MRNA THERAPEUTICS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2022-04-21 WO disclosed
WO-2022081694-A1 IN VIVO TARGETING OF FIBROSIS BY ANTI-CD5-TARGETED FAP-CAR T MRNA-LNP THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2022-04-21 WO disclosed
WO-2022081469-A1 INHIBITORS OF RAF KINASES KINNATE BIOPHARMA INC. (US) 2022-04-21 WO disclosed
US-20220119371-A1 COMPOUND, COMPOSITIONS, AND METHODS DENALI THERAPEUTICS INC. (US) 2022-04-21 US disclosed
US-20220119567-A1 NETWORK POLYMERS AND METHODS OF MAKING AND USING SAME NATIONAL SCIENCE FOUNDATION 2022-04-21 US disclosed
US-20220119409-A1 TRICYCLIC PYRIDONES AND PYRIMIDONES ERASCA, INC. 2022-04-21 US disclosed
US-20220119580-A1 POLYURETHANE/UREA MATERIALS FOLDAX, INC. 2022-04-21 US disclosed
US-20220118123-A1 COMBINATION OF AR ANTAGONISTS AND TARGETED THORIUM CONJUGATES BAYER AKTIENGESELLSCHAFT (DE) 2022-04-21 US disclosed
EP-3490982-B1 PHARMACEUTICAL COMPOUNDS ALMAC DISCOVERY LTD (GB) 2022-04-20 EP disclosed
US-11304929-B2 Tosylacetate based compounds and derivatives thereof as PHGDH inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-04-19 US disclosed
CN-108698992-B 2-cyanoisoindoline derivatives for the treatment of cancer 特殊治疗有限公司 2022-04-19 CN disclosed
CN-109476629-B Urea and thiourea substituted bicyclic derivatives as pesticides 先正达参股股份有限公司 2022-04-15 CN disclosed
CN-111356706-B Polymerization process 埃克森美孚化学专利公司 2022-04-15 CN disclosed
CN-114364382-A Formulations and methods of use of RBP4 inhibitors 倍亮生物有限责任公司 2022-04-15 CN disclosed
CN-114364363-A Silk hair care composition 自然进化公司 2022-04-15 CN disclosed
CN-114364666-A Substituted N-phenyl-N-semicarbazides pyrimidines and salts thereof and their use as herbicides 拜耳公司 2022-04-15 CN disclosed
US-20220112170-A1 INHIBITORS OF RAF KINASES Pierre Fabre Médicament (FR) 2022-04-14 US disclosed
US-20220110933-A1 METHODS OF TREATING DISEASE WITH MAGL INHIBITORS H. LUNDBECK A/S (DK) 2022-04-14 US disclosed
WO-2022073920-A1 OLIGOMERIC COMPOUND FOR DYSTROPHIN RESCUE IN DMD PATIENTS THROUGHOUT SKIPPING OF EXON-51 SQY THERAPEUTICS (FR) 2022-04-14 WO disclosed
US-20220110862-A1 TREATMENT OF COGNITIVE DYSFUNCTION WITH PYRROLOPYRIDINE-ANILINE COMPOUNDS NFLECTION THERAPEUTICS, INC. 2022-04-14 US disclosed
EP-3980015-A1 BROAD SPECTRUM ANTIVIRAL COMPOUNDS TARGETING THE SKI COMPLEX University of Maryland, Baltimore (US) 2022-04-13 EP disclosed
CN-110204544-B 2- (morpholin-4-yl) -1, 7-naphthyridine 拜耳制药股份公司 2022-04-12 CN disclosed
US-11299513-B2 Cyclative release of peptidic compounds CIRCLE PHARMA, INC. (US) 2022-04-12 US disclosed
CN-114302876-A NLRP3 inhibitor 英夫拉索姆有限公司 2022-04-08 CN disclosed
CN-114288294-A Compounds and methods for treating or preventing hematologic cancers 布罗德研究所股份有限公司 2022-04-08 CN disclosed
CN-109311001-B Organosilica polymer catalyst and method for producing same 埃克森美孚研究工程公司 2022-04-08 CN disclosed
US-20220106315-A1 SPIRO-CONDENSED PYRROLIDINE DERIVATIVES AS DEUBIQUITYLATING ENZYMES (DUB) INHIBITORS MISSION THERAPEUTICS LTD (GB) 2022-04-07 US disclosed
US-20220106289-A1 NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2022-04-07 US disclosed
EP-3319938-B1 SMALL MOLECULE INHIBITORS OF THE MCL-1 ONCOPROTEIN AND USES THEREOF UNIV MARYLAND (US) 2022-04-06 EP disclosed
CN-105682658-B Cancer therapy using PI3 kinase subtype modulators 无限药品公司 2022-04-05 CN disclosed
CN-114286677-A Heterocyclic compounds as modulators of beta-catenin/TCF 4 interaction 新加坡科技研究局 2022-04-05 CN disclosed
CN-108864149-B Purification of rapamycin derivatives 生物传感器国际集团有限公司 2022-04-05 CN disclosed
CN-110563773-B Planar chiral ferrocene compound, intermediate thereof, preparation method and application 中国科学院上海有机化学研究所 2022-04-01 CN disclosed
CN-110248947-B MAGL inhibitors H.隆德贝克有限公司 2022-04-01 CN disclosed
CN-110267963-B MAGL inhibitors H.隆德贝克有限公司 2022-04-01 CN disclosed
CN-108602823-B Spiro-condensed pyrrolidine derivatives as Deubiquitinase (DUB) inhibitors 特殊治疗有限公司 2022-04-01 CN disclosed
CN-114269746-A Spiro aromatic ring compound, preparation and application thereof 上海奕拓医药科技有限责任公司 2022-04-01 CN disclosed
CN-110267962-B MAGL inhibitors H.隆德贝克有限公司 2022-04-01 CN disclosed
US-20220102713-A1 AQUEOUS BASED POLYMERS FOR SILICON DOMINANT ANODES ENEVATE CORPORATION 2022-03-31 US disclosed
US-20220096513-A1 COMPOUNDS AND METHODS USEFUL FOR TREATING OR PREVENTING CANCERS THE BROAD INSTITUTE, INC. (US) 2022-03-31 US disclosed
EP-3972651-A2 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE Novartis AG (CH) 2022-03-30 EP disclosed
CN-107849013-B Cyanopyrrolidines as DUB inhibitors for the treatment of cancer 特殊治疗有限公司 2022-03-29 CN disclosed
CN-109790169-B Cyanopyrrolidine derivatives having activity as USP30 inhibitors 特殊治疗有限公司 2022-03-29 CN disclosed
CN-114258301-A Dual ATM and DNA-PK inhibitors for use in antitumor therapy 艾科思莱德制药公司 2022-03-29 CN disclosed
CN-108026141-B Ligands for orphan nuclear receptor Nur77 and uses thereof 艾凯奇(厦门)生物科技有限公司 2022-03-29 CN disclosed
US-11286263-B2 Macrocyclic fluorine substituted indole derivatives THE BROAD INSTITUTE, INC. (US) 2022-03-29 US disclosed
US-20220089593-A1 PDE9 INHIBITOR AND USE THEREOF TRANSTHERA SCIENCES (NANJING), INC. (CN) 2022-03-24 US disclosed
US-20220089539-A1 TUBULIN INHIBITORS LIN BIOSCIENCE INC. (TW) 2022-03-24 US disclosed
EP-3969442-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR KINASES Kinnate Biopharma Inc. (US) 2022-03-23 EP disclosed
US-11279689-B2 1-(3-(6-(3-hydroxynaphthalen-1-yl)benzofuran-2-yl)azetidin-1 yl)prop-2-en-1-one derivatives and similar compounds as KRAS G12C modulators for treating cancer ARAXES PHARMA LLC (US) 2022-03-22 US disclosed
CN-111867646-B Fluorescent polymer coated films for medical devices 斯特拉斯堡大学 2022-03-22 CN disclosed
CN-111704610-B Pyrrolylamido pyridone compounds, preparation method and application 上海凌达生物医药有限公司 2022-03-22 CN disclosed
CN-114206870-A Tricyclic AKR1C3 dependent KARS inhibitors 诺华股份有限公司 2022-03-18 CN disclosed
CN-114206463-A Lipid compounds and lipid nanoparticle compositions 苏州艾博生物科技有限公司 2022-03-18 CN disclosed
CN-114206827-A Lipid nanoparticle compositions 苏州艾博生物科技有限公司 2022-03-18 CN disclosed
CN-114195804-A Piperidine condensed ring compound, preparation method and application 上海凌达生物医药有限公司 2022-03-18 CN disclosed
CN-111057048-B Aminopyrazine/pyridine compound, preparation method and application 上海凌达生物医药有限公司 2022-03-18 CN disclosed
US-20220081392-A1 NOVEL CARBONYL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS Acuitas Therapeutics, Inc. (CA) 2022-03-17 US disclosed
WO-2022052924-A1 PREPARATION METHOD FOR CLASS OF NITROGEN-CONTAINING FUSED RING COMPOUNDS AND USE THEREOF 上海凌达生物医药有限公司 2022-03-17 WO disclosed
US-20220081409-A1 PDE9 INHIBITOR AND USE THEREOF TRANSTHERA SCIENCES (NANJING), INC. (CN) 2022-03-17 US disclosed
US-20220081407-A1 METHODS OF PREPARING SUBSTITUTED INDANES PELOTON THERAPEUTICS, INC. (US) 2022-03-17 US disclosed
EP-3966202-A1 THIANTHRENE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS Facebook Technologies, LLC. (US) 2022-03-16 EP disclosed
EP-3153023-B1 BENZOXAZOLE KINASE INHIBITORS AND METHODS OF USE TAKEDA PHARMACEUTICALS CO (JP) 2022-03-16 EP disclosed
EP-3613743-B1 PROCESSES FOR THE PREPARATION OF 1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE DERIVATIVES INTELLIKINE LLC (US) 2022-03-16 EP disclosed
US-11274083-B2 Substituted thiophenyl uracils, salts thereof and the use thereof as herbicidal agents SYNGENTA CROP PROTECTION AG (CH) 2022-03-15 US disclosed
US-11274093-B2 Fused bicyclic benzoheteroaromatic compounds and methods of use thereof ARAXES PHARMA LLC (US) 2022-03-15 US disclosed
CN-112868659-B Composition applicable to user equipment and application thereof 3M中国有限公司 2022-03-11 CN disclosed
CN-108350034-B Antimicrobial polymyxin derived compounds 莫纳什大学 2022-03-11 CN disclosed
CN-114174326-A Long-term stable adrenomedullin analogues and uses thereof 拜耳公司 2022-03-11 CN disclosed
US-20220072155-A1 NOVEL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS ACUITAS THERAPEUTICS INC (CA) 2022-03-10 US disclosed
EP-3962484-A1 INHIBITORS OF RAF KINASES Kinnate Biopharma Inc. (US) 2022-03-09 EP disclosed
EP-3565549-B1 SELECTIVE HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF HUMAN DISEASE SHUTTLE PHARMACEUTICALS INC (US) 2022-03-09 EP disclosed
EP-3700907-B1 NOVEL PYRAZOLO-PYRROLO-PYRIMIDINE-DIONE DERIVATIVES AS P2X3 INHIBITORS BAYER AG (DE) 2022-03-09 EP disclosed
EP-3963082-A1 METHODS OF MAKING OLIGOPOTENT AND UNIPOTENT PRECURSORS Transfusion Health LLC (US) 2022-03-09 EP disclosed
US-11267819-B2 Diamine derivatives as inhibitors of leukotriene A4 hydrolase Celltaxsis, LLC (US) 2022-03-08 US disclosed
CN-109496213-B Spiro compounds and methods of making and using the same H.隆德贝克有限公司 2022-03-04 CN disclosed
CN-114144520-A Enhanced nucleic acid polymerization by aromatic compounds 斯特拉托斯基因公司 2022-03-04 CN disclosed
CN-114144178-A Nicorandil derivatives 尤尼赛夫医疗公司 2022-03-04 CN disclosed
WO-2022046642-A1 COMPOUNDS AND COMPOSITIONS FOR DISRUPTING PROGRAMMED RIBOSOMAL FRAMESHIFTING YALE UNIVERSITY (US) 2022-03-03 WO disclosed
WO-2022047315-A1 COMPOUNDS AND FORMULATIONS FOR TREATING OPHTHALMIC DISEASES VIEWPOINT THERAPEUTICS, INC. (US) 2022-03-03 WO disclosed
CN-114106341-A Comb copolymer and preparation method and application thereof 广州立邦涂料有限公司 2022-03-01 CN disclosed
CN-109020887-B Amide compounds as agents for the prophylaxis and treatment of psychotic disorders 绍兴从零医药科技有限公司 2022-03-01 CN disclosed
US-11261184-B2 [1,6]naphthyridine compounds and derivatives as CDK8/CDK19 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-03-01 US disclosed
CN-114126615-A Opioid receptor antagonist prodrugs 尼萨姆实验室公司 2022-03-01 CN disclosed
CN-114127051-A Inhibitors of fibroblast growth factor receptor kinase 金耐特生物制药公司 2022-03-01 CN disclosed
CN-114106278-A Polyurethane/urea materials 联邦科学和工业研究组织 2022-03-01 CN disclosed
CN-114106088-A Bromomethylpyrazine-based drug conjugates and ADCs 联宁(苏州)生物制药有限公司 2022-03-01 CN disclosed
CN-114085198-A Lipid and lipid nanoparticle formulations for delivery of nucleic acids 爱康泰生治疗公司 2022-02-25 CN disclosed
CN-114096550-A Modified nucleosides and methods of synthesis thereof 斯微(上海)生物科技股份有限公司 2022-02-25 CN disclosed
WO-2022040241-A1 A3 ADENOSINE RECEPTOR AGONISTS FOR USE IN MEDICINE BIOINTERVENE, INC. (US) 2022-02-24 WO disclosed
EP-3955878-A1 CHEMICALLY LINKED SILK FIBROIN COATINGS AND METHODS OF MAKING AND USING THEREOF Evolved by Nature, Inc. (US) 2022-02-23 EP disclosed
EP-3955886-A1 SILK HAIR CARE COMPOSITIONS Evolved by Nature, Inc. (US) 2022-02-23 EP disclosed
EP-3956033-A1 BICYCLIC COMPOUNDS Vivace Therapeutics, Inc. (US) 2022-02-23 EP disclosed
EP-3432934-B1 PRODRUGS OF CYTOTOXIC AGENTS WITH ENZYMATICALLY CLEAVABLE GROUPS Bayer Pharma AG (DE) 2022-02-23 EP disclosed
CN-114075196-A Aromatic ring-lactam compound, preparation method and application thereof 上海凌达生物医药有限公司 2022-02-22 CN disclosed
US-11254637-B2 Conversion of lignin to ionic liquids NATIONAL TECHNOLOGY & ENGINEERING SOLUTIONS OF SANDIA, LLC (US) 2022-02-22 US disclosed
US-11254640-B2 N-substituted indoles and other heterocycles for treating brain disorders THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-02-22 US disclosed
CN-110256427-B 2- (morpholin-4-yl) -1, 7-naphthyridine 拜耳制药股份公司 2022-02-22 CN disclosed
CN-114057749-A Preparation method and application of irreversible alkyne heterocyclic compound FGFR inhibitor 药雅科技(上海)有限公司 2022-02-18 CN disclosed
CN-114053431-A Liposome composition of compound with STING agonistic activity, and preparation method and application thereof 四川科伦药物研究院有限公司 2022-02-18 CN disclosed
CN-114072207-A Bicyclic compounds 维瓦斯治疗公司 2022-02-18 CN disclosed
CN-114072144-A External phosphoinositide 3-kinase inhibitors 维瑟拉有限公司 2022-02-18 CN disclosed
CN-114072148-A Inhibitors of RAF kinase 金耐特生物制药公司 2022-02-18 CN disclosed
WO-2022034568-A1 TRIAZOLE-PYRIDINYL SUBSTITUTED AZACYCLOHEXYL ACETIC ACID COMPOUNDS AS LPA RECEPTOR ANTAGONISTS VIVA STAR BIOSCIENCES LIMITED (CN) 2022-02-17 WO disclosed
US-20220048950-A1 NICOTINIC ACETYLCHOLINE RECEPTOR PEPTIDE ANTAGONIST CONOTOXIN COMPOSITIONS AND RELATED METHODS GLO PHARMA, INC. 2022-02-17 US disclosed
US-20220052380-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH CYCLIC ORGANOSILICON CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2022-02-17 US disclosed
US-20220047612-A1 PRODRUGS OF ALOX-15 INHIBITORS AND METHODS OF USING THE SAME EMPIRICO INC. 2022-02-17 US disclosed
EP-3953376-A1 METHODS FOR SYNTHESIZING BETA-HOMOAMINO ACIDS Protagonist Therapeutics, Inc. (US) 2022-02-16 EP disclosed
EP-3953331-A1 PYRAZOLESULFONAMIDES AS ANTITUMOR AGENTS Peloton Therapeutics, Inc. (US) 2022-02-16 EP disclosed
CN-112457326-B Aromatic heterocyclic lactam compound, preparation method and application 上海凌达生物医药有限公司 2022-02-15 CN disclosed
CN-114040760-A Irreversible inhibitors of the MENIN-MLL interaction 拜欧米富士恩公司 2022-02-11 CN disclosed
CN-114031658-A Lymphatic prodrugs 莫纳什大学 2022-02-11 CN disclosed
US-20220040193-A1 FORMULATIONS OF PHOSPHOINOSITIDE 3-KINASE INHIBITORS BRIDGEBIO GENE THERAPY RESEARCH, INC. 2022-02-10 US disclosed
US-20220040285-A1 Nucleoside-Modified RNA For Inducing an Adaptive Immune Response UNIV PENNSYLVANIA (US) 2022-02-10 US disclosed
EP-3947476-A1 NON-CORE-SHELL POLYMER PARTICLES The University of Sydney (AU) 2022-02-09 EP disclosed
EP-3086815-B1 SULFONAMIDE-CONTAINING LINKAGE SYSTEMS FOR DRUG CONJUGATES ZYMEWORKS INC (CA) 2022-02-09 EP disclosed
EP-3728237-B1 SUBSTITUTED THIOPHENYLURACILS , THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS SYNGENTA CROP PROTECTION AG (CH) 2022-02-09 EP disclosed
EP-3164380-B1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2022-02-09 EP disclosed
EP-3728235-B1 SUBSTITUTED THIOPHENYLURACILS , THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS SYNGENTA CROP PROTECTION AG (CH) 2022-02-09 EP disclosed
EP-3193881-B1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2022-02-09 EP disclosed
EP-3947350-A1 SUBSTITUTED 2-HETEROARYLAMINOBENZENES AND THE SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS Bayer Aktiengesellschaft (DE) 2022-02-09 EP disclosed
CN-108347916-B Composition and method for reducing ice crystal formation 先时迈纳米生物科技股份有限公司 2022-02-08 CN disclosed
US-11242364-B1 Efficient and scalable syntheses of nicotinoyl ribosides and reduced nicotinoyl ribosides, modified derivatives thereof, phosphorylated analogs thereof, adenylyl dinucleotide conjugates thereof, and novel crystalline forms thereof ChromaDex Inc. (US) 2022-02-08 US disclosed
US-11242337-B2 Compounds useful for treating gastrointestinal tract disorders ARDELYX, INC. (US) 2022-02-08 US disclosed
US-20220031676-A1 METHODS OF TREATING DISEASE WITH MAGL INHIBITORS H. LUNDBECK A/S (DK) 2022-02-03 US disclosed
US-20220031685-A1 COMBINATION THERAPY FOR TREATING BLOOD CANCER SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2022-02-03 US disclosed
US-20220033397-A1 PHARMACEUTICAL COMPOUNDS AND THEIR USE AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 19 (USP19) ALMAC DISCOVERY LTD (GB) 2022-02-03 US disclosed
US-11236092-B2 Spiro-condensed pyrrolidine derivatives as deubiquitylating enzymes (DUB) inhibitors MISSION THERAPEUTICS LIMITED (GB) 2022-02-01 US disclosed
US-20220024936-A1 INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, INC. 2022-01-27 US disclosed
US-20220026803-A1 RESIST COMPOSITION AND PATTERNING PROCESS SHIN-ETSU CHEMICAL CO., LTD. (JP) 2022-01-27 US disclosed
US-20220024947-A1 Purification of Rapamycin Derivatives Using Temperature Induced Phase Separation BIOSENSORS INTERNATIONAL GROUP, LTD. (BM) 2022-01-27 US disclosed
US-20220025111-A1 NARROW ABSORPTION POLYMER NANOPARTICLES AND RELATED METHODS UNIVERSITY OF WASHINGTON (US) 2022-01-27 US disclosed
EP-3943490-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS Mission Therapeutics Limited (GB) 2022-01-26 EP disclosed
EP-3941922-A1 INHIBITORS OF RAF KINASES Kinnate Biopharma Inc. (US) 2022-01-26 EP disclosed
CN-111153901-B Nitrogen-containing fused heterocyclic SHP2 inhibitor compound, preparation method and application 上海凌达生物医药有限公司 2022-01-25 CN disclosed
CN-113956252-A PDE9 inhibitors and uses thereof 药捷安康(南京)科技股份有限公司 2022-01-21 CN disclosed
US-20220017522-A1 METHOD FOR PREPARING PYRROLOPYRIMIDINE COMPOUND AND APPLICATION THEREOF CINKATE PHARMACEUTICAL INTERMEDIATES CO., LTD. (CN) 2022-01-20 US disclosed
US-20220016115-A1 USP19 INHIBITORS FOR USE IN THERAPY ALMAC DISCOVERY LIMITED (GB) 2022-01-20 US disclosed
US-20220019015-A1 INORGANIC MATRIX NANOIMPRINT LITHOGRAPHS AND METHODS OF MAKING THEREOF META PLATFORMS TECHNOLOGIES, LLC 2022-01-20 US disclosed
US-20220017477-A1 BENZOTHIAZOLE AND RELATED COMPOUNDS SPINOGENIX, INC. 2022-01-20 US disclosed
US-20220016106-A1 COMPOUNDS AND METHODS USEFUL FOR TREATING OR PREVENTING HEMATOLOGICAL CANCERS THE BROAD INSTITUTE, INC. (US) 2022-01-20 US disclosed
US-20220017509-A1 GAS41 INHIBITORS AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-01-20 US disclosed
EP-3937938-A1 NICORANDIL DERIVATIVES Unicycive Therapeutics Inc. (US) 2022-01-19 EP disclosed
EP-3940456-A1 NANOIMPRINT LITHOGRAPHY GRATING AND OPTICAL COMPONENT COMPRISING SUCH GRATING Facebook Technologies, LLC (US) 2022-01-19 EP disclosed
EP-3939964-A1 COMBINATIONS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS Ardelyx, Inc. (US) 2022-01-19 EP disclosed
EP-3939588-A1 USES OF PHOSPHODIESTERASE INHIBITORS Transthera Sciences (Nanjing), Inc. (CN) 2022-01-19 EP disclosed
EP-3454945-B1 ASH1L INHIBITORS AND METHODS OF TREATMENT THEREWITH UNIV MICHIGAN REGENTS (US) 2022-01-19 EP disclosed
EP-3541822-B1 MAGL INHIBITORS H LUNDBECK AS (DK) 2022-01-19 EP disclosed
US-11225662-B2 Peptide oligonucleotide conjugates SAREPTA THERAPEUTICS, INC. (US) 2022-01-18 US disclosed
US-11225505-B2 Antimicrobial polymyxin derivative compounds MONASH UNIVERSITY (AU) 2022-01-18 US disclosed
CN-113929729-A Veratramine compound, preparation method and application thereof 上海医药工业研究院 2022-01-14 CN disclosed
CN-106255513-B Sulfonamide-containing linking systems for drug conjugates 酵活有限公司 2022-01-14 CN disclosed
CN-113933921-A Inorganic substrate nanoimprint lithography body and method for manufacturing same 脸谱科技有限责任公司 2022-01-14 CN disclosed
CN-113939544-A Non-core-shell polymer particles 悉尼大学 2022-01-14 CN disclosed
CN-111704611-B Aryl spiro SHP2 inhibitor compound, preparation method and application 上海凌达生物医药有限公司 2022-01-14 CN disclosed
CN-112300194-B Condensed ring pyridone compounds, preparation method and application 上海凌达生物医药有限公司 2022-01-14 CN disclosed
US-20220008386-A1 TOSYLACETATE BASED COMPOUNDS AND DERIVATIVES THEREOF AS PHGDH INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-01-13 US disclosed
US-20220009887-A1 CYANOARYL-ANILINE COMPOUNDS FOR TREATMENT OF DERMAL DISORDERS NFLECTION THERAPEUTICS, INC. 2022-01-13 US disclosed
WO-2022011313-A1 MODIFICATION OF METALLIC SURFACES WITH PHOSPHONIC ACIDS BIOLOGICAL DYNAMICS, INC. (US) 2022-01-13 WO disclosed
WO-2022010676-A1 SILICON ANODES WITH WATER-SOLUBLE MALEIC ANHYDRIDE-. AND/OR MALEIC ACID-CONTAINING POLYMERS/COPOLYMERS, DERIVATIVES, AND/OR COMBINATIONS (WITH OR WITHOUT ADDITIVES) AS BINDERS ENEVATE CORPORATION (US) 2022-01-13 WO disclosed
WO-2022010537-A1 GAS41 INHIBITORS AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2022-01-13 WO disclosed
US-20220008416-A1 PYRIDAZINONE COMPOUNDS AND THEIR USE AS DAAO INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2022-01-13 US disclosed
US-20220013768-A1 SILICON ANODES WITH WATER-SOLUBLE MALEIC ANHYDRIDE-, AND/OR MALEIC ACID-CONTAINING POLYMERS/COPOLYMERS, DERIVATIVES, AND/OR COMBINATIONS (WITH OR WITHOUT ADDITIVES) AS BINDERS ENEVATE CORPORATION 2022-01-13 US disclosed
WO-2022011043-A2 COMPOUNDS, COMPOSITIONS, AND METHODS FOR THE TREATMENT OF FIBROTIC DISEASES AND CANCER PURDUE RESEARCH FOUNDATION (US) 2022-01-13 WO disclosed
EP-3377487-B1 COMPOUNDS FOR MEDICINAL APPLICATIONS AusVir Therapeutics Pty Ltd (AU) 2022-01-12 EP disclosed
EP-3445752-B1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2022-01-12 EP disclosed
EP-3549963-B1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS KODIAK SCIENCES INC (US) 2022-01-12 EP disclosed
EP-3935037-A1 USE OF 8,9-DIHYDROCANNABIDIOL COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-01-12 EP disclosed
CN-113923988-A Substituted arylmethyl and heteroarylmethyl ureas, analogs thereof, and methods of using the same 爱彼特生物制药公司 2022-01-11 CN disclosed
US-11221336-B2 Encoded chromophoric polymer particles and methods of use thereof UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2022-01-11 US disclosed
WO-2022006331-A2 PYRIDINE-1,5-DIONES EXHIBITNG MNK INHIBITION AND THEIR METHOD OF USE 4E THERAPEUTICS, INC. (US) 2022-01-06 WO disclosed
US-20220002264-A1 PHARMACEUTICAL COMPOUNDS ALMAC DISCOVERY LIMITED (GB) 2022-01-06 US disclosed
WO-2022002838-A1 SUBSTITUTED HETEROARYLOXYPYRIDINES, THE SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2022-01-06 WO disclosed
WO-2022003200-A1 REDUCTION OF VIRAL INFECTIONS pHOxgen Limited (IE) 2022-01-06 WO disclosed
EP-3930718-A1 PYRAZOLOPYRIDINE COMPOUNDS FOR IRE1 INHIBITION Optikira LLC (US) 2022-01-05 EP disclosed
EP-3930722-A1 TREATMENT WITH P2X3 MODULATORS Bellus Health Cough Inc. (CA) 2022-01-05 EP disclosed
EP-3930759-A1 CYCLIC-AMP RESPONSE ELEMENT BINDING PROTEIN (CBP) AND/OR ADENOVIRAL E1A BINDING PROTEIN OF 300 KDA (P300) DEGRADATION COMPOUNDS AND METHODS OF USE Cullgen (Shanghai), Inc. (CN) 2022-01-05 EP disclosed
EP-3930712-A1 IMIDAZOLOPYRAZINE COMPOUNDS FOR IRE1 INHIBITION Optikira LLC (US) 2022-01-05 EP disclosed
EP-3930708-A1 N-SUBSTITUTED INDOLES AND OTHER HETEROCYCLES FOR TREATING BRAIN DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-01-05 EP disclosed
EP-3931189-A1 AZEPINO-INDOLES AND OTHER HETEROCYCLES FOR TREATING BRAIN DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-01-05 EP disclosed
CN-109575016-B PDE9 inhibitors and uses thereof 药捷安康(南京)科技股份有限公司 2022-01-04 CN disclosed
US-11214565-B2 Compound, compositions, and methods DENALI THERAPEUTICS INC. (US) 2022-01-04 US disclosed
US-11213031-B2 Tetrazolylpropyl derivatives and their use as fungicides BAYER AKTIENGESELLSCHAFT (DE) 2022-01-04 US disclosed
US-11213523-B2 Substituted pyrido[1,2-a]pyrrolo[1,2-d]pyrazines for treating viral infections GILEAD SCIENCES, INC. (US) 2022-01-04 US disclosed
US-11213520-B2 Phenylpyrazolylacetamide compounds and derivatives as CDK8/CDK19 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-01-04 US disclosed
US-11214542-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2022-01-04 US disclosed
US-11214557-B2 MAGL inhibitors H. LUNDBECK A/S (DK) 2022-01-04 US disclosed
CN-113874381-A Inhibitors of RAF kinase 金耐特生物制药公司 2021-12-31 CN disclosed
CN-113874341-A Process for preparing derivatives of 1, 1-dialkylethane-1, 2-diols as useful intermediates 科学与工业研究委员会 2021-12-31 CN disclosed
CN-113874507-A Nucleic acid vaccine for coronavirus 苏州艾博生物科技有限公司 2021-12-31 CN disclosed
CN-113874344-A Use of 8, 9-dihydrocannabidiol compounds 加利福尼亚大学董事会 2021-12-31 CN disclosed
CN-107922364-B Lipid and lipid nanoparticle formulations for delivery of nucleic acids 爱康泰生治疗公司 2021-12-31 CN disclosed
US-20210401814-A1 MACROCYCLIC TYROSINE KINASE INHIBITOR AND USES THEREOF Xuanzhu Biopharmaceutical Co., Ltd. (CN) 2021-12-30 US disclosed
US-20210402015-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS KODIAK SCIENCES INC (US) 2021-12-30 US disclosed
US-20210401835-A1 Methods of Treating Chronic Lymphocytic Leukemia and Small Lymphocytic Leukemia Using a BTK Inhibitor ACERTA PHARMA B.V. (NL) 2021-12-30 US disclosed
US-20210403802-A1 METAL OXIDE, METAL BRONZE AND POLYOXOMETALATE AS CHARGE STORAGE MATERIALS IN ELECTROCHROMIC DEVICE Furcifer Inc. (US) 2021-12-30 US disclosed
WO-2021258147-A1 HYDROGELS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2021-12-30 WO disclosed
WO-2021260443-A1 COMBINATIONS OF 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINES BAYER AKTIENGESELLSCHAFT (DE) 2021-12-30 WO disclosed
WO-2021262587-A1 QUATERNARY INDAZOLE GLUCOCORTICOID RECEPTOR ANTAGONISTS CORCEPT THERAPEUTICS INCORPORATED (US) 2021-12-30 WO disclosed
WO-2021262786-A1 PANK MODULATORS AND METHODS USING SAME YALE UNIVERSITY (US) 2021-12-30 WO disclosed
EP-3929204-A1 MODIFIED NUCLEOSIDE AND SYNTHETIC METHOD THEREFOR Stemirna Therapeutics Co., Ltd. (CN) 2021-12-29 EP disclosed
EP-3164509-B1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2021-12-29 EP disclosed
EP-3927339-A1 COMBINATION OF AR ANTAGONISTS AND TARGETED THORIUM CONJUGATES Bayer Aktiengesellschaft (DE) 2021-12-29 EP disclosed
US-11207420-B2 Cytotoxin and conjugate, uses of same and preparation method therefor SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2021-12-28 US disclosed
US-11208432-B2 Inhibitors of glucocorticoid receptor ORIC PHARMACEUTICALS, INC. (US) 2021-12-28 US disclosed
US-11208527-B2 Photoactive macromolecules and uses thereof BECKMAN COULTER, INC. (US) 2021-12-28 US disclosed
US-11208409-B2 Substituted xanthines and methods of use thereof HYDRA BIOSCIENCES, LLC (US) 2021-12-28 US disclosed
US-11208655-B2 Functionally-modified oligonucleotides and subunits thereof SAREPTA THERAPEUTICS, INC. (US) 2021-12-28 US disclosed
CN-113853219-A Antibody drug conjugates with linkers comprising hydrophilic groups 诺华股份有限公司 2021-12-28 CN disclosed
CN-113840600-A N-substituted indoles and other heterocyclic compounds for treating brain diseases 加利福尼亚大学董事会 2021-12-24 CN disclosed
US-20210395221-A1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS INC (US) 2021-12-23 US disclosed
US-20210395275-A1 COMPOSITIONS AND METHODS FOR SELECTIVE SEPARATION OF HYDROCARBON ISOMERS UNITED STATES DEPARTMENT OF ENERGY 2021-12-23 US disclosed
WO-2021255091-A1 1,3,4-OXADIAZOLES AND THEIR DERIVATIVES AS FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 2021-12-23 WO disclosed
WO-2021255070-A1 ACTIVE COMPOUND COMBINATIONS BAYER AKTIENGESELLSCHAFT (DE) 2021-12-23 WO disclosed
WO-2021255089-A1 1,3,4-OXADIAZOLE PYRIMIDINES AND 1,3,4-OXADIAZOLE PYRIDINES AS FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 2021-12-23 WO disclosed
WO-2021255169-A1 1,3,4-OXADIAZOLE PYRIMIDINES AS FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 2021-12-23 WO disclosed
US-20210395188-A1 LIPIDS FOR LIPID NANOPARTICLE DELIVERY OF ACTIVE AGENTS Acuitas Therapeutics, Inc. (CA) 2021-12-23 US disclosed
US-20210395244-A1 MITOGEN-ACTIVATED PROTEIN KINASE KINASE (MEK) DEGRADATION COMPOUNDS AND METHODS OF USE ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI 2021-12-23 US disclosed
WO-2021255170-A1 1,3,4-OXADIAZOLE PYRIMIDINES AS FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 2021-12-23 WO disclosed
WO-2021257669-A1 SYNTHESIS OF SUBSTITUTED ARYLMETHYLUREAS, ANALOGUES, AND CRYSTALLINE FORMS THEREOF AND METHODS OF USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2021-12-23 WO disclosed
US-20210395295-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. 2021-12-23 US disclosed
EP-3074385-B1 PIPERIDINE DERIVATIVES FOR USE IN THE TREATMENT OR PREVENTION OF PSYCHIATRIC AND NEUROLOGICAL CONDITIONS TAKEDA PHARMACEUTICALS CO (JP) 2021-12-22 EP disclosed
CN-113825756-A Substituted polycyclic carboxylic acids, analogs thereof, and methods of use thereof 爱彼特生物制药公司 2021-12-21 CN disclosed
CN-113816969-A Irinotecan compound, antibody drug conjugate thereof and application thereof 联宁(苏州)生物制药有限公司 2021-12-21 CN disclosed
US-11203600-B2 Kinase inhibitors and uses thereof DENALI THERAPEUTICS INC. (US) 2021-12-21 US disclosed
CN-108026046-B Substituted quinazoline compounds and their use as inhibitors of G12C mutant KRAS, HRAS and/or NRAS proteins 亚瑞克西斯制药公司 2021-12-21 CN disclosed
CN-113816990-A Modified amino acids and their use in ADCs 联宁(苏州)生物制药有限公司 2021-12-21 CN disclosed
CN-113813399-A Camptothecin compound, antibody drug conjugate thereof and application thereof 联宁(苏州)生物制药有限公司 2021-12-21 CN disclosed
CN-113801297-A Photosensitive macromolecules and uses thereof 拜克门寇尔特公司 2021-12-17 CN disclosed
CN-113801296-A Photosensitive macromolecules and uses thereof 拜克门寇尔特公司 2021-12-17 CN disclosed
US-20210386751-A1 TREATMENT WITH P2X3 MODULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.3) LIMITED (GB) 2021-12-16 US disclosed
US-20210389298-A1 Alzheimer's Disease Assay in a Living Patient PAIN THERAPEUTICS, INC. (US) 2021-12-16 US disclosed
US-20210388138-A1 DERIVATIZABLE MONOMERS AND POLYMERS, AND METHODS FOR MAKING AND USING SAME RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2021-12-16 US disclosed
WO-2021252494-A1 USE OF MULTI-KINASE INHIBITORS TO TREAT RNA VIRUS INFECTIONS ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2021-12-16 WO disclosed
WO-2021252709-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR TREATING, AMELIORATING, AND/OR PREVENTING SIGMA RECEPTOR RELATED DISEASES AND/OR DISORDERS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2021-12-16 WO disclosed
WO-2021250461-A1 SUBSTITUTED ISOQUINOLINYLMETHYL AMIDES, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2021-12-16 WO disclosed
WO-2021249995-A1 AZABICYCLYL-SUBSTITUTED HETEROCYCLES AS FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 2021-12-16 WO disclosed
US-20210386734-A1 DUAL MAGL AND FAAH INHIBITORS LUNDBECK LA JOLLA RESEARCH CENTER, INC. 2021-12-16 US disclosed
WO-2021252488-A1 INHIBITORS OF NEK7 KINASE Halia Therapeutics, Inc. (US) 2021-12-16 WO disclosed
WO-2021250466-A1 SUBSTITUTED (PHTHALAZIN-1-YLMETHYL)UREAS, SUBSTITUTED N-(PHTHALAZIN-1-YLMETHYL)AMIDES, AND ANALOGUES THEREOF ARBUTUS BIOPHARMA CORPORATION (CA) 2021-12-16 WO disclosed
EP-3441392-B1 A PHARMACEUTICAL COMPOSITION FOR ORAL ADMINISTRATION INTELLIKINE LLC (US) 2021-12-15 EP disclosed
EP-3921080-A1 CAPTURE OF FLUORINATED CARBON COMPOUNDS The University of Queensland (AU) 2021-12-15 EP disclosed
US-11198685-B2 Substituted ureas and methods of making and using same MEBIAS DISCOVERY, INC. (US) 2021-12-14 US disclosed
CN-113795254-A Pyrazolopyridine compounds for IRE1 inhibition 奥普提卡拉公司 2021-12-14 CN disclosed
CN-113784962-A Azacyclo-indoles and other heterocycles useful in the treatment of cerebral disorders 加利福尼亚大学董事会 2021-12-10 CN disclosed
CN-113784946-A Fluorene derived monomers and polymers for volume bragg gratings 脸谱科技有限责任公司 2021-12-10 CN disclosed
CN-108276410-B Anaplastic lymphoma kinase inhibitor and preparation method and application thereof 首药控股(北京)股份有限公司 2021-12-10 CN disclosed
US-20210379032-A1 HISTONE DEACETYLASE INHIBITORS FOR IMMUNOMODULATION IN TUMOR MICROENVIRONMENT Great Novel Therapeutics Biotech & Medicals Corporation (TW) 2021-12-09 US disclosed
US-20210379052-A1 QUINOLINE DERIVATIVE HAVING INDOLEAMINE-2,3-DIOXYGENASE INHIBITORY ACTIVITY SHENZHEN CHIPSCREEN BIOSCIENCES CO., LTD. (CN) 2021-12-09 US disclosed
US-20210380579-A1 PROTEOLYSIS TARGETING CHIMERA (PROTACS) AS DEGRADERS OF SMARCA2 AND /OR SMARCA4 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-12-09 US disclosed
US-20210380574-A1 ANNULATED 2-AMINO-3-CYANO THIOPHENES AND DERIVATIVES FOR THE TREATMENT OF CANCER VANDERBILT UNIVERSITY 2021-12-09 US disclosed
US-20210380595-A1 2-(2-ACRYLOYL-2,6-DIAZASPIRO[3.4]OCTAN-6-YL)-6-(1H-INDAZOL-4-YL)-BENZONITRILE DERIVATIVES AND RELATED COMPOUNDS AS INHIBITORS OF G12C MUTANT KRAS PROTEIN FOR INHIBITING TUMOR METASTASIS ARAXES PHARMA LLC (US) 2021-12-09 US disclosed
US-20210380562-A1 Novel Compounds MISSION THERAPEUTICS LIMITED (GB) 2021-12-09 US disclosed
US-20210379084-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. 2021-12-09 US disclosed
US-20210379064-A1 AXL INHIBITORS FOR USE IN COMBINATION THERAPY FOR PREVENTING, TREATING OR MANAGING METASTATIC CANCER MIDCAP FINANCIAL TRUST 2021-12-09 US disclosed
EP-3917915-A1 1,2,4-TRIAZIN-3(2H)-ONE COMPOUNDS FOR THE TREATMENT OF HYPERPROLIFERATIVE DISEASES Bayer Aktiengesellschaft (DE) 2021-12-08 EP disclosed
EP-3469601-B1 POLYMER-SILICA HYBRID PDOTS UNIV WASHINGTON (US) 2021-12-08 EP disclosed
EP-3918028-A1 QUANTUM DOTS AND PROCESSES FOR PREPARATION THEREOF The University of Queensland (AU) 2021-12-08 EP disclosed
CN-113754683-A Isotopically substituted spiroaromatic ring compounds and their use 上海奕拓医药科技有限责任公司 2021-12-07 CN disclosed
CN-112094269-B Saturated six-membered ring heterocyclic compound, preparation method and application 上海凌达生物医药有限公司 2021-12-07 CN disclosed
US-RE48842-E1 Pyrimido-pyrrolo-oxazine-dione compound inhibitors of the cystic fibrosis transmembrane conductance regulator protein and uses therefor THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-12-07 US disclosed
US-11192865-B2 Benzosulfonyl compounds VIVACE THERAPEUTICS, INC. (US) 2021-12-07 US disclosed
CN-110892001-B Electrochromic polymers and their synthesis and use 菲尔齐费尔公司 2021-12-03 CN disclosed
CN-113748108-A Thianthrene-derived monomers and polymers for volume bragg gratings 脸谱科技有限责任公司 2021-12-03 CN disclosed
CN-113748148-A Latent image for volume Bragg grating 脸谱科技有限责任公司 2021-12-03 CN disclosed
US-20210371855-A1 METHODS OF INHIBITING PROLIFERATIVE CELLS IDEAYA BIOSCIENCES, INC. 2021-12-02 US disclosed
WO-2021242505-A1 INHIBITORS OF NEK7 KINASE Halia Therapeutics, Inc. (US) 2021-12-02 WO disclosed
WO-2021239673-A1 SUBSTITUTED PYRROLINE-2-ONES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2021-12-02 WO disclosed
WO-2021239766-A1 ACTIVE COMPOUND COMBINATIONS BAYER AKTIENGESELLSCHAFT (DE) 2021-12-02 WO disclosed
US-20210369807-A1 BOTULINUM NEUROTOXIN-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING REGENERON PHARMACEUTICALS, INC. 2021-12-02 US disclosed
US-20210369724-A1 COMBINATION OF ATR KINASE INHIBITORS WITH 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2021-12-02 US disclosed
EP-3416960-B1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2021-12-01 EP disclosed
EP-3519412-B1 CYANOPYRROLIDINE DERIVATIVES WITH ACTIVITY AS INHIBITORS OF USP30 MISSION THERAPEUTICS LTD (GB) 2021-12-01 EP disclosed
EP-3915971-A1 PHENYL-S(O)N-PHENYLAMIDINES AND THE USE THEREOF AS FUNGICIDES Bayer Aktiengesellschaft (DE) 2021-12-01 EP disclosed
EP-3914589-A1 METHODS OF TREATING DISEASE WITH MAGL INHIBITORS H. Lundbeck A/S (DK) 2021-12-01 EP disclosed
EP-3915992-A1 PDE9 INHIBITOR AND USE THEREOF Transthera Sciences (Nanjing), Inc. (CN) 2021-12-01 EP disclosed
CN-113728029-A Thermally reversible and reconfigurable cross-linked polymers for volume bragg gratings 脸谱科技有限责任公司 2021-11-30 CN disclosed
CN-105979959-B Compounds and methods for inhibiting phosphate transport 阿德利克斯公司 2021-11-30 CN disclosed
CN-113727716-A Treatment with P2X3 modulators 贝卢斯医疗咳嗽病公司 2021-11-30 CN disclosed
US-11186554-B2 Non-fused tricyclic compounds VIVACE THERAPEUTICS, INC. (US) 2021-11-30 US disclosed
US-11186563-B2 Pd(II)-catalyzed enantioselective β-methylene C(sp3)—H bond activation THE SCRIPPS RESEARCH INSTITUTE (US) 2021-11-30 US disclosed
CN-113710661-A Compounds and methods for treating cancer 上海睿跃生物科技有限公司 2021-11-26 CN disclosed
CN-113698414-A Bioactive substance conjugate and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2021-11-26 CN disclosed
US-20210363123-A1 SLC26A3 INHIBITORS AND USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2021-11-25 US disclosed
US-20210363168-A1 EFFICIENT AND SCALABLE SYNTHESES OF NICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, MODIFIED DERIVATIVES THEREOF, PHOSPHORYLATED ANALOGS THEREOF, ADENYLYL DINUCLEOTIDE CONJUGATES THEREOF, AND NOVEL CRYSTALLINE FORMS THEREOF THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2021-11-25 US disclosed
US-20210363146-A1 TROPOMYOSIN RECEPTOR KINASE (TRK) DEGRADATION COMPOUNDS AND METHODS OF USE CULLGEN (SHANGHAI), INC. (CN) 2021-11-25 US disclosed
WO-2021233861-A1 AZABICYCLIC(THIO)AMIDES AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2021-11-25 WO disclosed
EP-3911653-A1 SUBSTITUTED POLYCYCLIC CARBOXYLIC ACIDS, ANALOGUES THEREOF, AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2021-11-24 EP disclosed
EP-3911632-A1 PRODRUGS OF ALOX-15 INHIBITORS AND METHODS OF USING THE SAME EMPIRICO INC. (US) 2021-11-24 EP disclosed
EP-3661925-B1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LTD (IE) 2021-11-24 EP disclosed
EP-3763712-B1 INDOLIZINE COMPOUNDS, PREPARATION METHOD AND USE THEREOF HAIHE BIOPHARMA CO LTD (CN) 2021-11-24 EP disclosed
CN-113683622-A Bioactive substance conjugate and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2021-11-23 CN disclosed
CN-107660199-B Piperazine carbamates and methods of making and using the same H.隆德贝克有限公司 2021-11-23 CN disclosed
CN-113677665-A Substituted 2-heteroarylaminobenzenes and their salts and their use as herbicides 拜耳公司 2021-11-19 CN disclosed
WO-2021228734-A1 TRIAZINE AND PYRIMIDINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2021-11-18 WO disclosed
WO-2021228939-A1 FLUOROGENIC DIMER COMPOUND, USEFUL AS A PROBE FOR DETECTION OF ENDOGENOUS RECEPTORS UNIVERSITE DE STRASBOURG (FR) 2021-11-18 WO disclosed
WO-2021231726-A1 ENPP1 MODULATORS AND USES THEREOF Vir Biotechnology, Inc. (US) 2021-11-18 WO disclosed
WO-2021229302-A1 SUBSTITUTED TRICYCLIC AMIDES, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2021-11-18 WO disclosed
WO-2021231892-A1 CERTAIN CHEMICAL COMPOSITIONS AND METHODS OF USE THEREOF ALGEN BIOTECHNOLOGIES, INC. (US) 2021-11-18 WO disclosed
US-20210353630-A1 1,2,4-TRIAZIN-3(2H)-ONE COMPOUNDS FOR THE TREATMENT OF HYPERPROLIFERATIVE DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2021-11-18 US disclosed
US-20210353555-A1 NANOPARTICLES BASED ON OPTIONALLY ALKOXYLATED POLY(ALKYL CYANOACRYLATES) HAVING A DEFINED DEGREE OF POLYMERIZATION AbbVie Deutschland GmbH & Co. KG (DE) 2021-11-18 US disclosed
US-20210355073-A1 COPPER NANOPARTICLE BASED CHEMOSELECTIVE REDUCTION BROWN UNIVERSITY 2021-11-18 US disclosed
US-20210355130-A1 INHIBITORS OF NEK7 KINASE Halia Therapeutics, Inc. 2021-11-18 US disclosed
EP-3908568-A1 LIPIDS FOR LIPID NANOPARTICLE DELIVERY OF ACTIVE AGENTS Acuitas Therapeutics, Inc. (CA) 2021-11-17 EP disclosed
CN-107531759-B Non-membrane disruptive p 53-activated stapled peptides 新加坡科技研究局 2021-11-16 CN disclosed
US-11174245-B2 Benzimidazole compounds and derivatives as EGFR inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-11-16 US disclosed
US-11174275-B2 Methods for the preparation of cyclopentaoxasilinones and cyclopentaoxaborininones and their use DREXEL UNIVERSITY (US) 2021-11-16 US disclosed
US-11174263-B2 Inhibitors of menin-MLL interaction BIOMEA FUSION, INC. (US) 2021-11-16 US disclosed
US-11174268-B2 Benzenesulfonamide compouds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2021-11-16 US disclosed
CN-113651831-A Bioactive substance conjugate and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2021-11-16 CN disclosed
CN-113660931-A Arylaniline and heteroarylaniline compounds for the treatment of skin cancer 恩福莱克逊治疗有限公司 2021-11-16 CN disclosed
CN-113645964-A Arylaniline and heteroarylaniline compounds for use in fetal marker therapy 恩福莱克逊治疗有限公司 2021-11-12 CN disclosed
CN-113646002-A Cyclic AMP response element binding protein (CBP) and/or 300KDA adenovirus E1A binding protein (P300) degradation compounds and methods of use 上海睿跃生物科技有限公司 2021-11-12 CN disclosed
CN-113636947-A Novel lipid and lipid nanoparticle formulations for delivery of nucleic acids 爱康泰生治疗公司 2021-11-12 CN disclosed
CN-108434197-B Compositions and methods for weight management 尤妮金公司 2021-11-12 CN disclosed
US-20210346391-A1 TREATMENT OF PRURITUS WITH P2X3 MODULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.3) LIMITED (GB) 2021-11-11 US disclosed
US-20210346382-A1 BTK Inhibitors to Treat Solid Tumors Through Modulation of the Tumor Microenvironment ACERTA PHARMA BV (NL) 2021-11-11 US disclosed
WO-2021226547-A2 TARGETED NEK7 INHIBITION FOR MODULATION OF THE NLRP3 INFLAMMASOME Halia Therapeutics, Inc. (US) 2021-11-11 WO disclosed
WO-2021226404-A1 USE OF IL-6 ANTIBODIES AND VEGF TRAPS, AND FUSION CONSTRUCTS AND CONJUGATES THEREOF KODIAK SCIENCES INC. (US) 2021-11-11 WO disclosed
WO-2021226247-A1 SYSTEMS AND METHODS FOR TYROSINASE-MEDIATED SITE-SPECIFIC PROTEIN CONJUGATION GENENTECH, INC. (US) 2021-11-11 WO disclosed
WO-2021224220-A1 PYRIDINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2021-11-11 WO disclosed
US-20210347806-A1 EFFICIENT AND SCALABLE SYNTHESES OF NICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, MODIFIED DERIVATIVES THEREOF, PHOSPHORYLATED ANALOGS THEREOF, ADENYLYL DINUCLEOTIDE CONJUGATES THEREOF, AND NOVEL CRYSTALLINE FORMS THEREOF THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2021-11-11 US disclosed
US-20210347804-A1 COMPOUNDS, COMPOSITIONS AND METHOD FOR COLORING EDIBLE MATERIALS THE PENN STATE RESEARCH FOUNDATION 2021-11-11 US disclosed
US-20210347737-A1 NOVEL COMPOUNDS INFLAZOME LIMITED (IE) 2021-11-11 US disclosed
US-20210347950-A1 POLYMER COMPOSITION BASF SE (DE) 2021-11-11 US disclosed
US-20210346369-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC. (US) 2021-11-11 US disclosed
EP-3906026-A1 IRREVERSIBLE INHIBITORS OF MENIN-MLL INTERACTION Biomea Fusion, LLC (US) 2021-11-10 EP disclosed
EP-3137169-B1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2021-11-10 EP disclosed
EP-3906029-A1 INHIBITORS OF MENIN-MLL INTERACTION Biomea Fusion, LLC (US) 2021-11-10 EP disclosed
CN-113620958-A Heterocyclic compounds for the treatment of PI 3K-gamma mediated disorders 无限药品股份有限公司 2021-11-09 CN disclosed
CN-108699057-B 5-substituted 2- (morpholin-4-yl) -1, 7-naphthyridines 拜耳医药股份公司 2021-11-09 CN disclosed
US-11168115-B2 Cyclic peptides as protein targeting agents CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2021-11-09 US disclosed
US-11166951-B2 Therapeutic combinations of a BTK inhibitor, a PI3K inhibitor, a JAK-2 inhibitor, and/or a BCL-2 inhibitor ACERTA PHARMA B.V. (NL) 2021-11-09 US disclosed
CN-113616656-A Heterocyclic compounds for the treatment of PI 3K-gamma mediated disorders 无限药品股份有限公司 2021-11-09 CN disclosed
CN-110809560-B Electrochromic polymer films with reduced self-bleaching behavior and enhanced cycling stability 菲尔齐费尔公司 2021-11-09 CN disclosed
CN-113631569-A Process for the synthesis of beta-homoamino acids 领导医疗有限公司 2021-11-09 CN disclosed
CN-110857300-B Condensed ring triazole compounds, preparation method and application 上海凌达生物医药有限公司 2021-11-05 CN disclosed
CN-108558889-B Bromodomain inhibitors 赛尔基因昆蒂赛尔研究公司 2021-11-05 CN disclosed
CN-108290992-B Polyurethane/urea materials 联邦科学和工业研究组织 2021-11-05 CN disclosed
CN-113603703-A Bioactive substance conjugate and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2021-11-05 CN disclosed
WO-2021222522-A1 CD73 INHIBITING 2,4-DIOXOPYRIMIDINE COMPOUNDS GILEAD SCIENCES, INC. (US) 2021-11-04 WO disclosed
WO-2021220132-A1 METHODS AND COMPOSITIONS FOR OCULAR CELL THERAPY NOVARTIS AG (CH) 2021-11-04 WO disclosed
US-20210344047-A1 Silicon-Based Energy Storage Devices With Fluorinated Polymer Containing Electrolyte Additives ENEVATE CORPORATION 2021-11-04 US disclosed
US-20210340534-A1 Mixed Tricyclo-DNA, 2'-Modified RNA Oligonucleotide Compositions and Uses Thereof SYNTHENA AG (CH) 2021-11-04 US disclosed
US-20210340547-A1 FIBROTIC TREATMENT MONASH UNIVERSITY (AU) 2021-11-04 US disclosed
US-20210339186-A1 MOF COMPOSITIONS FOR SELECTIVE SEPARATION OF HYDROCARBONS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2021-11-04 US disclosed
US-20210340313-A1 MULTICOLORED ELECTROCHROMIC POLYMER COMPOSITIONS AND METHODS OF MAKING AND USING THE SAME Furcifer Inc. (US) 2021-11-04 US disclosed
US-20210338653-A1 N-[2-(1 -BENZYLPIPERIDIN-4-YL)ETHYL]-4-(PYRAZIN-2-YL)-PIPERAZINE-1 -CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS MUSCARINIC RECEPTOR 4 (M4) ANTAGONISTS FOR TREATING NEUROLOGICAL DISEASES NEUROCRINE BIOSCIENCES, INC. 2021-11-04 US disclosed
US-20210343445-A1 POLYMER-SILICA HYBRID PDOTS AND METHODS OF USE THEREOF UNIVERSITY OF WASHINGTON (US) 2021-11-04 US disclosed
EP-3487850-B1 UREA AND THIOUREA SUBSTITUTED BICYCLES DERIVATIVES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2021-11-03 EP disclosed
US-11161834-B2 Methods of manufacturing of niraparib TESARO, INC. (US) 2021-11-02 US disclosed
US-11161852-B1 Inhibitors of NEK7 kinase Halia Therapeutics, Inc. (US) 2021-11-02 US disclosed
US-11165099-B2 Silicon-based energy storage devices with cyclic organosilicon containing electrolyte additives ENEVATE CORPORATION (US) 2021-11-02 US disclosed
US-11161856-B2 Spirocycle compounds and methods of making and using same H. LUNDBECK A/S (DK) 2021-11-02 US disclosed
US-11161849-B2 Inhibiting the transient receptor potential al ion channel ELI LILLY AND COMPANY (US) 2021-11-02 US disclosed
CN-109912599-B Chemical entities, compositions, and methods 英特利凯恩有限责任公司 2021-11-02 CN disclosed
CN-113563323-A Benzothiazolyl biaryl compounds, preparation method and application 上海凌达生物医药有限公司 2021-10-29 CN disclosed
US-20210332027-A1 ALKYNYL-SUBSTITUTED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF BEIJING INNOCARE PHARMA TECH CO., LTD. (CN) 2021-10-28 US disclosed
US-20210332020-A1 PHENYLSULFONYLUREA DERIVATIVES USEFUL AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2021-10-28 US disclosed
US-20210332012-A1 N-SUBSTITUTED INDOLES AND OTHER HETEROCYCLES FOR TREATING BRAIN DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA CORPORATION 2021-10-28 US disclosed
WO-2021217006-A1 (S)-2-AMINO-6-((3-AMINOPROPYL)AMINO)HEXANOIC ACID (APL) FOR USE IN THE TREATMENT OF NON-ALCOHOLIC STEATOHEPATITIS (NASH), LIVER INFLAMMATION, HEPATOCELLULAR BALLOONING, LIVER FIBROSIS AND STEATOSIS TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2021-10-28 WO disclosed
WO-2021214492-A1 METHOD OF SELECTING PATIENTS FOR TREATMENT WITH A COMBINATION OF AN AXL INHIBITOR AND AN IMMUNE CHECKPOINT MODULATOR BERGENBIO ASA (NO) 2021-10-28 WO disclosed
EP-2448569-B1 PHARMACOLOGY OF VISUAL CYCLE MODULATORS ACUCELA INC (US) 2021-10-27 EP disclosed
EP-3898620-A1 HETEROCYCLYL PYRIDAZINE AS FUNGICIDAL COMPOUNDS Bayer Aktiengesellschaft (DE) 2021-10-27 EP disclosed
EP-3898978-A2 NANOCAPSULES FOR THE DELIVERY OF CELL MODULATING AGENTS CSL Behring LLC (US) 2021-10-27 EP disclosed
EP-3010550-B1 CYCLIC PEPTIDES AS PROTEIN TARGETING AGENTS CALIFORNIA INST OF TECHN (US) 2021-10-27 EP disclosed
EP-3898612-A1 SUBSTITUTED PYRIDINYLOXYBENZENES AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL AGENTS Bayer Aktiengesellschaft (DE) 2021-10-27 EP disclosed
EP-3897154-A1 1,3,4-OXADIAZOLES AND THEIR DERIVATIVES AS NEW ANTIFUNGAL AGENTS Bayer Aktiengesellschaft (DE) 2021-10-27 EP disclosed
CN-108713023-B Glucocorticoid receptor inhibitors 欧瑞克制药公司 2021-10-26 CN disclosed
CN-107624115-B Botulinum neurotoxin specific capture agents, compositions, methods of use, and methods of manufacture 加州理工学院 2021-10-26 CN disclosed
US-11154554-B2 Therapeutic combinations of a MEK inhibitor and a BTK inhibitor Acera Pharma B.V. (NL) 2021-10-26 US disclosed
US-11155610-B2 Dual PDGF/VEGF antagonists KODIAK SCIENCES INC. (US) 2021-10-26 US disclosed
CN-109715632-B Macrocyclic indole derivatives 拜尔公开股份有限公司 2021-10-26 CN disclosed
CN-111295389-B Bioactive substance conjugate and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2021-10-22 CN disclosed
CN-113544270-A Nanocapsules for delivery of cell modulators 美国杰特贝林生物制品有限公司 2021-10-22 CN disclosed
CN-105102000-B Cancer therapy using PI3 kinase subtype modulators 无限药品公司 2021-10-22 CN disclosed
CN-109293652-B Substituted thiazole derivative and application thereof 四川科伦博泰生物医药股份有限公司 2021-10-22 CN disclosed
CN-113527299-A Nitrogen-containing condensed ring compounds, preparation method and application 上海凌达生物医药有限公司 2021-10-22 CN disclosed
WO-2021209490-A1 CYCLAMINEPHENYLAMINOQUINOLINES AS FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 2021-10-21 WO disclosed
WO-2021209486-A1 SPECIFICALLY SUBSTITUTED PYRROLINE-2-ONES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2021-10-21 WO disclosed
US-20210324006-A1 PEPTIDE COMPOSITIONS AND METHODS FOR INHIBITING NICOTINIC ACETYLCHOLINE RECEPTOR ACTIVITY GLO PHARMA, INC. 2021-10-21 US disclosed
US-20210323976-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD PHARMACEUTICALS, INC. 2021-10-21 US disclosed
US-20210322331-A1 NANOCAPSULES FOR THE DELIVERY OF CELL MODULATING AGENTS CSL BEHRING LLC (US) 2021-10-21 US disclosed
US-20210322432-A1 SELECTIVE P2X3 MODULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.3) LIMITED (GB) 2021-10-21 US disclosed
US-20210322408-A1 Methods of Treating Cancers, Immune and Autoimmune Diseases, and Inflammatory Diseases Based on BTK Occupancy and BTK Resynthesis Rate ACERTA PHARMA BV (NL) 2021-10-21 US disclosed
US-20210324063-A1 ANTIBODIES AND CONJUGATES THEREOF KODIAK SCIENCES INC. 2021-10-21 US disclosed
EP-3268362-B1 SUBSTITUTED PYRIDINES AND USES THEREOF PELOTON THERAPEUTICS INC (US) 2021-10-20 EP disclosed
EP-3356359-B1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC (US) 2021-10-20 EP disclosed
EP-3087091-B1 VAR2CSA-DRUG CONJUGATES ZYMEWORKS INC (CA) 2021-10-20 EP disclosed
EP-2367800-B9 SUBSTITUTED PYRIMIDINES FOR THE TREATMENT OF DISEASES SUCH AS CANCER IPHARMA H K LTD (HK) 2021-10-20 EP disclosed
EP-3893892-A1 ORGANIC COMPOUNDS Rutgers, the State University of New Jersey (US) 2021-10-20 EP disclosed
EP-3893645-A1 SUBSTITUTED ARYLMETHYLUREAS AND HETEROARYLMETHYLUREAS, ANALOGUES THEREOF, AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2021-10-20 EP disclosed
US-11149037-B2 Pyrazole MAGL inhibitors H. LUNDBECK A/S (DK) 2021-10-19 US disclosed
US-11148125-B2 Catalysts for olefin isomerization BRANDEIS UNIVERSITY (US) 2021-10-19 US disclosed
US-11147885-B2 ASH1L inhibitors and methods of treatment therewith THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2021-10-19 US disclosed
US-11147884-B2 Inhibitors of NHE-mediated antiport ARDELYX, INC. (US) 2021-10-19 US disclosed
CN-108699035-B Novel compounds 特殊治疗有限公司 2021-10-15 CN disclosed
CN-107709293-B Ligand activated meta C-H activation using transient mediators 斯克里普斯研究学院 2021-10-15 CN disclosed
US-20210317150-A1 CD73 INHIBITORS AND USES THEREOF PELOTON THERAPEUTICS, INC. (US) 2021-10-14 US disclosed
US-20210317128-A1 NOVEL PYRAZOLO-PYRROLO-PYRIMIDINE-DIONE DERIVATIVES AS P2X3 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2021-10-14 US disclosed
US-20210317127-A1 HETEROCYCLIC SPIRO COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF CANCER ARAXES PHARMA LLC (US) 2021-10-14 US disclosed
US-20210315999-A1 TROPOMYOSIN RECEPTOR KINASE (TRK) DEGRADATION COMPOUNDS AND METHODS OF USE CULLGEN (SHANGHAI), INC. (CN) 2021-10-14 US disclosed
US-20210317097-A1 NON-ATP/CATALYTIC SITE p38 MITOGEN ACTIVATED PROTEIN KINASE INHIBITORS UNIVERSITY OF MARYLAND, BALTIMORE 2021-10-14 US disclosed
EP-3890745-A1 SYNTHETIC DERIVATIVES OF CHOLIC ACID 7-SULFATE AND USES THEREOF President and Fellows of Harvard College (US) 2021-10-13 EP disclosed
EP-3890733-A1 NON-ATP/CATALYTIC SITE P38 MITOGEN ACTIVATED PROTEIN KINASE INHIBITORS University of Maryland, Baltimore (US) 2021-10-13 EP disclosed
EP-3890742-A1 PRODRUGS OF ANTI-CANCER AND ANTI-AUTOIMMUNE DISEASES THERAPEUTIC AGENTS, AND METHODS OF MAKING AND USE THEREOF University of Maryland, Baltimore (US) 2021-10-13 EP disclosed
CN-113498340-A Thienylaniline compounds for the treatment of skin diseases 恩福莱克逊治疗有限公司 2021-10-12 CN disclosed
US-11142682-B2 Metal oxide, metal bronze and polyoxometalate as charge storage materials in electrochromic device Furcifer Inc. (US) 2021-10-12 US disclosed
US-11142526-B2 Spirocycle compounds and methods of making and using same H. LUNDBECK A/S (DK) 2021-10-12 US disclosed
CN-108137639-B Nicotinamide mononucleotide derivative and application thereof 麦德龙国际生物科技有限责任公司 2021-10-08 CN disclosed
CN-113490663-A Pyridazine (thio) amides as fungicidal compounds 拜耳公司 2021-10-08 CN disclosed
CN-113476499-A Compositions and methods for weight management 尤妮金公司 2021-10-08 CN disclosed
WO-2021202540-A1 HSP70 INHIBITORS AND METHODS OF USING SAME THE WISTAR INSTITUTE (US) 2021-10-07 WO disclosed
WO-2021195716-A1 ANTIBIOTIC CONJUGATES MONASH UNIVERSITY (AU) 2021-10-07 WO disclosed
WO-2021202553-A1 CXCR5 ANTAGONISTS AND METHODS OF TREATING DISEASES OR DISORDERS USING SAME YALE UNIVERSITY (US) 2021-10-07 WO disclosed
WO-2021203131-A1 SUBSTITUTED PYRIMIDINES AND METHODS OF USE THERAVANCE BIOPHARMA R&D IP, LLC (US) 2021-10-07 WO disclosed
EP-3886844-A1 METHODS OF TREATING DISEASE WITH MAGL INHIBITORS H. Lundbeck A/S (DK) 2021-10-06 EP disclosed
EP-3887362-A1 PYRIDAZINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS Bayer Aktiengesellschaft (DE) 2021-10-06 EP disclosed
EP-3303317-B1 METHODS AND COMPOSITIONS FOR INHIBITING THE INTERACTION OF MENIN WITH MLL PROTEINS KURA ONCOLOGY INC (US) 2021-10-06 EP disclosed
EP-3179991-B1 THERAPEUTIC COMBINATIONS OF A BTK INHIBITOR AND A BCL-2 INHIBITOR ACERTA PHARMA BV (NL) 2021-10-06 EP disclosed
EP-3889237-A1 PHOTOACTIVE MACROMOLECULES AND USES THEREOF Beckman Coulter, Inc. (US) 2021-10-06 EP disclosed
EP-3887373-A1 COMPOUNDS AND METHODS OF USE THEREOF FOR TREATMENT OF CANCER Araxes Pharma LLC (US) 2021-10-06 EP disclosed
US-11136678-B2 Electrochemical oxidation of aliphatic and aromatic compounds MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2021-10-05 US disclosed
US-11136308-B2 Substituted quinazoline and quinazolinone compounds and methods of use thereof ARAXES PHARMA LLC (US) 2021-10-05 US disclosed
CN-108349936-B Compounds as muscarinic receptor 4 antagonists 纽罗克里生物科学有限公司 2021-10-01 CN disclosed
CN-107964016-B Thiophene derivatives 天津合美医药科技有限公司 2021-10-01 CN disclosed
CN-108530424-B Inhibitors of lysine-specific demethylase-1 赛尔基因昆蒂赛尔研究公司 2021-10-01 CN disclosed
CN-113474328-A Lipids for lipid nanoparticle delivery of active agents 爱康泰生治疗公司 2021-10-01 CN disclosed
CN-108059635-B Thiophene derivatives 天津合美医药科技有限公司 2021-10-01 CN disclosed
CN-113473986-A Nalidinone aniline compounds for the treatment of skin disorders 恩福莱克逊治疗有限公司 2021-10-01 CN disclosed
CN-113473860-A 1, 3, 4-oxadiazoles and derivatives thereof as novel antifungal agents 拜耳公司 2021-10-01 CN disclosed
CN-113473978-A Cyanoarene-aniline compounds for the treatment of skin diseases 恩福莱克逊治疗有限公司 2021-10-01 CN disclosed
CN-112300173-B Nitrogen-containing polycyclic compounds, preparation method and application 上海凌达生物医药有限公司 2021-10-01 CN disclosed
US-20210300904-A1 INHIBITORS OF RAF KINASES Pierre Fabre Médicament (FR) 2021-09-30 US disclosed
US-20210299109-A1 AGENTS FOR TREATING CANCER AND METHODS FOR IDENTIFYING SAID AGENTS MINERVA BIOTECHNOLOGIES CORPORATION 2021-09-30 US disclosed
WO-2021191197-A1 COMBINATION THERAPY COMPRISING AN AXL INHIBITOR BERGENBIO ASA (NO) 2021-09-30 WO disclosed
EP-3884935-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT Ardelyx, Inc. (US) 2021-09-29 EP disclosed
EP-3883646-A1 NLRP3 INHIBITORS Inflazome Limited (IE) 2021-09-29 EP disclosed
CN-113454079-A Heterocyclylpyridazines as fungicidal compounds 拜耳公司 2021-09-28 CN disclosed
US-11130748-B2 Compounds MISSION THERAPEUTICS LIMITED (GB) 2021-09-28 US disclosed
US-11129827-B2 Dual MAGL and FAAH inhibitors ABIDE THERAPEUTICS, INC. (US) 2021-09-28 US disclosed
US-11129828-B2 Pyridazinone compounds and their use as DAAO inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-09-28 US disclosed
US-11130827-B2 Polyethylene compositions and articles made therefrom EXXONMOBIL CHEMICAL PATENTS INC. (US) 2021-09-28 US disclosed
US-11130740-B2 Substituted 2,3-dihydro-1H-indene analogs and methods using same ARBUTUS BIOPHARMA CORPORATION (CA) 2021-09-28 US disclosed
US-11130782-B2 Nicotinic acetylcholine receptor peptide antagonist conotoxin compositions and related methods GLO PHARMA, INC. 2021-09-28 US disclosed
US-20210291156-A1 CATALYST COMPOSITIONS FOR HYDROFORMYLATION AND METHODS OF USE THEREOF NATIONAL SCIENCE FOUNDATION 2021-09-23 US disclosed
US-20210292718-A1 DIVERSE CARBENE TRANSFERASE ENZYME CATALYSTS DERIVED FROM A P450 ENZYME CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2021-09-23 US disclosed
US-20210292326-A1 Small-Molecule PI5P4K alpha/beta Inhibitors and Methods of Treatment Using Same UNIV YALE (US) 2021-09-23 US disclosed
US-20210292482-A1 NETWORK POLYMERS AND METHODS OF MAKING AND USING SAME THE REGENTS OF THE UNIV OF COLORADO A BODY CORPORTATE (US) 2021-09-23 US disclosed
US-20210292341-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2021-09-23 US disclosed
US-20210292330-A1 PYRROLIDINE-FUSED HETEROCYCLES ERASCA, INC. 2021-09-23 US disclosed
EP-3395818-B1 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES Bayer Pharma AG (DE) 2021-09-22 EP disclosed
US-11124537-B2 Inhibitors of glucocorticoid receptor ORIC PHARMACEUTICALS, INC. (US) 2021-09-21 US disclosed
US-11124601-B2 Electrochromic polymer and synthesis and uses thereof Furcifer Inc. (US) 2021-09-21 US disclosed
US-11123439-B2 Antibody drug conjugates (ADCS) and antibody prodrug conjugates (APDCS) with enzymatically cleavable groups BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-09-21 US disclosed
US-11123393-B2 Compositions and methods for joint health UNIGEN, INC. (US) 2021-09-21 US disclosed
US-11123352-B2 Testosterone ester triglyceride formulations ANTARES PHARMA, INC. (US) 2021-09-21 US disclosed
CN-112142735-B Condensed cyanopyridine compound, preparation method and application 上海凌达生物医药有限公司 2021-09-17 CN disclosed
WO-2021183970-A1 NON-ATP/CATALYTIC SITE P38 MITOGEN ACTIVATED PROTEIN KINASE INHIBITORS UNIVERSITY OF MARYLAND, BALTIMORE (US) 2021-09-16 WO disclosed
US-20210284972-A1 HOST CELLS AND METHODS USEFUL FOR PRODUCING UNNATURAL TERPENOIDS USING A NOVEL ARTIFICIAL METALLOENZYME UNITED STATES DEPARTMENT OF ENERGY 2021-09-16 US disclosed
US-20210283170-A1 METHODS AND COMPOUNDS FOR TREATMENT OF LYMPHOCYTE-RELATED DISEASES AND CONDITIONS SAREPTA THERAPEUTICS INC (US) 2021-09-16 US disclosed
US-20210284651-A1 Spiropiperidine Derivatives CEPHALON LLC 2021-09-16 US disclosed
US-20210284631-A1 CYANO-SUBSTITUTED HETEROCYCLES WITH ACTIVITY AS INHIBITORS OF USP30 MISSION THERAPEUTICS LIMITED (GB) 2021-09-16 US disclosed
EP-3877811-A1 CURABLE FORMULATION WITH HIGH REFRACTIVE INDEX AND ITS APPLICATION IN SURFACE RELIEF GRATING USING NANOIMPRINTING LITHOGRAPHY Facebook Technologies, LLC. (US) 2021-09-15 EP disclosed
EP-3877430-A1 POLYETHYLENE COMPOSITIONS AND ARTICLES MADE THEREFROM ExxonMobil Chemical Patents Inc. (US) 2021-09-15 EP disclosed
EP-3878853-A1 NITROGEN-CONTAINING FUSED HETEROCYCLIC SHP2 INHIBITOR COMPOUND, PREPARATION METHOD, AND USE Shanghai Ringene BioPharma Co., Ltd. (CN) 2021-09-15 EP disclosed
EP-3877356-A1 BICYCLIC COMPOUNDS Vivace Therapeutics, Inc. (US) 2021-09-15 EP disclosed
EP-3878850-A1 NOVEL BENZYLAMINO SUBSTITUTED QUINAZOLINES AND DERIVATIVES AS SOS1 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2021-09-15 EP disclosed
EP-3878854-A1 MACROCYCLIC TYROSINE KINASE INHIBITOR AND USES THEREOF Shandong Xuanzhu Pharma Co., Ltd. (CN) 2021-09-15 EP disclosed
CN-113395965-A USP19 inhibitors for treatment 阿尔麦克探索有限公司 2021-09-14 CN disclosed
CN-113396145-A PFKFB3 inhibitors and uses thereof 盖罗发现有限责任公司 2021-09-14 CN disclosed
CN-113395963-A non-ATP/catalytic site p38 mitogen-activated protein kinase inhibitors 马里兰大学巴尔的摩分校 2021-09-14 CN disclosed
US-11118179-B2 Mixed tricyclo-DNA, 2′-modified RNA oligonucleotide compositions and uses thereof SYNTHENA AG (CH) 2021-09-14 US disclosed
US-11116778-B2 Prodrugs of ALOX-15 inhibitors and methods of using the same EMPIRICO INC. (US) 2021-09-14 US disclosed
US-11118204-B2 Switchable ionic liquids for biomass pretreatment and enzymatic hydrolysis NATIONAL TECHNOLOGY & ENGINEERING SOLUTIONS OF SANDIA, LLC (US) 2021-09-14 US disclosed
US-11117878-B2 Benzothiazole and related compounds SPINOGENIX, INC. (US) 2021-09-14 US disclosed
US-11117915-B2 Antibacterial aminoglycoside analogs Cipla USA, Inc. (US) 2021-09-14 US disclosed
US-11118197-B2 High gravity, fed-batch ionic liquid based process for deconstructing biomass NATIONAL TECHNOLOGY & ENGINEERING SOLUTIONS OF SANDIA, LLC (US) 2021-09-14 US disclosed
WO-2021176045-A1 IMIDAZOTRIAZINES ACTING ON CANCER VIA INHIBITION OF CDK12 BAYER AKTIENGESELLSCHAFT (DE) 2021-09-10 WO disclosed
WO-2021176049-A1 PYRAZOLOPYRAZINES ACTING ON CANCERS VIA INHIBITION OF CDK12 BAYER AKTIENGESELLSCHAFT (DE) 2021-09-10 WO disclosed
WO-2021178684-A1 CAR AND NRF2 DUAL ACTIVATOR AGENTS FOR CYCLOPHOSPHAMIDE-BASED AND DOXORUBICIN-BASED TREATMENTS OF CANCER UNIVERSITY OF MARYLAND, BALTIMORE (US) 2021-09-10 WO disclosed
CN-113383272-A Curable formulations with high refractive index and their use in surface relief gratings using nanoimprint lithography 脸谱科技有限责任公司 2021-09-10 CN disclosed
CN-111592541-B Macrocyclic kinase inhibitors and uses thereof 山东轩竹医药科技有限公司 2021-09-10 CN disclosed
CN-113382736-A Compounds, compositions and methods for treating androgen mediated diseases 加利福尼亚大学董事会 2021-09-10 CN disclosed
CN-110229151-B Indolizine compound, preparation method and application thereof 上海海和药物研究开发股份有限公司 2021-09-10 CN disclosed
CN-108619141-B Antibacterial composition and application thereof 山东轩竹医药科技有限公司 2021-09-10 CN disclosed
US-20210277022-A1 MACROCYCLIC CHLORINE SUBSTITUTED INDOLE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-09-09 US disclosed
US-20210276974-A1 SUBSTITUTED 2-HETEROARYLOXYPYRIDINES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2021-09-09 US disclosed
EP-3874556-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH PHOSPHAZENE CONTAINING ELECTROLYTE ADDITIVES Enevate Corporation (US) 2021-09-08 EP disclosed
EP-3873479-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR TREATMENT OF ANDROGEN-MEDIATED DISEASE The Regents of the University of California (US) 2021-09-08 EP disclosed
CN-113365696-A Pharmaceutical compounds and their use as inhibitors of ubiquitin-specific protease 19(USP19) 阿尔麦克探索有限公司 2021-09-07 CN disclosed
CN-113354811-A Oxazoline polymer with side chain containing amino and/or hydroxyl, preparation method and application thereof 华东理工大学 2021-09-07 CN disclosed
US-11110103-B2 Inhibitors of glucocorticoid receptor ORIC PHARMACEUTICALS, INC. (US) 2021-09-07 US disclosed
US-11114660-B1 Silicon anodes with water-soluble maleic anhydride-, and/or maleic acid-containing polymers/copolymers, derivatives, and/or combinations (with or without additives) as binders ENEVATE CORPORATION (US) 2021-09-07 US disclosed
US-11111259-B2 Acylsulfonamide derivatives for treating senescence-associated diseases and disorders UNITY BIOTECHNOLOGY, INC. (US) 2021-09-07 US disclosed
US-11110177-B2 ASH1L degraders and methods of treatment therewith THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2021-09-07 US disclosed
US-11111352-B2 Methods of producing organosilica materials and uses thereof EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2021-09-07 US disclosed
US-11111325-B2 Polymerization processes EXXONMOBIL CHEMICAL PATENTS INC. (US) 2021-09-07 US disclosed
CN-108601769-B Pyrazole compounds and methods of making and using the same H.隆德贝克有限公司 2021-09-03 CN disclosed
CN-113348165-A 1,2, 4-triazin-3 (2H) -one compounds for the treatment of hyperproliferative diseases 拜耳股份有限公司 2021-09-03 CN disclosed
CN-113347971-A Methods of treating diseases with MAGL inhibitors H.隆德贝克有限公司 2021-09-03 CN disclosed
CN-113348181-A DC-SIGN antibody conjugates comprising a STING agonist 诺华股份有限公司 2021-09-03 CN disclosed
CN-108368028-B Novel lipid and lipid nanoparticle formulations for delivery of nucleic acids 爱康泰生治疗公司 2021-09-03 CN disclosed
CN-113330005-A Methods of treating diseases with MAGL inhibitors H.隆德贝克有限公司 2021-08-31 CN disclosed
CN-113318113-A Use of fibroblast growth factor receptor inhibitors 南京药捷安康生物科技有限公司 2021-08-31 CN disclosed
CN-113302187-A Substituted pyridyloxybenzenes and their salts and their use as herbicides 拜耳公司 2021-08-24 CN disclosed
CN-110372550-B Aryl ethers and their use 佩洛通治疗公司 2021-08-24 CN disclosed
CN-113302175-A Bicyclic compounds 维瓦斯治疗公司 2021-08-24 CN disclosed
CN-107281490-B Compositions and methods for weight management 尤妮金公司 2021-08-20 CN disclosed
US-20210253598-A1 ARYL ANNULATED MACROCYCLIC INDOLE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-08-19 US disclosed
US-20210253628-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR TREATMENT OF ANDROGEN-MEDIATED DISEASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-08-19 US disclosed
WO-2021161105-A1 P2X3 MODULATORS BELLUS HEALTH COUGH INC. (CA) 2021-08-19 WO disclosed
WO-2021160873-A1 NANOPARTICLES ENCAPSULATING SMALL MOLECULES ETH ZURICH (CH) 2021-08-19 WO disclosed
US-20210251991-A1 SUBSTITUTED 2,2'-BIPYRIMIDINYL COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2021-08-19 US disclosed
US-20210253595-A1 2-Aminopyrimidine Derivative and Preparation Method and Use Thereof ETERN BIOPHARMA (SHANGHAI) CO., LTD. (CN) 2021-08-19 US disclosed
US-20210253614-A1 COMPOSITIONS AND METHODS FOR INHIBITING CD73 PELOTON THERAPEUTICS, INC. (US) 2021-08-19 US disclosed
EP-3863640-A1 TREATMENT OF PRURITUS WITH P2X3 ANTAGONISTS Bellus Health Cough Inc. (CA) 2021-08-18 EP disclosed
EP-3515897-B1 PIPERAZINE CARBAMATES AS MODULATORS OF MAGL AND/OR ABHD6 AND THEIR USE H LUNDBECK AS (DK) 2021-08-18 EP disclosed
CN-113262175-A Skin care compositions and methods of use thereof 尤尼根公司 2021-08-17 CN disclosed
CN-110950876-B Furanolactam compounds, preparation method and application 上海凌达生物医药有限公司 2021-08-17 CN disclosed
US-11090302-B2 Methods of treating chronic lymphocytic leukemia and small lymphocytic leukemia using a BTK inhibitor ACERTA PHARMA B.V. (NL) 2021-08-17 US disclosed
US-11090309-B2 Anti-thrombotic agents and methods of use thereof TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2021-08-17 US disclosed
US-11091488-B2 1-cyano-pyrrolidine derivatives as inhibitors of USP30 MISSION THERAPEUTICS LIMITED (GB) 2021-08-17 US disclosed
US-11091473-B2 Compounds for pain treatment, compositions comprising same, and methods of using same ACADIA PHARMACEUTICALS INC. (US) 2021-08-17 US disclosed
CN-110964012-B Fused heterocyclic biaryl benzyl alcohol compound, preparation method and application 上海凌达生物医药有限公司 2021-08-13 CN disclosed
US-20210249689-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ELECTROLYTE CONTAINING CYANATE BASED COMPOUNDS ENEVATE CORPORATION 2021-08-12 US disclosed
US-20210244755-A1 METHODS FOR TREATING CANCERS BY PRODRUGS OF CLOFARABINE BoYen Therapeutics, Inc. (TW) 2021-08-12 US disclosed
US-20210246155-A1 Metallocene Synthesis Process EXXONMOBIL CHEMICAL PATENTS INC. 2021-08-12 US disclosed
US-20210246266-A1 HIGH DYNAMIC RANGE TWO-STAGE PHOTOPOLYMERS NATIONAL SCIENCE FOUNDATION 2021-08-12 US disclosed
US-20210246135-A1 INHIBITORS OF RAF KINASES Pierre Fabre Médicament (FR) 2021-08-12 US disclosed
US-20210246614-A1 WATER RESISTANT MATERIALS FOR FOOD-SAFE USES JL DARLING LLC (US) 2021-08-12 US disclosed
WO-2021158366-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ELECTROLYTE CONTAINING CYANATE BASED COMPOUNDS ENEVATE CORPORATION (US) 2021-08-12 WO disclosed
WO-2021158481-A1 SUBSTITUTED 1,1'-BIPHENYL COMPOUNDS AND METHODS USING SAME ARBUTUS BIOPHARMA, INC. (US) 2021-08-12 WO disclosed
US-11084825-B2 Substituted pyridines as irreversible inhibitors of menin-MLL interaction BIOMEA FUSION, LLC (US) 2021-08-10 US disclosed
US-11084793-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2021-08-10 US disclosed
US-11084932-B2 Phenylethynylnaphthalene dyes and methods for their use Sony Group Corporation (JP) 2021-08-10 US disclosed
US-11084821-B2 Cyanopyrrolidine derivatives with activity as inhibitors of USP30 MISSION THERAPEUTICS LIMITED (GB) 2021-08-10 US disclosed
US-11087900-B2 Polymer-silica hybrid Pdots and methods of use thereof UNIVERSITY OF WASHINGTON (US) 2021-08-10 US disclosed
CN-113226321-A Pyrazolyl compounds and methods of use thereof 阿利安制药有限责任公司 2021-08-06 CN disclosed
CN-113227092-A Compounds and methods of use thereof for treating cancer 亚瑞克西斯制药公司 2021-08-06 CN disclosed
US-20210238154-A1 OXADIAZOLE COMPOUNDS VIVACE THERAPEUTICS, INC. 2021-08-05 US disclosed
US-20210238196-A1 SPIRO AROMATIC RING COMPOUND AND APPLICATION THEREOF ETERN BIOPHARMA (SHANGHAI) CO., LTD. (CN) 2021-08-05 US disclosed
US-20210238221-A1 TRIPTOLIDE DERIVATIVE AND PREPARATION METHOD THEREFOR AND USE THEREOF CINKATE PHARMACEUTICAL INTERMEDIATES CO., LTD. (CN) 2021-08-05 US disclosed
US-20210238161-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2021-08-05 US disclosed
WO-2021151976-A1 [(1,4,5-TRISUBSTITUTED-1H-PYRAZOL-3-YL)SULFANYL]ACETIC ACID DERIVATIVES, SALTS THEREOF, AND USE THEREOF AS HERBICIDAL INGREDIENTS BAYER AKTIENGESELLSCHAFT (DE) 2021-08-05 WO disclosed
WO-2021152390-A1 COMPOSITIONS FOR THE TREATMENT OF ANGIOLIPOMA RAZIEL THERAPEUTICS LTD. (IL) 2021-08-05 WO disclosed
WO-2021155253-A1 ANAT INHIBITORS AND METHODS OF USE THEREOF Atomwise Inc. (US) 2021-08-05 WO disclosed
WO-2021152481-A1 HYBRID POLYETHER ETHER KETONE POLYMERS KING ABDULLAH UNIVERSITY OF SCIENCE AND TECHNOLOGY (SA) 2021-08-05 WO disclosed
WO-2021154966-A1 COMPOUNDS AND COMPOSITIONS FOR USE IN TREATING SKIN DISORDERS KAMARI PHARMA LTD. (IL) 2021-08-05 WO disclosed
WO-2021155062-A1 WATER RESISTANT MATERIALS FOR FOOD-SAFE USES JL DARLING LLC (US) 2021-08-05 WO disclosed
EP-2972258-B1 PURIFICATION OF RAPAMYCIN DERIVATIVES BIOSENSORS INT GROUP LTD (BM) 2021-08-04 EP disclosed
EP-3858813-A1 QUINOLONE DERIVATIVE HAVING INDOLEAMINE-2,3-DIOXYGENASE INHIBITED ACTIVITY Shenzhen Chipscreen Biosciences Co., Ltd. (CN) 2021-08-04 EP disclosed
CN-113207291-A 2- (2-acryloyl-2, 6-diazaspiro [3.4] oct-6-yl) -6- (1H-indazol-4-yl) benzonitrile derivatives and related compounds as inhibitors of G12C mutant KRAS protein for inhibiting tumor metastasis 亚瑞克西斯制药公司 2021-08-03 CN disclosed
US-11077107-B2 Triazolopyrazine BOEHRINGER INGELHEIM INTERNATIONAL GMBH 2021-08-03 US disclosed
US-11078171-B2 Non-ATP/catalytic site p38 mitogen activated protein kinase inhibitors UNIVERSITY OF MARYLAND, BALTIMORE (US) 2021-08-03 US disclosed
US-11078162-B2 Processes for preparing AG-10, its intermediates, and salts thereof Eidos Therapeutics, Inc. (US) 2021-08-03 US disclosed
CN-113194977-A Nicotinamide acetylcholine receptor peptide antagonist conotoxin compositions and related methods 格罗制药公司 2021-07-30 CN disclosed
CN-113185740-A Method for improving antibacterial activity and biocompatibility of substrate surface 华东理工大学 2021-07-30 CN disclosed
CN-108778270-B Antibacterial composition and application thereof 吉林四环制药有限公司 2021-07-30 CN disclosed
CN-113195492-A Novel compound with three-fused ring structure, preparation method and application thereof 信达生物制药(苏州)有限公司 2021-07-30 CN disclosed
US-20210230116-A1 1,4-Substituted Piperidine Derivatives CEPHALON LLC 2021-07-29 US disclosed
US-20210228563-A1 METHODS OF TREATING RBP4 RELATED DISEASES WITH TRIAZOLOPYRIDINES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2021-07-29 US disclosed
US-20210230157-A1 PAIN TREATING COMPOUNDS AND USES THEREOF BIONOMICS LIMITED (AU) 2021-07-29 US disclosed
US-20210228565-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC. (US) 2021-07-29 US disclosed
US-20210230165-A1 MODULATORS OF ION CHANNEL RECEPTORS AND USES THEREOF BIONOMICS LIMITED (AU) 2021-07-29 US disclosed
EP-3853590-A1 NARROW ABSORPTION POLYMER NANOPARTICLES AND RELATED METHODS University of Washington (US) 2021-07-28 EP disclosed
EP-3852911-A2 SYSTEMS AND METHODS FOR MANUFACTURING LIPID NANOPARTICLES AND LIPOSOMES Acuitas Therapeutics, Inc. (CA) 2021-07-28 EP disclosed
EP-3052485-B1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS INC (US) 2021-07-28 EP disclosed
EP-3852766-A1 COMBINATION THERAPY FOR TREATING BLOOD CANCER SignalChem Lifesciences Corporation (CA) 2021-07-28 EP disclosed
EP-3853210-A1 ANTIBACTERIAL COMPOUNDS Forge Therapeutics, Inc. (US) 2021-07-28 EP disclosed
US-11075408-B2 Silicon-based energy storage devices with fluorinated polymer containing electrolyte additives ENEVATE CORPORATION (US) 2021-07-27 US disclosed
US-11071788-B2 Antibody drug conjugates of kinesin spindel protein (KSP) inhibitors with antiB7H3-antibodies BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-07-27 US disclosed
US-11072793-B2 DsRNA molecules comprising oligonucleotide analogs having modified intersubunit linkages and/or terminal groups SAREPTA THERAPEUTICS, INC. (US) 2021-07-27 US disclosed
US-11071771-B2 Butyrylcholinesterase zwitterionic polymer conjugates KODIAK SCIENCES INC. (US) 2021-07-27 US disclosed
US-11071749-B2 Oligonucleotide analogues targeting human LMNA SAREPTA THERAPEUTICS, INC. (US) 2021-07-27 US disclosed
CN-113166155-A Macrocyclic tyrosine kinase inhibitors and uses thereof 山东轩竹医药科技有限公司 2021-07-23 CN disclosed
CN-113164490-A Treatment of pruritis with P2X3 antagonists 贝卢斯医疗咳嗽病公司 2021-07-23 CN disclosed
CN-113166077-A Antibacterial compounds 福至治疗公司 2021-07-23 CN disclosed
CN-113149941-A Ether compound and pharmaceutical application thereof in preventing and treating diabetes and metabolic syndrome 中国科学院上海药物研究所 2021-07-23 CN disclosed
CN-113164381-A Pharmaceutical compositions and methods relating to otic therapeutic agents 频率医疗公司 2021-07-23 CN disclosed
CN-113164763-A NLRP3 inhibitor 英夫拉索姆有限公司 2021-07-23 CN disclosed
WO-2021144162-A1 PROCESS FOR PREPARING CYCLIC CARBONATES WITH AN EXOCYCLIC VINYLIDENE GROUP BASF SE (DE) 2021-07-22 WO disclosed
US-20210221835-A1 CARBON-MONOXIDE-RELEASING MOLECULES AND THERAPEUTIC APPLICATIONS THEREOF GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2021-07-22 US disclosed
US-20210221781-A1 FATTY ACID ANALOGUES AND METHODS OF USE LIN BIOSCIENCE INC. (TW) 2021-07-22 US disclosed
US-20210226251-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ELECTROLYTE CONTAINING CROWN ETHER BASED COMPOUNDS ENEVATE CORPORATION 2021-07-22 US disclosed
US-20210221796-A1 ANTIBACTERIAL COMPOUNDS BLACKSMITH MEDICINES, INC. 2021-07-22 US disclosed
US-20210222257-A1 BIOMARKERS OF RESPONSE TO HIF-2-ALPHA INHIBITION IN CANCER AND METHODS FOR THE USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2021-07-22 US disclosed
US-20210221790-A1 ABHD12 INHIBITORS AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2021-07-22 US disclosed
US-20210221813-A1 4,6 DIHYDROPYRROLO [3,4-C] PYRAZOLE-5 (1H)-CARBONITRILE DERIVATES FOR TREATING CANCER MISSION THERAPEUTICS LIMITED (AE) 2021-07-22 US disclosed
EP-3851444-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR Oric Pharmaceuticals, Inc. (US) 2021-07-21 EP disclosed
EP-3851469-A1 POLYURETHANE/UREA MATERIALS Commonwealth Scientific and Industrial Research Organisation (AU) 2021-07-21 EP disclosed
EP-3849990-A2 MOF COMPOSITIONS FOR SELECTIVE SEPARATION OF HYDROCARBONS Rutgers, The State University of New Jersey (US) 2021-07-21 EP disclosed
US-11066513-B2 Multicolored electrochromic polymer compositions and methods of making and using the same Furcifer Inc. (US) 2021-07-20 US disclosed
US-11066465-B2 Antibodies and conjugates thereof KODIAK SCIENCES INC. (US) 2021-07-20 US disclosed
US-11066365-B2 1-cyano-pyrrolidine compounds as USP30 inhibitors MISSION THERAPEUTICS LIMITED (GB) 2021-07-20 US disclosed
US-20210218059-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH CARBOXYLIC ETHER, CARBOXYLIC ACID BASED SALT, OR ACRYLATE ELECTROLYTE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2021-07-15 US disclosed
US-20210214375-A1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2021-07-15 US disclosed
EP-3277677-B9 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS MISSION THERAPEUTICS LTD (GB) 2021-07-14 EP disclosed
EP-3846806-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS Pipeline Therapeutics, Inc. (US) 2021-07-14 EP disclosed
US-11059819-B2 Fused hetero-hetero bicyclic compounds and methods of use thereof JANSSEN BIOTECH, INC. (US) 2021-07-13 US disclosed
US-11059805-B2 Alkynyl-substituted heterocyclic compound, preparation method therefor and medical use thereof BEIJING INNOCARE PHARMA TECH CO., LTD. (CN) 2021-07-13 US disclosed
US-11059822-B2 MAGL inhibitors H. LUNDBECK A/S (DK) 2021-07-13 US disclosed
WO-2021138215-A1 TREATMENT OF CANCER WITH CDK12/13 INHIBITORS KINNATE BIOPHARMA INC. (US) 2021-07-08 WO disclosed
US-20210206735-A1 MAGL INHIBITORS LUNDBECK LA JOLLA RESEARCH CENTER, INC. (US) 2021-07-08 US disclosed
US-20210205284-A1 THERAPEUTIC COMPOUNDS CELGENE QUANTICEL RESEARCH, INC. (US) 2021-07-08 US disclosed
US-20210205762-A1 CURABLE POLY(RTIL)-BASED MIXED-MATRIX MEMBRANES AND METHODS USING SAME THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2021-07-08 US disclosed
US-20210205304-A1 AXL KINASE INHIBITORS AND USE OF THE SAME SUMITOMO DAINIPPON PHARMA ONCOLOGY, INC. (US) 2021-07-08 US disclosed
US-20210205291-A1 NITROGENOUS HETEROCYCLIC AMIDE DERIVATIVE, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL APPLICATION SICHUAN HAISCO PHARMACEUTICAL CO., LTD. (CN) 2021-07-08 US disclosed
EP-3844158-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS SODIUM CHANNEL INHIBITORS Xenon Pharmaceuticals Inc. (CA) 2021-07-07 EP disclosed
EP-3844150-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2021-07-07 EP disclosed
CN-106794362-B Carbon monoxide-releasing molecules for therapeutic applications and methods of making and using the same 乔治亚州立大学研究基金会股份有限公司 2021-07-06 CN disclosed
US-11053237-B2 Process for the manufacture of 6-alkynyl-pyridine derivatives BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-07-06 US disclosed
US-11053213-B2 Pharmaceutical compounds ALMAC DISCOVERY LIMITED (GB) 2021-07-06 US disclosed
US-11053242-B2 [9,10-dimethoxy-3-(2-methylpropyl)-1H,2H,3H,4H,6H,7H,11BH-pyrido-[2,1-a]isoquinolin-2-yl]methanol and compounds, compositions and methods relating thereto NEUROCRINE BIOSCIENCES, INC. (US) 2021-07-06 US disclosed
US-11053221-B2 Substituted pyrimidines for inhibiting embryonic leucine zipper kinase activity ARRIEN PHARMACEUTICALS LLC (US) 2021-07-06 US disclosed
US-11053342-B2 Polyurethane/urea materials COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2021-07-06 US disclosed
CN-108368089-B Deubiquitinase inhibitor 特殊治疗有限公司 2021-07-06 CN disclosed
US-11053198-B2 1-cyano-pyrrolidine compounds as USP30 inhibitors MISSION THERAPEUTICS LIMITED (GB) 2021-07-06 US disclosed
CN-113061132-A Condensed ring lactam compound, preparation method and application 上海凌达生物医药有限公司 2021-07-02 CN disclosed
US-20210198708-A1 CONVERSION OF SUGARS TO IONIC LIQUIDS UNITED STATES DEPARTMENT OF ENERGY 2021-07-01 US disclosed
WO-2021130638-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS CARNA BIOSCIENCES, INC. (JP) 2021-07-01 WO disclosed
US-20210198288-A1 PENICILLIN-BINDING PROTEIN INHIBITORS VenatoRx Pharmaceuticals, Inc. 2021-07-01 US disclosed
EP-3842427-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS Mission Therapeutics Limited (GB) 2021-06-30 EP disclosed
US-11046682-B2 Fused heterocyclic derivatives, their preparation methods thereof and medical uses thereof BEIJING INNOCARE PHARMA TECH CO., LTD. (CN) 2021-06-29 US disclosed
US-11046711-B2 Purification of rapamycin derivatives using temperature induced phase separation BIOSENSORS INTERNATIONAL GROUP, LTD. (BM) 2021-06-29 US disclosed
US-11046707-B2 Spiropiperidine derivatives 89BIO LTD (IL) 2021-06-29 US disclosed
US-11046679-B2 Indoleamine 2,3-dioxygenase inhibitor and application NANJING TRANSTHERA BIOSCIENCES CO. LTD. (CN) 2021-06-29 US disclosed
US-20210188869-A1 INHIBITORS OF KRAS G12C ARAXES PHARMA LLC 2021-06-24 US disclosed
US-20210186953-A1 NHE3-BINDING COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. (US) 2021-06-24 US disclosed
US-20210186943-A1 OTIC FORMULATIONS FOR DRUG-INDUCED OTOTOXICITY SPIRAL THERAPEUTICS INC. 2021-06-24 US disclosed
WO-2021127404-A1 TRICYCLIC PYRIDONES AND PYRIMIDONES ERASCA, INC. (US) 2021-06-24 WO disclosed
WO-2021127356-A1 Substituted Bicyclic and Tricyclic Ureas and Amides, Analogues Thereof, and Methods Using Same ARBUTUS BIOPHARMA, INC. (US) 2021-06-24 WO disclosed
WO-2021122728-A1 1,5-DIPHENYLPYRAZOLYL-3-OXYALKYL ACIDS AND 1-PHENYL-5-THIENYLPYRAZOLYL-3-OXYALKYL ACIDS AND THE USE THEREOF FOR CONTROL OF UNDESIRED PLANT GROWTH BAYER AKTIENGESELLSCHAFT (DE) 2021-06-24 WO disclosed
WO-2021126341-A1 METHODS OF TREATING VASCULAR LESIONS AND MALFORMATIONS Blaze Bioscience, Inc. (US) 2021-06-24 WO disclosed
WO-2021123074-A1 METHODS OF SEQUENCING BY SYNTHESIS USING A CONSECUTIVE LABELING SCHEME F. HOFFMANN-LA ROCHE AG (CH) 2021-06-24 WO disclosed
US-20210194056-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ELECTROLYTE CONTAINING SULFONATE OR CARBOXYLATE SALT BASED COMPOUNDS ENEVATE CORPORATION 2021-06-24 US disclosed
EP-3837242-A1 NOVEL SULFONEUREA COMPOUNDS Inflazome Limited (IE) 2021-06-23 EP disclosed
EP-3256484-B1 NON-MEMBRANE DISRUPTIVE P53 ACTIVATING STAPLED PEPTIDES AGENCY SCIENCE TECH & RES (SG) 2021-06-23 EP disclosed
EP-3836917-A1 NOVEL SULFONAMIDEUREA COMPOUNDS Inflazome Limited (IE) 2021-06-23 EP disclosed
EP-3837243-A1 NOVEL SULFONEUREA COMPOUNDS Inflazome Limited (IE) 2021-06-23 EP disclosed
EP-3837301-A1 POLYMER COMPOSITION BASF SE (DE) 2021-06-23 EP disclosed
US-11040038-B2 Methods for treating diseases associated with abnormal ACVR1 expression and ACVR1 inhibitors for use in the same SUMITOMO DAINIPPON PHARMA ONCOLOGY, INC. (US) 2021-06-22 US disclosed
US-11040970-B2 VMAT2 inhibitor compounds and compositions thereof NEUROCRINE BIOSCIENCES, INC. (US) 2021-06-22 US disclosed
US-11040945-B2 Tubulin inhibitors LIN BIOSCIENCE PTY LTD. 2021-06-22 US disclosed
US-11040112-B2 Lipids and lipid nanoparticle formulations for delivery of nucleic acids Acuitas Therapeutics, Inc. (CA) 2021-06-22 US disclosed
CN-113004788-A Surface finishing composition 3M中国有限公司 2021-06-22 CN disclosed
CN-112996518-A WD40 repeat domain protein 5(WDR5) degradation/disruption compounds and methods of use 西奈山伊坎医学院 2021-06-18 CN disclosed
WO-2021119554-A1 COMPOSITIONS AND METHODS FOR POTENTIATING IMMUNE ACTIVITY KUMQUAT BIOSCIENCES INC. (US) 2021-06-17 WO disclosed
WO-2021113922-A1 IMPROVED METHOD FOR PREPARING N-(BENZENESULFONYL)-L-PROLYL- L-O-(1-PYRROLIDINYLCARBONYL)TYROSINE COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2021-06-17 WO disclosed
US-20210179524-A1 ANTIMALARIAL COMPOSITIONS AND USES THEREOF SCRIPPS RESEARCH INST (US) 2021-06-17 US disclosed
US-20210179616-A1 AZABICYCLO AND DIAZEPINE DERIVATIVES ALCON INC. (CH) 2021-06-17 US disclosed
US-20210179612-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION 2021-06-17 US disclosed
US-20210177851-A1 NOVEL BENZYLAMINO SUBSTITUTED QUINAZOLINES AND DERIVATIVES AS SOS1 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2021-06-17 US disclosed
US-20210179557-A1 SUBSTITUTED TETRAHYDROCYCLOPENTA[C]PYRROLES, SUBSTITUTED DIHYDROPYRROLIZINES, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2021-06-17 US disclosed
US-20210184258-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ELECTROLYTE CONTAINING DIHYDROFURANONE BASED COMPOUND ENEVATE CORPORATION 2021-06-17 US disclosed
EP-3833353-A1 SMALL-MOLECULE PI5P4K ALPHA/BETA INHIBITORS AND METHODS OF TREATMENT USING SAME Yale University (US) 2021-06-16 EP disclosed
EP-3833348-A1 TRANSGLUTAMINASE 2 (TG2) INHIBITORS SITARI PHARMA, INC (US) 2021-06-16 EP disclosed
EP-3430012-B1 4,6-DIHYDROPYRROLO[3,4-C]PYRAZOLE-5(1H)-CARBONITRILE DERIVATIVES FOR TREATING CANCER MISSION THERAPEUTICS LTD (GB) 2021-06-16 EP disclosed
EP-3429994-B1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER MISSION THERAPEUTICS LTD (GB) 2021-06-16 EP disclosed
CN-107973741-B Synthesis method of 1H-pyrrole-2, 5-diketone derivative 重庆文理学院 2021-06-15 CN disclosed
CN-112969472-A Methods and compositions for ocular cell therapy 诺华股份有限公司 2021-06-15 CN disclosed
CN-112970141-A Silicon-based energy storage device with electrolyte additive containing phosphazene 新强能电池公司 2021-06-15 CN disclosed
US-11034719-B2 7-dehydrocholesterol derivatives and methods using same UNIVERSITY OF ROCHESTER (US) 2021-06-15 US disclosed
US-11034686-B2 Aminopyridine derivatives as TAM family kinase inhibitors SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2021-06-15 US disclosed
US-11034667-B2 Selective histone deacetylase inhibitors for the treatment of human disease SHUTTLE PHARMACEUTICALS, INC. (US) 2021-06-15 US disclosed
US-11033539-B2 Compounds of formulas (VII), (VIII), (IX), (XI), (XII), (XIII), and (XIV) as muscarinic receptor 4(M4) antagonists for treating neurological diseases NEUROCRINE BIOSCIENCES, INC. (US) 2021-06-15 US disclosed
US-11034685-B2 Aminopyridine derivatives as TAM family kinase inhibitors SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2021-06-15 US disclosed
CN-112939982-A Alkyne heterocyclic BTK inhibitor and preparation method and application thereof 药雅科技(上海)有限公司 2021-06-11 CN disclosed
US-20210172957-A1 METHODS AND SYSTEMS FOR ANALYSIS USING POLYMER DOTS UNIVERSITY OF WASHINGTON (US) 2021-06-10 US disclosed
US-20210171435-A1 Methods for the Treatment of Diabetic Retinopathy and other Ophthalmic Diseases ACUCELA INC. 2021-06-10 US disclosed
WO-2021113682-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION (US) 2021-06-10 WO disclosed
US-20210171531-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION 2021-06-10 US disclosed
US-20210170043-A1 DC-SIGN ANTIBODY CONJUGATES COMPRISING STING AGONISTS CHINOOK THERAPEUTICS, INC. 2021-06-10 US disclosed
WO-2021113686-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION (US) 2021-06-10 WO disclosed
WO-2021113690-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION (US) 2021-06-10 WO disclosed
WO-2021113698-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION (US) 2021-06-10 WO disclosed
US-20210171512-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION 2021-06-10 US disclosed
US-20210171537-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2021-06-10 US disclosed
US-20210171461-A1 MASP-2 INHIBITORS AND METHODS OF USE OMEROS CORPORATION 2021-06-10 US disclosed
EP-3351248-B1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX INC (US) 2021-06-09 EP disclosed
EP-3829580-A1 HETEROCYCLIC SPIRO COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF CANCER Araxes Pharma LLC (US) 2021-06-09 EP disclosed
EP-3829570-A1 SUBSTITUTED TETRAHYDROCYCLOPENTA[C]PYRROLES, SUBSTITUTED DIHYDROPYRROLIZINES, ANALOGUES THEREOF, AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2021-06-09 EP disclosed
EP-3831383-A1 BROMODOMAIN INHIBITORS Celgene Quanticel Research, Inc. (US) 2021-06-09 EP disclosed
US-11028066-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2021-06-08 US disclosed
CN-111171049-B Tyrosine kinase inhibitors and uses thereof 山东轩竹医药科技有限公司 2021-06-04 CN disclosed
US-20210163480-A1 TRANSGLUTAMINASE 2 (TG2) INHIBITORS SITARI PHARMA, INC. 2021-06-03 US disclosed
WO-2021108023-A1 PENICILLIN-BINDING PROTEIN INHIBITORS VenatoRx Pharmaceuticals, Inc. (US) 2021-06-03 WO disclosed
WO-2021108282-A1 AROMATIC SUBSTITUTED METHANE-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS FACEBOOK TECHNOLOGIES, LLC (US) 2021-06-03 WO disclosed
WO-2021108204-A1 AROMATIC SUBSTITUTED ETHANE-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS FACEBOOK TECHNOLOGIES, LLC (US) 2021-06-03 WO disclosed
WO-2021108232-A1 ANTHRAQUINONE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS FACEBOOK TECHNOLOGIES, LLC (US) 2021-06-03 WO disclosed
WO-2021108191-A1 AROMATIC SUBSTITUTED ALKANE-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS FACEBOOK TECHNOLOGIES, LLC (US) 2021-06-03 WO disclosed
WO-2021105115-A1 SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION BAYER AKTIENGESELLSCHAFT (DE) 2021-06-03 WO disclosed
WO-2021105101-A1 [(1,5-DIPHENYL-1H-1,2,4-TRIAZOL-3-YL)OXY]ACETIC ACID DERIVATIVES AND SALTS THEREOF, CROP PROTECTION COMPOSITIONS COMPRISING THEM, METHODS FOR PRODUCING THEM AND USE THEREOF AS SAFENERS BAYER AKTIENGESELLSCHAFT (DE) 2021-06-03 WO disclosed
WO-2021105117-A1 SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION BAYER AKTIENGESELLSCHAFT (DE) 2021-06-03 WO disclosed
WO-2021105116-A1 SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION BAYER AKTIENGESELLSCHAFT (DE) 2021-06-03 WO disclosed
WO-2021108597-A1 THIOPHOSPHATE AND PHOSPHINE SULFIDE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS FACEBOOK TECHNOLOGIES, LLC (US) 2021-06-03 WO disclosed
US-20210161889-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CONTINEUM THERAPEUTICS, INC. 2021-06-03 US disclosed
US-20210167361-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ANHYDRIDE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2021-06-03 US disclosed
US-20210161837-A1 METHODS FOR TREATING CANCER WITH RORGAMMA INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-06-03 US disclosed
US-20210163412-A1 NOVEL SULFONEUREA COMPOUNDS INFLAZOME LIMITED (IE) 2021-06-03 US disclosed
US-20210162406-A1 MODIFICATION OF SURFACE PROPERTIES OF MICROFLUIDIC DEVICES BIO RAD LABORATORIES (US) 2021-06-03 US disclosed
US-20210167423-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ELECTROLYTE CONTAINING A BENZOYL PEROXIDE BASED COMPOUND ENEVATE CORPORATION 2021-06-03 US disclosed
EP-3826684-A1 METHODS FOR TREATING DISEASES ASSOCIATED WITH ABNORMAL ACVR1 EXPRESSION AND ACVR1 INHIBITORS FOR USE IN THE SAME Sumitomo Dainippon Pharma Oncology, Inc. (US) 2021-06-02 EP disclosed
EP-3828179-A1 CYANOPYRROLIDINES AS DUB MODULATORS Mission Therapeutics Limited (GB) 2021-06-02 EP disclosed
CN-112888675-A Novel sulfonylurea compound 英夫拉索姆有限公司 2021-06-01 CN disclosed
CN-111690031-B Glucocorticoid receptor inhibitors 欧瑞克制药公司 2021-06-01 CN disclosed
CN-112888681-A Tropomyosin Receptor Kinase (TRK) degrading compounds and methods of use 上海睿跃生物科技有限公司 2021-06-01 CN disclosed
CN-112868659-A Composition applicable to user equipment and application thereof 3M中国有限公司 2021-06-01 CN disclosed
US-11020417-B2 Methods and compounds for treatment of lymphocyte-related diseases and conditions SAREPTA THERAPEUTICS, INC (US) 2021-06-01 US disclosed
US-11021463-B2 Therapeutic inhibitory compounds ATTUNE PHARMACEUTICALS, INC. (US) 2021-06-01 US disclosed
US-11021470-B2 2-substituted quinazoline compounds comprising a substituted heterocyclic group and methods of use thereof ARAXES PHARMA LLC (US) 2021-06-01 US disclosed
US-11021510-B2 Prodrugs of clofarabine BoYen Therapeutics, Inc. (TW) 2021-06-01 US disclosed
US-11021471-B2 Antibacterial compounds FORGE THERAPEUTICS, INC. (US) 2021-06-01 US disclosed
US-11020380-B2 Therapeutic compounds CELGENE QUANTICEL RESEARCH, INC. (US) 2021-06-01 US disclosed
US-11020731-B2 Catalysts for selective coupling of olefins, and methods of making and using same RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2021-06-01 US disclosed
CN-112851587-A Alkyne heterocyclic compound for treating cancer and preparation method and application thereof 药雅科技(上海)有限公司 2021-05-28 CN disclosed
WO-2021099842-A1 PENTAFLUOROBENZENESULFONAMIDE DERIVATIVES AND USES THEREOF 2692372 ONTARIO INC. (CA) 2021-05-27 WO disclosed
WO-2021102204-A1 HETEROARYL COMPOUNDS VIVACE THERAPEUTICS, INC. (US) 2021-05-27 WO disclosed
WO-2021101903-A1 DUAL ANDROGEN RECEPTOR/AKR1C3 INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-05-27 WO disclosed
WO-2021102468-A1 SUBSTITUTED 1,5-NAPHTHYRIDINES OR QUINOLINES AS ALK5 INHIBITORS THERAVANCE BIOPHARMA R&D IP, LLC (US) 2021-05-27 WO disclosed
US-20210155615-A1 INDENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION AQUINOX PHARMACEUTICALS (CANADA) INC. (CA) 2021-05-27 US disclosed
US-20210155639-A1 THIOPHOSPHATE AND PHOSPHINE SULFIDE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2021-05-27 US disclosed
US-20210155581-A1 AROMATIC SUBSTITUTED ETHANE-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2021-05-27 US disclosed
US-20210155599-A1 AROMATIC SUBSTITUTED ALKANE-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2021-05-27 US disclosed
US-20210154179-A1 SUBSTITUTED PYRIDINES AND METHODS OF USE THERAVANCE BIOPHARMA R&D IP, LLC (US) 2021-05-27 US disclosed
US-20210155964-A1 AMMONIUM BASED IONIC LIQUIDS USEFUL FOR LIGNOCELLULOSIC PROCESSING UNITED STATES DEPARTMENT OF ENERGY 2021-05-27 US disclosed
US-20210155590-A1 ISOINDOLE DERIVATIVE TIANJIN HEMAY PHARMACEUTICAL CO., LTD. (CN) 2021-05-27 US disclosed
US-20210155584-A1 AROMATIC SUBSTITUTED METHANE-CORE MONOMERS AND POLYMERS THEREOF FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2021-05-27 US disclosed
US-20210155601-A1 INHIBITORS FOR SOLUBLE EPOXIDE HYDROLASE (SEH) AND FATTY ACID AMIDE HYDROLASE (FAAH) THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2021-05-27 US disclosed
US-20210155585-A1 ANTHRAQUINONE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2021-05-27 US disclosed
US-20210155629-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS CONTINEUM THERAPEUTICS, INC. 2021-05-27 US disclosed
EP-3823465-A2 COMPOUNDS, COMPOSITIONS, AND METHODS FOR COLORING EDIBLE MATERIALS Ziegler, Gregory Ray (US) 2021-05-26 EP disclosed
CN-108290861-B 1-cyano-pyrrolidine derivatives as USP30 inhibitors 特殊治疗有限公司 2021-05-25 CN disclosed
US-11014960-B2 Amino acid and peptide conjugates and uses thereof AUCKLAND UNISERVICES LIMITED (NZ) 2021-05-25 US disclosed
US-11015002-B2 Polymerization processes EXXONMOBIL CHEMICAL PATENTS INC. (US) 2021-05-25 US disclosed
US-11013726-B2 Substituted pyridinone-containing trycyclic compounds, and methods using same ARBUTUS BIOPHARMA CORPORATION (CA) 2021-05-25 US disclosed
US-11014912-B2 Cyanopyrrolidine derivatives with activity as inhibitors of USP30 MISSION THERAPEUTICS LIMITED (GB) 2021-05-25 US disclosed
US-11013741-B1 AXL kinase inhibitors and use of the same SUMITOMO DAINIPPON PHARMA ONCOLOGY, INC. (US) 2021-05-25 US disclosed
US-20210147371-A1 OXADIAZOLINE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2021-05-20 US disclosed
US-20210147349-A1 PHENYLSULFONYLUREA DERIVATIVES USEFUL AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2021-05-20 US disclosed
WO-2021097075-A1 SUBSTITUTED ISOINDOLONYL 2,2'-BIPYRIMIDINYL COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA, INC. (US) 2021-05-20 WO disclosed
EP-3519397-B1 CYANO-SUBTITUTED HETEROCYCLES WITH ACTIVITY AS INHIBITORS OF USP30 MISSION THERAPEUTICS LTD (GB) 2021-05-19 EP disclosed
EP-3380536-B1 A POLYMERIC COMPOSITION AGENCY SCIENCE TECH & RES (SG) 2021-05-19 EP disclosed
US-11008596-B2 Cytochrome P450 BM3 enzyme variants for preparation of cyclopropanes CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2021-05-18 US disclosed
US-11007245-B2 Botulinum neurotoxin-specific capture agents, compositions, and methods of using and making INDI MOLECULAR, INC. (US) 2021-05-18 US disclosed
US-11007274-B2 Compounds for medicinal applications AusVir Therapeutics Pty Ltd (AU) 2021-05-18 US disclosed
US-11007186-B2 Methods of treating RBP4 related diseases with triazolopyridines BELITE BIO, INC (KY) 2021-05-18 US disclosed
US-11008297-B2 Bio-based, multi-aromatic compounds, and methods of making and using same ROWAN UNIVERSITY (US) 2021-05-18 US disclosed
CN-106967257-B Method of forming polythiophene polysulfonate complexes 新加坡科技研究局 2021-05-18 CN disclosed
CN-112805292-A Modified nucleoside and synthetic method thereof 斯微(上海) 生物科技有限公司 2021-05-14 CN disclosed
US-20210139897-A1 OLIGONUCLEOTIDE ANALOGUES HAVING MODIFIED INTERSUBUNIT LINKAGES AND/OR TERMINAL GROUPS SAREPTA THERAPEUTICS, INC. 2021-05-13 US disclosed
US-20210139460-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2021-05-13 US disclosed
US-20210139896-A1 Peptide Oligonucleotide Conjugates JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2021-05-13 US disclosed
EP-3271352-B1 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME H LUNDBECK AS (DK) 2021-05-12 EP disclosed
EP-3817745-A1 PROTEIN TYROSINE KINASE 6 (PTK6) DEGRADATION / DISRUPTION COMPOUNDS AND METHODS OF USE Icahn School of Medicine at Mount Sinai (US) 2021-05-12 EP disclosed
CN-112789040-A Transglutaminase 2(TG2) inhibitors 思达利医药公司 2021-05-11 CN disclosed
CN-107693797-B Peptide oligonucleotide conjugates 萨勒普塔医疗公司 2021-05-11 CN disclosed
CN-112778336-A Nitrogen-containing fused ring STING regulator compounds, preparation method and application 上海凌达生物医药有限公司 2021-05-11 CN disclosed
CN-112789264-A Novel sulfonylurea compound 英夫拉索姆有限公司 2021-05-11 CN disclosed
US-11001564-B2 Substituted chromane-8-carboxamide compounds and analogues thereof, and methods using same ARBUTUS BIOPHARMA CORPORATION (CA) 2021-05-11 US disclosed
US-11001601-B2 Compounds, compositions and methods for coloring edible materials THE PENN STATE RESEARCH FOUNDATION (US) 2021-05-11 US disclosed
US-11001568-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2021-05-11 US disclosed
US-11001570-B2 6-amino-quinolinone compounds and derivatives as BCL6 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-05-11 US disclosed
CN-110878052-B FXR agonist-containing compound and preparation method and application thereof 山东大学 2021-05-07 CN disclosed
WO-2021087408-A1 OTIC FORMULATIONS FOR DRUG-INDUCED OTOTOXICITY OTONOMY, INC. (US) 2021-05-06 WO disclosed
US-20210130359-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2021-05-06 US disclosed
US-20210130329-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2021-05-06 US disclosed
US-20210130354-A1 MULTI-KINASE INHIBITOR COMPOUND, AND CRYSTAL FORM AND USE THEREOF TRANSTHERA SCIENCES (NANJING), INC. (CN) 2021-05-06 US disclosed
US-20210130340-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASES KINNATE BIOPHARMA INC. 2021-05-06 US disclosed
US-20210135288-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH WITH METAL SULFIDE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2021-05-06 US disclosed
US-20210128488-A1 LIPIDS FOR USE IN LIPID NANOPARTICLE FORMULATIONS Acuitas Therapeutics, Inc. (CA) 2021-05-06 US disclosed
US-20210130366-A1 PDE9 INHIBITOR AND USE THEREOF TRANSTHERA SCIENCES (NANJING), INC. (CN) 2021-05-06 US disclosed
WO-2021083383-A1 NITROGEN-CONTAINING FUSED CYCLIC COMPOUND AS STING REGULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海凌达生物医药有限公司 2021-05-06 WO disclosed
US-20210128572-A1 COMBINATION OF ATR KINASE INHIBITORS WITH PARP INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-05-06 US disclosed
US-20210130338-A1 Heparanase Inhibitors and Use Thereof Beta Therapeutics Pty Ltd (AU) 2021-05-06 US disclosed
US-20210128723-A1 COMBINATION OF ATR KINASE INHIBITORS AND PD-1/PD-L1 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-05-06 US disclosed
EP-3813819-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASES Kinnate Biopharma Inc. (US) 2021-05-05 EP disclosed
EP-3813784-A1 PRC1 INHIBITORS AND METHODS OF TREATMENT THEREWITH The Regents Of The University Of Michigan (US) 2021-05-05 EP disclosed
EP-3071591-B1 ANTIMICROBIAL PEPTIDOMIMETICS AGENCY SCIENCE TECH & RES (SG) 2021-05-05 EP disclosed
CN-107847765-B 1, 4-substituted piperidine derivatives 89生物有限公司 2021-05-04 CN disclosed
CN-112724349-A Novel polymers and uses thereof 立邦涂料(中国)有限公司 2021-04-30 CN disclosed
CN-112740018-A Narrow absorbing polymeric nanoparticles and related methods 华盛顿大学 2021-04-30 CN disclosed
CN-107936024-B Anaplastic lymphoma kinase inhibitor and preparation method and application thereof 北京赛林泰医药技术有限公司 2021-04-30 CN disclosed
CN-112739349-A Combination therapy for the treatment of leukemia 圣诺康生命科学公司 2021-04-30 CN disclosed
US-20210122703-A1 LIPIDS FOR USE IN LIPID NANOPARTICLE FORMULATIONS Acuitas Therapeutics, Inc. (CA) 2021-04-29 US disclosed
US-20210122739-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LIMITED (IE) 2021-04-29 US disclosed
US-20210122773-A1 HETEROATOMIC-BASED HOLE-TRANSPORT MATERIALS SIGMA-ALDRICH CO. LLC 2021-04-29 US disclosed
WO-2021081375-A1 INHIBITORS OF RAF KINASES KINNATE BIOPHARMA INC. (US) 2021-04-29 WO disclosed
WO-2021081380-A1 PEROVSKITE NANOCRYSTAL COMPOSITIONS QUANTUM ADVANCED SOLUTIONS LTD (GB) 2021-04-29 WO disclosed
WO-2021078811-A1 NOVEL HETEROCYCLIC COMPOUNDS FLORATEK PHARMA AG (CH) 2021-04-29 WO disclosed
US-20210122702-A1 LIPIDS FOR USE IN LIPID NANOPARTICLE FORMULATIONS Acuitas Therapeutics, Inc. (CA) 2021-04-29 US disclosed
US-20210122730-A1 GLUCOCORTICOID RECEPTOR MODULATORS ORIC PHARMACEUTICALS, INC. 2021-04-29 US disclosed
US-20210122716-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2021-04-29 US disclosed
EP-3810589-A1 SUBSTITUTED 2-HETEROARYLOXYPYRIDINES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS Bayer Aktiengesellschaft (DE) 2021-04-28 EP disclosed
EP-3810588-A1 SUBSTITUTED 4-HETEROARYLOXYPYRIDINES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS Bayer Aktiengesellschaft (DE) 2021-04-28 EP disclosed
EP-3810146-A1 OTIC FORMULATIONS FOR DRUG-INDUCED OTOTOXICITY Otonomy, Inc. (US) 2021-04-28 EP disclosed
EP-3811974-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS Infinity Pharmaceuticals, Inc. (US) 2021-04-28 EP disclosed
EP-3169325-B1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS INC (US) 2021-04-28 EP disclosed
EP-3810145-A1 WD40 REPEAT DOMAIN PROTEIN 5 (WDR5) DEGRADATION / DISRUPTION COMPOUNDS AND METHODS OF USE Icahn School of Medicine at Mount Sinai (US) 2021-04-28 EP disclosed
EP-3810109-A1 COMPOSITIONS AND METHODS FOR INHIBITING CD73 Peloton Therapeutics, Inc. (US) 2021-04-28 EP disclosed
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CN-112714646-A Protein tyrosine kinase 6(PTK6) degradation/disruption compounds and methods of use 西奈山伊坎医学院 2021-04-27 CN disclosed
CN-112707893-A 1-cyanopyrrolidine compounds as USP30 inhibitors 特殊治疗有限公司 2021-04-27 CN disclosed
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WO-2021077066-A1 LIPID AND LIPID NANOPARTICLE FORMULATION FOR DRUG DELIVERY THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2021-04-22 WO disclosed
WO-2021077067-A1 LIPID NANOPARTICLES AND FORMULATIONS THEREOF FOR CAR MRNA DELIVERY THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2021-04-22 WO disclosed
WO-2021074227-A1 2-METHYL-AZA-QUINAZOLINES BAYER AKTIENGESELLSCHAFT (DE) 2021-04-22 WO disclosed
US-20210113562-A1 PIM KINASE INHIBITORS FOR TREATMENT OF MYELOPROLIFERATIVE NEOPLASMS AND FIBROSIS ASSOCIATED WITH CANCER SUMITOMO PHARMA AMERICA, INC. 2021-04-22 US disclosed
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EP-3806850-A2 METHODS OF INHIBITING PROLIFERATIVE CELLS Ideaya Biosciences, Inc. (US) 2021-04-21 EP disclosed
EP-3806856-A1 VMAT2 INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS RELATING THERETO Neurocrine Biosciences, Inc. (US) 2021-04-21 EP disclosed
EP-3807281-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2021-04-21 EP disclosed
EP-3251675-B1 PREVENTION OR TREATMENT OF URIC ACID OR GOUT DISEASE SHANTON PHARMA PTE LTD (SG) 2021-04-21 EP disclosed
EP-3464289-B1 ULTRA-POTENT VINCA ALKALOIDS: ADDED MOLECULAR COMPLEXITY FURTHER DISRUPTS THE TUBULIN DIMER-DIMER INTERFACE SCRIPPS RESEARCH INST (US) 2021-04-21 EP disclosed
EP-3233866-B1 PYRAZOLOPYRIDINAMINES AS MKNK1 AND MKNK2 INHIBITORS Bayer Pharma AG (DE) 2021-04-21 EP disclosed
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US-10981893-B2 Therapeutic inhibitory compounds ATTUNE PHARMACEUTICALS, INC. (US) 2021-04-20 US disclosed
US-10981932-B2 Macrocyclic indole derivatives BAYER AKTIENGESELLSCHAFT (DE) 2021-04-20 US disclosed
CN-112661696-A Green synthesis method of multi-aryl substituted methanol 华东理工大学 2021-04-16 CN disclosed
CN-112672995-A Novel sulfonamide urea compounds 英夫拉索姆有限公司 2021-04-16 CN disclosed
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WO-2021071843-A1 MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS Pipeline Therapeutics, Inc. (US) 2021-04-15 WO disclosed
WO-2021072265-A1 METHODS OF TREATING AN EYE DISORDER KODIAK SCIENCES INC. (US) 2021-04-15 WO disclosed
US-20210107896-A1 Macrophage Migration Inhibitory Factor Inhibitors, and Methods of Making and Using Same UNIV YALE (US) 2021-04-15 US disclosed
EP-3804723-A1 COMBINATION THERAPY BerGenBio ASA (NO) 2021-04-14 EP disclosed
EP-3802551-A1 PENICILLIN-BINDING PROTEIN INHIBITORS Venatorx Pharmaceuticals, Inc. (US) 2021-04-14 EP disclosed
EP-3802524-A1 COMPOUNDS FOR PAIN TREATMENT, COMPOSITIONS COMPRISING SAME, AND METHODS OF USING SAME Cersci Therapeutics, Inc. (US) 2021-04-14 EP disclosed
EP-3802471-A1 SYNTHESIS OF E,E-FARNESOL, FARNESYL ACETATE AND SQUALENE FROM FARNESENE VIA FARNESYL CHLORIDE Amyris, Inc. (US) 2021-04-14 EP disclosed
EP-3443049-B1 PHOTOACTIVE MACROMOLECULES AND USES THEREOF BECKMAN COULTER INC (US) 2021-04-14 EP disclosed
EP-3598218-B1 METAL OXIDE, METAL BRONZE AND POLYOXOMETALATE AS CHARGE STORAGE MATERIALS IN ELECTROCHROMIC DEVICE FURCIFER INC (US) 2021-04-14 EP disclosed
EP-3207031-B1 ATAXIA TELENGIECTASIA AND RAD3-RELATED (ATR) PROTEIN KINASE INHIBITORS Atrin Pharmaceuticals LLC (US) 2021-04-14 EP disclosed
EP-3523291-B1 CYANO-SUBSTITUTED HETEROCYCLES WITH ACTIVITY AS INHIBITORS OF USP30 MISSION THERAPEUTICS LTD (GB) 2021-04-14 EP disclosed
US-10975071-B2 Inhibitors of KRAS G12C mutant proteins ARAXES PHARMA LLC (US) 2021-04-13 US disclosed
US-10975101-B2 Ultra-potent vinca alkaloids: added molecular complexity further disrupts the tublin dimer-dimer interface THE SCRIPPS RESEARCH INSTITUTE (US) 2021-04-13 US disclosed
US-10975096-B2 Synthesis of polycyclic-carbamoylpyridone compounds GILEAD SCIENCES, INC. (US) 2021-04-13 US disclosed
US-10975123-B2 Mutant Akt-specific capture agents, compositions, and methods of using and making CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2021-04-13 US disclosed
US-10978739-B2 Silicon-based energy storage devices with carboxylic ether, carboxylic acid based salt, or acrylate electrolyte containing electrolyte additives ENEVATE CORPORATION (US) 2021-04-13 US disclosed
CN-112654632-A Hexahydro-1H-cyclopenta [ alpha ] phenanthrene derivatives useful for the treatment of pain and inflammation 塔罗制药公司 2021-04-13 CN disclosed
CN-112638381-A Muscarinic acetylcholine M1 receptor antagonists 帕珀莱恩医疗公司 2021-04-09 CN disclosed
CN-112638387-A VMAT2 inhibitor compounds, compositions, and methods related thereto 纽罗克里生物科学有限公司 2021-04-09 CN disclosed
CN-112638898-A Heteroaryl substituted sulfonamide compounds and their use as sodium channel inhibitors 泽农医药公司 2021-04-09 CN disclosed
CN-112638879-A Heteroaryl substituted sulfonamide compounds and their use as therapeutic agents 泽农医药公司 2021-04-09 CN disclosed
CN-112638373-A Cyclin-dependent kinase inhibitors 金耐特生物制药公司 2021-04-09 CN disclosed
CN-112638376-A Substituted tetrahydrocyclopenta [ c ] pyrroles, substituted dihydropyrrolizines, analogs thereof and methods of use thereof 爱彼特生物制药公司 2021-04-09 CN disclosed
CN-112638927-A Gemcitabine prodrugs 治愈生物医药公司 2021-04-09 CN disclosed
US-20210100238-A1 COMPOSITIONS AND METHODS FOR REDUCING ICE CRYSTAL FORMATION X-THERMA, INC. (US) 2021-04-08 US disclosed
US-20210101868-A1 Substituted 3-Dialkylaminomethyl-Piperidin-4-yl-Benzamides and Methods of Making and Using Same MEBIAS DISCOVERY, INC. 2021-04-08 US disclosed
US-20210101906-A2 BIOACTIVE CONJUGATE, PREPARATION METHOD THEREFOR AND USE THEREOF SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2021-04-08 US disclosed
US-20210101912-A1 NEW SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2021-04-08 US disclosed
US-20210101936-A1 CYCLIC PEPTIDES AS PROTEIN TARGETING AGENTS CALIFORNIA INSTITUTE OF TECHNOLOGY 2021-04-08 US disclosed
EP-3800186-A1 CYANOPYRROLIDINES AS DUB INHIBITORS FOR THE TREATMENT OF CANCER Mission Therapeutics Limited (GB) 2021-04-07 EP disclosed
CN-109942665-B Triptolide derivative and preparation method and application thereof 欣凯医药化工中间体(上海)有限公司 2021-04-06 CN disclosed
US-10968215-B2 Pyrido five-element aromatic ring compound, preparation method therefor and use thereof SHANGHAI HAIHE PHARMACEUTICAL CO., LTD. (CN) 2021-04-06 US disclosed
WO-2021058458-A1 PROCESS COMPRISING THE USE OF NEW IRIDIUM CATALYSTS FOR ENANTIOSELECTIVE HYDROGENATION OF 4-SUBSTITUTED 1,2-DIHYDROQUINOLINES BAYER AKTIENGESELLSCHAFT (DE) 2021-04-01 WO disclosed
WO-2021058457-A1 IMPROVED ENANTIOSELECTIVE HYDROGENATION OF 4-SUBSTITUTED 1,2-DIHYDROQUINOLINES IN PRESENCE OF A CHIRAL IRIDIUM CATALYST AND AN ADDITIVE BAYER AKTIENGESELLSCHAFT (DE) 2021-04-01 WO disclosed
US-20210098827-A1 Silicon-Based Energy Storage Devices With Electrolyte Containing Dimethoxyethane Based Compound ENEVATE CORPORATION 2021-04-01 US disclosed
US-20210095248-A1 METHOD OF INHIBITING TAU PHOSPHORYLATION PAIN THERAPEUTICS, INC. 2021-04-01 US disclosed
CN-112584833-A Heterocyclic spiro compounds and methods of use thereof for treating cancer 亚瑞克西斯制药公司 2021-03-30 CN disclosed
US-10960005-B2 Treatment of relapsed and/or refractory solid tumors and non-hodgkin's lymphomas CELGENE QUANTICEL RESEARCH, INC. (US) 2021-03-30 US disclosed
US-10959984-B2 Methods for treating cancer with RORγ inhibitors THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-03-30 US disclosed
WO-2021053205-A1 CHROMENE-4-ONE DERIVATIVES AS BRAIN-DERIVED NEUROTROPHIC FACTOR (BDNF) MIMETICS FLORATEK PHARMA AG (CH) 2021-03-25 WO disclosed
US-20210087143-A1 AGENTS FOR DIFFERENTIATING STEM CELLS AND TREATING CANCER MINERVA BIOTECHNOLOGIES CORP (US) 2021-03-25 US disclosed
US-20210085656-A1 SUBSTITUTED DIHYDROIMIDAZOPYRIDINEDIONES AS MKNK1 AND MKNK2 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-03-25 US disclosed
US-20210085682-A1 FATTY LIVER DISEASE TREATMENT USING GLUCOCORTICOID AND MINERALOCORTICOID RECEPTOR ANTAGONISTS CORCEPT THERAPEUTICS, INC. 2021-03-25 US disclosed
US-20210087151-A1 SUBSTITUTED THIOPHENYL URACILS, SALTS THEREOF AND THE USE THEREOF AS HERBICIDAL AGENTS SYNGENTA CROP PROTECTION AG (CH) 2021-03-25 US disclosed
WO-2021055705-A1 BIAMINOQUINOLINES AND NANOFORMULATIONS FOR CANCER TREATMENT THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-03-25 WO disclosed
WO-2021055560-A1 FLUORINATED ELECTROLYTE ADDITIVES E3TRIGEN, INC. (US) 2021-03-25 WO disclosed
WO-2021053617-A1 MLL1 INHIBITORS AND ANTI-CANCER AGENTS NOVARTIS AG (CH) 2021-03-25 WO disclosed
EP-3793550-A2 SUBSTITUTED 2,2'-BIPYRIMIDINYL COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2021-03-24 EP disclosed
EP-3793551-A1 OXADIAZOLE COMPOUNDS Vivace Therapeutics, Inc. (US) 2021-03-24 EP disclosed
EP-3793547-A1 MAGL INHIBITORS H. Lundbeck A/S (DK) 2021-03-24 EP disclosed
EP-3793552-A1 ABHD12 INHIBITORS AND METHODS OF MAKING AND USING SAME The Scripps Research Institute (US) 2021-03-24 EP disclosed
CN-112543753-A Indene derivatives useful for treating pain and inflammation 塔罗制药公司 2021-03-23 CN disclosed
CN-107922345-B Arylsulfonamide compounds as carbonic anhydrase inhibitors and their therapeutic use 圣诺康生命科学公司 2021-03-23 CN disclosed
US-10957898-B2 Silicon-based energy storage devices with anhydride containing electrolyte additives ENEVATE CORPORATION (US) 2021-03-23 US disclosed
US-10954328-B2 Polymerization processes EXXONMOBIL CHEMICAL PATENTS INC. (US) 2021-03-23 US disclosed
US-10954391-B2 Water soluble fluorescent or colored dyes and methods for their use SONY CORPORATION (JP) 2021-03-23 US disclosed
US-10955419-B2 Methods and systems for analysis using polymer dots UNIVERSITY OF WASHINGTON (US) 2021-03-23 US disclosed
US-10957938-B2 Sodium-ion electrolyte composition DEAKIN UNIVERSITY (AU) 2021-03-23 US disclosed
CN-112533581-A PRC1 inhibitors and methods of treatment therewith 密歇根大学董事会 2021-03-19 CN disclosed
CN-112533913-A Novel compounds 英夫拉索姆有限公司 2021-03-19 CN disclosed
CN-112533602-A AXL kinase inhibitors and uses thereof 大日本住友制药肿瘤公司 2021-03-19 CN disclosed
CN-112533905-A Indene derivatives useful for treating pain and inflammation 塔罗制药公司 2021-03-19 CN disclosed
US-20210078963-A1 SELECTIVE HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF HUMAN DISEASE SHUTTLE PHARMACEUTICALS, INC. 2021-03-18 US disclosed
US-20210079018-A1 MACROCYCLIC FLUORINE SUBSTITUTED INDOLE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-03-18 US disclosed
US-20210077427-A1 ALKOXY COMPOUNDS FOR DISEASE TREATMENT ACUCELA INC. 2021-03-18 US disclosed
WO-2021048626-A1 COMPOSITIONS FOR THE TREATMENT OF SOLID TUMORS RAZIEL THERAPEUTICS LTD. (IL) 2021-03-18 WO disclosed
US-20210079039-A1 COMPOSITIONS AND METHODS FOR THE SELECTIVE DELIVERY OF THERAPEUTIC AND IMAGING AGENTS AVELAS ACQUISITION CORPORATION 2021-03-18 US disclosed
EP-3359542-B1 SPIRO[3H-INDOLE-3,2´-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2021-03-17 EP disclosed
EP-3791875-A1 METHOD FOR INHIBITING GROWTH OF CANCER CELLS Pain Therapeutics, Inc. (US) 2021-03-17 EP disclosed
CN-112512597-A Methods for treating diseases associated with aberrant ACVR1 expression and ACVR1 inhibitors useful therefor 大日本住友制药肿瘤公司 2021-03-16 CN disclosed
US-10947176-B2 Antimalarial compositions and uses thereof THE SCRIPPS RESEARCH INSTITUTE (US) 2021-03-16 US disclosed
CN-109526219-B Benzenesulfonamides and their use as therapeutic agents 泽农医药公司 2021-03-12 CN disclosed
WO-2021045686-A1 HETEROCYCLIC COMPOUNDS AS MODULATORS OF BETA-CATENIN / TCF4 INTERACTION AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2021-03-11 WO disclosed
WO-2021043966-A1 NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2021-03-11 WO disclosed
WO-2021042169-A1 NITRIFICATION INHIBITORS THE UNIVERSITY OF MELBOURNE (AU) 2021-03-11 WO disclosed
US-20210069201-A1 SELECTIVE P2X3 MODULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.3) LIMITED (GB) 2021-03-11 US disclosed
US-20210070715-A1 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE SUMITOMO PHARMA AMERICA, INC. 2021-03-11 US disclosed
US-20210070748-A1 INHIBITORS OF BRUTONS TYROSINE KINASE PHARMACYCLICS LLC (US) 2021-03-11 US disclosed
US-20210070773-A1 4-HYDROXYPIPERIDINE DERIVATIVES AND THEIR USE AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 19 (USP19) ALMAC DISCOVERY LIMITED (GB) 2021-03-11 US disclosed
EP-3134410-B1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL LILLY CO ELI (US) 2021-03-10 EP disclosed
EP-3283077-B1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RES INC (US) 2021-03-10 EP disclosed
EP-3787629-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASES Kinnate Biopharma Inc. (US) 2021-03-10 EP disclosed
EP-3788041-A1 NOVEL COMPOUNDS Inflazome Limited (IE) 2021-03-10 EP disclosed
CN-112469725-A Penicillin binding protein inhibitors 维纳拓尔斯制药公司 2021-03-09 CN disclosed
CN-112457326-A Aromatic heterocyclic lactam compound, preparation method and application 上海凌达生物医药有限公司 2021-03-09 CN disclosed
CN-112469720-A Dual ATM and DNA-PK inhibitors for use in antitumor therapy 艾科思莱德制药公司 2021-03-09 CN disclosed
CN-112469712-A Substituted 2-heteroaryloxypyridines and their salts and their use as herbicides 拜耳公司 2021-03-09 CN disclosed
US-10940146-B2 NHE3-binding compounds and methods for inhibiting phosphate transport ARDELYX, INC. (US) 2021-03-09 US disclosed
US-10941160-B2 Bromodomain inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2021-03-09 US disclosed
US-10941162-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2021-03-09 US disclosed
CN-112441980-A Pyrazole derivatives for FGFR inhibitor and preparation method thereof 上海奕拓医药科技有限责任公司 2021-03-05 CN disclosed
WO-2021037219-A1 PYRAZOLE DERIVATIVE FOR FGFR INHIBITOR AND PREPARATION METHOD THEREFOR 上海奕拓医药科技有限责任公司 2021-03-04 WO disclosed
US-20210062251-A1 ENHANCEMENT OF NUCLEIC ACID POLYMERIZATION BY AROMATIC COMPOUNDS Roche Sequencing Solutions, Inc. 2021-03-04 US disclosed
US-20210060022-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS INFINITY PHARMACEUTICALS, INC. 2021-03-04 US disclosed
US-20210061834-A1 NOVEL PRECATALYST SCAFFOLDS FOR CROSS-COUPLING REACTIONS, AND METHODS OF MAKING AND USING SAME NATIONAL SCIENCE FOUNDATION 2021-03-04 US disclosed
EP-3596064-B1 TOSYLACETATE BASED COMPOUNDS AND DERIVATIVES THEREOF AS PHGDH INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2021-03-03 EP disclosed
EP-3784229-A2 SLC26A3 INHIBITORS AND USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-03-03 EP disclosed
EP-3786166-A1 2-AMINOPYRIMIDINE DERIVATIVE, PREPARATION METHOD AND USE THEREOF Etern Biopharma (Shanghai) Co., Ltd. (CN) 2021-03-03 EP disclosed
US-10934253-B2 Therapeutic compounds and methods UNIVERSITY OF TASMANIA (AU) 2021-03-02 US disclosed
US-10934322-B2 B-vitamin and amino acid conjugates of nicotinoyl ribosides and reduced nicotinoyl ribosides, derivatives thereof, and methods of preparation thereof ChromaDex Inc. (US) 2021-03-02 US disclosed
US-10934568-B2 Conversion of sugars to ionic liquids NATIONAL TECHNOLOGY & ENGINEERING SOLUTIONS OF SANDIA, LLC (US) 2021-03-02 US disclosed
US-10934531-B2 Method for enantioselective carbene C—H insertion using an iron-containing protein catalyst CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2021-03-02 US disclosed
US-10934376-B2 Polyethylene compositions and films made therefrom EXXONMOBIL CHEMICAL PATENTS INC. (US) 2021-03-02 US disclosed
CN-107406548-B Compositions and methods for treating hyperkalemia 阿德利克斯公司 2021-03-02 CN disclosed
CN-112430250-A Lymphatic prodrugs 莫纳什大学 2021-03-02 CN disclosed
CN-108884068-B 1-cyano-pyrrolidine derivatives as DUB inhibitors 特殊治疗有限公司 2021-02-26 CN disclosed
US-20210053969-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASES KINNATE BIOPHARMA INC. 2021-02-25 US disclosed
US-20210053975-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES FORWARD THERAPEUTICS, INC. 2021-02-25 US disclosed
US-20210053989-A1 PYRIMIDINE-FUSED CYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF SHANGHAI BLUERAY BIOPHARMA CO., LTD. (CN) 2021-02-25 US disclosed
US-20210053953-A1 A COMPOUND, A REACTION PRODUCT OF SAID COMPOUND AND PRODUCTION METHODS THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2021-02-25 US disclosed
US-20210053988-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2021-02-25 US disclosed
US-20210052585-A1 SUBSTITUTED 1,1'-BIPHENYL COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2021-02-25 US disclosed
WO-2021035096-A1 COMPOSITIONS AND METHODS FOR TARGETING CELLULAR MOLECULES KUMQUAT BIOSCIENCES INC. (US) 2021-02-25 WO disclosed
WO-2021032883-A1 COMBINATION THERAPY OF A PATIENT SUBGROUP BERGENBIO ASA (NO) 2021-02-25 WO disclosed
WO-2021032591-A1 MACROCYCLIC SULFONYLUREA DERIVATIVES USEFUL AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2021-02-25 WO disclosed
WO-2021032588-A1 MACROCYCLIC SULFONYLAMIDE DERIVATIVES USEFUL AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2021-02-25 WO disclosed
US-20210053960-A1 PYRAZOLE MAGL INHIBITORS H. LUNDBECK A/S (DK) 2021-02-25 US disclosed
US-20210052532-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF INSULIN RESISTANCE TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2021-02-25 US disclosed
US-20210054003-A1 Methods for the preparation of cyclopentaoxasilinones and cyclopentaoxaborininones and their use DREXEL UNIVERSITY 2021-02-25 US disclosed
EP-3783001-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS Gilead Sciences, Inc. (US) 2021-02-24 EP disclosed
EP-3781565-A1 2-METHYL-AZA-QUINAZOLINES Bayer Pharma Aktiengesellschaft (DE) 2021-02-24 EP disclosed
EP-3781194-A1 COMPOSITIONS AND METHODS FOR THE SELECTIVE DELIVERY OF THERAPEUTIC AND IMAGING AGENTS Avelas Biosciences, Inc. (US) 2021-02-24 EP disclosed
EP-3782983-A1 ISOINDOLE DERIVATIVE Tianjin Hemay Pharmaceutical Co., Ltd. (CN) 2021-02-24 EP disclosed
EP-3277677-B1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS MISSION THERAPEUTICS LTD (GB) 2021-02-24 EP disclosed
EP-3434674-B1 ((4-(2-OXOIMIDAZOLIDINE-1-YL)PYRIMIDIN-2-YL)AMINE DERIVATIVES AS MUTANT IDH INHIBITORS FOR TREATING CANCER SHANGHAI HAIHE PHARMACEUTICAL CO LTD (CN) 2021-02-24 EP disclosed
CN-112390832-A Metal complex, intermediate, preparation method and application thereof 中国科学院上海有机化学研究所 2021-02-23 CN disclosed
CN-112390904-A Polyethylene containing polar functional group and preparation method thereof 中国科学院上海有机化学研究所 2021-02-23 CN disclosed
CN-112390838-A Modified nucleoside and synthetic method thereof 斯微(上海)生物科技有限公司 2021-02-23 CN disclosed
US-10927202-B2 Polyethylene compositions and articles made therefrom EXXONMOBIL CHEMICAL PATENTS INC. (US) 2021-02-23 US disclosed
US-10927203-B2 Polyethylene compositions and articles made therefrom EXXONMOBIL CHEMICAL PATENTS INC. (US) 2021-02-23 US disclosed
US-10927125-B2 Substituted cinnolines as inhibitors of KRAS G12C ARAXES PHARMA LLC (US) 2021-02-23 US disclosed
US-10927205-B2 Polymerization processes and polymers made therefrom EXXONMOBIL CHEMICAL PATENTS INC. (US) 2021-02-23 US disclosed
US-10927110-B2 Cyano-subtituted heterocycles with activity as inhibitors of USP30 MISSION THERAPEUTICS LIMITED (GB) 2021-02-23 US disclosed
US-10927105-B1 Pyrazole MAGL inhibitors LUNDBECK LA JOLLA RESEARCH CENTER, INC. (US) 2021-02-23 US disclosed
US-10927111-B2 Inhibitors of RAF kinases KINNATE BIOPHARMA INC. (US) 2021-02-23 US disclosed
US-10927355-B2 Method for producing an organosilicon product CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2021-02-23 US disclosed
CN-112384507-A Substituted 4-heteroaryloxypyridines and their salts and their use as herbicides 拜耳公司 2021-02-19 CN disclosed
CN-106604997-B Inhibitors of lysine-specific demethylase-1 赛尔基因昆蒂赛尔研究公司 2021-02-19 CN disclosed
CN-108473632-B Polymeric compositions 新加坡科技研究局 2021-02-19 CN disclosed
CN-107531738-B Niacinetoside or nicotinamide riboside compositions, reduced derivatives thereof and uses thereof 可劳迈戴斯有限公司 2021-02-19 CN disclosed
CN-107922405-B Compound with ERK kinase inhibitory activity, preparation method and application thereof 中国科学院上海药物研究所 2021-02-19 CN disclosed
CN-112384508-A Tricyclic ASK1 inhibitor and application thereof 山东轩竹医药科技有限公司 2021-02-19 CN disclosed
US-20210047302-A1 NOVEL COMPOUNDS INFLAZOME LIMITED (IE) 2021-02-18 US disclosed
US-20210046030-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF INSULIN RESISTANCE TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2021-02-18 US disclosed
US-20210046069-A1 PENTAFLUOROSULFANYL-SUBSTITUTED AMIDE DERIVATIVES, PREPARATION METHODS THEREOF AND MEDICAL USES THEREOF BEIJING INNOCARE PHARMA TECH CO., LTD. (CN) 2021-02-18 US disclosed
WO-2021028419-A1 SUBSTITUTED 3-(2-HETEROARYLOXYPHENYL)ISOXAZOLINES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2021-02-18 WO disclosed
WO-2021028421-A1 SUBSTITUTED (2-HETEROARYLOXYPHENYL)ISOXAZOLINES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2021-02-18 WO disclosed
WO-2021028854-A1 PIPERIDINYL-METHYL-PURINEAMINES AS NSD2 INHIBITORS AND ANTI-CANCER AGENTS NOVARTIS AG (CH) 2021-02-18 WO disclosed
WO-2021027614-A1 MODIFIED NUCLEOSIDE AND SYNTHESIS METHOD THEREFOR 斯微(上海)生物科技有限公司 2021-02-18 WO disclosed
EP-3774836-A1 HEXADECAHYDRO-1H-CYCLOPENTA[A]PHENANTHRENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION Aquinox Pharmaceuticals (Canada) Inc. (CA) 2021-02-17 EP disclosed
EP-3774748-A1 OXADIAZOLINE DERIVATIVES Bayer Aktiengesellschaft (DE) 2021-02-17 EP disclosed
EP-3773560-A1 PIM KINASE INHIBITORS FOR TREATMENT OF MYELOPROLIFERATIVE NEOPLASMS AND FIBROSIS ASSOCIATED WITH CANCER Sumitomo Dainippon Pharma Oncology, Inc. (US) 2021-02-17 EP disclosed
EP-3774709-A1 METHODS OF REDUCING INFLAMMATION OF THE DIGESTIVE SYSTEM WITH INHIBITORS OF HIF-2-ALPHA Peloton Therapeutics, Inc. (US) 2021-02-17 EP disclosed
EP-3778584-A1 PRODUCTION PROCESS OF 2-CHLORO-4-HETEROARYL-PYRIMIDINE DERIVATIVES ARIAD Pharmaceuticals, Inc. (US) 2021-02-17 EP disclosed
EP-3394049-B1 CYANOPYRROLIDINE DERVIVATIVES AS INHBITORS FOR DUBS MISSION THERAPEUTICS LTD (GB) 2021-02-17 EP disclosed
EP-3331894-B1 NICOTINAMIDE MONONUCLEOTIDE DERIVATIVES AND THEIR USES METRO INT BIOTECH LLC (US) 2021-02-17 EP disclosed
EP-3558979-B1 NOVEL BENZYLAMINO SUBSTITUTED QUINAZOLINES AND DERIVATIVES AS SOS1 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2021-02-17 EP disclosed
EP-3774746-A1 INDENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION Aquinox Pharmaceuticals (Canada) Inc. (CA) 2021-02-17 EP disclosed
EP-3492106-B1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX INC (US) 2021-02-17 EP disclosed
EP-3773591-A1 AXL KINASE INHIBITORS AND USE OF THE SAME Sumitomo Dainippon Pharma Oncology, Inc. (US) 2021-02-17 EP disclosed
US-10918643-B2 No-donors for the treatment of cerebrovascular vasospasms after brain hemorrhage WESTFAELISCHE WILHELMS-UNIVERSITAET MUENSTER (DE) 2021-02-16 US disclosed
US-10919913-B2 Spiro[3H-indole-3,2′-pyrrolidin]-2(1H)-one compounds and derivatives as MDM2-p53 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-02-16 US disclosed
US-10919850-B2 Covalent inhibitors of KRas G12C ARAXES PHARMA LLC (US) 2021-02-16 US disclosed
US-10919875-B2 Substituted 4-benzyl and 4-benzoyl piperidine derivatives 89BIO LTD (IL) 2021-02-16 US disclosed
US-10919914-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2021-02-16 US disclosed
US-10921674-B2 Electrochromic polymer thin films having reduced self-bleaching behavior and enhanced cycling stability Furcifer Inc. (US) 2021-02-16 US disclosed
US-10919038-B2 Modification of surface properties of microfluidic devices BIO-RAD LABORATORIES, INC. (US) 2021-02-16 US disclosed
CN-109908356-B Cyanoacrylate material loaded with antitumor drug 中国人民解放军军事医学科学院毒物药物研究所 2021-02-12 CN disclosed
US-20210040065-A1 NOVEL COMPOUNDS INFLAZOME LIMITED (IE) 2021-02-11 US disclosed
US-20210038628-A1 NANOPARTICLE COMPOSITIONS JANUARY THERAPEUTICS, INC. (US) 2021-02-11 US disclosed
WO-2021026257-A1 PRODRUGS OF ALOX-15 INHIBITORS AND METHODS OF USING THE SAME EMPIRICO INC. (US) 2021-02-11 WO disclosed
WO-2021025976-A1 SUBSTITUTED CYCLOPROPYL-2,2'-BIPYRIMIDINYL COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA, INC. (US) 2021-02-11 WO disclosed
CN-106661229-B Organosilicon ligands for quantum dots 纳米系统公司 2021-02-09 CN disclosed
CN-108117534-B Benzo-oxygenated aliphatic cyclomethylamines 华东理工大学 2021-02-05 CN disclosed
CN-107531613-B Benzo-aliphatic ring-substituted alkylamine compound and application thereof 华东理工大学 2021-02-05 CN disclosed
US-20210030772-A1 PRODRUGS OF ALOX-15 INHIBITORS AND METHODS OF USING THE SAME EMPIRICO INC. 2021-02-04 US disclosed
US-20210030005-A1 BENZOXABOROLE COMPOSITIONS HAVING A GROWTH ENHANCING EFFECT 5METIS, INC. 2021-02-04 US disclosed
US-20210032264-A1 INDENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION AQUINOX PHARMACEUTICALS (CANADA) INC. (CA) 2021-02-04 US disclosed
WO-2021022078-A1 DUAL ATM AND DNA-PK INHIBITORS FOR USE IN ANTI-TUMOR THERAPY XRAD THERAPEUTICS, INC. (US) 2021-02-04 WO disclosed
WO-2021018287-A1 SPIROAROMATIC COMPOUND, PREPARATION AND APPLICATION THEREOF 上海奕拓医药科技有限责任公司 2021-02-04 WO disclosed
CN-112300196-A Piperidine condensed ring compound, preparation method and application 上海凌达生物医药有限公司 2021-02-02 CN disclosed
CN-112300194-A Condensed ring pyridone compounds, preparation method and application 上海凌达生物医药有限公司 2021-02-02 CN disclosed
CN-112300173-A Nitrogen-containing polycyclic compounds, preparation method and application 上海凌达生物医药有限公司 2021-02-02 CN disclosed
US-10907184-B2 Ammonium based ionic liquids useful for lignocellulosic processing NATIONAL TECHNOLOGY & ENGINEERING SOLUTIONS OF SANDIA, LLC (US) 2021-02-02 US disclosed
US-10905702-B2 Inhibition of galectin 3 binding to the airway epithelial surface to treat or prevent septic shock resulting from influenza and subsequent pneumococcal pneumonia infection UNIVERSITY OF MARYLAND, BALTIMORE (US) 2021-02-02 US disclosed
CN-112300160-A Spiro aromatic ring compound, preparation and application thereof 上海奕拓医药科技有限责任公司 2021-02-02 CN disclosed
CN-112300159-A Dual ATM and DNA-PK inhibitors for use in antitumor therapy 艾科思莱德制药公司 2021-02-02 CN disclosed
CN-107484415-B 1-cyanopyrrolidine compounds as USP30 inhibitors 特殊治疗有限公司 2021-01-29 CN disclosed
CN-107709470-B Super bright dimeric or polymeric dyes 索尼公司 2021-01-29 CN disclosed
CN-112280553-A Encoded chromophoric polymer particles 华盛顿大学商业中心 2021-01-29 CN disclosed
CN-112292184-A Nanoparticle compositions 詹纽瑞治疗公司 2021-01-29 CN disclosed
US-20210023095-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. 2021-01-28 US disclosed
US-20210024501-A1 COVALENT INHIBITORS OF KRAS ARAXES PHARMA LLC 2021-01-28 US disclosed
US-20210024571-A1 HEXADECAHYDRO-1H-CYCLOPENTA[A]PHENANTHRENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION AQUINOX PHARMACEUTICALS (CANADA) INC. (CA) 2021-01-28 US disclosed
US-20210024457-A1 DIAMIDE ANTIMICROBIAL AGENTS BROWN UNIVERSITY 2021-01-28 US disclosed
WO-2021013800-A1 SUBSTITUTED N-PHENYL-N-AMINOUARCILS AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2021-01-28 WO disclosed
WO-2021013799-A1 SUBSTITUTED N-PHENYL URACILS, SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2021-01-28 WO disclosed
WO-2021013978-A1 TARGETED RADIOPHARMACEUTICALS FOR THE DIAGNOSIS AND TREATMENT OF PROSTATE CANCER BAYER AS (NO) 2021-01-28 WO disclosed
EP-3521399-B1 ENCODED CHROMOPHORIC POLYMER PARTICLES UNIV WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2021-01-27 EP disclosed
US-10899860-B2 Polymerization processes and polymers made therefrom EXXONMOBIL CHEMICAL PATENTS INC. (US) 2021-01-26 US disclosed
US-10899739-B2 Macrophage migration inhibitory factor inhibitors, and methods of making and using same YALE UNIVERSITY (US) 2021-01-26 US disclosed
US-10898487-B2 Benzylamino substituted quinazolines and derivatives as SOS1 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-01-26 US disclosed
US-10899737-B2 Piperazine carbamates and methods of making and using same LUNDBECK LA JOLLA RESEARCH CENTER, INC. (US) 2021-01-26 US disclosed
CN-112262116-A Synthesis of E, E-farnesol, farnesyl acetate and squalene from farnesene via farnesyl chloride 阿迈瑞斯公司 2021-01-22 CN disclosed
CN-112262142-A Benzenesulfonamide compounds and their use as therapeutic agents 泽农医药公司 2021-01-22 CN disclosed
CN-112262145-A 2-aminopyrimidine derivatives, preparation method and application thereof 上海奕拓医药科技有限责任公司 2021-01-22 CN disclosed
US-20210017100-A1 ORGANIC REACTIONS CARRIED OUT IN AQUEOUS SOLUTION IN THE PRESENCE OF A HYDROXYALKYL(ALKYL)CELLULOSE OR AN ALKYLCELLULOSE AbbVie Deutschland GmbH & Co. KG (DE) 2021-01-21 US disclosed
US-20210017219-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. 2021-01-21 US disclosed
US-20210017174-A1 IDENTIFICATION AND USE OF ERK5 INHIBITOR BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-01-21 US disclosed
US-20210015764-A1 METHODS OF REDUCING INFLAMMATION OF THE DIGESTIVE SYSTEM WITH INHIBITORS OF HIF-2- ALPHA PELOTON THERAPEUTICS INC. (US) 2021-01-21 US disclosed
WO-2021011796-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASES KINNATE BIOPHARMA INC. (US) 2021-01-21 WO disclosed
WO-2021009568-A1 BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF 2692372 ONTARIO, INC. (CA) 2021-01-21 WO disclosed
US-20210017220-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. 2021-01-21 US disclosed
US-20210017186-A1 SUBSTITUTED 2-PYRIDONE TRICYCLIC COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2021-01-21 US disclosed
EP-3349747-B1 NO-DONORS FOR THE TREATMENT OF CEREBROVASCULAR VASOSPASMS AFTER BRAIN HEMORRHAGE UNIV MUENSTER WESTFAELISCHE WILHELMS (DE) 2021-01-20 EP disclosed
EP-3458441-B1 PROCESS FOR THE MANUFACTURE OF 6-ALKYNYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM INT (DE) 2021-01-20 EP disclosed
EP-3765158-A1 NANOPARTICLE COMPOSITIONS January Therapeutics, Inc. (US) 2021-01-20 EP disclosed
CN-105873564-B Skin care compositions and methods of use thereof 尤尼根公司 2021-01-19 CN disclosed
US-10894788-B2 Inhibitors of cyclin-dependent kinases KINNATE BIOPHARMA INC. (US) 2021-01-19 US disclosed
US-10894802-B2 Precatalyst scaffolds for cross-coupling reactions, and methods of making and using same YALE UNIVERSITY (US) 2021-01-19 US disclosed
CN-112236139-A PIM kinase inhibitors for the treatment of myeloproliferative tumors and cancer-associated fibrosis 大日本住友制药肿瘤公司 2021-01-15 CN disclosed
WO-2021007236-A1 NON-NATIVE O-GLCNAC MODIFICATION OF PEPTIDE HORMONES YIELDS POTENT GPCR AGONISTS WITH IMPROVED SERUM STABILITY UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2021-01-14 WO disclosed
WO-2021005586-A1 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS NOVARTIS AG (CH) 2021-01-14 WO disclosed
WO-2021007172-A1 FORMULATIONS OF RBP4 INHIBITORS AND METHODS OF USE BELITE BIO, LLC (US) 2021-01-14 WO disclosed
US-20210008076-A1 NANOPARTICLE COMPOSITIONS JANUARY THERAPEUTICS, INC. 2021-01-14 US disclosed
US-20210013536-A1 MEMBRANES FOR AQUEOUS REDOX FLOW BATTERIES FIRST-CITIZENS BANK & TRUST COMPANY 2021-01-14 US disclosed
US-20210009521-A1 ENANTIOSELECTIVE HYDROGENATION OF 4-SUBSTITUTED 1,2-DIHYDROQUINOLINES IN PRESENCE OF A CHIRAL IRIDIUM CATALYST BAYER AKTIENGESELLSCHAFT (DE) 2021-01-14 US disclosed
US-20210009585-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2021-01-14 US disclosed
US-20210007999-A1 NANOPARTICLE COMPOSITIONS JANUARY THERAPEUTICS, INC. 2021-01-14 US disclosed
US-20210009520-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2021-01-14 US disclosed
US-20210008043-A1 Substituted Chromenones, IRE1 Inhibitors, and Methods of Using Same NATIONAL INSTITUTES OF HEALTH 2021-01-14 US disclosed
US-20210009588-A1 NOVEL BENZYLAMINO SUBSTITUTED PYRIDOPYRIMIDINONES AND DERIVATIVES AS SOS1 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2021-01-14 US disclosed
EP-3763367-A1 PYRIDINE-PYRAZOLE DERIVATIVES AS HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2021-01-13 EP disclosed
EP-3761984-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF INSULIN RESISTANCE Temple University - Of The Commonwealth System of Higher Education (US) 2021-01-13 EP disclosed
EP-3762381-A1 SERINE THREONINE KINASE (AKT) DEGRADATION / DISRUPTION COMPOUNDS AND METHODS OF USE Icahn School of Medicine at Mount Sinai (US) 2021-01-13 EP disclosed
EP-3763712-A1 INDOLIZINE COMPOUNDS, PREPARATION METHOD AND USE THEREOF Shanghai Haihe Pharmaceutical Co., Ltd. (CN) 2021-01-13 EP disclosed
EP-3761985-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF INSULIN RESISTANCE Temple University - Of The Commonwealth System of Higher Education (US) 2021-01-13 EP disclosed
EP-3762365-A1 METHODS AND COMPOSITIONS OF ISOINDOLINE-1,3-DIONE AND ISOINDOLE PRODRUGS USEFUL FOR TREATING CANCER, ULCERATIVE COLITIS AND RELATED INFLAMMATORY DISEASES Amgen (Europe) GmbH (CH) 2021-01-13 EP disclosed
EP-3762379-A1 IDENTIFICATION AND USE OF ERK5 INHIBITORS Bayer Aktiengesellschaft (DE) 2021-01-13 EP disclosed
CN-112218860-A Substituted phenylthiouracils, their salts and their use as herbicides 先正达农作物保护股份公司 2021-01-12 CN disclosed
CN-112218533-A Nanoparticle compositions 詹纽瑞治疗公司 2021-01-12 CN disclosed
CN-112218873-A Metallocene synthesis method 埃克森美孚化学专利公司 2021-01-12 CN disclosed
US-10888853-B2 Cinchonium betaine catalysts and methods of using same BRANDEIS UNIVERSITY (US) 2021-01-12 US disclosed
US-10889591-B2 PDE9 inhibitor and use thereof NANJING TRANSTHERA BIOSCIENCES CO. LTD. (CN) 2021-01-12 US disclosed
US-10889586-B2 Multi-kinase inhibitor compound, and crystal form and use thereof NANJING TRANSTHERA BIOSCIENCES CO. LTD. (CN) 2021-01-12 US disclosed
US-10888562-B1 2021-01-12 US disclosed
CN-112204025-A Compounds for the treatment of pain, compositions comprising the same and methods of using the same 瑟赛治疗公司 2021-01-08 CN disclosed
CN-107098908-B Preparation method and application of pyrrolopyrimidine compound 欣凯医药科技(上海)有限公司 2021-01-08 CN disclosed
CN-112203679-A IL-6 antibodies and fusion constructs and conjugates thereof 科达制药股份有限公司 2021-01-08 CN disclosed
US-20210002324-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. 2021-01-07 US disclosed
US-20210002274-A1 NOVEL COMPOUNDS INFLAZOME LIMITED (IE) 2021-01-07 US disclosed
US-20210002469-A1 TOUGH, HEALABLE COMPOSITES DISPLAYING STRESS RELAXATION AT THE RESIN-FILLER INTERFACE NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2021-01-07 US disclosed
US-20210002233-A1 PKM2 MODULATORS AND METHODS FOR THEIR USE SUMITOMO PHARMA ONCOLOGY, INC. 2021-01-07 US disclosed
US-20210000837-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2021-01-07 US disclosed
US-20210003916-A1 POSITIVE RESIST COMPOSITION AND PATTERNING PROCESS SHIN-ETSU CHEMICAL CO., LTD. (JP) 2021-01-07 US disclosed
EP-3759090-A1 NOVEL COMPOUNDS Inflazome Limited (IE) 2021-01-06 EP disclosed
EP-3760639-A1 ZWITTERIONIC POLYMER CONJUGATES Kodiak Sciences Inc. (US) 2021-01-06 EP disclosed
EP-3758801-A1 PHENYLSULFONYLUREA DERIVATIVES USEFUL AS NLRP3 INHIBITORS Inflazome Limited (IE) 2021-01-06 EP disclosed
EP-3759073-A1 SULFONAMIDE DERIVATES AS NLRP3 INHIBITORS Inflazome Limited (IE) 2021-01-06 EP disclosed
EP-3758737-A1 IL-6 ANTIBODIES AND FUSION CONSTRUCTS AND CONJUGATES THEREOF Kodiak Sciences Inc. (US) 2021-01-06 EP disclosed
EP-3759089-A1 NOVEL COMPOUNDS Inflazome Limited (IE) 2021-01-06 EP disclosed
EP-3758490-A1 NANOPARTICLE COMPOSITIONS January Therapeutics, Inc. (US) 2021-01-06 EP disclosed
EP-3759227-A1 IMPROVED METHOD FOR THE SYNTHESIS OF TRYPTOPHAN ANALOGS IN AQUEOUS SOLVENTS AT REDUCED TEMPERATURES California Institute of Technology (US) 2021-01-06 EP disclosed
EP-3759102-A1 NOVEL COMPOUNDS Inflazome Limited (IE) 2021-01-06 EP disclosed
EP-3759103-A1 NOVEL COMPOUNDS Inflazome Limited (IE) 2021-01-06 EP disclosed
EP-3758495-A1 NANOPARTICLE COMPOSITIONS January Therapeutics, Inc. (US) 2021-01-06 EP disclosed
EP-3759077-A1 NOVEL COMPOUNDS Inflazome Limited (IE) 2021-01-06 EP disclosed
EP-3759078-A1 NOVEL COMPOUNDS Inflazome Limited (IE) 2021-01-06 EP disclosed
EP-3759084-A1 PHENYLSULFONYLUREA DERIVATIVES USEFUL AS NLRP3 INHIBITORS Inflazome Limited (IE) 2021-01-06 EP disclosed
EP-3107898-B1 1,2-SUBSTITUTED CYCLOPENTANES AS OREXIN RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICALS CO (JP) 2021-01-06 EP disclosed
EP-3377110-B1 NANOPARTICLES BASED ON OPTIONALLY ALKOXYLATED POLY(ALKYL CYANOACRYLATES) HAVING A DEFINED DEGREE OF POLYMERIZATION ABBVIE DEUTSCHLAND (DE) 2021-01-06 EP disclosed
CN-108290893-B Dihydroperidinone derivatives, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2021-01-05 CN disclosed
CN-107793395-B Fibroblast growth factor receptor inhibitors and uses thereof 南京药捷安康生物科技有限公司 2021-01-05 CN disclosed
US-10881660-B2 Fatty liver disease treatment using glucocorticoid and mineralocorticoid receptor antagonists CORCEPT THERAPEUTICS, INC. (US) 2021-01-05 US disclosed
US-10882866-B1 Spiro[3H-indole-3,2′-pyrrolidin]-2(1H)-one compounds and derivatives as MDM2-P53 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2021-01-05 US disclosed
US-10882847-B2 Inhibitors of KRAS G12C mutant proteins ARAXES PHARMA LLC (US) 2021-01-05 US disclosed
CN-112176418-A High-flux compound library construction and screening method and reaction device 中国科学院上海有机化学研究所 2021-01-05 CN disclosed
CN-107454903-B Water-soluble fluorescent or colored dyes containing conjugated groups 索尼公司 2021-01-01 CN disclosed
US-20200407340-A1 SULFONAMIDE DERIVATES AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2020-12-31 US disclosed
US-20200407375-A1 PROTECTIVE GROUPS AND METHODS FOR PROTECTING BENZOXABOROLES OR OXABOROLES UNIVERSITY OF THE SCIENCES (US) 2020-12-31 US disclosed
US-20200405730-A1 PI3KGAMMA INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-12-31 US disclosed
WO-2020263703-A1 ENHANCEMENT OF NUCLEIC ACID POLYMERIZATION BY AROMATIC COMPOUNDS STRATOS GENOMICS, INC. (US) 2020-12-30 WO disclosed
WO-2020260252-A1 NEW MACROCYCLIC COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-12-30 WO disclosed
WO-2020264120-A1 PI3KGAMMA INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-12-30 WO disclosed
WO-2020264128-A1 METHODS AND COMPOSITIONS RELATED TO PRINTED CELLULAR NICHES FOR PRESERVING AND CONTROLLING SYNTHETIC MICROBIAL CONSORTIA BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2020-12-30 WO disclosed
EP-3755317-A1 PROTEIN ARGININE METHYLTRANSFERASE 5 (PRMT5) DEGRADATION / DISRUPTION COMPOUNDS AND METHODS OF USE Icahn School of Medicine at Mount Sinai (US) 2020-12-30 EP disclosed
EP-3755694-A1 NEW BENZIMIDAZOLE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS Boehringer Ingelheim International GmbH (DE) 2020-12-30 EP disclosed
EP-3455226-B1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME LUNDBECK LA JOLLA RESEARCH CENTER INC (US) 2020-12-30 EP disclosed
EP-3368582-B1 POLYURETHANE/UREA MATERIALS COMMW SCIENT IND RES ORG (AU) 2020-12-30 EP disclosed
CN-112154146-A Serine threonine kinase (AKT) degradation/disruption compounds and methods of use 西奈山伊坎医学院 2020-12-29 CN disclosed
CN-112154147-A Substituted phenylthiouracils, their salts and their use as herbicides 先正达农作物保护股份公司 2020-12-29 CN disclosed
CN-112142735-A Condensed cyanopyridine compound, preparation method and application 上海凌达生物医药有限公司 2020-12-29 CN disclosed
US-10875842-B2 Inhibitors of KRAS G12C mutant proteins ARAXES PHARMA LLC (US) 2020-12-29 US disclosed
CN-112135818-A 4-hydroxypiperidine derivatives and their use as inhibitors of ubiquitin-specific protease 19(USP19) 阿尔麦克探索有限公司 2020-12-25 CN disclosed
CN-112125901-A Inhibitors of lysine-specific demethylase-1 赛尔基因昆蒂赛尔研究公司 2020-12-25 CN disclosed
US-20200399270-A1 INDOLIZINE COMPOUNDS, PREPARATION METHOD AND USE THEREOF HAIHE BIOPHARMA CO., LTD. (CN) 2020-12-24 US disclosed
US-20200399266-A1 SERINE THREONINE KINASE (AKT) DEGRADATION / DISRUPTION COMPOUNDS AND METHODS OF USE ICAHN SCHOOL MED MOUNT SINAI (US) 2020-12-24 US disclosed
US-20200397798-A1 COMBINATION THERAPIES WITH FARNESOID X RECEPTOR (FXR) MODULATORS AKARNA THERAPEUTICS, LTD. (GB) 2020-12-24 US disclosed
US-20200399243-A1 NOVEL COMPOUNDS INFLAZOME LIMITED (IE) 2020-12-24 US disclosed
US-20200399242-A1 NOVEL COMPOUNDS INFLAZOME LIMITED (IE) 2020-12-24 US disclosed
WO-2020254197-A1 ADRENOMEDULLIN-ANALOGUES FOR LONG-TERM STABILIZATION AND THEIR USE BAYER AKTIENGESELLSCHAFT (DE) 2020-12-24 WO disclosed
WO-2020254451-A1 ANTICANCER COMBINATION THERAPY BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-12-24 WO disclosed
WO-2020257733-A1 HISTONE DEMETHYLASE INHIBITORS FOR TREATING CANCERS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2020-12-24 WO disclosed
WO-2020257734-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR TREATING, AMELIORATING, OR PREVENTING BACTERIAL INFECTIONS BAYLOR COLLEGE OF MEDICINE (US) 2020-12-24 WO disclosed
WO-2020254489-A1 BENZYLPHENYL HYDROXYISOXAZOLINES AND ANALOGUES AS NEW ANTIFUNGAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-12-24 WO disclosed
WO-2020254490-A1 PHENOXYPHENYL HYDROXYISOXAZOLINES AND ANALOGUES AS NEW ANTIFUNGAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-12-24 WO disclosed
EP-3753941-A1 PYRIMIDINE-FUSED CYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Shanghai Blueray Biopharma Co., Ltd. (CN) 2020-12-23 EP disclosed
US-10870634-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-12-22 US disclosed
CN-112105364-A Compositions and methods for treating insulin resistance 坦普尔大学 2020-12-18 CN disclosed
CN-107001945-B Aromatic hydrogenation catalyst and use thereof 埃克森美孚研究工程公司 2020-12-18 CN disclosed
CN-112105355-A ABHD12 inhibitors and methods of making and using the same 斯克利普斯研究所 2020-12-18 CN disclosed
CN-112094269-A Saturated six-membered ring heterocyclic compound, preparation method and application 上海凌达生物医药有限公司 2020-12-18 CN disclosed
US-20200390100-A1 SUBSTITUTED N-HETEROCYCLYL- AND N-HETEROARYL-TETRAHYDROPYRIMIDINONES AND THE SALTS THEREOF, AND THE USE OF SAME AS HERBICIDAL ACTIVE SUBSTANCES BAYER AG (DE) 2020-12-17 US disclosed
US-20200392075-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF INSULIN RESISTANCE UNIV TEMPLE (US) 2020-12-17 US disclosed
US-20200390792-A1 MODIFIED OLIGOMERIC COMPOUNDS COMPRISING TRICYCLO-DNA NUCLEOSIDES AND USES THEREOF SYNTHENA AG (CH) 2020-12-17 US disclosed
US-20200392136-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL ELI LILLY AND COMPANY 2020-12-17 US disclosed
US-20200392082-A1 METHODS AND COMPOSITIONS OF ISOINDOLINE-1,3-DIONE AND ISOINDOLE PRODRUGS USEFUL FOR TREATING CANCER, ULCERATIVE COLITIS AND RELATED INFLAMMATORY DISEASES PRO-ONICS PHARMACEUTCIALS LLC 2020-12-17 US disclosed
EP-3508482-B1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR AND USE THEREOF NANJING TRANSTHERA BIOSCIENCES CO LTD (CN) 2020-12-16 EP disclosed
CN-112088006-A Compositions and methods for treating insulin resistance 坦普尔大学 2020-12-15 CN disclosed
CN-112088001-A MAGL inhibitors 隆德贝克拉荷亚研究中心有限公司 2020-12-15 CN disclosed
CN-109721599-B Amino-substituted nitrogen-containing fused ring compound and preparation method and application thereof 上海凌达生物医药有限公司 2020-12-15 CN disclosed
US-10865384-B2 2,4,5-tri-substituted azole-based casein kinase 1 inhibitors as inducers for cardiomyogenesis AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2020-12-15 US disclosed
US-10865310-B2 Ultra bright dimeric or polymeric dyes SONY CORPORATION OF AMERICA (US) 2020-12-15 US disclosed
US-10864202-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2020-12-15 US disclosed
US-20200388880-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ELECTROLYTE ADDITIVE COMPOUNDS ENEVATE CORPORATION 2020-12-10 US disclosed
US-20200388881-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH FUNCTIONAL THIOPHENE COMPOUNDS OR DERIVATIVES OF THIOPHENE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2020-12-10 US disclosed
US-20200388876-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH SILICON CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2020-12-10 US disclosed
US-20200388885-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH LIPO2F2 SALT-CONTAINING ELECTROLYTE FORMULATIONS ENEVATE CORPORATION 2020-12-10 US disclosed
US-20200383985-A1 Inhibitors of Protease Activated Receptor-2 MONASH UNIVERSITY (AU) 2020-12-10 US disclosed
US-20200383991-A1 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2020-12-10 US disclosed
US-20200385364-A1 FUSED N-HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC 2020-12-10 US disclosed
US-20200385409-A1 BENZOXABOROLE COMPOUNDS AND FORMULATIONS THEREOF Boragen, Inc. 2020-12-10 US disclosed
US-20200388836-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH FUNCTIONAL TERTHIOPHENE COMPOUND OR THIOPHENE OLIGOMER COMPOUND CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2020-12-10 US disclosed
US-20200388837-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH SILYL AMINE COMPOUNDS OR DERIVATIVES OF SILYL AMINE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2020-12-10 US disclosed
US-20200388882-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH FLUORINATED ELECTROLYTE FORMULATIONS ENEVATE CORPORATION 2020-12-10 US disclosed
US-20200388879-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH FUNCTIONALIZED LINEAR SULFONATE ESTER DERIVATIVE COMPOUND CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2020-12-10 US disclosed
US-20200385388-A1 PROCESSES FOR PREPARING ISOQUINOLINONES AND SOLID FORMS OF ISOQUINOLINONES INFINITY PHARMACEUTICALS, INC. 2020-12-10 US disclosed
WO-2020245097-A1 SUBSTITUTED PYRIDINYLOXYPYRIDINES AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-12-10 WO disclosed
WO-2020247540-A1 ADENOSINE ANALOGS FOR THE TREATMENT OF DISEASE BIOINTERVENE, INC. (US) 2020-12-10 WO disclosed
WO-2020247546-A1 ADENOSINE ANALOGS FOR THE TREATMENT OF DISEASE BIOINTERVENE, INC. (US) 2020-12-10 WO disclosed
WO-2020247860-A1 BROAD SPECTRUM ANTIVIRAL COMPOUNDS TARGETING THE SKI COMPLEX UNIVERSITY OF MARYLAND, BALTIMORE (US) 2020-12-10 WO disclosed
WO-2020247928-A1 PHOTOPOLYMERIZABLE THERMOPLASTICS AND METHODS OF MAKING AND USING SAME THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2020-12-10 WO disclosed
EP-3747868-A1 SUBSTITUTED PHENOXYPYRIDINES, THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS Bayer AG (DE) 2020-12-09 EP disclosed
EP-3747867-A1 SUBSTITUTED PYRIDINYLOXYANILINES, THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS Bayer AG (DE) 2020-12-09 EP disclosed
EP-3746445-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL ELI LILLY AND COMPANY (US) 2020-12-09 EP disclosed
EP-3746430-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES Padforward LLC (US) 2020-12-09 EP disclosed
EP-3747865-A1 PENTAFLUOROSULFANYL-SUBSTITUTED AMIDE COMPOUND, PREPARATION METHOD THEREFOR, AND MEDICAL APPLICATION THEREOF Beijing InnoCare Pharma Tech Co., Ltd. (CN) 2020-12-09 EP disclosed
EP-3344243-B1 COMPOUNDS AND METHODS USEFUL FOR TREATING OR PREVENTING HEMATOLOGICAL CANCERS BROAD INST INC (US) 2020-12-09 EP disclosed
EP-3747472-A1 THERAPEUTIC COMBINATIONS OF A CD19 INHIBITOR AND A BTK INHIBITOR Acerta Pharma B.V. (NL) 2020-12-09 EP disclosed
CN-111592525-B Spiro aromatic ring compound and application thereof 上海奕拓医药科技有限责任公司 2020-12-08 CN disclosed
US-10858343-B2 Inhibitors of KRAS G12C mutant proteins ARAXES PHARMA LLC (US) 2020-12-08 US disclosed
US-10858316-B2 Small molecule inhibitors of the MCL-1 oncoprotein and uses thereof UNIVERSITY OF MARYLAND, BALTIMORE (US) 2020-12-08 US disclosed
US-10858338-B2 Inhibitors for soluble epoxide hydrolase (SEH) and fatty acid amide hydrolase (FAAH) THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-12-08 US disclosed
CN-112040947-A NSD family inhibitors and methods of treatment therewith 密歇根大学董事会 2020-12-04 CN disclosed
US-20200377553-A1 ANTIBODY SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING CALIFORNIA INSTITUTE OF TECHNOLOGY 2020-12-03 US disclosed
US-20200377476-A1 NEW BENZIMIDAZOLE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-12-03 US disclosed
WO-2020243008-A1 SENSORS AND METHODS FOR RAPID MICROBIAL DETECTION BAMBU VAULT LLC (US) 2020-12-03 WO disclosed
WO-2020023910-A9 METHODS FOR TREATING DISEASES ASSOCIATED WITH ABNORMAL ACVR1 EXPRESSION AND ACVR1 INHIBITORS FOR USE IN THE SAME SUMITOMO DAINIPPON PHARMA ONCOLOGY, INC. (US) 2020-12-03 WO disclosed
EP-3743126-A1 FLUORESCENT POLYMERIC COATING FILM FOR MEDICAL DEVICES Université de Strasbourg (FR) 2020-12-02 EP disclosed
EP-3310773-B1 SUBSTITUTED 4-BENZYL AND 4-BENZOYL PIPERIDINE DERIVATIVES 89BIO LTD (IL) 2020-12-02 EP disclosed
EP-3160952-B1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2020-12-02 EP disclosed
EP-3283462-B1 FUSED-TRICYCLIC INHIBITORS OF KRAS AND METHODS OF USE THEREOF ARAXES PHARMA LLC (US) 2020-12-02 EP disclosed
CN-107108522-B Benzimidazol-2-amines as mIDH1 inhibitors 德国癌症研究中心 2020-12-01 CN disclosed
US-10851057-B2 1,4-substituted piperidine derivatives 89BIO LTD (IL) 2020-12-01 US disclosed
US-10849898-B2 Treatment of relapsed and/or refractory solid tumors and non-Hodgkin's lymphomas CELGENE QUANTICEL RESEARCH, INC. (US) 2020-12-01 US disclosed
CN-107501297-B Phenothiazine-pyridine compounds and uses thereof 香港中文大学 2020-12-01 CN disclosed
US-RE48335-E1 Polymyxin derivatives as antimicrobial compounds MONASH UNIVERSITY (AU) 2020-12-01 US disclosed
CN-112011002-A Method for controlled radical polymerization and apparatus for controlled radical polymerization 立邦工业涂料(上海)有限公司 2020-12-01 CN disclosed
CN-112004537-A Selective histone deacetylase inhibitors for the treatment of human diseases 穿梭药业公司 2020-11-27 CN disclosed
CN-112004790-A Novel indoleamine 2, 3-dioxygenase inhibitor and preparation method and application thereof 信达生物制药(苏州)有限公司 2020-11-27 CN disclosed
US-20200369658-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2020-11-26 US disclosed
WO-2020236524-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR KINASES KINNATE BIOPHARMA INC. (US) 2020-11-26 WO disclosed
WO-2020236556-A1 METHODS OF PREPARING MACROCYCLIC INDOLES THE BROAD INSTITUTE, INC. (US) 2020-11-26 WO disclosed
WO-2020236841-A2 ANTIBODY DRUG CONJUGATES HAVING LINKERS COMPRISING HYDROPHILIC GROUPS NOVARTIS AG (CH) 2020-11-26 WO disclosed
WO-2020236825-A2 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE NOVARTIS AG (CH) 2020-11-26 WO disclosed
WO-2020236817-A2 MCL-1 INHIBITOR ANTIBODY-DRUG CONJUGATES AND METHODS OF USE NOVARTIS AG (CH) 2020-11-26 WO disclosed
US-20200369633-A1 DIHYDROOXADIAZINONES BAYER AKTIENGESELLSCHAFT (DE) 2020-11-26 US disclosed
US-20200369639-A1 TRICYCLO-DNA NUCLEOSIDE PRECURSORS AND PROCESSES FOR PREPARING THE SAME SYNTHENA AG (CH) 2020-11-26 US disclosed
US-20200373620-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ETHER CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORP (US) 2020-11-26 US disclosed
US-20200369695-A1 ORGANOPHOSPHATE DERIVATIVES JANUARY THERAPEUTICS, INC. 2020-11-26 US disclosed
EP-3740472-A1 TRICYCLO-DNA NUCLEOSIDE PRECURSORS AND PROCESSES FOR PREPARING THE SAME Synthena AG (CH) 2020-11-25 EP disclosed
EP-3741749-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2020-11-25 EP disclosed
EP-3741742-A1 METHODS FOR THE TREATMENT OF DIABETIC RETINOPATHY AND OTHER OPHTHALMIC DISEASES Acucela Inc. (US) 2020-11-25 EP disclosed
US-10844054-B2 Compounds for pain treatment, compositions comprising same, and methods of using same CERSCI THERAPEUTICS, INC. (US) 2020-11-24 US disclosed
CN-111983219-A Polymer dot compositions and related methods 华盛顿大学商业中心 2020-11-24 CN disclosed
US-10844079-B2 Spiro aromatic ring compound and application thereof ETERN BIOPHARMA (SHANGHAI) CO., LTD. (CN) 2020-11-24 US disclosed
US-20200361895-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LIMITED (IE) 2020-11-19 US disclosed
US-20200361894-A1 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS NATIONAL YANG MING CHIAO TUNG UNIVERSITY (TW) 2020-11-19 US disclosed
US-20200361927-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2020-11-19 US disclosed
EP-3519385-B1 CYANOPYRROLIDINE DERIVATIVES WITH ACTIVITY AS INHIBITORS OF USP30 MISSION THERAPEUTICS LTD (GB) 2020-11-18 EP disclosed
EP-3738960-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2020-11-18 EP disclosed
EP-3737376-A1 SELECTIVE HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF HUMAN DISEASE Shuttle Pharmaceuticals, Inc. (US) 2020-11-18 EP disclosed
US-10836761-B2 Cinchonine-derived catalysts and methods of using same BRANDEIS UNIVERSITY (US) 2020-11-17 US disclosed
US-10836789-B2 Inhibitors of glucocorticoid receptor ORIC PHARMACEUTICALS, INC. (US) 2020-11-17 US disclosed
US-10836688-B2 Organic reactions carried out in aqueous solution in the presence of a hydroxyalkyl(alkyl)cellulose or an alkylcellulose ABBVIE INC. (US) 2020-11-17 US disclosed
US-10836728-B2 Substituted 3-dialkylaminomethyl-piperidin-4-yl-benzamides and methods of making and using same MEBIAS DISCOVERY, INC. (US) 2020-11-17 US disclosed
WO-2020227264-A1 FLUORENE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS FACEBOOK TECHNOLOGIES, LLC (US) 2020-11-12 WO disclosed
WO-2020227296-A1 THERMALLY REVERSIBLE AND REORGANIZABLE CROSSLINKING POLYMERS FOR VOLUME BRAGG GRATINGS FACEBOOK TECHNOLOGIES, LLC (US) 2020-11-12 WO disclosed
WO-2020227020-A1 INHIBITORS OF RAF KINASES KINNATE BIOPHARMA INC. (US) 2020-11-12 WO disclosed
WO-2020227305-A1 LATENT IMAGING FOR VOLUME BRAGG GRATINGS FACEBOOK TECHNOLOGIES, LLC (US) 2020-11-12 WO disclosed
WO-2020227325-A1 HETEROBIFUNCTIONAL COMPOUNDS AS DEGRADERS OF HPK1 ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2020-11-12 WO disclosed
WO-2020227276-A1 THIANTHRENE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS FACEBOOK TECHNOLOGIES, LLC (US) 2020-11-12 WO disclosed
US-20200354594-A1 THERMALLY REVERSIBLE AND REORGANIZABLE CROSSLINKING POLYMERS FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2020-11-12 US disclosed
US-20200354341-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS SYGNATURE DISCOVERY LIMITED (GB) 2020-11-12 US disclosed
US-20200354325-A1 BENZOSULFONYL COMPOUNDS VIVACE THERAPEUTICS, INC. 2020-11-12 US disclosed
US-20200354354-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2020-11-12 US disclosed
US-20200352966-A1 NICOTINAMIDE MONONUCLEOTIDE DERIVATIVES AND THEIR USES METROBIOTECH, LLC 2020-11-12 US disclosed
US-20200355997-A1 THIANTHRENE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2020-11-12 US disclosed
US-20200352915-A1 CAR ACTIVATOR AGENTS FOR CYCLOPHOSPHAMIDE-BASED TREATMENTS OF CANCER NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2020-11-12 US disclosed
US-20200354311-A1 FLUORENE DERIVATIZED MONOMERS AND POLYMERS FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2020-11-12 US disclosed
US-20200354496-A1 LATENT IMAGING FOR VOLUME BRAGG GRATINGS META PLATFORMS TECHNOLOGIES, LLC 2020-11-12 US disclosed
US-20200354367-A1 COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-11-12 US disclosed
EP-3736279-A1 NOVEL PRECATALYST SCAFFOLDS FOR CROSS-COUPLING REACTIONS, AND METHODS OF MAKING AND USING SAME Yale University (US) 2020-11-11 EP disclosed
EP-3735409-A1 ENHANCEMENT OF NUCLEIC ACID POLYMERIZATION BY AROMATIC COMPOUNDS Stratos Genomics Inc. (US) 2020-11-11 EP disclosed
EP-3735404-A1 ASK1 INHIBITOR COMPOUNDS AND USES THEREOF Seal Rock Therapeutics, Inc. (US) 2020-11-11 EP disclosed
US-10829464-B2 Benzoheterocyclic alkylamine compounds and use thereof EAST CHINA UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2020-11-10 US disclosed
US-10829458-B2 Substituted quinazoline compounds and methods of use thereof ARAXES PHARMA LLC (US) 2020-11-10 US disclosed
US-10829440-B2 Antibacterial compounds and methods of making and using same BROWN UNIVERSITY (US) 2020-11-10 US disclosed
US-10829792-B2 Biocatalytic synthesis of strained carbocycles CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2020-11-10 US disclosed
US-10829487-B2 Benzylamino substituted pyridopyrimidinones and derivatives as SOS1 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-11-10 US disclosed
CN-111909083-A Histone demethylase inhibitors 赛尔基因昆蒂赛尔研究公司 2020-11-10 CN disclosed
CN-111902399-A Enantioselective hydrogenation of 4-substituted 1, 2-dihydroquinolines in the presence of chiral iridium catalysts 拜耳公司 2020-11-06 CN disclosed
CN-107108554-B 1-cyclohexyl-2-phenylaminobenzimidazole as MIDH1 inhibitor for treating tumors 德国癌症研究中心 2020-11-06 CN disclosed
CN-106660987-B Inhibitors of lysine-specific demethylase-1 赛尔基因昆蒂赛尔研究公司 2020-11-06 CN disclosed
US-20200347248-A1 PHOTO-CLEAVABLE PRIMER COMPOSITIONS AND METHODS OF USE ENVISTA (US) 2020-11-05 US disclosed
US-20200347009-A1 BICYCLIC COMPOUNDS VIVACE THERAPEUTICS, INC. 2020-11-05 US disclosed
US-20200345717-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC. (US) 2020-11-05 US disclosed
US-20200347052-A1 INHIBITORS OF RAF KINASES Pierre Fabre Médicament (FR) 2020-11-05 US disclosed
US-20200347247-A1 SURFACE PRIMER COMPOSITIONS AND METHODS OF USE ENVISTA (US) 2020-11-05 US disclosed
US-20200347075-A1 BIOACTIVE CONJUGATE, PREPARATION METHOD THEREFOR AND USE THEREOF SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2020-11-05 US disclosed
US-20200347061-A1 CLASS OF AMINO-SUBSTITUTED NITROGEN-CONTAINING FUSED RING COMPOUNDS, PREPARATION METHOD THEREFOR, AND USE THEREOF SHANGHAI RINGENE BIOPHARMA CO., LTD. (CN) 2020-11-05 US disclosed
US-20200347243-A1 FLUORESCENT POLYMERIC COATING FILM FOR MEDICAL DEVICES UNIVERSITE DE STRASBOURG (FR) 2020-11-05 US disclosed
WO-2020223530-A1 GEMCITABINE PRODRUGS CURE BIOPHARMA INC. (US) 2020-11-05 WO disclosed
WO-2020223517-A1 METHODS OF MAKING OLIGOPOTENT AND UNIPOTENT PRECURSORS TRANSFUSION HEALTH, LLC (US) 2020-11-05 WO disclosed
US-10822312-B2 Substituted quinazoline compounds and methods of use ARAXES PHARMA LLC (US) 2020-11-03 US disclosed
US-10821103-B2 Substituted pyridinone-containing trycyclic compounds, and methods using same ARBUTUS BIOPHARMA CORPORATION (CA) 2020-11-03 US disclosed
US-10822434-B2 Catalyst systems and polymerization processes for using the same EXXONMOBIL CHEMICAL PATENTS INC. (US) 2020-11-03 US disclosed
CN-107814798-B 3-substituted acrylic acid compound and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2020-11-03 CN disclosed
CN-106458996-B Fused pyrimidines as inhibitors of the p97 complex 克里弗生物科学公司 2020-11-03 CN disclosed
CN-105820103-B N-benzoyloxy-substituted benzopyrroline-2-ketone derivative and application thereof 北京韩美药品有限公司 2020-11-03 CN disclosed
CN-111885914-A Compositions and methods for producing expanded hematopoietic stem cells using fluorene derivatives 投资健康有限责任公司 2020-11-03 CN disclosed
CN-111848573-A Benzothiophene amide compounds, and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2020-10-30 CN disclosed
CN-111867646-A Fluorescent polymer coated films for medical devices 斯特拉斯堡大学 2020-10-30 CN disclosed
US-20200339541-A1 ALKYNYL-SUBSTITUTED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF BEIJING INNOCARE PHARMA TECH CO., LTD. (CN) 2020-10-29 US disclosed
US-20200340024-A1 METHODS AND ENZYME CATALYSTS FOR THE SYNTHESIS OF NON-CANONICAL AMINO ACIDS CALIFORNIA INSTITUTE OF TECHNOLOGY 2020-10-29 US disclosed
WO-2020216701-A1 ACYL SULFONAMIDES FOR TREATING CANCER BAYER AKTIENGESELLSCHAFT (DE) 2020-10-29 WO disclosed
EP-3727386-A1 INHIBITORS OF PROTEASE ACTIVATED RECEPTOR-2 Takeda Pharmaceutical Company Limited (JP) 2020-10-28 EP disclosed
EP-3728254-A1 NOVEL BENZYLAMINO SUBSTITUTED PYRIDOPYRIMIDINONES AND DERIVATIVES AS SOS1 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2020-10-28 EP disclosed
EP-3727677-A1 METHODS OF PRODUCING ORGANOSILICA MATERIALS AND USES THEREOF ExxonMobil Research and Engineering Company (US) 2020-10-28 EP disclosed
EP-3728235-A1 SUBSTITUTED THIOPHENYL URACILS, SALTS THEREOF AND THE USE THEREOF AS HERBICIDAL AGENTS Syngenta Crop Protection AG (CH) 2020-10-28 EP disclosed
EP-3728237-A1 SUBSTITUTED THIOPHENYL URACILS, SALTS THEREOF AND THE USE THEREOF AS HERBICIDAL AGENTS Syngenta Crop Protection AG (CH) 2020-10-28 EP disclosed
EP-3728214-A1 SUBSTITUTED N-HETEROCYCLYL- AND N-HETEROARYL-TETRAHYDROPYRIMIDINONES AND THE SALTS THEREOF, AND THE USE OF SAME AS HERBICIDAL ACTIVE SUBSTANCES Bayer Aktiengesellschaft (DE) 2020-10-28 EP disclosed
CN-111825595-A Sodium channel blockers 山东轩竹医药科技有限公司 2020-10-27 CN disclosed
CN-107074787-B Inhibitors of lysine-specific demethylase-1 赛尔基因昆蒂赛尔研究公司 2020-10-27 CN disclosed
US-10815229-B1 Benzenesulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2020-10-27 US disclosed
US-10815234-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-10-27 US disclosed
CN-111808135-A Functionally modified oligonucleotides and subunits thereof 萨勒普塔医疗公司 2020-10-23 CN disclosed
CN-107531709-B Beta-lactamase inhibitor and use thereof 吉林四环制药有限公司 2020-10-23 CN disclosed
US-20200331888-A1 1-CYANO-PYRROLIDINE DERIVATIVES AS DUB INHIBITORS MISSION THERAPEUTICS LIMITED (GB) 2020-10-22 US disclosed
US-20200331874-A1 NON-ATP/CATALYTIC SITE p38 MITOGEN ACTIVATED PROTEIN KINASE INHIBITORS UNIVERSITY OF MARYLAND, BALTIMORE 2020-10-22 US disclosed
US-20200331850-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LIMITED (IE) 2020-10-22 US disclosed
US-20200331886-A1 NOVEL COMPOUNDS INFLAZOME LIMITED (IE) 2020-10-22 US disclosed
WO-2020214854-A1 SILK HAIR CARE COMPOSITIONS EVOLVED BY NATURE, INC. (US) 2020-10-22 WO disclosed
WO-2020214734-A1 BICYCLIC COMPOUNDS VIVACE THERAPEUTICS, INC. (US) 2020-10-22 WO disclosed
WO-2019222431-A9 OXADIAZOLE COMPOUNDS VIVACE THERAPEUTICS, INC. (US) 2020-10-22 WO disclosed
WO-2020214860-A1 CHEMICALLY LINKED SILK FIBROIN COATINGS AND METHODS OF MAKING AND USING THEREOF EVOLVED BY NATURE, INC. (US) 2020-10-22 WO disclosed
EP-3193851-B1 COMBINATION THERAPIES FOR TREATMENT OF CANCER ARAXES PHARMA LLC (US) 2020-10-21 EP disclosed
EP-3725798-A1 BIOACTIVE CONJUGATE, PREPARATION METHOD THEREFOR AND USE THEREOF Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-10-21 EP disclosed
US-10807982-B2 Bromodomain inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-10-20 US disclosed
CN-111801314-A ASK1 inhibitor compounds and uses thereof 西尔洛克治疗公司 2020-10-20 CN disclosed
CN-111801321-A tricyclic-DNA nucleoside precursors and methods for their preparation 新特纳股份公司 2020-10-20 CN disclosed
US-10807956-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-10-20 US disclosed
US-10808053-B2 Polyethylene compositions and articles made therefrom EXXONMOBIL CHEMICAL PATENTS INC. (US) 2020-10-20 US disclosed
US-10807948-B2 Aromatic compounds and uses thereof PELOTON THERAPEUTICS, INC. (US) 2020-10-20 US disclosed
US-10811727-B2 Silicon-based energy storage devices with ether containing electrolyte additives ENEVATE CORPORATION (US) 2020-10-20 US disclosed
US-10808005-B2 Ligand for orphan nuclear receptor Nur77 and uses thereof IXMEDICINE (XIAMEN) BIOLOGICAL TECHNOLOGY COMPANY LIMITED (CN) 2020-10-20 US disclosed
US-20200325168-A9 WITHANOLIDES USEFUL FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES ARNA THERAPEUTICS INC. (CA) 2020-10-15 US disclosed
WO-2020210139-A1 PYRAZOLESULFONAMIDES AS ANTITUMOR AGENTS PELOTON THERAPEUTICS, INC. (US) 2020-10-15 WO disclosed
EP-3720430-A1 BENZOCARBONYL COMPOUNDS Vivace Therapeutics, Inc. (US) 2020-10-14 EP disclosed
EP-3720436-A1 TUBULIN INHIBITORS Lin Bioscience, Pty Ltd. (AU) 2020-10-14 EP disclosed
EP-3720439-A1 NSD FAMILY INHIBITORS AND METHODS OF TREATMENT THEREWITH The Regents Of The University Of Michigan (US) 2020-10-14 EP disclosed
EP-3464224-B1 PROCESS FOR PREPARING 2,3-UNSATURATED ALCOHOLS BASF SE (DE) 2020-10-14 EP disclosed
EP-3464296-B1 ISOTHIAZOLOPYRIDONES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND/OR PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2020-10-14 EP disclosed
EP-3179990-B1 FATTY ACID SYNTHASE INHIBITOR FOR USE IN THE TREATMENT OF DRUG RESISTANT CANCER SAGIMET BIOSCIENCES INC (US) 2020-10-14 EP disclosed
EP-2928471-B1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2020-10-14 EP disclosed
CN-111771001-A Enhanced nucleic acid polymerization by aromatic compounds 斯特拉托斯基因公司 2020-10-13 CN disclosed
CN-111763217-A Thieno-nitrogen heterocyclic compound, preparation method and application 上海凌达生物医药有限公司 2020-10-13 CN disclosed
CN-107667090-B Pesticidally active oxime and hydrazone derivatives 先正达参股股份有限公司 2020-10-09 CN disclosed
US-20200317696-A1 ULTRA-POTENT VINA ALKALOIDS: ADDED MOLECULAR COMPLEXITY FURTHER DISRUPTS THE TUBLIN DIMER-DIMER INTERFACE NATIONAL INSTITUTES OF HEALTH 2020-10-08 US disclosed
US-20200317695-A1 SPIRO AROMATIC RING COMPOUND AND APPLICATION THEREOF ETERN BIOPHARMA (SHANGHAI) CO., LTD. (CN) 2020-10-08 US disclosed
US-20200315174-A1 SUBSTITUTED THIOPHENYL URACILS, SALTS THEREOF AND THE USE THEREOF AS HERBICIDAL AGENTS SYNGENTA CROP PROTECTION AG (CH) 2020-10-08 US disclosed
US-20200317709-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS Cipla USA, Inc. 2020-10-08 US disclosed
US-20200317690-A1 NOVEL ISOTHIAZOLOPYRIDONES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND/OR PLANT GROWTH REGULATORS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2020-10-08 US disclosed
WO-2020198789-A1 NON-CORE-SHELL POLYMER PARTICLES THE UNIVERSITY OF SYDNEY (AU) 2020-10-08 WO disclosed
WO-2020200154-A1 A CLASS OF THIOPHENE FUSED N-HETEROCYCLIES, PREPARATION METHOD AND USE 上海凌达生物医药有限公司 2020-10-08 WO disclosed
US-20200317637-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LIMITED (IE) 2020-10-08 US disclosed
EP-3409669-B1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD PHARMA INC (US) 2020-10-07 EP disclosed
EP-3716981-A1 COMPOUNDS FOR TREATING NEAR VISION DISORDERS Viewpoint Therapeutics, Inc. (US) 2020-10-07 EP disclosed
EP-3716766-A1 BENZOXABOROLE COMPOUNDS AND FORMULATIONS THEREOF Boragen, Inc. (US) 2020-10-07 EP disclosed
EP-3718573-A1 CHROMOPHORIC POLYMER DOTS WITH NARROW-BAND EMISSION University of Washington Through Its Center for Commercialization (US) 2020-10-07 EP disclosed
CN-108290872-B Cyanopyrrolidine derivatives as DUBs inhibitors 特殊治疗有限公司 2020-10-02 CN disclosed
US-20200308181-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELLTAXIS, LLC 2020-10-01 US disclosed
WO-2020198682-A1 METHODS FOR SYNTHESIZING β-HOMOAMINO ACIDS PROTAGONIST THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2020198058-A1 INHIBITORS OF RAF KINASES KINNATE BIOPHARMA INC. (US) 2020-10-01 WO disclosed
WO-2020193474-A1 SUBSTITUTED 2-HETEROARYLAMINOBENZENES AND THE SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-10-01 WO disclosed
US-20200312481-A1 POLYMER-SILICA HYBRID PDOTS AND METHODS OF USE THEREOF UNIVERSITY OF WASHINGTON 2020-10-01 US disclosed
US-20200308155-A1 Substituted Ureas and Methods of Making and Using Same MEBIAS DISCOVERY, INC. 2020-10-01 US disclosed
US-20200306370-A1 AMINO ACID AND PEPTIDE CONJUGATES AND CONJUGATION PROCESS AUCKLAND UNISERVICES LTD (NZ) 2020-10-01 US disclosed
CN-111727185-A Substituted N-heterocyclyl-and N-heteroaryltetrahydropyrimidines and their salts and their use as herbicidal active substances 拜耳公司 2020-09-29 CN disclosed
CN-111727042-A Tubulin inhibitors 仁新医药私人有限公司 2020-09-29 CN disclosed
US-10787483-B2 Antimicrobial peptidomimetics AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2020-09-29 US disclosed
US-10786480-B2 Combination therapy of a HIF-2-α inhibitor and an immunotherapeutic agent and uses thereof PELOTON THERAPEUTICS, INC. (US) 2020-09-29 US disclosed
US-10787668-B2 Fibrotic treatment MONASH UNIVERSITY (AU) 2020-09-29 US disclosed
CN-111704611-A Aryl spiro SHP2 inhibitor compound, preparation method and application 上海凌达生物医药有限公司 2020-09-25 CN disclosed
CN-111704610-A Pyrrolylamido pyridone compounds, preparation method and application 上海凌达生物医药有限公司 2020-09-25 CN disclosed
US-20200299285-A1 CARBOXYLIC ACID, ACYL SULFONAMIDE AND ACYL SULFAMIDE-DERIVATIZED BICYCLIC AZA-HETEROAROMATICS AS SELECTIVE MCL-1 INHIBITORS AND AS DUAL MCL-1/BCL-2 INHIBITORS UNIVERSITY OF MARYLAND, BALTIMORE 2020-09-24 US disclosed
US-20200299287-A1 AMINOPYRIDINE DERIVATIVES AS TAM FAMILY KINASE INHIBITORS SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2020-09-24 US disclosed
US-20200297727-A1 TREATMENT OF RELAPSED AND/OR REFRACTORY SOLID TUMORS AND NON-HODGKIN'S LYMPHOMAS CELGENE QUANTICEL RESEARCH, INC. (US) 2020-09-24 US disclosed
US-20200299288-A1 AMINOPYRIDINE DERIVATIVES AS TAM FAMILY KINASE INHIBITORS SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2020-09-24 US disclosed
WO-2020190890-A1 NICORANDIL DERIVATIVES Unicycive Therapeutics Inc. (US) 2020-09-24 WO disclosed
WO-2020187123-A1 PYRROLE AMIDOPYRIDONE COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海凌达生物医药有限公司 2020-09-24 WO disclosed
EP-3464267-B1 NEW PHENYLPYRAZOLYLACETAMIDE COMPOUNDS AND DERIVATIVES AS CDK8/CDK19 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2020-09-23 EP disclosed
EP-3712151-A1 SPIRO AROMATIC RING COMPOUND AND APPLICATION THEREOF Etern Biopharma (Shanghai) Co., Ltd. (CN) 2020-09-23 EP disclosed
EP-3710502-A1 POLYMERIZATION PROCESSES ExxonMobil Chemical Patents Inc. (US) 2020-09-23 EP disclosed
EP-3710447-A1 ARYL ANNULATED MACROCYCLIC INDOLE DERIVATIVES Bayer Aktiengesellschaft (DE) 2020-09-23 EP disclosed
EP-3710456-A1 MACROCYCLIC INDOLE DERIVATIVES The Broad Institute, Inc. (US) 2020-09-23 EP disclosed
EP-3710448-A1 MACROCYCLIC CHLORINE SUBSTITUTED INDOLE DERIVATIVES Bayer Aktiengesellschaft (DE) 2020-09-23 EP disclosed
EP-3710449-A1 MACROCYCLIC FLUORINE SUBSTITUTED INDOLE DERIVATIVES AS MCL-1 INHIBITORS, FOR USE IN THE TREATMENT OF CANCER The Broad Institute, Inc. (US) 2020-09-23 EP disclosed
EP-3710450-A1 MACROCYCLIC CHLORINE SUBSTITUTED INDOLE DERIVATIVES Bayer Aktiengesellschaft (DE) 2020-09-23 EP disclosed
EP-3710451-A1 SUBSTITUTED MACROCYCLIC INDOLE DERIVATIVES Bayer Aktiengesellschaft (DE) 2020-09-23 EP disclosed
EP-3710432-A1 TETRAZOLYLPROPYL DERIVATIVES AND THEIR USE AS FUNGICIDES Bayer Aktiengesellschaft (DE) 2020-09-23 EP disclosed
US-10781200-B2 Therapeutic inhibitory compounds ATTUNE PHARMACEUTICALS, INC. (US) 2020-09-22 US disclosed
US-10781211-B2 Spirocycle compounds and methods of making and using same LUNDBECK LA JOLLA RESEARCH CENTER, INC. (US) 2020-09-22 US disclosed
CN-111698991-A Inhibitors of protease activated receptor-2 武田药品工业株式会社 2020-09-22 CN disclosed
CN-111690031-A Glucocorticoid receptor inhibitors 欧瑞克制药公司 2020-09-22 CN disclosed
CN-107438606-B [9, 10-dimethoxy-3- (2-methylpropyl) -1H,2H,3H,4H,6H,7H,11 BH-pyrido- [2,1-A ] isoquinolin-2-yl ] methanol and compounds, compositions, and methods related thereto 纽罗克里生物科学有限公司 2020-09-18 CN disclosed
US-20200291060-A1 NOVEL 7-DEHYDROCHOLESTEROL DERIVATIVES AND METHODS USING SAME WOMEN & INFANTS HOSPITAL OF RHODE ISLAND 2020-09-17 US disclosed
US-20200291023-A1 MAGL INHIBITORS H. LUNDBECK A/S (DK) 2020-09-17 US disclosed
WO-2020182076-A1 USES OF PHOSPHODIESTERASE INHIBITORS 南京药捷安康生物科技有限公司 2020-09-17 WO disclosed
WO-2020182929-A1 SUBSTITUTED UREAS AND DERIVATIVES AS NEW ANTIFUNGAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-09-17 WO disclosed
WO-2020185661-A1 USE OF 8,9-DIHYDROCANNABIDIOL COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-09-17 WO disclosed
US-20200291050-A1 ACYLSULFONAMIDE DERIVATIVES FOR TREATING SENESCENCE-ASSOCIATED DISEASES AND DISORDERS UNITY BIOTECHNOLOGY, INC. 2020-09-17 US disclosed
US-20200291020-A1 NEW [1,6]NAPHTHYRIDINE COMPOUNDS AND DERIVATIVES AS CDK8/CDK19 INHIBITORS BOEHRINGER INGELHEIM RCV GMBH & CO. KG (AT) 2020-09-17 US disclosed
US-20200291058-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. 2020-09-17 US disclosed
US-20200289528-A1 Testosterone Ester Triglyceride Formulations ANTARES PHARMA, INC. (US) 2020-09-17 US disclosed
US-20200291003-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS SYGNATURE DISCOVERY LIMITED (GB) 2020-09-17 US disclosed
US-20200291164-A1 DYNAMIC COVALENT THERMOSET NANOCOMPOSITES AND USES THEREOF NATIONAL SCIENCE FOUNDATION 2020-09-17 US disclosed
US-20200289458-A1 TOPICAL FORMULATIONS OF CANNABINOIDS AND USE THEREOF IN THE TREATMENT OF PAIN INMED PHARMACEUTICALS INC (CA) 2020-09-17 US disclosed
EP-3555063-B1 6-AMINO-QUINOLINONE COMPOUNDS AND DERIVATIVES AS BCL6 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2020-09-16 EP disclosed
EP-3707137-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS Inflazome Limited (IE) 2020-09-16 EP disclosed
EP-3706736-A1 ASH1L DEGRADERS AND METHODS OF TREATMENT THEREWITH The Regents of the University of Michigan (US) 2020-09-16 EP disclosed
EP-3707134-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS Inflazome Limited (IE) 2020-09-16 EP disclosed
EP-3706737-A1 ASH1L INHIBITORS AND METHODS OF TREATMENT THEREWITH The Regents of the University of Michigan (US) 2020-09-16 EP disclosed
EP-3708565-A1 PYRIMIDINYLOXYPHENYLAMIDINES AND THE USE THEREOF AS FUNGICIDES Bayer AG (DE) 2020-09-16 EP disclosed
CN-111658653-A Use of phosphodiesterase inhibitors 南京药捷安康生物科技有限公司 2020-09-15 CN disclosed
US-10774078-B2 Compounds MISSION THERAPEUTICS LTD (GB) 2020-09-15 US disclosed
US-10772893-B2 2-(morpholin-4-yl)-1,7-naphthyridines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2020-09-15 US disclosed
CN-111655666-A Anti-inflammatory, anti-cancer and anti-angiogenic compounds, pharmaceutical compositions and methods of making and using the same 麦迪康制药公司 2020-09-11 CN disclosed
CN-111655035-A Benzoxaborole compounds and formulations thereof 博瑞金股份有限公司 2020-09-11 CN disclosed
CN-111655257-A ASH1L inhibitors and methods of treatment therewith 密歇根大学董事会 2020-09-11 CN disclosed
CN-111655693-A Inhibition of transient receptor potential A1 ion channels 伊莱利利公司 2020-09-11 CN disclosed
CN-111643512-A Niacinetoside or nicotinamide riboside compositions, reduced derivatives thereof and uses thereof 可劳迈戴斯有限公司 2020-09-11 CN disclosed
US-20200283372-A1 LIPIDS FOR LIPID NANOPARTICLE DELIVERY OF ACTIVE AGENTS Acuitas Therapeutics, Inc. (CA) 2020-09-10 US disclosed
EP-3270951-B1 BOTULINUM NEUROTOXIN-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING CALIFORNIA INST OF TECHN (US) 2020-09-09 EP disclosed
EP-3003309-B1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS INFINITY PHARMACEUTICALS INC (US) 2020-09-09 EP disclosed
EP-3704117-A1 AZABICYCLO AND DIAZEPINE DERIVATIVES FOR TREATING OCULAR DISORDERS ALCON INC. (CH) 2020-09-09 EP disclosed
EP-3705480-A1 CLASS OF AMINO-SUBSTITUTED NITROGEN-CONTAINING FUSED RING COMPOUNDS, PREPARATION METHOD THEREFOR, AND USE THEREOF Rudong Ringene Pharmaceuticals, Co. Ltd (CN) 2020-09-09 EP disclosed
US-10770197-B2 Polymer-silica hybrid Pdots and methods of use thereof UNIVERSITY OF WASHINGTON (US) 2020-09-08 US disclosed
US-10766903-B2 Piperidine derivatives as inhibitors of ubiquitin specific protease 7 ALMAC DISCOVERY LIMITED (GB) 2020-09-08 US disclosed
US-10766865-B2 PKM2 modulators and methods for their use SUMITOMO DAINIPPON PHARMA ONCOLOGY, INC. (US) 2020-09-08 US disclosed
US-10766902-B2 Wee-1 inhibiting pyrazolopyrimidinone compounds ALMAC DISCOVERY LIMITED (GB) 2020-09-08 US disclosed
CN-106660982-B Histone demethylase inhibitors 赛尔基因昆蒂赛尔研究公司 2020-09-08 CN disclosed
CN-107722036-B Thiophene derivatives 天津合美医药科技有限公司 2020-09-04 CN disclosed
US-20200277251-A1 NOVEL ANTIBACTERIAL COMPOUNDS AND METHODS OF MAKING AND USING SAME NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2020-09-03 US disclosed
US-20200276211-A1 COMPOUNDS FOR TREATING NEAR VISION DISORDERS VIEWPOINT THERAPEUTICS INC (US) 2020-09-03 US disclosed
US-20200277598-A1 Peptide Oligonucleotide Conjugates JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2020-09-03 US disclosed
US-20200275660-A1 TETRAZOLYLPROPYL DERIVATIVES AND THEIR USE AS FUNGICIDES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2020-09-03 US disclosed
US-10759806-B2 Isotopologues of isoquinolinone and quinazolinone compounds and uses thereof as PI3K kinase inhibitors INFINITY PHARMACEUTICALS, INC. (US) 2020-09-01 US disclosed
US-10760078-B2 Oligonucleotide analogues having modified intersubunit linkages and/or terminal groups SAREPTA THERAPEUTICS, INC. (US) 2020-09-01 US disclosed
US-10760052-B2 Method of inhibiting tau phosphorylation Cassava Science, Inc. (US) 2020-09-01 US disclosed
CN-111592541-A Macrocyclic kinase inhibitors and uses thereof 山东轩竹医药科技有限公司 2020-08-28 CN disclosed
CN-111592525-A Spiro aromatic ring compound and application thereof 上海奕拓医药科技有限责任公司 2020-08-28 CN disclosed
CN-111592534-A Novel compounds 特殊治疗有限公司 2020-08-28 CN disclosed
CN-111601601-A Selective P2X3 modulators 贝卢斯医疗咳嗽病公司 2020-08-28 CN disclosed
US-20200271427-A1 LEUCO DYE SHOOTING TARGETS JL DARLING LLC 2020-08-27 US disclosed
US-20200270272-A1 PURIFICATION OF RAPAMYCIN DERIVATIVES USING TEMPERATURE INDUCED PHASE SEPARATION JOHNSON MATTHEY PHARMACEUTICAL MATERIALS, INC. D/B/A JOHNSON MATTHEY PHARMA SERVICES 2020-08-27 US disclosed
US-20200270227-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2020-08-27 US disclosed
US-20200268741-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC. (US) 2020-08-27 US disclosed
EP-3699184-A1 TRIPTOLIDE DERIVATIVE AND PREPARATION METHOD THEREFOR AND USE THEREOF Cinkate Pharmaceutical Intermediates Co., Ltd. (CN) 2020-08-26 EP disclosed
EP-3054956-B1 METHOD FOR INHIBITING GROWTH OF CANCER CELLS PAIN THERAPEUTICS INC (US) 2020-08-26 EP disclosed
EP-3097092-B1 FUSED PYRIMIDINES AS INHIBITORS OF P97 COMPLEX CLEAVE BIOSCIENCES INC (US) 2020-08-26 EP disclosed
CN-107438613-B Compounds and methods for preventing or treating sensory hair cell death 华盛顿大学 2020-08-25 CN disclosed
US-10752628-B2 Compounds and methods for treating synovial sarcomas THE BROAD INSTITUTE, INC. (US) 2020-08-25 US disclosed
US-10752625-B2 Method of making tetrahydronaphthyridinyl nonanoic acid compounds SCIFLUOR LIFE SCIENCES, INC. (US) 2020-08-25 US disclosed
US-10751344-B2 Carbon monoxide-releasing molecules for therapeutic applications and methods for the preparation and use thereof GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2020-08-25 US disclosed
US-10752927-B2 Method for the synthesis of tryptophan analogs in aqueous solvents at reduced temperatures CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2020-08-25 US disclosed
US-10752623-B2 Heteroaryl-substituted sulfonamide compounds and their use as sodium channel inhibitors XENON PHARMACEUTICALS INC. (CA) 2020-08-25 US disclosed
US-10752594-B2 JAK1 and ALK2 inhibitors and methods for their use SUMITOMO DAINIPPON PHARMA ONCOLOGY, INC. (US) 2020-08-25 US disclosed
CN-111587256-A Catalyst system and polymerization process using the same 埃克森美孚化学专利公司 2020-08-25 CN disclosed
CN-111557942-A Treatment of fatty liver disease using glucocorticoid and mineralocorticoid receptor antagonists 科赛普特治疗学股份有限公司 2020-08-21 CN disclosed
CN-111566104-A Spiro aromatic ring compound and application thereof 上海奕拓医药科技有限责任公司 2020-08-21 CN disclosed
US-20200262838-A1 1-CYANO-PYRROLIDINE DERIVATIVES AS INHIBITORS OF USP30 MISSION THERAPEUTICS LIMITED (GB) 2020-08-20 US disclosed
US-20200261590-A1 FACTOR VIII ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC. 2020-08-20 US disclosed
US-20200261432-A1 SUBSTITUTED PYRIDINONE-CONTAINING TRYCYCLIC COMPOUNDS, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2020-08-20 US disclosed
US-20200262834-A1 [9,10-DIMETHOXY-3-(2-METHYLPROPYL)-1H,2H,3H,4H,6H,7H,11BH-PYRIDO-[2,1-A]ISOQUINOLIN-2-YL]METHANOL AND COMPOUNDS, COMPOSITIONS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES, INC. 2020-08-20 US disclosed
US-20200262905-A1 DUAL PDGF/VEGF ANTAGONISTS KODIAK SCIENCES INC. (US) 2020-08-20 US disclosed
EP-3377060-B1 PYRAZOLE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND USES THEREOF LUNDBECK LA JOLLA RESEARCH CENTER INC (US) 2020-08-19 EP disclosed
EP-3197870-B1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC (US) 2020-08-19 EP disclosed
CN-107106562-B Treatment of fatty liver disease using glucocorticoid and mineralocorticoid receptor antagonists 科赛普特治疗学股份有限公司 2020-08-18 CN disclosed
CN-111548313-A Guanidine compounds as medicine for preventing and treating chronic pain 绍兴从零医药科技有限公司 2020-08-18 CN disclosed
US-10744139-B2 Inhibitors of fibroblast growth factor receptor and use thereof NANJING TRANSTHERA BIOSCIENCES CO. LTD. (CN) 2020-08-18 US disclosed
US-10745673-B2 Heme protein catalysts for carbon-boron bond formation in vitro and in vivo CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2020-08-18 US disclosed
US-10745392-B2 Benzenesulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2020-08-18 US disclosed
US-10744205-B2 Antibody drug conjugates of kinesin spindel protein (KSP) inhibitors with anti-CD123-antibodies BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2020-08-18 US disclosed
US-10745385-B2 Covalent inhibitors of KRAS ARAXES PHARMA LLC (US) 2020-08-18 US disclosed
CN-108084125-B Benzoheterocyclylalkylamines and their use 华东理工大学 2020-08-18 CN disclosed
CN-111542318-A ASH1L degradants and methods of treatment therewith 密歇根大学董事会 2020-08-14 CN disclosed
CN-111542324-A Cytotoxic agents and conjugates thereof, methods of making and uses thereof 四川科伦博泰生物医药股份有限公司 2020-08-14 CN disclosed
CN-111542315-A Benzosulfonyl compounds 维瓦斯治疗公司 2020-08-14 CN disclosed
US-20200255413-A1 ANTIBACTERIAL COMPOUNDS BLACKSMITH MEDICINES, INC. 2020-08-13 US disclosed
US-20200255434-A1 INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, INC. 2020-08-13 US disclosed
US-20200255427-A1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2020-08-13 US disclosed
US-20200255371-A1 COMPOSITIONS AND METHODS OF MAKING EXPANDED HEMATOPOIETIC STEM CELLS USING DERIVATIVES OF FLUORENE IMMUNEBRIDGE LLC 2020-08-13 US disclosed
US-20200253954-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC. (US) 2020-08-13 US disclosed
WO-2020160626-A1 CAPTURE OF FLUORINATED CARBON COMPOUNDS THE UNIVERSITY OF QUEENSLAND (AU) 2020-08-13 WO disclosed
WO-2020163334-A1 CURABLE FORMULATION WITH HIGH REFRACTIVE INDEX AND ITS APPLICATION IN SURFACE RELIEF GRATING USING NANOIMPRINTING LITHOGRAPHY FACEBOOK TECHNOLOGIES, LLC (US) 2020-08-13 WO disclosed
EP-3691642-A1 NEW [1,6]NAPHTHYRIDINE COMPOUNDS AND DERIVATIVES AS CDK8/CDK19 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2020-08-12 EP disclosed
EP-3692020-A1 NOVEL COMPOUNDS Inflazome Limited (IE) 2020-08-12 EP disclosed
EP-3691623-A1 BENZOSULFONYL COMPOUNDS Vivace Therapeutics, Inc. (US) 2020-08-12 EP disclosed
EP-3527573-B1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES INC (US) 2020-08-12 EP disclosed
US-10736897-B2 Compounds and methods of use thereof for treatment of cancer ARAXES PHARMA LLC (US) 2020-08-11 US disclosed
US-10738297-B2 3D printable hydrogel materials UNIVERSITY OF WASHINGTON (US) 2020-08-11 US disclosed
CN-106188175-B Treatment of klebsiella pneumoniae infections with antibacterial aminoglycoside compounds 轩竹(北京)医药科技有限公司 2020-08-11 CN disclosed
CN-104411831-B Boronic acid conjugates of oligonucleotide analogs 萨勒普塔医疗公司 2020-08-11 CN disclosed
CN-111526877-A Compounds and compositions for IRE1 inhibition 奥普提卡拉公司 2020-08-11 CN disclosed
CN-111518100-A Cyclopropenoarylbenzofuran substituted nitrogen heteroaryl compound and application thereof 上海青煜医药科技有限公司 2020-08-11 CN disclosed
CN-111527090-A Novel pyrazolo-pyrrolo-pyrimidine-dione derivatives as P2X3 inhibitors 拜耳公司 2020-08-11 CN disclosed
CN-107207735-B Organosilica material 埃克森美孚研究工程公司 2020-08-07 CN disclosed
CN-111511781-A Catalyst system and polymerization process using the same 埃克森美孚化学专利公司 2020-08-07 CN disclosed
CN-111511465-A Method for producing organosilica materials and uses thereof 埃克森美孚研究工程公司 2020-08-07 CN disclosed
WO-2020154775-A1 QUANTUM DOTS AND PROCESSES FOR PREPARATION THEREOF THE UNIVERSITY OF QUEENSLAND (AU) 2020-08-06 WO disclosed
WO-2020157199-A1 ANNULATED DIHYDROPYRIDAZINONE COMPOUNDS AS ANTI-CANCER COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2020-08-06 WO disclosed
WO-2020157236-A1 PYRIDYL SUBSTITUTED DIHYDROOXADIAZINONES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-06 WO disclosed
WO-2020157201-A1 OXADIAZINONE COMPOUNDS FOR THE TREATMENT OF HYPERPROLIFERATIVE DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-06 WO disclosed
WO-2020157194-A1 1,2,4-TRIAZIN-3(2H)-ONE COMPOUNDS FOR THE TREATMENT OF HYPERPROLIFERATIVE DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-06 WO disclosed
WO-2020157189-A1 1,2,4-TRIAZIN-6(1H)-ONE COMPOUNDS FOR THE TREATMENT OF HYPERPROLIFERATIVE DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-06 WO disclosed
US-20200247816-A1 TOPICAL PHOSPHOINOSITIDE 3-KINASE INHIBITORS NAVIRE PHARMA, INC. 2020-08-06 US disclosed
US-20200246474-A1 ASH1L INHIBITORS AND METHODS OF TREATMENT THEREWITH THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2020-08-06 US disclosed
US-20200246330-A1 ANTI-INFLAMMATORY, ANTI-CANCER, AND ANTI-ANGIOGENIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF MAKING AND USING THEREOF MEDICON PHARMACEUTICALS, INC. (US) 2020-08-06 US disclosed
US-20200247756-A1 PROCESSES FOR PREPARING AG-10, ITS INTERMEDIATES, AND SALTS THEREOF Ferro Therapeutics, Inc. 2020-08-06 US disclosed
US-20200249568-A1 CURABLE FORMULATION WITH HIGH REFRACTIVE INDEX AND ITS APPLICATION IN SURFACE RELIEF GRATING USING NANOIMPRINTING LITHOGRAPHY META PLATFORMS TECHNOLOGIES, LLC 2020-08-06 US disclosed
US-20200247783-A1 6-PHENYL-4,5-DIHYDROPYRIDAZIN-3(2H)-ONE DERIVATIVES AS PDE3A AND PDE3B INHIBITORS FOR TREATING CANCER BAYER AKTIENGESELLSCHAFT (DE) 2020-08-06 US disclosed
US-20200247803-A1 SPIRO-CONDENSED PYRROLIDINE DERIVATIVES AS DEUBIQUITYLATING ENZYMES (DUB) INHIBITORS MISSION THERAPEUTICS LIMITED (GB) 2020-08-06 US disclosed
EP-3689876-A1 PDE9 INHIBITOR AND USE THEREOF Nanjing Transthera Biosciences Co. Ltd. (CN) 2020-08-05 EP disclosed
EP-3687972-A1 ANTI-INFLAMMATORY, ANTI-CANCER, AND ANTI-ANGIOGENIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF MAKING AND USING THEREOF Medicon Pharmaceuticals, Inc. (US) 2020-08-05 EP disclosed
EP-3041513-B1 FACTOR VIII ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC (US) 2020-08-05 EP disclosed
US-10730867-B2 Inhibitors of KRAS G12C mutant proteins ARAXES PHARMA LLC (US) 2020-08-04 US disclosed
US-10730825-B2 Methods for the treatment of diabetic retinopathy and other ophthalmic diseases ACUCELA INC. (US) 2020-08-04 US disclosed
US-10729670-B2 Compositions and methods for treatment of insulin resistance Temple University—Of The Commonwealth Systems Of Higher Education (US) 2020-08-04 US disclosed
US-10729680-B2 5-substituted 2-(morpholin-4-yl)-1,7-naphthyridines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2020-08-04 US disclosed
US-10730994-B2 Synthesis of polycarbonate siloxane diols AORTECH INTERNATIONAL PLC (GB) 2020-08-04 US disclosed
CN-106414480-B Polymyxin derivatives as antimicrobial compounds 莫纳什大学 2020-08-04 CN disclosed
CN-111491634-A Organic phosphate derivatives 詹纽瑞治疗公司 2020-08-04 CN disclosed
CN-106488910-B Inhibitors of KRAS G12C 亚瑞克西斯制药公司 2020-07-31 CN disclosed
CN-111471059-A PDE9 inhibitors and uses thereof 南京药捷安康生物科技有限公司 2020-07-31 CN disclosed
WO-2020154683-A1 METHODS OF TREATING DISEASE WITH MAGL INHIBITORS LUNDBECK LA JOLLA RESEARCH CENTER, INC. (US) 2020-07-30 WO disclosed
US-20200237766-A1 PKM2 ACTIVATORS IN COMBINATION WITH REACTIVE OXYGEN SPECIES FOR TREATMENT OF CANCER SUMITOMO PHARMA ONCOLOGY, INC. 2020-07-30 US disclosed
US-20200239632-A1 NOVEL PEPTOID POLYMERS AND METHODS OF USE X-THERMA, INC. (US) 2020-07-30 US disclosed
US-20200239435-A1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS, INC. 2020-07-30 US disclosed
EP-2970341-B1 POLYHEDRAL OLIGOMERIC SILSESQUIOXANE NANOCRYSTAL STABILIZATION LIGANDS NANOSYS INC (US) 2020-07-29 EP disclosed
EP-3310441-B1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES 89BIO LTD (IL) 2020-07-29 EP disclosed
EP-3328384-B1 FIBROTIC TREATMENT UNIV MONASH (AU) 2020-07-29 EP disclosed
EP-3684368-A2 SELECTIVE P2X3 MODULATORS Bellus Health Cough Inc. (CA) 2020-07-29 EP disclosed
EP-3684353-A1 TOPICAL FORMULATIONS OF CANNABINOIDS AND USE THEREOF IN THE TREATMENT OF PAIN Inmed Pharmaceuticals Inc. (CA) 2020-07-29 EP disclosed
US-10723759-B2 Inhibitors of glucocorticoid receptor ORIC PHARMACEUTICALS, INC. (US) 2020-07-28 US disclosed
US-10723725-B2 Aminopyridine derivatives as TAM family kinase inhibitors SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2020-07-28 US disclosed
US-10723738-B2 Inhibitors of KRAS G12C mutant proteins ARAXES PHARMA LLC (US) 2020-07-28 US disclosed
US-10723844-B2 Polyurethane/urea compositions COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2020-07-28 US disclosed
CN-111454165-A Novel lipid and lipid nanoparticle formulations for delivery of nucleic acids 爱康泰生治疗公司 2020-07-28 CN disclosed
CN-111465626-A Polyethylene compositions and films made therefrom 埃克森美孚化学专利公司 2020-07-28 CN disclosed
CN-111448299-A Odorants and compositions comprising odorants 丝趣科尔卡有限公司 2020-07-24 CN disclosed
CN-111448226-A Polymerization process 埃克森美孚化学专利公司 2020-07-24 CN disclosed
CN-111447939-A Method for preparing conjugate 四川科伦博泰生物医药股份有限公司 2020-07-24 CN disclosed
CN-111448223-A Polyethylene compositions and articles made therefrom 埃克森美孚化学专利公司 2020-07-24 CN disclosed
WO-2020150366-A1 SUBSTITUTED POLYCYCLIC CARBOXYLIC ACIDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2020-07-23 WO disclosed
WO-2020150265-A1 PRODRUGS OF ALOX-15 INHIBITORS AND METHODS OF USING THE SAME EMPIRICO INC. (US) 2020-07-23 WO disclosed
US-20200231549-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2020-07-23 US disclosed
US-20200230148-A1 SELECTIVE P2X3 MODULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.3) LIMITED (GB) 2020-07-23 US disclosed
US-20200235415-A1 MEMBRANE ELECTRODE ASSEMBLY WITH FLUORO ALKYL COMPOUND ADDITIVE BALLARD POWER SYSTEMS (CA) 2020-07-23 US disclosed
US-20200231542-A1 CYANOPYRROLIDINES AS DUB INHIBITORS FOR THE TREATMENT OF CANCER MISSION THERAPEUTICS LIMITED (GB) 2020-07-23 US disclosed
EP-3417851-B1 ARYL ETHERS AND USES THEREOF PELOTON THERAPEUTICS INC (US) 2020-07-22 EP disclosed
EP-3209646-B1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS DEUTSCHES KREBSFORSCHUNGSZENTRUM STIFTUNG DES OEFFENTLICHEN RECHTS (DE) 2020-07-22 EP disclosed
US-10717929-B2 Ionic liquid flame retardants IONIC FLAME RETARDANT INC. (US) 2020-07-21 US disclosed
US-10717798-B2 Polymeric composition AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2020-07-21 US disclosed
US-10717742-B2 Spiro[3H-indole-3,2′-pyrrolidin]-2(1H)-one compounds and derivatives as MDM2-P53 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-07-21 US disclosed
US-10716959-B2 Polymer-flavonoid conjugates and hydrogels for biomedical applications AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2020-07-21 US disclosed
CN-111433336-A Odorants and compositions comprising odorants 丝趣科尔卡有限公司 2020-07-17 CN disclosed
US-20200222304-A1 Skin Care Compositions and Methods of Use Thereof UNIGEN, INC. (US) 2020-07-16 US disclosed
US-20200222384-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE, INC. 2020-07-16 US disclosed
WO-2020146805-A1 LIPIDS FOR LIPID NANOPARTICLE DELIVERY OF ACTIVE AGENTS Acuitas Therapeutics, Inc. (CA) 2020-07-16 WO disclosed
WO-2020143626-A1 PDE9 INHIBITOR AND USE THEREOF 南京药捷安康生物科技有限公司 2020-07-16 WO disclosed
US-20200223866-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES, INC. 2020-07-16 US disclosed
US-20200223853-A1 IRREVERSIBLE INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, LLC 2020-07-16 US disclosed
EP-2536485-B1 A SUBSTRATE FOR IMMOBILIZING FUNCTIONAL SUBSTANCES AND METHOD FOR PREPARING THE SAME TEMASEK POLYTECHNIC (SG) 2020-07-15 EP disclosed
EP-3680240-A1 ASYMMETRIC PHASE TRANSFER CATALYSIS MERCK SHARP & DOHME CORP. (US) 2020-07-15 EP disclosed
CN-111407750-A Methods for treating brain cancer 有联生技股份有限公司 2020-07-14 CN disclosed
US-10710981-B2 Alkynyl-substituted heterocyclic compound, preparation method therefor and medical use thereof BEIJING INNOCARE PHARMA TECH CO., LTD. (CN) 2020-07-14 US disclosed
CN-111410659-A PDE9 inhibitors and uses thereof 南京药捷安康生物科技有限公司 2020-07-14 CN disclosed
CN-111407751-A Methods for treating inflammatory disorders 有联生技股份有限公司 2020-07-14 CN disclosed
CN-111407749-A Methods for treating neurodegenerative disorders 有联生技股份有限公司 2020-07-14 CN disclosed
CN-106604746-B Fatty acid synthetase inhibitors for the treatment of drug resistant cancers 3-V生物科学股份有限公司 2020-07-10 CN disclosed
CN-107872956-B Synergistic antifungal composition containing benzoxaborole 宾夕法尼亚州研究基金会 2020-07-10 CN disclosed
US-20200214999-A1 Method for Treating an Inflammatory Disorder ALLIANZ PHARMASCIENCE LTD. 2020-07-09 US disclosed
US-20200214998-A1 Method for Treating a Brain Cancer ALLIANZ PHARMASCIENCE LTD. (TW) 2020-07-09 US disclosed
US-20200215062-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2020-07-09 US disclosed
US-20200215064-A1 COMBINATION THERAPY WITH AXL INHIBITOR AND IMMUNE CHECKPOINT MODULATOR OR ONCOLYTIC VIRUS BERGENBIO ASA (NO) 2020-07-09 US disclosed
WO-2020142557-A1 IRREVERSIBLE INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, LLC (US) 2020-07-09 WO disclosed
WO-2020142559-A1 INHIBITORS OF MENIN-MLL INTERACTION BIOMEA FUSION, LLC (US) 2020-07-09 WO disclosed
US-20200216389-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LIMITED (IE) 2020-07-09 US disclosed
US-20200216401-A1 NOVEL SYRINGOLIN ANALOGUES AND METHODS OF MAKING AND USING SAME UNIV BROWN (US) 2020-07-09 US disclosed
US-20200215035-A1 MICROTUBULE POLYMERIZATION INHIBITOR PRODRUGS AND METHODS OF USING THE SAME UNIVERSITY OF MARYLAND, BALTIMORE 2020-07-09 US disclosed
US-20200214997-A1 Method for Treating a Neurodegenerative Disorder Annji Pharmaceutical Co., Ltd. (TW) 2020-07-09 US disclosed
US-20200216420-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2020-07-09 US disclosed
EP-3677257-A1 METHOD FOR TREATING AN INFLAMMATORY DISORDER WITH A SUBSTITUTED PHENYL-PROPENAL MOIETY Allianz Pharmascience Ltd (TW) 2020-07-08 EP disclosed
EP-3677256-A1 METHOD FOR TREATING A NEURODEGENERATIVE DISORDER WITH A SUBSTITUTED PHENYL-PROPENAL MOITEY Allianz Pharmascience Ltd (TW) 2020-07-08 EP disclosed
EP-3675847-A1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME Lundbeck La Jolla Research Center, Inc. (US) 2020-07-08 EP disclosed
EP-3677255-A1 METHOD FOR TREATING A BRAIN CANCER WITH A SUBSTITUTED PHENYL-PROPENAL MOIETY Allianz Pharmascience Ltd (TW) 2020-07-08 EP disclosed
EP-3675868-A1 TESTOSTERONE ESTER TRIGLYCERIDE FORMULATIONS Antares Pharma, Inc. (US) 2020-07-08 EP disclosed
EP-3675848-A1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME Lundbeck La Jolla Research Center, Inc. (US) 2020-07-08 EP disclosed
EP-3675858-A2 COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION Optikira LLC (US) 2020-07-08 EP disclosed
EP-3074390-B1 AMINOPYRIDINE DERIVATIVES AS TAM FAMILY KINASE INHIBITORS SIGNALCHEM LIFESCIENCES CORP (CA) 2020-07-08 EP disclosed
US-10702608-B2 Factor VIII zwitterionic polymer conjugates KODIAK SCIENCES INC. (US) 2020-07-07 US disclosed
CN-106795191-B Novel precatalyst scaffolds for crosslinking reactions and methods of making and using same 耶鲁大学 2020-07-03 CN disclosed
WO-2020139748-A1 METHODS OF TREATING INFLAMMATORY BOWEL DISEASES THAT TARGET RIPK2 CEDARS-SINAI MEDICAL CENTER (US) 2020-07-02 WO disclosed
US-20200207780-A1 NOVEL COMPOUNDS AND USES THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2020-07-02 US disclosed
US-20200206292-A1 Compositions and Methods for Managing or Improving Bone Disorders, Joint Disorders, Cartilage Disorders, or a Combination Thereof UNIGEN, INC. (US) 2020-07-02 US disclosed
US-20200207803-A1 CYCLATIVE RELEASE OF PEPTIDIC COMPOUNDS CIRCLE PHARMA, INC. 2020-07-02 US disclosed
WO-2020139807-A2 NANOCAPSULES FOR THE DELIVERY OF CELL MODULATING AGENTS CSL BEHRING L.L.C. (US) 2020-07-02 WO disclosed
EP-3408258-B1 ORGANIC REACTIONS CARRIED OUT IN AQUEOUS SOLUTION IN THE PRESENCE OF A HYDROXYALKYL(ALKYL)CELLULOSE OR AN ALKYLCELLULOSE ABBVIE DEUTSCHLAND (DE) 2020-07-01 EP disclosed
US-10696698-B2 Surface primer compositions and methods of use ORMCO CORPORATION 2020-06-30 US disclosed
US-10694739-B2 Compositions and methods for reducing ice crystal formation X-THERMA, INC. (US) 2020-06-30 US disclosed
US-10696635-B2 Versatile ligand for palladium-catalyzed meta-C—H functionalizations of aromatic substrates THE SCRIPPS RESEARCH INSTITUTE (US) 2020-06-30 US disclosed
CN-111356705-A Polymerization process 埃克森美孚化学专利公司 2020-06-30 CN disclosed
CN-111356706-A Polymerization process 埃克森美孚化学专利公司 2020-06-30 CN disclosed
CN-111349128-A Flavonol derivative and preparation method and application thereof 上海医药工业研究院 2020-06-30 CN disclosed
CN-111344316-A Polyethylene compositions and articles made therefrom 埃克森美孚化学专利公司 2020-06-26 CN disclosed
WO-2020127780-A1 HETEROCYCLYL PYRIDAZINE AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2020-06-25 WO disclosed
WO-2020127974-A1 1,3,4-OXADIAZOLES AND THEIR DERIVATIVES AS NEW ANTIFUNGAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-06-25 WO disclosed
WO-2020132072-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH CYCLIC ORGANOSILICON CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION (US) 2020-06-25 WO disclosed
WO-2020132057-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ANHYDRIDE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION (US) 2020-06-25 WO disclosed
US-20200199122-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2020-06-25 US disclosed
US-20200203711-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ANHYDRIDE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2020-06-25 US disclosed
US-20200203764-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH CYCLIC ORGANOSILICON CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2020-06-25 US disclosed
US-20200197390-A1 METHODS OF TREATING METABOLIC DISEASES WITH FUSED BICYCLIC PYRAZOLES BELITE BIO, INC (KY) 2020-06-25 US disclosed
US-20200199171-A1 NOVEL STEROIDS AND METHODS OF MANUFACTURE TRUSTEES OF DARTMOUTH COLLEGE 2020-06-25 US disclosed
US-20200199087-A1 BIO-BASED, MULTI-AROMATIC COMPOUNDS, AND METHODS OF MAKING AND USING SAME ROWAN UNIVERSITY 2020-06-25 US disclosed
US-20200199126-A1 CYANOPYRROLIDINE DERIVATIVES WITH ACTIVITY AS INHIBITORS OF USP30 MISSION THERAPEUTICS LIMITED (GB) 2020-06-25 US disclosed
WO-2020126746-A1 SUBSTITUTED PYRIDINYLOXYBENZENES AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-06-25 WO disclosed
EP-3668833-A1 LIPIDS FOR USE IN LIPID NANOPARTICLE FORMULATIONS Acuitas Therapeutics, Inc. (CA) 2020-06-24 EP disclosed
EP-3668843-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS Inflazome Limited (IE) 2020-06-24 EP disclosed
EP-3668840-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS Inflazome Limited (IE) 2020-06-24 EP disclosed
EP-3668601-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS Inflazome Limited (IE) 2020-06-24 EP disclosed
EP-3668842-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS Inflazome Limited (IE) 2020-06-24 EP disclosed
EP-3668599-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS Inflazome Limited (IE) 2020-06-24 EP disclosed
EP-3668862-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS Inflazome Limited (IE) 2020-06-24 EP disclosed
EP-3668861-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS Inflazome Limited (IE) 2020-06-24 EP disclosed
EP-3670505-A1 SUBSTITUTED PYRIDINYLOXYBENZENES, THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS Bayer AG (DE) 2020-06-24 EP disclosed
US-10689407-B2 Photo-cleavable primer compositions and methods of use ENVISTA (US) 2020-06-23 US disclosed
US-10689399-B2 Substituted 3,4,5,6,8,10,14,14a-octahydro-2h-2,6-methanopyrido[1′,2′:4,5]pyrazino[2,1-b][1,3]oxazocines and methods for treating viral infections GILEAD SCIENCES, INC. (US) 2020-06-23 US disclosed
US-10687531-B2 Urea and thiourea substituted bicycles derivatives as pesticides SYNGENTA PARTICIPATIONS AG (CH) 2020-06-23 US disclosed
US-10689373-B2 1,2-substituted cyclopentanes as orexin receptor antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2020-06-23 US disclosed
US-10689381-B2 Vinblastine 20″ amides: synthetic analogs that maintain or improve potency and simultaneously overcome Pgp-derived efflux and resistance THE SCRIPPS RESEARCH INSTITUTE (US) 2020-06-23 US disclosed
US-10689411-B2 Efficient and scalable syntheses of nicotinoyl ribosides and reduced nicotinoyl ribosides, modified derivatives thereof, phosphorylated analogs thereof, adenylyl dinucleotide conjugates thereof, and novel crystalline forms thereof THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2020-06-23 US disclosed
US-10689356-B2 Inhibitors of KRAS G12C mutant proteins ARAXES PHARMA LLC (US) 2020-06-23 US disclosed
US-10689345-B2 1-cyano-pyrrolidine compounds as USP30 inhibitors MISSION THERAPEUTICS LIMITED (GB) 2020-06-23 US disclosed
CN-111315733-A Novel sulfonamide carboxamide compounds 英夫拉索姆有限公司 2020-06-19 CN disclosed
CN-106659914-B Inhibitors of lysine-specific demethylase-1 赛尔基因昆蒂赛尔研究公司 2020-06-19 CN disclosed
CN-111303152-A Polycyclic-carbamoylpyridone compounds and their pharmaceutical use 吉利德科学公司 2020-06-19 CN disclosed
WO-2020123674-A1 SUBSTITUTED ARYLMETHYLUREAS AND HETEROARYLMETHYLUREAS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2020-06-18 WO disclosed
US-20200190031-A1 ARYL ETHERS AND USES THEREOF PELOTON THERAPEUTICS, INC. (US) 2020-06-18 US disclosed
US-20200188536-A1 CHLOROTOXIN CONJUGATES AND METHODS OF USE THEREOF Blaze Bioscience, Inc. 2020-06-18 US disclosed
WO-2020123847-A1 ORGANIC COMPOUNDS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2020-06-18 WO disclosed
US-20200190059-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES TAKEDA PHARMACEUTICALS CO (JP) 2020-06-18 US disclosed
US-20200188336-A1 PHARMACOLOGY OF VISUAL CYCLE MODULATORS ACUCELA INC. 2020-06-18 US disclosed
EP-3209660-B1 1-CYCLOHEXYL-2-PHENYLAMINOBENZIMIDAZOLES AS MIDH1 INHIBITORS FOR THE TREATMENT OF TUMORS DEUTSCHES KREBSFORSCHUNGSZENTRUM STIFTUNG DES OEFFENTLICHEN RECHTS (DE) 2020-06-17 EP disclosed
EP-2825536-B1 BIS-QUARTERNARY CINCHONA ALKALOID SALTS AS ASYMMETRIC PHASE TRANSFER CATALYSTS MERCK SHARP & DOHME (US) 2020-06-17 EP disclosed
EP-3230325-B1 METHODS OF SEPARATING AROMATIC COMPOUNDS FROM LUBE BASE STOCKES EXXONMOBIL RES & ENG CO (US) 2020-06-17 EP disclosed
EP-2989089-B1 ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS AND USES THEREOF - III MERCK SHARP & DOHME (US) 2020-06-17 EP disclosed
US-10683269-B2 2-cyanoisoindoline derivatives for treating cancer MISSION THERAPEUTICS LIMITED (GB) 2020-06-16 US disclosed
US-10683324-B2 7-dehydrocholesterol derivatives and methods using same UNIVERSITY OF ROCHESTER (US) 2020-06-16 US disclosed
CN-111282598-A Novel precatalyst scaffolds for crosslinking reactions and methods of making and using same 耶鲁大学 2020-06-16 CN disclosed
US-10683283-B2 Substituted ureas and methods of making and using same MEBIAS DISCOVERY, INC. (US) 2020-06-16 US disclosed
CN-111295389-A Bioactive substance conjugate and preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2020-06-16 CN disclosed
US-10682352-B2 Compound having mutant IDH inhibitory activity, preparation method and use thereof SHANGHAI HAIHE PHARMACEUTICAL CO., LTD. (CN) 2020-06-16 US disclosed
CN-111278872-A Polyethylene compositions and articles made therefrom 埃克森美孚化学专利公司 2020-06-12 CN disclosed
WO-2020118194-A1 NON-ATP/CATALYTIC SITE p38 MITOGEN ACTIVATED PROTEIN KINASE INHIBITORS UNIVERSITY OF MARYLAND, BALTIMORE (US) 2020-06-11 WO disclosed
WO-2020117945-A1 SYNTHETIC DERIVATIVES OF CHOLIC ACID 7-SULFATE AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2020-06-11 WO disclosed
WO-2020117938-A1 PRODRUGS OF ANTI-CANCER AND ANTI-AUTOIMMUNE DISEASES THERAPEUTIC AGENTS, AND METHODS OF MAKING AND USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2020-06-11 WO disclosed
WO-2020117755-A1 COMPOSITIONS AND METHODS FOR TREATING BIOFILMS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-06-11 WO disclosed
US-20200181131-A1 INDOLEAMINE 2,3-DIOXYGENASE INHIBITOR AND APPLICATION NANJING TRANSTHERA BIOSCIENCES CO. LTD. (CN) 2020-06-11 US disclosed
US-20200179529-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME AND PREPARATION METHOD THEREFOR SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2020-06-11 US disclosed
US-20200181317-A1 Bisphenol A-Free Crosslinked Polymer Composition WARNER BABCOCK INSTITUTE FOR GREEN CHEMISTRY, LLC (US) 2020-06-11 US disclosed
US-20200181117-A1 SUBSTITUTED 3-HETEROARYLOXY-1H-PYRAZOLES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2020-06-11 US disclosed
US-20200181086-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS MISSION THERAPEUTICS LIMITED (GB) 2020-06-11 US disclosed
US-20200181123-A1 2-SUBSTITUTED QUINAZOLINE COMPOUNDS COMPRISING A SUBSTITUTED HETEROCYCLIC GROUP AND METHODS OF USE THEREOF ARAXES PHARMA LLC 2020-06-11 US disclosed
EP-3661917-A1 6-PHENYL-4,5-DIHYDROPYRIDAZIN-3(2H)-ONE DERIVATIVES AS PDE3A AND PDE3B INHIBITORS FOR TREATING CANCER Bayer Aktiengesellschaft (DE) 2020-06-10 EP disclosed
EP-3661925-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS Inflazome Limited (IE) 2020-06-10 EP disclosed
EP-3661505-A1 BENZOTHIAZOLE AND RELATED COMPOUNDS Spinogenix, Inc. (US) 2020-06-10 EP disclosed
EP-3661560-A1 COMBINATION OF ATR KINASE INHIBITORS AND PD-1/PD-L1 INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2020-06-10 EP disclosed
EP-3661513-A1 ORGANOPHOSPHATE DERIVATIVES January Therapeutics, Inc. (US) 2020-06-10 EP disclosed
EP-3661517-A1 DIHYDROOXADIAZINONES Bayer Aktiengesellschaft (DE) 2020-06-10 EP disclosed
US-10675286-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2020-06-09 US disclosed
US-10675355-B2 VAR2CSA-drug conjugates VAR2 PHARMACEUTICALS APS (DK) 2020-06-09 US disclosed
CN-111247147-A Azabicyclo and diazepatriene derivatives useful for treating ocular disorders 爱尔康公司 2020-06-05 CN disclosed
US-20200172506-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2020-06-04 US disclosed
US-20200170241-A1 NOVEL SUPERCOOLING METHODS FOR PRESERVATION OF BIOLOGICAL SAMPLES X-THERMA, INC. (US) 2020-06-04 US disclosed
WO-2020113071-A1 COMPOUNDS AND METHODS OF USE THEREOF FOR TREATMENT OF CANCER ARAXES PHARMA LLC (US) 2020-06-04 WO disclosed
WO-2020112905-A1 METHODS OF TREATING DISEASE WITH MAGL INHIBITORS LUNDBECK LA JOLLA RESEARCH CENTER, INC. (US) 2020-06-04 WO disclosed
US-20200172516-A1 Novel Compounds MISSION THERAPEUTICS LIMITED (GB) 2020-06-04 US disclosed
US-20200171179-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS KODIAK SCIENCES INC. 2020-06-04 US disclosed
US-20200172485-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2020-06-04 US disclosed
US-20200172491-A1 SUBSTITUTED 5-(HET-)ARYLPYRAZOLAMIDES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2020-06-04 US disclosed
WO-2020109391-A1 PYRIDAZINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2020-06-04 WO disclosed
EP-3659591-A1 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES Kodiak Sciences Inc. (US) 2020-06-03 EP disclosed
EP-3658567-A1 CYCLATIVE RELEASE OF PEPTIDIC COMPOUNDS Circle Pharma, Inc. (US) 2020-06-03 EP disclosed
US-10669234-B2 Cyanopyrrolidines as dub inhibitors for the treatment of cancer MISSION THERAPEUTICS LIMITED (GB) 2020-06-02 US disclosed
US-10668064-B2 Polycyclic-carbamoylpyridone compounds and their pharmaceutical use GILEAD SCIENCES, INC. (US) 2020-06-02 US disclosed
CN-106795096-B Novel lipid and lipid nanoparticle formulations for delivery of nucleic acids 爱康泰生治疗公司 2020-05-29 CN disclosed
CN-111212647-A Dihydroxadiazinones 拜耳股份有限公司 2020-05-29 CN disclosed
US-20200163946-A1 THERAPEUTIC COMPOUNDS CELGENE QUANTICEL RESEARCH, INC. (US) 2020-05-28 US disclosed
US-20200165224-A1 METHODS AND COMPOSITIONS FOR INHIBITING THE INTERACTION OF MENIN WITH MLL PROTEINS WELLSPRING BIOSCIENCES LLC 2020-05-28 US disclosed
US-20200165213-A1 SUBSTITUTED 2,3-DIHYDRO-1H-INDENE ANALOGS AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2020-05-28 US disclosed
EP-3204395-B1 NOVEL PRECATALYST SCAFFOLDS FOR CROSS-COUPLING REACTIONS, AND METHODS OF MAKING AND USING SAME UNIV YALE (US) 2020-05-27 EP disclosed
EP-3160956-B1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2020-05-27 EP disclosed
EP-3655393-A1 SUBSTITUTED 5-(HET-)ARYLPYRAZOLAMIDES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES Bayer CropScience Aktiengesellschaft (DE) 2020-05-27 EP disclosed
EP-3655402-A1 SUBSTITUTED 3-HETEROARYLOXY-1H-PYRAZOLES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES Bayer CropScience Aktiengesellschaft (DE) 2020-05-27 EP disclosed
US-10662184-B2 Benzenesulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2020-05-26 US disclosed
US-10661262-B2 Aromatic hydrogenation catalysts and uses thereof EXXONMOBIL RESEARCH & ENGINEERING COMPANY (US) 2020-05-26 US disclosed
CN-111196816-A Seven-membered ring compound and application thereof in preventing and treating diabetes and metabolic syndrome 中国科学院上海药物研究所 2020-05-26 CN disclosed
WO-2020102707-A1 COPPER NANOPARTICLE BASED CHEMOSELECTIVE REDUCTION BROWN UNIVERSITY (US) 2020-05-22 WO disclosed
US-20200158724-A1 POLYMER DOT COMPOSITIONS AND RELATED METHODS UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION 2020-05-21 US disclosed
US-20200155609-A1 COMPOSITIONS AND METHODS OF MAKING EXPANDED HEMATOPOIETIC STEM CELLS USING PTEN INHIBITORS TRANSFUSION HEALTH LLC 2020-05-21 US disclosed
US-20200157089-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2020-05-21 US disclosed
US-20200157068-A1 BENZOTHIAZOLE AND RELATED COMPOUNDS SPINOGENIX, INC. 2020-05-21 US disclosed
US-20200157077-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2020-05-21 US disclosed
US-20200157123-A1 PENICILLIN-BINDING PROTEIN INHIBITORS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2020-05-21 US disclosed
EP-3652235-A1 ELECTROCHROMIC POLYMER AND SYNTHESIS AND USES THEREOF Furcifer Inc. (US) 2020-05-20 EP disclosed
EP-3652111-A1 ELECTROCHROMIC POLYMER THIN FILMS HAVING REDUCED SELF-BLEACHING BEHAVIOR AND ENHANCED CYCLING STABILITY Furcifer Inc. (US) 2020-05-20 EP disclosed
EP-2797635-B1 CHROMOPHORIC POLYMER DOTS WITH NARROW-BAND EMISSION UNIV WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2020-05-20 EP disclosed
US-10655012-B2 Process for the preparation of polyurethane solutions based on silicon-polycarbonate diols AORTECH INTERNATIONAL PLC (GB) 2020-05-19 US disclosed
US-10654830-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-05-19 US disclosed
US-10654853-B2 Spiro-condensed pyrrolidine derivatives as deubiquitylating enzymes (DUB) inhibitors MISSION THERAPEUTICS LIMITED (GB) 2020-05-19 US disclosed
CN-111171049-A Tyrosine kinase inhibitors and uses thereof 山东轩竹医药科技有限公司 2020-05-19 CN disclosed
US-10654810-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2020-05-19 US disclosed
US-10654852-B2 Antibiotics and methods of using same THE BROAD INSTITUTE, INC. (US) 2020-05-19 US disclosed
CN-111163773-A Benzothiazoles and related compounds 斯皮诺吉尼克斯公司 2020-05-15 CN disclosed
CN-111153901-A Nitrogen-containing fused heterocyclic SHP2 inhibitor compound, preparation method and application 如东凌达生物医药科技有限公司 2020-05-15 CN disclosed
US-20200148653-A1 MAGL INHIBITORS H. LUNDBECK A/S (DK) 2020-05-14 US disclosed
US-20200147119-A1 OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2020-05-14 US disclosed
US-20200147593-A1 Cinchonium betaine catalysts and methods of using same BRANDEIS UNIVERSITY 2020-05-14 US disclosed
US-20200148703-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2020-05-14 US disclosed
US-20200148610-A1 ORGANIC REACTIONS CARRIED OUT IN AQUEOUS SOLUTION IN THE PRESENCE OF A HYDROXYALKYL(ALKYL)CELLULOSE OR AN ALKYLCELLULOSE ABBVIE INC. 2020-05-14 US disclosed
EP-3649112-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS Inflazome Limited (IE) 2020-05-13 EP disclosed
CN-111138412-A Spiro aromatic ring compound and application thereof 上海奕拓医药科技有限责任公司 2020-05-12 CN disclosed
US-10647798-B2 Spray-dried olefin polymerization catalyst compositions and polymerization processes for using the same EXXONMOBIL CHEMICAL PATENTS, INC. (US) 2020-05-12 US disclosed
US-10647703-B2 Inhibitors of KRAS G12C mutant proteins ARAXES PHARMA LLC (US) 2020-05-12 US disclosed
US-10646488-B2 Conjugates of cereblon binding compounds and G12C mutant KRAS, HRAS or NRAS protein modulating compounds and methods of use thereof ARAXES PHARMA LLC (US) 2020-05-12 US disclosed
US-10646495-B2 Testosterone ester triglyceride formulations ANTARES PHARMA, INC. (US) 2020-05-12 US disclosed
CN-111132964-A Glucocorticoid receptor modulators 欧瑞克制药公司 2020-05-08 CN disclosed
CN-111132673-A Non-fused tricyclic compounds 维瓦斯治疗公司 2020-05-08 CN disclosed
CN-111132973-A Substituted 3-heteroaryloxy-1H-pyrazoles and their salts and their use as herbicidal active substances 拜耳作物科学股份公司 2020-05-08 CN disclosed
CN-111132974-A Novel sulfonamide carboxamide compounds 英夫拉索姆有限公司 2020-05-08 CN disclosed
US-20200144672-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH PHOSPHORUS CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2020-05-07 US disclosed
US-20200138970-A1 ANTIBODY DRUG CONJUGATES OF KINESIN SPINDEL PROTEIN (KSP) INHIBITORS WITH ANTIB7H3-ANTIBODIES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2020-05-07 US disclosed
US-20200140487-A1 PEPTIDE LIBRARIES WITH NON-CANONICAL AMINO ACIDS REGENERON PHARMACEUTICALS, INC. 2020-05-07 US disclosed
US-20200138828-A1 Anti-thrombotic Agents and Methods of Use Thereof UNIV TEMPLE (US) 2020-05-07 US disclosed
US-10639286-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2020-05-05 US disclosed
US-10640498-B2 Compounds MISSION THERAPEUTICS LIMITED (GB) 2020-05-05 US disclosed
CN-107033157-B Bisbenzylisoquinoline derivative and application thereof in preparing medicament for treating or preventing tumor 贵州省中国科学院天然产物化学重点实验室 2020-05-05 CN disclosed
CN-111107903-A Novel sulfonamide carboxamide compounds 英夫拉索姆有限公司 2020-05-05 CN disclosed
CN-111087612-A Phosphorus-containing flame-retardant nylon and preparation method and application thereof 今创景新材料科技(上海)有限公司 2020-05-01 CN disclosed
CN-111093773-A Sulfonylureas and sulfonylthioureas as NLRP3 inhibitors 英夫拉索姆有限公司 2020-05-01 CN disclosed
CN-111087796-A Phosphorus-containing copolymerized nylon and preparation method and application thereof 今创景新材料科技(上海)有限公司 2020-05-01 CN disclosed
US-20200131194-A1 FMS-LIKE TYROSINE KINASE INHIBITORS Sagabio Co., Ltd. (TW) 2020-04-30 US disclosed
US-20200131474-A1 METHODS AND COMPOSITIONS FOR OCULAR CELL THERAPY NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2020-04-30 US disclosed
US-20200131170-A1 Compounds for Pain Treatment, Compositions Comprising Same, and Methods of Using Same CERSCI THERAPEUTICS, INC. 2020-04-30 US disclosed
US-20200131154-A1 PYRAZOLYL COMPOUNDS AND METHODS OF USE THEREOF ARRIEN PHARMACEUTICALS LLC 2020-04-30 US disclosed
US-20200136185-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH PHOSPHAZENE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2020-04-30 US disclosed
US-20200131119-A1 THERAPEUTIC COMPOUNDS AND METHODS UNIVERSITY OF TASMANIA (AU) 2020-04-30 US disclosed
US-20200131304-A1 MULTICOLORED ELECTROCHROMIC POLYMER COMPOSITIONS AND METHODS OF MAKING AND USING THE SAME Furcifer Inc. (US) 2020-04-30 US disclosed
US-20200131173-A1 VMAT2 INHIBITOR COMPOUNDS AND COMPOSITIONS THEREOF NEUROCRINE BIOSCIENCES, INC. 2020-04-30 US disclosed
EP-3641760-A1 NOVEL ANTIBACTERIAL COMPOUNDS AND METHODS OF MAKING AND USING SAME Brown University (US) 2020-04-29 EP disclosed
EP-3641741-A1 MICROTUBULE POLYMERIZATION INHIBITOR PRODRUGS AND METHODS OF USING THE SAME University of Maryland, Baltimore (US) 2020-04-29 EP disclosed
EP-3383859-B1 1-CYANO-PYRROLIDINE DERIVATIVES AS INHIBITORS OF USP30 MISSION THERAPEUTICS LTD (GB) 2020-04-29 EP disclosed
US-10632209-B2 ASH1L inhibitors and methods of treatment therewith THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2020-04-28 US disclosed
CN-111057048-A Aminopyrazine/pyridine compound, preparation method and application 如东凌达生物医药科技有限公司 2020-04-24 CN disclosed
WO-2020081583-A1 NICOTINIC ACETYLCHOLINE RECEPTOR PEPTIDE ANTAGONIST CONOTOXIN COMPOSITIONS AND RELATED METHODS Glo Pharma, LLC (US) 2020-04-23 WO disclosed
WO-2020078933-A1 PROTEOLYSIS TARGETING CHIMERA (PROTACS) AS DEGRADERS OF SMARCA2 AND/OR SMARCA4 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-04-23 WO disclosed
WO-2020078788-A1 COMBINATION OF ATR KINASE INHIBITORS WITH 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE COMPOUNDS BAYER AKTIENGESELLSCHAFT (DE) 2020-04-23 WO disclosed
WO-2020081938-A1 LIPIDS FOR LIPID NANOPARTICLE DELIVERY OF ACTIVE AGENTS Acuitas Therapeutics, Inc. (CA) 2020-04-23 WO disclosed
WO-2020080979-A1 PFKFB3 INHIBITORS AND THEIR USES GERO DISCOVERY LIMITED LIABILITY COMPANY (RU) 2020-04-23 WO disclosed
US-20200121678-A1 PYRIDAZINONE COMPOUNDS AND THEIR USE AS DAAO INHIBITORS TAKEDA PHARMACEUTICALS CO (JP) 2020-04-23 US disclosed
US-20200123313-A1 ELECTROCHROMIC POLYMER AND SYNTHESIS AND USES THEREOF Furcifer Inc. (US) 2020-04-23 US disclosed
US-20200121809-A1 LIPID NANOPARTICLE FORMULATIONS Acuitas Therapeutics, Inc. (CA) 2020-04-23 US disclosed
EP-3640241-A1 BROMODOMAIN INHIBITORS Celgene Quanticel Research, Inc. (US) 2020-04-22 EP disclosed
EP-2844636-B1 METHODS FOR THE TREATMENT OF PROLIFERATIVE DIABETIC RETINOPATHY ACUCELA INC (US) 2020-04-22 EP disclosed
EP-3638239-A1 METHODS OF TREATING RBP4 RELATED DISEASES WITH TRIAZOLOPYRIDINES Belite Bio, Inc (KY) 2020-04-22 EP disclosed
EP-3638238-A1 METHODS OF TREATING METABOLIC DISEASES WITH FUSED BICYCLIC PYRAZOLES Belite Bio, Inc (KY) 2020-04-22 EP disclosed
CN-111050765-A Spiro compounds and methods of making and using the same 隆德贝克拉荷亚研究中心有限公司 2020-04-21 CN disclosed
US-10626104-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2020-04-21 US disclosed
US-10626103-B2 Inhibitor of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2020-04-21 US disclosed
CN-111032034-A Spiro compounds and methods of making and using the same 隆德贝克拉荷亚研究中心有限公司 2020-04-17 CN disclosed
US-20200115709-A1 Functionally-Modified Oligonucleotides And Subunits Thereof JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2020-04-16 US disclosed
US-20200113905-A1 TREATMENT OF RELAPSED AND/OR REFRACTORY SOLID TUMORS AND NON-HODGKIN'S LYMPHOMAS CELGENE QUANTICEL RESEARCH, INC. (US) 2020-04-16 US disclosed
US-20200115404-A1 CD73 INHIBITORS AND USES THEREOF PELOTON THERAPEUTICS INC. 2020-04-16 US disclosed
US-20200115384-A1 PDE9 INHIBITOR AND USE THEREOF TRANSTHERA SCIENCES (NANJING), INC. (CN) 2020-04-16 US disclosed
US-20200115414-A1 NICOTINIC ACETYLCHOLINE RECEPTOR PEPTIDE ANTAGONIST CONOTOXIN COMPOSITIONS AND RELATED METHODS GLO PHARMA, INC. 2020-04-16 US disclosed
US-20200115363-A1 QUINAZOLINE DERIVATIVES AS MODULATORS OF MUTANT KRAS, HRAS OR NRAS ARAXES PHARMA LLC 2020-04-16 US disclosed
EP-3033335-B1 PYRIDINONES BOEHRINGER INGELHEIM INT (DE) 2020-04-15 EP disclosed
EP-3634404-A1 PYRAZOLE MAGL INHIBITORS Lundbeck La Jolla Research Center, Inc. (US) 2020-04-15 EP disclosed
EP-3636639-A1 INHIBITORS OF KRAS G12C Araxes Pharma LLC (US) 2020-04-15 EP disclosed
CN-111000898-A Compositions and methods for joint health 尤妮金公司 2020-04-14 CN disclosed
US-10617680-B2 Therapeutic compounds CELGENE QUANTICEL RESEARCH, INC. (US) 2020-04-14 US disclosed
WO-2020070050-A1 FUNGICIDAL 5-SUBSTITUTED IMIDAZOL-1-YL CARBINOL DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2020-04-09 WO disclosed
US-20200108052-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2020-04-09 US disclosed
US-20200108070-A2 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR AND USE THEREOF NANJING TRANSTHERA BIOSCIENCES CO. LTD. (CN) 2020-04-09 US disclosed
WO-2020072602-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING OTIC THERAPEUTIC AGENTS AND RELATED METHODS Frequency Therapeutics, Inc. (US) 2020-04-09 WO disclosed
US-20200109287-A1 WATER SOLUBLE FLUORESCENT OR COLORED DYES AND METHODS FOR THEIR USE Sony Group Corporation (JP) 2020-04-09 US disclosed
US-20200109120-A1 PKM2 MODULATORS AND METHODS FOR THEIR USE SUMITOMO PHARMA ONCOLOGY, INC. 2020-04-09 US disclosed
EP-3630746-A1 COMPOUNDS AND METHODS OF USE THEREOF FOR TREATMENT OF CANCER Araxes Pharma LLC (US) 2020-04-08 EP disclosed
EP-3630956-A1 COMPOSITIONS AND METHODS OF MAKING EXPANDED HEMATOPOIETIC STEM CELLS USING PTEN INHIBITORS Transfusion Health, LLC (US) 2020-04-08 EP disclosed
EP-3630744-A1 PYRAZOLE MAGL INHIBITORS Lundbeck La Jolla Research Center, Inc. (US) 2020-04-08 EP disclosed
EP-3252038-B1 N-BENZOATE GROUP SUBSTITUTED BENZOPYRROLINE-2-ONE DERIVATIVE AND USE THEREOF BEIJING HANMI PHARMACEUTICAL CO LTD (CN) 2020-04-08 EP disclosed
EP-3630782-A1 PENICILLIN-BINDING PROTEIN INHIBITORS Venatorx Pharmaceuticals, Inc. (US) 2020-04-08 EP disclosed
EP-3630783-A1 PENICILLIN-BINDING PROTEIN INHIBITORS Venatorx Pharmaceuticals, Inc. (US) 2020-04-08 EP disclosed
EP-3630747-A1 QUINAZOLINE DERIVATIVES AS MODULATORS OF MUTANT KRAS, HRAS OR NRAS Araxes Pharma LLC (US) 2020-04-08 EP disclosed
EP-3630745-A2 COVALENT INHIBITORS OF KRAS Araxes Pharma LLC (US) 2020-04-08 EP disclosed
US-10610857-B2 Cinchonium betaine catalysts and methods of using same BRANDEIS UNIVERSITY (US) 2020-04-07 US disclosed
US-10611775-B2 Thiophene derivatives TIANJIN HEMAY PHARMACEUTICAL CO., LTD. (CN) 2020-04-07 US disclosed
US-10611723-B2 Ligand-enabled meta-C-H activation using a transient mediator THE SCRIPPS RESEARCH INSTITUTE (US) 2020-04-07 US disclosed
US-10611763-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-04-07 US disclosed
US-10612056-B2 Beta-substituted non-canonical amino acids CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2020-04-07 US disclosed
CN-110964012-A Fused heterocyclic biaryl benzyl alcohol compound, preparation method and application 如东凌达生物医药科技有限公司 2020-04-07 CN disclosed
CN-110950876-A Furanolactam compounds, preparation method and application 如东凌达生物医药科技有限公司 2020-04-03 CN disclosed
CN-110950842-A Quinoline derivatives having indoleamine-2, 3-dioxygenase inhibitory activity 深圳微芯生物科技股份有限公司 2020-04-03 CN disclosed
CN-110959008-A Penicillin binding protein inhibitors 维纳拓尔斯制药公司 2020-04-03 CN disclosed
WO-2020061617-A1 OPTICAL DATA STORAGE MATERIAL AND METHOD ROYAL MELBOURNE INSTITUTE OF TECHNOLOGY (AU) 2020-04-02 WO disclosed
WO-2020063727-A1 TRICYCLIC RING ASK1 INHIBITORS AND USE THEREOF 山东轩竹医药科技有限公司 2020-04-02 WO disclosed
WO-2020063976-A1 FUSED HETEROCYCLIC BIARYL BENZYL ALCOHOL COMPOUND, PREPARATION METHOD, AND USE 如东凌达生物医药科技有限公司 2020-04-02 WO disclosed
WO-2020063618-A1 QUINOLONE DERIVATIVE HAVING INDOLEAMINE-2,3-DIOXYGENASE INHIBITED ACTIVITY 深圳微芯生物科技股份有限公司 2020-04-02 WO disclosed
US-20200102331-A1 PENICILLIN-BINDING PROTEIN INHIBITORS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2020-04-02 US disclosed
WO-2020064260-A1 SUBSTITUTED 5-(SULFANYL)-3,4-DIHYDRO-2H-PYRROL-4-CARBOXAMIDES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2020-04-02 WO disclosed
US-20200102321-A1 SUBSTITUTED QUINAZOLINES AS INHIBITORS OF KRAS G12C ARAXES PHARMA LLC 2020-04-02 US disclosed
EP-3057617-B1 NANOPARTICLE-CONTAINING HYDROGELS AGENCY SCIENCE TECH & RES (SG) 2020-04-01 EP disclosed
US-10603270-B2 Skin care compositions and methods of use thereof UNIGEN, INC. (US) 2020-03-31 US disclosed
CN-107674086-B Polycyclic-carbamoylpyridone compounds and their pharmaceutical use 吉利德科学公司 2020-03-31 CN disclosed
CN-105742702-B Rechargeable lithium battery 三星SDI株式会社 2020-03-31 CN disclosed
CN-110945697-A Membrane electrode assembly with fluorocarbon additives 百拉得动力系统公司 2020-03-31 CN disclosed
CN-110945005-A Modified oligomeric compounds comprising tricyclic DNA nucleosides and uses thereof 新特纳股份公司 2020-03-31 CN disclosed
CN-110945001-A FMS-like tyrosine kinase inhibitors 三日月生技股份有限公司 2020-03-31 CN disclosed
US-20200093936-A1 Therapeutic Targeting of Lipid Nanoparticles THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2020-03-26 US disclosed
US-20200095272-A1 PRODRUGS OF CLOFARABINE BoYen Therapeutics, Inc. (TW) 2020-03-26 US disclosed
US-20200093852-A1 Methods of Treating Ocular Disorders Beta Therapeutics Pty Ltd (AU) 2020-03-26 US disclosed
WO-2020061216-A1 COMBINATION THERAPY FOR TREATING BLOOD CANCER SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2020-03-26 WO disclosed
US-20200095236-A1 ANTIBACTERIAL COMPOUNDS BLACKSMITH MEDICINES, INC. 2020-03-26 US disclosed
WO-2020061375-A1 ANTIBACTERIAL COMPOUNDS FORGE THERAPEUTICS, INC. (US) 2020-03-26 WO disclosed
WO-2020060937-A1 NARROW ABSORPTION POLYMER NANOPARTICLES AND RELATED METHODS UNIVERSITY OF WASHINGTON (US) 2020-03-26 WO disclosed
WO-2020060873-A2 MOF COMPOSITIONS FOR SELECTIVE SEPARATION OF HYDROCARBONS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2020-03-26 WO disclosed
WO-2020061426-A2 SYSTEMS AND METHODS FOR MANUFACTURING LIPID NANOPARTICLES AND LIPOSOMES Acuitas Therapeutics, Inc. (CA) 2020-03-26 WO disclosed
US-20200095241-A1 SUBSTITUTED 1,2,4-THIADIAZOLYLPYRROLONES AND 1,2,4-THIADIAZOLYLHYDANTOINS AND SALTS THEREOF AND USE THEREOF AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2020-03-26 US disclosed
EP-3193880-B1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL LILLY CO ELI (US) 2020-03-25 EP disclosed
EP-3624797-A1 KINASE INHIBITORS AND USES THEREOF Denali Therapeutics Inc. (US) 2020-03-25 EP disclosed
EP-3625200-A1 BIO-BASED, MULTI-AROMATIC COMPOUNDS, AND METHODS OF MAKING AND USING SAME Rowan University (US) 2020-03-25 EP disclosed
CN-110903275-A Process for producing iobitridol, intermediate therefor, and process for producing the same 苏州科伦药物研究有限公司 2020-03-24 CN disclosed
US-10597425-B2 Anti-GP41 antibody-specific capture agents, compositions, and methods of using and making CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2020-03-24 US disclosed
US-10597368-B2 Syringolin analogues and methods of making and using same BROWN UNIVERSITY (US) 2020-03-24 US disclosed
US-10597406-B2 Purification of rapamycin derivatives using temperature induced phase separation BIOSENSORS INTERNATIONAL GROUP, LTD. (BM) 2020-03-24 US disclosed
CN-110914256-A Novel sulfonamide carboxamide compounds 英夫拉索姆有限公司 2020-03-24 CN disclosed
CN-110913858-A Kinase inhibitors and uses thereof 戴纳立制药公司 2020-03-24 CN disclosed
US-10597366-B2 Aryl ethers and uses thereof PELOTON THERAPEUTICS, INC. (US) 2020-03-24 US disclosed
US-10597376-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2020-03-24 US disclosed
US-10597379-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-03-24 US disclosed
US-10597365-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-03-24 US disclosed
CN-107082782-B Substituted xanthines and methods of use thereof 海德拉生物科学有限责任公司 2020-03-20 CN disclosed
US-20200087322-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2020-03-19 US disclosed
US-20200085823-A1 METHODS FOR TREATING DISEASES ASSOCIATED WITH ABNORMAL ACVR1 EXPRESSION AND ACVR1 INHIBITORS FOR USE IN THE SAME SUMITOMO PHARMA ONCOLOGY, INC. 2020-03-19 US disclosed
US-20200087319-A1 Kinase Inhibitors and Uses Thereof DENALI THERAPEUTICS INC. (US) 2020-03-19 US disclosed
US-20200087304-A1 PYRAZOLE MAGL INHIBITORS H. LUNDBECK A/S (DK) 2020-03-19 US disclosed
EP-3621461-A1 METHODS AND ENZYME CATALYSTS FOR THE SYNTHESIS OF NON-CANONICAL AMINO ACIDS California Institute of Technology (US) 2020-03-18 EP disclosed
EP-3197883-B1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2020-03-18 EP disclosed
EP-3621961-A2 ANTIBACTERIAL COMPOUNDS Forge Therapeutics, Inc. (US) 2020-03-18 EP disclosed
EP-3621962-A2 ANTIBACTERIAL COMPOUNDS Forge Therapeutics, Inc. (US) 2020-03-18 EP disclosed
US-10590075-B2 Cyanopyrrolidine derivatives as inhibitors for DUBs MISSION THERAPEUTICS LIMITED (GB) 2020-03-17 US disclosed
CN-107001339-B Novel compounds 特殊治疗有限公司 2020-03-17 CN disclosed
CN-110892001-A Electrochromic polymers and their synthesis and use 菲尔齐费尔公司 2020-03-17 CN disclosed
CN-110891941-A Substituted 5- (hetero) arylpyrazolamides and their salts and their use as herbicidally active substances 拜耳作物科学股份公司 2020-03-17 CN disclosed
US-10588907-B2 Methods and compositions for inhibiting the interaction of menin with MLL proteins KURA ONCOLOGY, INC. (US) 2020-03-17 US disclosed
CN-110878052-A FXR agonist-containing compound and preparation method and application thereof 山东大学 2020-03-13 CN disclosed
CN-110878048-A Anilines as psychotropic disorders 中国科学院上海药物研究所 2020-03-13 CN disclosed
US-20200081398-A1 PHOTOSENSITIVE POLYMERS FOR VOLUME HOLOGRAPHY META PLATFORMS TECHNOLOGIES, LLC 2020-03-12 US disclosed
US-20200079754-A1 INHIBITORS OF BRUTONS TYROSINE KINASE PHARMACYCLICS LLC (US) 2020-03-12 US disclosed
US-20200079765-A1 SUBSTITUTED HETEROARYL PYRROLONES AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES BAYER AKTIENGESELLSCHAFT (DE) 2020-03-12 US disclosed
EP-3620053-A1 FUNGICIDAL ACTIVE COMPOUND COMBINATIONS Bayer Aktiengesellschaft (DE) 2020-03-11 EP disclosed
EP-3618818-A1 NON-FUSED TRICYCLIC COMPOUNDS Vivace Therapeutics, Inc. (US) 2020-03-11 EP disclosed
CN-105828838-B Hydrogel containing nanoparticles 新加坡科技研究局 2020-03-10 CN disclosed
US-10583161-B2 Compositions and methods for managing or improving bone disorders, joint disorders, cartilage disorders, or a combination thereof UNIGEN, INC. (US) 2020-03-10 US disclosed
US-10583137-B2 Triazole DAGLα inhibitors THE SCRIPPS RESEARCH INSTITUTE (US) 2020-03-10 US disclosed
CN-110869358-A Covalent inhibitors of KRAS 亚瑞克西斯制药公司 2020-03-06 CN disclosed
CN-110869357-A Compounds and methods of use thereof for treating cancer 亚瑞克西斯制药公司 2020-03-06 CN disclosed
US-20200071436-A1 Polymerization Processes and Polymers Made Therefrom EXXONMOBIL CHEMICAL PATENTS INC. 2020-03-05 US disclosed
US-20200069668-A1 Therapeutic Combinations of an IRAK4 Inhibitor and a BTK Inhibitor ACERTA PHARMA BV (NL) 2020-03-05 US disclosed
US-20200071437-A1 Polymerization Processes and Polymers Made Therefrom EXXONMOBIL CHEMICAL PATENTS INC. 2020-03-05 US disclosed
US-20200071332-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2020-03-05 US disclosed
US-20200071313-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS SODIUM CHANNEL INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2020-03-05 US disclosed
US-20200069796-A1 Therapeutic Combinations of a BTK Inhibitor, a PI3K Inhibitor, a JAK-2 Inhibitor, a PD-1 Inhibitor, and/or a PD-L1 Inhibitor ACERTA PHARMA BV (NL) 2020-03-05 US disclosed
US-20200071288-A1 SELECTIVE HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF HUMAN DISEASE SHUTTLE PHARMACEUTICALS, INC. 2020-03-05 US disclosed
US-20200071297-A1 NEW 6-AMINO-QUINOLINONE COMPOUNDS AND DERIVATIVES AS BCL6 INHIBITORS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2020-03-05 US disclosed
WO-2020047487-A1 METHODS FOR TREATING CANCER WITH RORGAMMA INHIBITORS AND STATINS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-03-05 WO disclosed
WO-2020047323-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2020-03-05 WO disclosed
WO-2020047312-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS SODIUM CHANNEL INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2020-03-05 WO disclosed
EP-3013789-B1 AMINO ACID AND PEPTIDE CONJUGATES AND CONJUGATION PROCESS AUCKLAND UNISERVICES LTD (NZ) 2020-03-04 EP disclosed
EP-2753613-B1 DERIVATIVES OF XANTHONE COMPOUNDS AGENCY SCIENCE TECH & RES (SG) 2020-03-04 EP disclosed
EP-3617204-A1 INDOLEAMINE 2,3-DIOXYGENASE INHIBITOR AND APPLICATION Nanjing Transthera Biosciences Co. Ltd. (CN) 2020-03-04 EP disclosed
EP-3615513-A1 METHODS OF MANUFACTURING OF NIRAPARIB Tesaro Inc. (US) 2020-03-04 EP disclosed
EP-3615502-A1 THERAPEUTIC COMPOUNDS AND METHODS University Of Tasmania (AU) 2020-03-04 EP disclosed
EP-3617221-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME, AND PREPARATION METHOD THEREFOR Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed
EP-3615080-A1 ANTIBODY CONJUGATES COMPRISING STING AGONIST Novartis AG (CH) 2020-03-04 EP disclosed
EP-3615510-A1 NOVEL CARBONYL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS Acuitas Therapeutics, Inc. (CA) 2020-03-04 EP disclosed
EP-3615537-A2 6-6 FUSED BICYCLIC HETEROARYL COMPOUNDS AND THEIR USE AS LATS INHIBITORS Novartis AG (CH) 2020-03-04 EP disclosed
US-10577349-B2 Quinolinones as inhibitors of translation initiation complex Sanford Burnham Prebys Medical Discovery Institute (US) 2020-03-03 US disclosed
US-10576144-B2 Amino acid and peptide conjugates and conjugation process AUCKLAND UNISERVICES LIMITED (NZ) 2020-03-03 US disclosed
US-10576453-B2 Membrane fabrication methods using organosilica materials and uses thereof EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2020-03-03 US disclosed
US-10577308-B2 Sodium channel modulators The Florey Institute (AU) 2020-03-03 US disclosed
US-10576064-B2 Spiro[3H-indole-3,2′-pyrrolidin]-2(1H)-one compounds and derivatives as MDM2-P53 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-03-03 US disclosed
CN-110857300-A Condensed ring triazole compounds, preparation method and application 如东凌达生物医药科技有限公司 2020-03-03 CN disclosed
US-20200062761-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC 2020-02-27 US disclosed
US-20200062721-A1 NON-FUSED TRICYCLIC COMPOUNDS VIVACE THERAPEUTICS, INC. 2020-02-27 US disclosed
WO-2020038458-A1 CLASS OF FUSED RING TRIAZOLE COMPOUND, PREPARATION METHOD, AND USE 如东凌达生物医药科技有限公司 2020-02-27 WO disclosed
WO-2020041051-A1 GEMCITABINE PRODRUGS CURE BIOPHARMA INC. (US) 2020-02-27 WO disclosed
WO-2020041050-A1 GEMCITABINE PRODRUGS CURE BIOPHARMA INC. (US) 2020-02-27 WO disclosed
US-20200062768-A1 CX3CR1 Small Molecule Antagonists, and Methods Using Same DREXEL UNIVERSITY 2020-02-27 US disclosed
EP-3612546-A1 MODIFIED OLIGOMERIC COMPOUNDS COMPRISING TRICYCLO-DNA NUCLEOSIDES AND USES THEREOF Synthena AG (CH) 2020-02-26 EP disclosed
EP-3612522-A1 THERAPEUTIC COMPOUNDS Celgene Quanticel Research, Inc. (US) 2020-02-26 EP disclosed
EP-3612532-A1 VMAT2 INHIBITOR COMPOUNDS AND COMPOSITIONS THEREOF Neurocrine Biosciences, Inc. (US) 2020-02-26 EP disclosed
EP-3613743-A1 PROCESSES FOR THE PREPARATION OF 1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE DERIVATIVES Intellikine, LLC (US) 2020-02-26 EP disclosed
US-10570106-B2 MAGL inhibitors LUNDBECK LA JOLLA RESEARCH CENTER, INC. (US) 2020-02-25 US disclosed
CN-110831933-A Quinazoline derivatives as modulators of mutated KRAS, HRAS or NRAS 亚瑞克西斯制药公司 2020-02-21 CN disclosed
US-20200055892-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. 2020-02-20 US disclosed
US-20200054764-A1 MEDICAL USE OF ANTI-C MET ANTIBODY-CYTOTOXIC DRUG CONJUGATE Suzhou Suncadia Biopharmaceuticals Co., Ltd. (CN) 2020-02-20 US disclosed
US-20200055837-A1 METHODS OF MANUFACTURING OF NIRAPARIB TESARO, INC. 2020-02-20 US disclosed
WO-2020035465-A1 NOVEL SULFONEUREA COMPOUNDS INFLAZOME LIMITED (IE) 2020-02-20 WO disclosed
WO-2020035464-A1 NOVEL SULFONAMIDEUREA COMPOUNDS INFLAZOME LIMITED (IE) 2020-02-20 WO disclosed
WO-2020035300-A1 POLYMER COMPOSITION BASF SE (DE) 2020-02-20 WO disclosed
WO-2020035466-A1 NOVEL SULFONEUREA COMPOUNDS INFLAZOME LIMITED (IE) 2020-02-20 WO disclosed
EP-3610010-A2 COMPLEMENT FACTOR D ANTAGONIST ANTIBODIES AND CONJUGATES THEREOF Kodiak Sciences Inc. (US) 2020-02-19 EP disclosed
EP-3609872-A1 GLUCOCORTICOID RECEPTOR MODULATORS Oric Pharmaceuticals, Inc. (US) 2020-02-19 EP disclosed
EP-3254678-B1 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC (US) 2020-02-19 EP disclosed
EP-3303285-B1 PESTICIDALLY ACTIVE OXIME AND HYDRAZONE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2020-02-19 EP disclosed
EP-3417852-B1 ARYL ETHERS AND USES THEREOF PELOTON THERAPEUTICS INC (US) 2020-02-19 EP disclosed
EP-3150203-B1 COMPOUNDS WITH (1E,6E)-1,7-BIS-(3,4- DIMETHOXYPHENYL)-4,4-DISSTITUTED-HEPA-1,6-DIENE-3,5-DI-ONE STRUCTURAL SCAFFOLD,THEIR BIOLOGICAL ACTIVITY, AND USES THEREOF ALLIANZ PHARMASCIENCE LTD (TW) 2020-02-19 EP disclosed
US-10562915-B2 Bromodomain inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-02-18 US disclosed
US-10562859-B2 Aryl sulfonamide compounds as carbonic anhydrase inhibitors and their therapeutic use SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2020-02-18 US disclosed
US-10562882-B2 Piperidine derivatives for use in the treatment or prevention of psychiatric and neurological conditions TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2020-02-18 US disclosed
CN-110809560-A Electrochromic polymer films with reduced self-bleaching behavior and enhanced cycling stability 菲尔齐费尔公司 2020-02-18 CN disclosed
CN-110799492-A Novel carbonyl lipid and lipid nanoparticle formulations for delivery of nucleic acids 爱康泰生治疗公司 2020-02-14 CN disclosed
CN-110799218-A Antibody conjugates comprising STING agonists 诺华股份有限公司 2020-02-14 CN disclosed
US-20200046838-A1 LIPIDS FOR DELIVERY OF ACTIVE AGENTS Acuitas Therapeutics, Inc. (CA) 2020-02-13 US disclosed
US-20200048243-A1 CINCHONINE-DERIVED CATALYSTS AND METHODS OF USING SAME BRANDEIS UNIVERSITY (US) 2020-02-13 US disclosed
US-20200048228-A1 ALVOCIDIB PRODRUGS AND THEIR USE AS PROTEIN KINASE INHIBITORS SUMITOMO PHARMA ONCOLOGY, INC. 2020-02-13 US disclosed
US-20200048301-A1 EPOXY-(METH)ACRYLATE MONOMERS AND POLYMERS AND METHODS OF MAKING AND USING THE SAME ROWAN UNIVERSITY 2020-02-13 US disclosed
US-20200047169-A1 CATALYSTS FOR OLEFIN ISOMERIZATION BRANDEIS UNIVERSITY (US) 2020-02-13 US disclosed
WO-2020033784-A1 TRANSGLUTAMINASE 2 (TG2) INHIBITORS SITARI PHARMA, INC. (US) 2020-02-13 WO disclosed
WO-2020033823-A1 SMALL-MOLECULE PI5P4K ALPHA/BETA INHIBITORS AND METHODS OF TREATMENT USING SAME YALE UNIVERSITY (US) 2020-02-13 WO disclosed
EP-3606743-A1 COATING FOR RECYCLABLE PAPER JL Darling LLC (US) 2020-02-12 EP disclosed
EP-3608325-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE Gilead Sciences, Inc. (US) 2020-02-12 EP disclosed
EP-3094687-B1 WATER SOLUBLE FLUORESCENT OR COLORED DYES SONY CORP (JP) 2020-02-12 EP disclosed
CN-107207524-B Bisbenzylisoquinoline derivatives, preparation method thereof and application thereof in treatment and prevention of liver diseases 贵州省中国科学院天然产物化学重点实验室 2020-02-07 CN disclosed
CN-107072985-B Therapeutic inhibiting compounds 莱福斯希医药公司 2020-02-07 CN disclosed
CN-110770236-A VMAT2 inhibitor compounds and compositions thereof 纽罗克里生物科学有限公司 2020-02-07 CN disclosed
CN-110769689-A Novel supercooling method for preserving biological samples 先时迈纳米生物科技股份有限公司 2020-02-07 CN disclosed
WO-2020028706-A1 HETEROCYCLIC SPIRO COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF CANCER ARAXES PHARMA LLC (US) 2020-02-06 WO disclosed
US-20200038475-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. (US) 2020-02-06 US disclosed
US-20200039963-A1 PRC1 INHIBITORS AND METHODS OF TREATMENT THEREWITH NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2020-02-06 US disclosed
US-20200039941-A1 CXCR4 CHEMOKINE RECEPTOR MODULATORS NATIONAL INSTITUTES OF HEALTH 2020-02-06 US disclosed
EP-3601267-A1 2-METHYL-QUINAZOLINES Bayer Pharma Aktiengesellschaft (DE) 2020-02-05 EP disclosed
EP-3601307-A1 CROSS-COUPLING REACTION CATALYSTS, AND METHODS OF MAKING AND USING SAME Yale University (US) 2020-02-05 EP disclosed
EP-3600273-A1 CD73 INHIBITORS AND USES THEREOF Peloton Therapeutics, Inc. (US) 2020-02-05 EP disclosed
EP-3604271-A1 PEPTIDES FOR AMINO ACID AND PEPTIDE CONJUGATES AND CONJUGATION PROCESS Auckland Uniservices Limited (NZ) 2020-02-05 EP disclosed
EP-3601216-A1 SUBSTITUTED DIHYDROINDENE-4-CARBOXAMIDES AND ANALOGS THEREOF, AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2020-02-05 EP disclosed
EP-3600451-A1 AGENTS FOR DIFFERENTIATING STEM CELLS AND TREATING CANCER Minerva Biotechnologies Corporation (US) 2020-02-05 EP disclosed
EP-3236940-B1 COMPOSITIONS AND METHODS FOR TREATING HYPERKALEMIA ARDELYX INC (US) 2020-02-05 EP disclosed
US-10548896-B2 Treatment of relapsed and/or refractory solid tumors and non-Hodgkin's lymphomas CELGENE QUANTICEL RESEARCH, INC. (US) 2020-02-04 US disclosed
US-10550122-B2 Solid forms of (S)-3-(1-(9H-purin-6-ylamino)ethyl)-8-chloro-2-phenylisoquinolin-1(2H)-one and methods of use thereof INFINITY PHARMACEUTICALS, INC. (US) 2020-02-04 US disclosed
US-10550221-B2 Electrochromic polymer and synthesis and uses thereof Furcifer Inc. (US) 2020-02-04 US disclosed
US-10550084-B2 Substituted 1-hydroxy-pyridin-2(1H)-ones, and methods of making and using same ARBUTUS BIOPHARMA CORPORATION (CA) 2020-02-04 US disclosed
US-10548913-B2 Nicotinamide mononucleotide derivatives and their uses METRO INTERNATIONAL BIOTECH, LLC (US) 2020-02-04 US disclosed
CN-110753684-A Method for producing nilapali 特沙诺有限公司 2020-02-04 CN disclosed
CN-110734436-A Pyrimidine or pyrazine ring compounds and application thereof 上海青煜医药科技有限公司 2020-01-31 CN disclosed
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WO-2020020816-A1 NOVEL TRIAZOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2020-01-30 WO disclosed
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CN-105452269-B Compositions and methods for joint health 尤妮金公司 2020-01-10 CN disclosed
CN-110678456-A Pyrazole MAGL inhibitors 隆德贝克拉荷亚研究中心有限公司 2020-01-10 CN disclosed
CN-105828820-B Bromodomain inhibitors 赛尔基因昆蒂赛尔研究公司 2020-01-07 CN disclosed
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CN-110662753-A Cross-coupling reaction catalysts and methods of making and using the same 耶鲁大学 2020-01-07 CN disclosed
CN-110655520-A Pyrimido-cyclic compounds, process for their preparation and their use 上海青煜医药科技有限公司 2020-01-07 CN disclosed
CN-110662542-A Efficient and scalable synthesis of nicotinyl nucleosides and reduced nicotinyl nucleosides, modified derivatives thereof, phosphorylated analogs thereof, adenosine dinucleotide conjugates thereof, and novel crystalline forms thereof 英国贝尔法斯特女王大学 2020-01-07 CN disclosed
WO-2020002091-A1 SUBSTITUTED THIAZOLYLPYRROLONES, SALTS THEREOF AND THE USE THEREOF AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-01-02 WO disclosed
WO-2020002089-A1 SUBSTITUTED 2-HETEROARYLOXYPYRIDINES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-01-02 WO disclosed
WO-2020002085-A1 SUBSTITUTED 4-HETEROARYLOXYPYRIDINES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-01-02 WO disclosed
WO-2020002090-A1 SUBSTITUTED THIAZOLYLPYRROLONES, SALTS THEREOF AND THE USE THEREOF AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-01-02 WO disclosed
WO-2020002087-A1 SUBSTITUTED 3-HETEROARYLOXYPYRIDINES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-01-02 WO disclosed
WO-2020002083-A1 SUBSTITUTED HETEROCYCLIC PYRROLONES AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2020-01-02 WO disclosed
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CN-110582480-A Therapeutic compounds and methods 塔斯马尼亚大学 2019-12-17 CN disclosed
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CN-110573511-A 6-6 fused bicyclic heteroaryl compounds and their use as LATS inhibitors 诺华股份有限公司 2019-12-13 CN disclosed
CN-110563722-A pyridine or pyridazine ring compound and application thereof 上海青煜医药科技有限公司 2019-12-13 CN disclosed
CN-110551105-A substituted triazoles useful as AXL inhibitors RIGEL PHARMACEUTICALS INC 2019-12-10 CN disclosed
WO-2019227173-A1 STABLE PROTEIN LIGANDS AS ANTI-INFECTIVE AGENTS MONASH UNIVERSITY (AU) 2019-12-05 WO disclosed
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CN-110498769-A IDO inhibitor and application NANJING TRANSTHERA BIOSCIENCES CO LTD 2019-11-26 CN disclosed
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EP-3043784-B9 ARYL ETHERS AND USES THEREOF PELOTON THERAPEUTICS INC (US) 2019-11-20 EP disclosed
EP-3322702-B1 CYANOPYRROLIDINES AS DUB INHIBITORS FOR THE TREATMENT OF CANCER MISSION THERAPEUTICS LTD (GB) 2019-11-20 EP disclosed
EP-3222620-B1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO LTD (CN) 2019-11-20 EP disclosed
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EP-3565811-A1 INHIBITORS OF NHE-MEDIATED ANTIPORT Ardelyx, Inc. (US) 2019-11-13 EP disclosed
EP-3565808-A1 COMPOUNDS USEFUL FOR TREATING GASTROINTESTINAL TRACT DISORDERS Ardelyx, Inc. (US) 2019-11-13 EP disclosed
EP-3565549-A1 SELECTIVE HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF HUMAN DISEASE Shuttle Pharmaceuticals, Inc. (US) 2019-11-13 EP disclosed
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CN-110430877-A Compositions and methods for treating androgen-independent cancer UNIV CALIFORNIA 2019-11-08 CN disclosed
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EP-3562893-A1 MODIFICATION OF SURFACE PROPERTIES OF MICROFLUIDIC DEVICES Bio-Rad Laboratories, Inc. (US) 2019-11-06 EP disclosed
EP-2701505-B1 FORMULATION COMPONENT SYNGENTA LTD (GB) 2019-11-06 EP disclosed
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US-10463663-B2 Pyridazinone compounds and their use as DAAO inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2019-11-05 US disclosed
US-20190330202-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2019-10-31 US disclosed
US-20190330261-A1 LIGAND FOR ORPHAN NUCLEAR RECEPTOR NUR77 AND USES THEREOF XIAMEN UNIVERSITY (CN) 2019-10-31 US disclosed
US-20190330212-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL ELI LILLY AND COMPANY 2019-10-31 US disclosed
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EP-3558976-A1 SUBSTITUTED AZOLYLPYRROLONES AND AZOLYLHYDANTOINES AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES Bayer CropScience Aktiengesellschaft (DE) 2019-10-30 EP disclosed
EP-3402795-B1 5-SUBSTITUTED 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES Bayer Pharma AG (DE) 2019-10-30 EP disclosed
EP-3558975-A1 SUBSTITUTED HETEROARYL PYRROLONES AND SALTS THEREOF AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES Bayer CropScience Aktiengesellschaft (DE) 2019-10-30 EP disclosed
EP-3558979-A1 NOVEL BENZYLAMINO SUBSTITUTED QUINAZOLINES AND DERIVATIVES AS SOS1 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2019-10-30 EP disclosed
EP-3558986-A1 SUBSTITUTED 1,2,4-THIADIAZOLYL PYRROLONES AND 1,2,4-THIADIAZOLYL HYDANTOINES AND SALTS THEREOF AND USE THEREOF AS HERBICIDES Bayer CropScience Aktiengesellschaft (DE) 2019-10-30 EP disclosed
EP-3559120-A1 AQUEOUS POLYMER COMPOSITION Commonwealth Scientific and Industrial Research Organisation (AU) 2019-10-30 EP disclosed
EP-3558386-A1 PRODRUGS OF CYTOTOXIC ACTIVE AGENTS HAVING ENZYMATICALLY CLEAVABLE GROUPS Bayer Aktiengesellschaft (DE) 2019-10-30 EP disclosed
CN-110386921-A Fibroblast growth factor acceptor inhibitor compound 南京药捷安康生物科技有限公司 2019-10-29 CN disclosed
CN-110392571-A Substituted 3-dialkylaminomethyl-piperidin-4-yl-benzamides and methods of making and using the same 梅比斯发现公司 2019-10-29 CN disclosed
US-10456395-B2 Substituted dipyrido[1,2-a:1′,2′-d]pyrazines for treating viral infections GILEAD SCIENCES, INC. (US) 2019-10-29 US disclosed
US-20190322684-A1 THIOPHENE DERIVATIVES TIANJIN HEMAY PHARMACEUTICAL CO., LTD. (CN) 2019-10-24 US disclosed
US-20190322624-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS MISSION THERAPEUTICS LIMITED (GB) 2019-10-24 US disclosed
US-20190322667-A1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2019-10-24 US disclosed
WO-2019204364-A1 COMPOSITIONS AND METHODS FOR THE SELECTIVE DELIVERY OF THERAPEUTIC AND IMAGING AGENTS AVELAS BIOSCIENCES, INC. (US) 2019-10-24 WO disclosed
WO-2019201255-A1 ISOINDOLE DERIVATIVE 天津合美医药科技有限公司 2019-10-24 WO disclosed
WO-2019201848-A1 2-METHYL-AZA-QUINAZOLINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-10-24 WO disclosed
EP-2972349-B1 POLYMER DOT COMPOSITIONS AND RELATED METHODS UNIV WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2019-10-23 EP disclosed
EP-3555063-A1 NEW 6-AMINO-QUINOLINONE COMPOUNDS AND DERIVATIVES AS BCL6 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2019-10-23 EP disclosed
EP-3554505-A1 METHODS OF TREATING OCULAR DISORDERS Beta Therapeutics Pty. Ltd. (AU) 2019-10-23 EP disclosed
CN-110357888-A Heterocycle phosphodiesterase inhibitors and application thereof 南京药捷安康生物科技有限公司 2019-10-22 CN disclosed
US-20190314524-A1 NOVEL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS ACUITAS THERAPEUTICS INC (CA) 2019-10-17 US disclosed
US-20190315710-A1 Pd(II)-catalyzed Enantioselective Beta-Methylene C(sp3)–H Bond Activation THE SCRIPPS RESEARCH INSTITUTE 2019-10-17 US disclosed
US-20190315798-A1 WITHANOLIDES USEFUL FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES IMSTAR THERAPEUTICS INC (CA) 2019-10-17 US disclosed
US-20190315703-A1 BENZOHETEROCYCLIC ALKYLAMINE COMPOUNDS AND USE THEREOF EAST CHINA UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2019-10-17 US disclosed
US-20190314369-A1 Methods of Treating Cancers, Immune and Autoimmune Diseases, and Inflammatory Diseases Based on BTK Occupancy and BTK Resynthesis Rate ACERTA PHARMA BV (NL) 2019-10-17 US disclosed
US-20190314347-A1 SUBSTITUTED PYRIDINONE-CONTAINING TRYCYCLIC COMPOUNDS, AND METHODS USING SAME ARBUTUS BIOPHARMA, INC. 2019-10-17 US disclosed
WO-2019200254-A1 PIM KINASE INHIBITORS FOR TREATMENT OF MYELOPROLIFERATIVE NEOPLASMS AND FIBROSIS ASSOCIATED WITH CANCER TOLERO PHARMACEUTICALS, INC. (US) 2019-10-17 WO disclosed
WO-2019197371-A1 OXADIAZOLINE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2019-10-17 WO disclosed
EP-3551628-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Celtaxsys Inc. (US) 2019-10-16 EP disclosed
EP-3551608-A1 PENDANT AMINES AND DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Celtaxsys Inc. (US) 2019-10-16 EP disclosed
EP-3551611-A1 MONAMINE AND MONOAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Celtaxsys Inc. (US) 2019-10-16 EP disclosed
EP-3551626-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2019-10-16 EP disclosed
EP-3551169-A1 DELIVERY OF TARGET SPECIFIC NUCLEASES Sangamo Therapeutics, Inc. (US) 2019-10-16 EP disclosed
EP-3552630-A1 NHE3-BINDING COMPOUNDS FOR INHIBITING PHOSPHATE TRANSPORT Ardelyx, Inc. (US) 2019-10-16 EP disclosed
EP-2970543-B1 ALKYL-ACID LIGANDS FOR NANOCRYSTALS NANOSYS INC (US) 2019-10-16 EP disclosed
US-10444243-B2 Encoded chromophoric polymer particles and methods of use thereof UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2019-10-15 US disclosed
US-10442772-B2 Benzimidazol-2-amines as mIDH1 inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-10-15 US disclosed
CN-110325542-A The pro-drug of clofarabine 劳伦斯·I·吴 2019-10-11 CN disclosed
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WO-2019195751-A1 INDENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION AQUINOX PHARMACEUTICALS (CANADA) INC. (CA) 2019-10-10 WO disclosed
WO-2019195753-A1 AXL KINASE INHIBITORS AND USE OF THE SAME TOLERO PHARMACEUTICALS, INC. (US) 2019-10-10 WO disclosed
WO-2019195692-A1 HEXADECAHYDRO-1H-CYCLOPENTA[A]PHENANTHRENE DERIVATIVES USEFUL IN TREATING PAIN AND INFLAMMATION AQUINOX PHARMACEUTICALS (CANADA) INC. (CA) 2019-10-10 WO disclosed
WO-2019195135-A1 SUBSTITUTED CHROMENONES, IRE1 INHIBITORS, AND METHODS OF USING SAME THE WISTAR INSTITUTE (US) 2019-10-10 WO disclosed
US-20190308967-A1 PROCESS FOR THE MANUFACTURE OF 6-ALKYNYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2019-10-10 US disclosed
US-20190307743-A1 OPIOID RECEPTOR ANTAGONIST PRODRUGS NIRSUM LABORATORIES, INC. 2019-10-10 US disclosed
US-20190308989-A1 OPIOID RECEPTOR ANTAGONIST PRODRUGS NIRSUM LABORATORIES, INC. 2019-10-10 US disclosed
US-20190308988-A1 OPIOID RECEPTOR ANTAGONIST PRODRUGS NIRSUM LABORATORIES, INC. 2019-10-10 US disclosed
EP-2739678-B1 GLASS FILLED COPOLYMER PRODUCTS FOR THIN WALL AND HIGH SURFACE GLOSS ARTICLES SABIC GLOBAL TECHNOLOGIES BV (NL) 2019-10-09 EP disclosed
EP-3169721-B1 SILICONE LIGANDS FOR QUANTUM DOTS NANOSYS INC (US) 2019-10-09 EP disclosed
EP-3549963-A2 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS Kodiak Sciences Inc. (US) 2019-10-09 EP disclosed
EP-3549581-A2 COMPOUNDS WITH (1E, 6E)-1,7-BIS-(3,4-DIMETHOXYPHENYL)-4,4-DISSTITUTED-HEPA-1,6-DIENE-3,5-DIONE STRUCTURAL SCAFFOLD, THEIR BIOLOGICAL ACTIVITY, AND USES THEREOF Allianz Pharmascience Ltd (TW) 2019-10-09 EP disclosed
US-10435563-B2 Water soluble fluorescent or colored dyes and methods for their use SONY CORPORATION (JP) 2019-10-08 US disclosed
US-10435375-B2 CXCR4 chemokine receptor modulators NORTHWESTERN UNIVERSITY (US) 2019-10-08 US disclosed
US-10435514-B2 Organosilica materials, methods of making, and uses thereof EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2019-10-08 US disclosed
CN-110312730-A Cytotoxin and conjugate, its Use and preparation method 四川科伦博泰生物医药股份有限公司 2019-10-08 CN disclosed
WO-2019191624-A1 SUBSTITUTED 1,1'-BIPHENYL COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA, INC. (US) 2019-10-03 WO disclosed
WO-2019191227-A1 METHODS OF REDUCING INFLAMMATION OF THE DIGESTIVE SYSTEM WITH INHIBITORS OF HIF-2-ALPHA PELOTON THERAPEUTICS, INC. (US) 2019-10-03 WO disclosed
EP-3546454-A1 BENZOHETEROCYCLYL ALKYLAMINE COMPOUND AND USE THEREOF East China University of Science and Technology (CN) 2019-10-02 EP disclosed
EP-3545974-A1 MEDICAL USE OF ANTI-C MET ANTIBODY-CYTOTOXIC DRUG CONJUGATE Suzhou Suncadia Biopharmaceuticals Co., Ltd. (CN) 2019-10-02 EP disclosed
EP-3055290-B1 INHIBITORS OF KRAS G12C ARAXES PHARMA LLC (US) 2019-10-02 EP disclosed
CN-110294742-A And ring class ASK1 inhibitor and its application 山东轩竹医药科技有限公司 2019-10-01 CN disclosed
US-10428072-B2 Inhibiting the transient receptor potential A1 ion channel ELI LILLY AND COMPANY (US) 2019-10-01 US disclosed
US-10428064-B2 Fused-tricyclic inhibitors of KRAS and methods of use thereof ARAXES PHARMA LLC (US) 2019-10-01 US disclosed
CN-110291073-A Heparanase inhibitors and application thereof 贝塔医疗私人有限公司 2019-09-27 CN disclosed
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US-20190290644-A1 Methods of Treating Chronic Lymphocytic Leukemia and Small Lymphocytic Leukemia Using a BTK Inhibitor ACERTA PHARMA B.V. (NL) 2019-09-26 US disclosed
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WO-2019183140-A1 TOUGH, HEALABLE COMPOSITES DISPLAYING STRESS RELAXATION AT THE RESIN-FILLER INTERFACE THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2019-09-26 WO disclosed
EP-3541820-A1 MAGL INHIBITORS Abide Therapeutics, Inc. (US) 2019-09-25 EP disclosed
EP-3541822-A1 MAGL INHIBITORS Abide Therapeutics, Inc. (US) 2019-09-25 EP disclosed
EP-3541821-A1 MAGL INHIBITORS Abide Therapeutics, Inc. (US) 2019-09-25 EP disclosed
EP-3543207-A1 WESTERN BLOT ANALYSIS USING POLYMER DOTS University Of Washington Through Its Center For Commercialization (US) 2019-09-25 EP disclosed
CN-105793249-B Piperidine derivatives for the treatment or prevention of psychiatric and neurological disorders 武田药品工业株式会社 2019-09-24 CN disclosed
US-20190282568-A1 DUAL MAGL AND FAAH INHIBITORS LUNDBECK LA JOLLA RESEARCH CENTER, INC. 2019-09-19 US disclosed
US-20190282661-A1 METHODS OF TREATING BREAST CANCER Blaze Bioscience, Inc. 2019-09-19 US disclosed
US-20190282535-A1 COMBINATION THERAPY OF A HIF-2-ALPHA INHIBITOR AND AN IMMUNOTHERAPEUTIC AGENT AND USES THEREOF PELOTON THERAPEUTICS, INC. 2019-09-19 US disclosed
US-20190284138-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS MISSION THERAPEUTICS LIMITED (GB) 2019-09-19 US disclosed
US-20190284144-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC 2019-09-19 US disclosed
US-20190284343-A1 POLYURETHANE/UREA COMPOSITIONS FOLDAX, INC. 2019-09-19 US disclosed
WO-2019178528-A1 NANOPARTICLE COMPOSITIONS JANUARY THERAPEUTICS, INC. (US) 2019-09-19 WO disclosed
WO-2019177937-A1 SUBSTITUTED 2-PYRIDONE TRICYCLIC COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA, INC. (US) 2019-09-19 WO disclosed
EP-3538099-A1 EFFICIENT AND SCALABLE SYNTHESES OF NICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, MODIFIED DERIVATIVES THEREOF, PHOSPHORYLATED ANALOGS THEREOF, ADENYLYL DINUCLEOTIDE CONJUGATES THEREOF, AND NOVEL CRYSTALLINE FORMS THEREOF The Queen's University of Belfast (GB) 2019-09-18 EP disclosed
EP-3074482-B1 ENCODED CHROMOPHORIC POLYMER PARTICLES UNIV WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2019-09-18 EP disclosed
US-10414750-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2019-09-17 US disclosed
US-10413536-B2 6-alkyny-pyridine derivatives BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2019-09-17 US disclosed
US-10414771-B2 Compounds useful for inhibiting metastasis from cancer and methods using same DREXEL UNIVERSITY (US) 2019-09-17 US disclosed
US-10414757-B2 2-substituted quinazoline compounds comprising a substituted heterocyclic group and methods of use thereof ARAXES PHARMA LLC (US) 2019-09-17 US disclosed
CN-110229157-A Pyrimido 5-membered aromatic heterocycle class compound, preparation method and the usage 上海海和药物研究开发有限公司 2019-09-13 CN disclosed
US-20190275028-A1 NHE3-BINDING COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. (US) 2019-09-12 US disclosed
US-20190274968-A1 NUCLEOSIDE-MODIFIED RNA FOR INDUCING AN ADAPTIVE IMMUNE RESPONSE NIH - DEITR 2019-09-12 US disclosed
US-20190276805-A1 METHOD FOR ENANTIOSELECTIVE CARBENE C-H INSERTION USING AN IRON-CONTAINING PROTEIN CATALYST CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2019-09-12 US disclosed
WO-2019170543-A1 IDENTIFICATION AND USE OF ERK5 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2019-09-12 WO disclosed
WO-2019170063-A1 INDOLIZINE COMPOUNDS, PREPARATION METHOD AND USE THEREOF 上海海和药物研究开发有限公司 2019-09-12 WO disclosed
WO-2019170750-A1 METHODS AND COMPOSITIONS OF ISOINDOLINE-1,3-DIONE AND ISOINDOLE PRODRUGS USEFUL FOR TREATING CANCER, ULCERATIVE COLITIS AND RELATED INFLAMMATORY DISEASES CELGENE INTERNATIONAL II SARL (CH) 2019-09-12 WO disclosed
WO-2019173633-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF INSULIN RESISTANCE TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2019-09-12 WO disclosed
WO-2019173640-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF INSULIN RESISTANCE TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2019-09-12 WO disclosed
WO-2019143560-A9 METHODS FOR PROMOTING MITOCHONDRIAL BIOGENESIS IN NEURAL CELLS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-09-12 WO disclosed
WO-2019173516-A1 SERINE THREONINE KINASE (AKT) DEGRADATION / DISRUPTION COMPOUNDS AND METHODS OF USE ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2019-09-12 WO disclosed
WO-2019173814-A1 PROTECTIVE GROUPS AND METHODS FOR PROTECTING BENZOXABOROLES OR OXABOROLES UNIVERSITY OF THE SCIENCES (US) 2019-09-12 WO disclosed
EP-3534903-A1 SUBSTITUTED PYRIDINONE-CONTAINING TRICYCLIC COMPOUNDS, AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2019-09-11 EP disclosed
US-20190270708-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS MISSION THERAPEUTICS LIMITED (GB) 2019-09-05 US disclosed
US-20190271016-A1 METHOD FOR THE SYNTHESIS OF TRYPTOPHAN ANALOGS IN AQUEOUS SOLVENTS AT REDUCED TEMPERATURES CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2019-09-05 US disclosed
US-20190269718-A1 METHODS FOR ADVERSELY AFFECTING BIOFILMS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2019-09-05 US disclosed
US-20190271686-A1 ALZHEIMER'S DISEASE ASSAY IN A LIVING PATIENT PAIN THERAPEUTICS, INC. 2019-09-05 US disclosed
US-20190269785-A1 CYTOTOXIC AND ANTI-MITOTIC COMPOUNDS, AND METHODS OF USING THE SAME ZYMEWORKS BC INC. (CA) 2019-09-05 US disclosed
US-20190270806-A1 IL-6 ANTIBODIES AND FUSION CONSTRUCTS AND CONJUGATES THEREOF KODIAK SCIENCES INC. 2019-09-05 US disclosed
EP-3532103-A1 LIPID NANOPARTICLE FORMULATIONS Acuitas Therapeutics, Inc. (CA) 2019-09-04 EP disclosed
EP-3532097-A1 NUCLEOSIDE-MODIFIED RNA FOR INDUCING AN ADAPTIVE IMMUNE RESPONSE The Trustees Of The University Of Pennsylvania (US) 2019-09-04 EP disclosed
EP-3253766-B1 COMPOUNDS AND METHODS FOR PREVENTING OR TREATING SENSORY HAIR CELL DEATH UNIV WASHINGTON (US) 2019-09-04 EP disclosed
US-10399994-B2 Compounds and methods for preventing or treating sensory hair cell death UNIVERSITY OF WASHINGTON (US) 2019-09-03 US disclosed
US-10399953-B2 Preparation of furan fatty acids from 5-(chloromethyl)furfural THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-09-03 US disclosed
US-10399986-B2 Inhibitors of leukotriene A4 hydrolase CELTAXSYS, INC. (US) 2019-09-03 US disclosed
US-10398721-B2 Methods for treating progeroid laminopathies using oligonucleotide analogues targeting human LMNA SAREPTA THERAPEUTICS, INC. (US) 2019-09-03 US disclosed
US-10399982-B2 Substituted xanthines and methods of use thereof HYDRA BIOSCIENCES, INC. (US) 2019-09-03 US disclosed
US-20190263748-A1 CONVERSION OF LIGNIN TO IONIC LIQUIDS NATIONAL TECHNOLOGY & ENGINEERING SOLUTIONS OF SANDIA, LLC 2019-08-29 US disclosed
US-20190263953-A1 Polyethylene Compositions and Articles Made Therefrom EXXONMOBIL CHEMICAL PATENTS INC. 2019-08-29 US disclosed
US-20190262342-A1 COMBINATION THERAPIES FOR TREATMENT OF CANCER ARAXES PHARMA LLC 2019-08-29 US disclosed
US-20190263783-A1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS, INC. 2019-08-29 US disclosed
US-20190263738-A1 PROCESS FOR PREPARING 2,3-UNSATURATED ALCOHOLS BASF SE (DE) 2019-08-29 US disclosed
US-20190263818-A1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS, INC. 2019-08-29 US disclosed
WO-2019162228-A1 1-(5-SUBSTITUTED IMIDAZOL-1-YL)BUT-3-EN DERIVATIVES AND THEIR USE AS FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 2019-08-29 WO disclosed
WO-2019162323-A1 NEW BENZIMIDAZOLE COMPOUNDS AND DERIVATIVES AS EGFR INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2019-08-29 WO disclosed
WO-2019165189-A1 PROTEIN ARGININE METHYLTRANSFERASE 5 (PRMT5) DEGRADATION / DISRUPTION COMPOUNDS AND METHODS OF USE ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2019-08-29 WO disclosed
EP-3529254-A1 PRODRUGS OF CLOFARABINE Wu, Laurence I. (TW) 2019-08-28 EP disclosed
CN-110177822-A The synthesis of polycarbonate siloxane glycol 奥特克国际公开有限公司 2019-08-27 CN disclosed
US-10392380-B2 Compounds MISSION THERAPEUTICS LIMITED (GB) 2019-08-27 US disclosed
CN-110156770-A Aminopyrazole derivatives as TAM race kinase inhibitor 圣诺康生命科学公司 2019-08-23 CN disclosed
US-20190256527-A1 Purification of Rapamycin Derivatives Using Temperature Induced Phase Separation JOHNSON MATTHEY PHARMACEUTICAL MATERIALS, INC. D/B/A JOHNSON MATTHEY PHARMA SERVICES 2019-08-22 US disclosed
US-20190256518-A1 PIPERIDINE DERIVATIVES AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 7 GENETECH, INC. 2019-08-22 US disclosed
US-20190255155-A1 BUTYRYLCHOLINESTERASE ZWITTERIONIC POLYMER CONJUGATES OLIGASIS, LLC 2019-08-22 US disclosed
US-20190256552-A1 Amino Acid and Peptide Conjugates and Uses Thereof AUCKLAND UNISERVICES LIMITED (NZ) 2019-08-22 US disclosed
US-20190256494-A1 PYRAZOLE COMPOUNDS AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2019-08-22 US disclosed
EP-3105209-B1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS Bayer Pharma AG (DE) 2019-08-21 EP disclosed
EP-3527573-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS Gilead Sciences, Inc. (US) 2019-08-21 EP disclosed
US-10385057-B2 Pyrazole compounds and methods of making and using same LUNDBECK LA JOLLA RESEARCH CENTER, INC. (US) 2019-08-20 US disclosed
US-10385062-B2 Thiophene derivatives TIANJIN HEMAY BIO-TECH CO., LTD. (CN) 2019-08-20 US disclosed
US-10385047-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2019-08-20 US disclosed
US-10385051-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2019-08-20 US disclosed
US-10383831-B2 2,4,6-trialkoxystryl aryl sulfones, sulfonamides and carboxamides, and methods of preparation and use Temple University—Of the Commonwealth System of Higher Education (US) 2019-08-20 US disclosed
US-10385007-B2 Monamine and monoamine derivatives as inhibitors of leukotriene A4 hydrolase CELTAXSYS, INC. (US) 2019-08-20 US disclosed
US-10385024-B2 Compounds and methods for inhibiting NHE-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders ARDELYX, INC. (US) 2019-08-20 US disclosed
CN-110128998-A A kind of allyl organic silicon potting adhesive and preparation method thereof 矽时代材料科技股份有限公司 2019-08-16 CN disclosed
US-20190248815-A1 ORGANIC MAGNESIUM PHOSPHIDE AND MANUFACTURING METHOD THEREOF, ORGANIC MAGNESIUM PHOSPHIDE COMPLEX AND MANUFACTURING METHOD THEREOF, AND MANUFACTURING METHOD OF ORGANIC PHOSPHORUS COMPOUND USING SAID PHOSPHIDE HOKKO CHEMICAL INDUSTRY CO., LTD. (JP) 2019-08-15 US disclosed
US-20190248795-A1 WEE-1 INHIBITING PYRAZOLOPYRIMIDINONE COMPOUNDS ALMAC DISCOVERY LIMITED (GB) 2019-08-15 US disclosed
WO-2019154120-A1 CYTOTOXIC AGENT AND CONJUGATE THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-08-15 WO disclosed
WO-2019157013-A1 COMPOSITIONS AND METHODS FOR SELECTIVE SEPARATION OF HYDROCARBON ISOMERS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2019-08-15 WO disclosed
US-20190249179-A1 FIBROTIC TREATMENT MONASH UNIVERSITY (AU) 2019-08-15 US disclosed
EP-3523315-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR Oric Pharmaceuticals, Inc. (US) 2019-08-14 EP disclosed
EP-3523289-A1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF RAS AND METHODS OF USE THEREOF Araxes Pharma LLC (US) 2019-08-14 EP disclosed
EP-3524602-A1 PYRIDO FIVE-ELEMENT AROMATIC RING COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Haihe Pharmaceutical Co., Ltd. (CN) 2019-08-14 EP disclosed
US-10376481-B2 Compounds and methods for inhibiting NHE-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders ARDELYX, INC. (US) 2019-08-13 US disclosed
US-10377743-B2 Inhibitors of RAS and methods of use thereof ARAXES PHARMA LLC (US) 2019-08-13 US disclosed
US-10376535-B2 Therapy for malignant disease UNIVERSITY OF ROCHESTER (US) 2019-08-13 US disclosed
WO-2019152883-A1 INHIBITORS OF PROTEIN ARGININE DEIMINASES PADFORWARD LLC (US) 2019-08-08 WO disclosed
WO-2019152641-A1 BENZOXABOROLE COMPOSITIONS HAVING A GROWTH ENHANCING EFFECT Boragen, Inc. (US) 2019-08-08 WO disclosed
WO-2019152465-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL ELI LILLY AND COMPANY (US) 2019-08-08 WO disclosed
WO-2019149116-A1 METHOD FOR PREPARING CONJUGATE 四川科伦博泰生物医药股份有限公司 2019-08-08 WO disclosed
US-20190240223-A1 TREATMENT OF RELAPSED AND/OR REFRACTORY SOLID TUMORS AND NON-HODGKIN'S LYMPHOMAS CELGENE CORPORATION (US) 2019-08-08 US disclosed
US-20190240212-A1 METHODS OF TREATING RBP4 RELATED DISEASES WITH TRIAZOLOPYRIDINES THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2019-08-08 US disclosed
US-20190241890-A1 METHODS AND COMPOSITIONS FOR MANIPULATING TRANSLATION OF PROTEIN ISOFORMS FROM ALTERNATIVE INITIATION START SITES SAREPTA THERAPEUTICS INC (US) 2019-08-08 US disclosed
US-20190240219-A1 TRIAZOLOPYRAZINE BOEHRINGER INGELHEIM INT (DE) 2019-08-08 US disclosed
US-20190240203-A1 NOVEL ANTIBIOTICS AND METHODS OF USING SAME THE BROAD INSTITUTE, INC. (US) 2019-08-08 US disclosed
US-20190240217-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2019-08-08 US disclosed
US-20190240222-A1 TREATMENT OF RELAPSED AND/OR REFRACTORY SOLID TUMORS AND NON-HODGKIN'S LYMPHOMAS CELGENE CORPORATION (US) 2019-08-08 US disclosed
EP-3519412-A1 CYANOPYRROLIDINE DERIVATIVES WITH ACTIVITY AS INHIBITORS OF USP30 Mission Therapeutics Limited (GB) 2019-08-07 EP disclosed
EP-3521399-A1 ENCODED CHROMOPHORIC POLYMER PARTICLES University of Washington through its Center for Commercialization (US) 2019-08-07 EP disclosed
EP-3519816-A1 COMPOUNDS FOR INCREASING NEURAL PLASTICITY The Regents of the University of California (US) 2019-08-07 EP disclosed
EP-3519402-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS Araxes Pharma LLC (US) 2019-08-07 EP disclosed
EP-3519397-A1 CYANO-SUBTITUTED HETEROCYCLES WITH ACTIVITY AS INHIBITORS OF USP30 Mission Therapeutics Limited (GB) 2019-08-07 EP disclosed
US-10370386-B2 Substituted quinolines as inhibitors of KRAS G12C ARAXES PHARMA LLC (US) 2019-08-06 US disclosed
CN-110090308-A The method for preparing conjugate 四川科伦博泰生物医药股份有限公司 2019-08-06 CN disclosed
CN-110092750-A Amides compound that Pentafluorosulfanyl replaces, preparation method and its in application pharmaceutically 北京诺诚健华医药科技有限公司 2019-08-06 CN disclosed
CN-110088096-A Piperidine derivatives as inhibitors of ubiquitin-specific protease 7 阿尔麦克探索有限公司 2019-08-02 CN disclosed
WO-2019145532-A1 FLUORESCENT POLYMERIC COATING FILM FOR MEDICAL DEVICES UNIVERSITE DE STRASBOURG (FR) 2019-08-01 WO disclosed
WO-2019147865-A1 A METHOD FOR ENANTIOSELECTIVE CARBENE C-H INSERTION USING AN IRON-CONTAINING PROTEIN CATALYST CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2019-08-01 WO disclosed
US-20190233394-A1 PHARMACEUTICAL COMPOUNDS ALMAC DISCOVERY LIMITED (GB) 2019-08-01 US disclosed
US-20190231775-A1 Methods of Blocking the CXCR-4/SDF-1 Signaling Pathway With Inhibitors of Bruton's Tyrosine Kinase ACERTA PHARMA BV (NL) 2019-08-01 US disclosed
EP-3517146-A1 FLUORESCENT POLYMERIC COATING FILM FOR MEDICAL DEVICES Université de Strasbourg (FR) 2019-07-31 EP disclosed
EP-3517535-A1 ALKYNYL-SUBSTITUTED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF Beijing InnoCare Pharma Tech Co., Ltd. (CN) 2019-07-31 EP disclosed
EP-3516061-A1 MIXED TRICYCLO-DNA, 2'-MODIFIED RNA OLIGONUCLEOTIDE COMPOSITIONS AND USES THEREOF Synthena AG (CH) 2019-07-31 EP disclosed
EP-3515897-A1 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME Abide Therapeutics, Inc. (US) 2019-07-31 EP disclosed
EP-3194387-B1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2019-07-31 EP disclosed
EP-2831042-B1 HETEROARYL COMPOUNDS WITH A-CYCLIC BRIDGING UNIT INTERVET INT BV (NL) 2019-07-31 EP disclosed
US-10363290-B2 Butyrylcholinesterase zwitterionic polymer conjugates KODIAK SCIENCES INC. (US) 2019-07-30 US disclosed
US-10363239-B2 Method for inhibiting growth of cancer cells PAIN THERAPEUTICS (US) 2019-07-30 US disclosed
US-10363249-B2 Fatty acid synthase inhibitor for use in the treatment of drug resistant cancer 3-V BIOSCIENCES, INC. (US) 2019-07-30 US disclosed
WO-2019143560-A1 METHODS FOR PROMOTING MITOCHONDRIAL BIOGENESIS IN NEURAL CELLS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-07-25 WO disclosed
WO-2019142053-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2019-07-25 WO disclosed
WO-2019142135-A1 TRICYCLO-DNA NUCLEOSIDE PRECURSORS AND PROCESSES FOR PREPARING THE SAME SYNTHENA AG (CH) 2019-07-25 WO disclosed
US-20190223438-A1 UREA AND THIOUREA SUBSTITUTED BICYCLES DERIVATIVES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2019-07-25 US disclosed
US-20190225593-A1 SUBSTITUTED CHROMANE-8-CARBOXAMIDE COMPOUNDS AND ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORP (CA) 2019-07-25 US disclosed
EP-2864420-B1 SILICONE LIGANDS FOR STABILIZING QUANTUM DOT FILMS NANOSYS INC (US) 2019-07-24 EP disclosed
EP-3512840-A1 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS Tseng, Yufeng, Jane (US) 2019-07-24 EP disclosed
US-10358447-B2 Substituted 2-N-hydroxy-1,3-dioxo-1,2,3,4-tetrahydronaphthyridines, and methods of making and using same ARBUTUS BIOPHARMA CORPORATION (CA) 2019-07-23 US disclosed
US-20190218215-A1 CYANO-SUBTITUTED HETEROCYCLES WITH ACTIVITY AS INHIBITORS OF USP30 MISSION THERAPEUTICS LIMITED (GB) 2019-07-18 US disclosed
US-20190218554-A1 Mixed Tricyclo-DNA, 2'-Modified RNA Oligonucleotide Compositions and Uses Thereof SYNTHENA AG (CH) 2019-07-18 US disclosed
US-20190218212-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD PHARMACEUTICALS, INC. 2019-07-18 US disclosed
US-20190218246-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. 2019-07-18 US disclosed
US-20190218551-A1 OLIGONUCLEOTIDE ANALOGUES HAVING MODIFIED INTERSUBUNIT LINKAGES AND/OR TERMINAL GROUPS JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2019-07-18 US disclosed
EP-3511319-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Celgene Quanticel Research, Inc. (US) 2019-07-17 EP disclosed
US-10351580-B2 Acene-based transmitter molecules for photon upconversion THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-07-16 US disclosed
US-10351639-B2 Organosilica materials for use as adsorbents for oxygenate removal EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2019-07-16 US disclosed
US-10350205-B2 Dual MAGL and FAAH inhibitors ABIDE THERAPEUTICS, INC. (US) 2019-07-16 US disclosed
US-10351590-B2 Withanolides useful for the treatment of neurodegenerative diseases IMSTAR THERAPEUTICS INC. (CA) 2019-07-16 US disclosed
US-10351550-B2 Substituted quinazoline compounds and methods of use thereof ARAXES PHARMA LLC (US) 2019-07-16 US disclosed
US-20190211010-A1 PYRIDO FIVE-ELEMENT AROMATIC RING COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF HAIHE BIOPHARMA CO. LTD. (CN) 2019-07-11 US disclosed
US-20190209591-A1 Therapeutic Combinations of a Proteasome Inhibitor and a BTK Inhibitor ACERTA PHARMA BV (NL) 2019-07-11 US disclosed
US-20190212326-A1 Method for the Selection of Patients and Kit ALLIANZ PHARMASCIENCE LTD. (TW) 2019-07-11 US disclosed
US-20190209564-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR AND USE THEREOF NANJING TRANSTHERA BIOSCIENCES CO LTD (CN) 2019-07-11 US disclosed
US-20190211367-A1 VIVO AND IN VITRO OLEFIN CYCLOPROPANATION CATALYZED BY HEME ENZYMES CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2019-07-11 US disclosed
US-20190210997-A1 ALKYNYL-SUBSTITUTED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF BEIJING INNOCARE PHARMA TECH CO., LTD. (CN) 2019-07-11 US disclosed
WO-2019136025-A1 ASK1 INHIBITOR COMPOUNDS AND USES THEREOF Seal Rock Therapeutics, Inc. (US) 2019-07-11 WO disclosed
WO-2019135975-A1 ENHANCEMENT OF NUCLEIC ACID POLYMERIZATION BY AROMATIC COMPOUNDS STRATOS GENOMICS INC. (US) 2019-07-11 WO disclosed
EP-3508855-A1 METHOD FOR THE SELECTION OF PATIENTS AND KIT Allianz Pharmascience Ltd (TW) 2019-07-10 EP disclosed
EP-3506983-A1 SUBSTITUTED UREAS AND METHODS OF MAKING AND USING SAME Mebias Discovery LLC (US) 2019-07-10 EP disclosed
EP-3508482-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR AND USE THEREOF Nanjing Transthera Biosciences Co. Ltd. (CN) 2019-07-10 EP disclosed
US-10344281-B2 Functionally-modified oligonucleotides and subunits thereof SAREPTA THERAPEUTICS, INC. (US) 2019-07-09 US disclosed
US-10343992-B2 1-cyano-pyrrolidine compounds as USP30 inhibitors Missions Therapeutics Limited (GB) 2019-07-09 US disclosed
US-20190207113-A1 POLYTHIOPHENE DERIVATIVE, COMPOSITE AND MANUFACTURE METHOD THEREOF SHENZHEN CHINA STAR OPTOELECTRONICS TECHNOLOGY CO., LTD. (CN) 2019-07-04 US disclosed
US-20190202766-A1 ANTIMALARIAL COMPOSITIONS AND USES THEREOF THE SCRIPPS RESEARCH INSTITUTE 2019-07-04 US disclosed
US-20190202835-A1 ISOTOPOLOGUES OF ISOQUINOLINONE AND QUINAZOLINONE COMPOUNDS AND USES THEREOF AS PI3K KINASE INHIBITORS TWELVE THERAPEUTICS, INC. 2019-07-04 US disclosed
US-20190202801-A1 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2019-07-04 US disclosed
EP-3505517-A1 FUSED HETEROCYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF Beijing InnoCare Pharma Tech Co., Ltd. (CN) 2019-07-03 EP disclosed
EP-3504251-A1 NETWORK POLYMERS AND METHODS OF MAKING AND USING SAME The Regents of the University of Colorado, a Body Corporate (US) 2019-07-03 EP disclosed
EP-2887964-B1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX INC (US) 2019-07-03 EP disclosed
EP-2822938-B1 RODENTICIDAL NORBORMIDE ANALOGUES LANDCARE RES NEW ZEALAND LIMITED (NZ) 2019-07-03 EP disclosed
EP-3229953-B1 COATING METHOD USING ORGANOSILICA MATERIAL, COATED SUBSTRATE, AND GAS SEPARATION PROCESS EMPLOYING SAID SUBSTRATE EXXONMOBIL RES & ENG CO (US) 2019-07-03 EP disclosed
EP-2558538-B1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS KODIAK SCIENCES INC (US) 2019-07-03 EP disclosed
US-10336709-B2 Lp-PLA2 inhibitors ABIDE THERAPEUTICS, INC (US) 2019-07-02 US disclosed
CN-109956927-A Benzimidazoles derivative, preparation method and its in application pharmaceutically 北京诺诚健华医药科技有限公司 2019-07-02 CN disclosed
US-10335402-B2 Sulfonyl piperidine derivatives and their use for treating prokineticin mediated gastrointestinal disorders TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2019-07-02 US disclosed
US-10336691-B2 Pesticidally active oxime and hydrazone derivatives SYNGENTA PARTICIPATIONS AG (CH) 2019-07-02 US disclosed
US-10335388-B2 Combination therapy of a HIF-2-alpha inhibitor and an immunotherapeutic agent and uses thereof PELOTON THERAPEUTICS, INC. (US) 2019-07-02 US disclosed
US-10336727-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2019-07-02 US disclosed
US-20190194195-A1 METHOD OF MAKING TETRAHYDRONAPHTHYRIDINYL NONANOIC ACID COMPOUNDS FELIQS CORPORATION (JP) 2019-06-27 US disclosed
US-20190194161-A1 INHIBITOR OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2019-06-27 US disclosed
US-20190194178-A1 SUBSTITUTED UREAS AND METHODS OF MAKING AND USING SAME MEBIAS DISCOVERY LLC 2019-06-27 US disclosed
US-20190194414-A1 METHODS OF PRODUCING ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RES & ENG CO (US) 2019-06-27 US disclosed
US-20190192454-A1 METHODS FOR TREATING CANCER WITH RORGAMMA INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-06-27 US disclosed
US-20190194184-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2019-06-27 US disclosed
US-20190194162-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2019-06-27 US disclosed
US-20190192462-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF INSULIN RESISTANCE TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2019-06-27 US disclosed
US-20190192521-A1 Methods of Treating Arid1A-Mutated Cancers With HDAC6 Inhibitors and EZH2 Inhibitors WISTAR INST (US) 2019-06-27 US disclosed
US-20190194192-A1 NOVEL BENZYLAMINO SUBSTITUTED PYRIDOPYRIMIDINONES AND DERIVATIVES AS SOS1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2019-06-27 US disclosed
EP-3180342-B1 PYRROLO[3,2-D]PYRIMIDINE-2,4(3H,5H)-DIONE DERIVATIVES HYDRA BIOSCIENCES INC (US) 2019-06-26 EP disclosed
US-10329299-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2019-06-25 US disclosed
US-10328074-B2 Substituted [1,2,4]triazolo[4,3-a]pyrazines as BRD4 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2019-06-25 US disclosed
US-10328080-B2 Therapeutic combination of PI3K inhibitor and a BTK inhibitor Acerta Pharma, B.V. (NL) 2019-06-25 US disclosed
US-10328077-B2 Treatment of relapsed and/or refractory solid tumors and non-hodgkin's lymphomas CELGENE CORPORATION (US) 2019-06-25 US disclosed
CN-109908356-A Load the alpha-cyanoacrylate ester material of anti-tumor drug 中国人民解放军军事医学科学院毒物药物研究所 2019-06-21 CN disclosed
CN-109913203-A Chromophoric polymers point with narrow emission 华盛顿大学商业中心 2019-06-21 CN disclosed
WO-2019115338-A1 PROCESS FOR THE PREPARATION OF (5-CYANO-IMIDAZOL-1-YL)ETHANONE DERIVATIVES AND INTERMEDIATES USEFUL THEREFOR BAYER AKTIENGESELLSCHAFT (DE) 2019-06-20 WO disclosed
US-20190186026-A1 ELECTROCHEMICAL OXIDATION OF ALIPHATIC AND AROMATIC COMPOUNDS MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2019-06-20 US disclosed
US-20190190069-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH LINEAR CARBONATE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2019-06-20 US disclosed
US-20190190070-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH CARBOXYLIC ETHER, CARBOXYLIC ACID BASED SALT, OR ACRYLATE ELECTROLYTE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2019-06-20 US disclosed
US-20190183865-A1 NSD FAMILY INHIBITORS AND METHODS OF TREATMENT THEREWITH THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2019-06-20 US disclosed
US-20190183816-A1 ALKOXY COMPOUNDS FOR DISEASE TREATMENT ACUCELA INC. 2019-06-20 US disclosed
US-20190185461-A1 BENZOCYCLIC DERIVATIVE HAVING B2-RECEPTOR AGONIST ACTIVITY AND M3-RECEPTOR ANTAGONIST ACTIVITY AND MEDICAL USE THEREOF SICHUAN HAISCO PHARMACEUTICAL CO., LTD. (CN) 2019-06-20 US disclosed
US-20190185472-A1 FUSED HETEROCYCLIC DERIVATIVES, THEIR PREPARATION METHODS THEREOF AND MEDICAL USES THEREOF BEIJING INNOCARE PHARMA TECH CO., LTD. (CN) 2019-06-20 US disclosed
EP-3496721-A1 TREATMENT OF RELAPSED AND/OR REFRACTORY SOLID TUMORS AND NON-HODGKIN'S LYMPHOMAS Celgene Corporation (US) 2019-06-19 EP disclosed
EP-3497092-A1 SUBSTITUTED PYRAZOLINYL DERIVATES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND/OR PLANT GROWTH REGULATORS Bayer CropScience Aktiengesellschaft (DE) 2019-06-19 EP disclosed
US-10323038-B2 Pyrazole compounds and methods of making and using same ABIDE THERAPEUTICS, INC. (US) 2019-06-18 US disclosed
US-10322132-B2 Prevention or treatment of uratic or gouty diseases SHANTON PHARMA CO., LTD (CN) 2019-06-18 US disclosed
US-10322108-B2 N-benzoate group substituted benzopyrroline-2-one derivative and use thereof Beijing Hanmi Pharmaceutical Co., Ltd. (CN) 2019-06-18 US disclosed
US-10322995-B2 Substituted cyano cycloalkyl penta-2,4-dienes, cyano cycloalkyl pent-2-en-4-ynes, cyano heterocyclyl penta-2,4-dienes and cyano heterocyclyl pent-2-en-4-ynes as active substances against abiotic plant stress BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2019-06-18 US disclosed
WO-2019113236-A1 BENZOCARBONYL COMPOUNDS VIVACE THERAPEUTICS, INC. (US) 2019-06-13 WO disclosed
WO-2019113532-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH FLUORINATED CYCLIC COMPOUND CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION (US) 2019-06-13 WO disclosed
US-20190181441-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH FLUORINATED CYCLIC COMPOUND CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2019-06-13 US disclosed
WO-2019113518-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH LINEAR CARBONATE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION (US) 2019-06-13 WO disclosed
WO-2019113530-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ETHER CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION (US) 2019-06-13 WO disclosed
WO-2019113469-A1 NSD FAMILY INHIBITORS AND METHODS OF TREATMENT THEREWITH THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2019-06-13 WO disclosed
WO-2019113528-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH CARBOXYLIC ETHER, CARBOXYLIC ACID BASED SALT, OR ACRYLATE ELECTROLYTE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION (US) 2019-06-13 WO disclosed
WO-2019113242-A1 TUBULIN INHIBITORS Lin BioScience, LLC (US) 2019-06-13 WO disclosed
US-20190181502-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH ETHER CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2019-06-13 US disclosed
US-20190181501-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH CYCLIC CARBONATE CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2019-06-13 US disclosed
US-20190181500-A1 SILICON-BASED ENERGY STORAGE DEVICES WITH FLUORINATED POLYMER CONTAINING ELECTROLYTE ADDITIVES ENEVATE CORPORATION 2019-06-13 US disclosed
US-20190167816-A1 METHODS FOR PREVENTING OR TREATING FIBROTIC DISEASES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-06-06 US disclosed
US-20190166840-A1 SUBSTITUTED PYRAZOLINYL DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND/OR PLANT GROWTH REGULATORS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2019-06-06 US disclosed
US-20190169128-A1 SUBSTITUTED 1-HYDROXY-PYRIDIN-2(1H)-ONES, AND METHODS OF MAKING AND USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2019-06-06 US disclosed
US-20190169127-A1 TUBULIN INHIBITORS LIN BIOSCIENCE INC. (TW) 2019-06-06 US disclosed
US-20190169185-A1 SUBSTITUTED 2-N-HYDROXY-1,3-DIOXO-1,2,3,4-TETRAHYDRONAPHTHYRIDINES, AND METHODS OF MAKING AND USING SAME ARBUTUS BIOPHARMA, INC. 2019-06-06 US disclosed
US-20190169611-A1 dsRNA MOLECULES COMPRISING OLIGONUCLEOTIDE ANALOGS HAVING MODIFIED INTERSUBUNIT LINKAGES AND/OR TERMINAL GROUPS JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2019-06-06 US disclosed
US-20190169209-A1 NEW SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2019-06-06 US disclosed
EP-3492106-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT Ardelyx, Inc. (US) 2019-06-05 EP disclosed
EP-3009436-B1 KINASE INHIBITORS AND METHODS OF USE INTELLIKINE LLC (US) 2019-06-05 EP disclosed
EP-2968440-B1 CYTOTOXIC AND ANTI-MITOTIC COMPOUNDS, AND METHODS OF USING THE SAME ZYMEWORKS INC (CA) 2019-06-05 EP disclosed
US-10308637-B2 Therapeutic inhibitory compounds LIFESCI PHARMACEUTICALS, INC. (BB) 2019-06-04 US disclosed
US-10308635-B2 1-sulfonyl piperidine derivatives as modulators of prokineticin receptors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2019-06-04 US disclosed
US-20190159457-A1 Combinatorial Compositions of Benzoxaboroles and Biologic Agents 5METIS, INC. 2019-05-30 US disclosed
US-20190161437-A1 PENDANT AMINES AND DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS INC (US) 2019-05-30 US disclosed
US-20190161567-A1 Polyethylene Compositions and Films Made Therefrom EXXONMOBIL CHEMICAL PATENTS INC. 2019-05-30 US disclosed
US-20190161523-A1 METHODS OF TREATMENT USING CHLOROTOXIN CONJUGATES Blaze Bioscience, Inc. 2019-05-30 US disclosed
US-20190161471-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS INC (US) 2019-05-30 US disclosed
US-20190161559-A1 Catalyst Systems and Polymerization Processes for Using the Same EXXONMOBIL CHEMICAL PATENTS INC. 2019-05-30 US disclosed
EP-2240452-B1 1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE DERIVATIVES AS PI3 KINASE MODULATORS, THEIR COMPOSITIONS AND USES INTELLIKINE LLC (US) 2019-05-29 EP disclosed
EP-3487850-A1 UREA AND THIOUREA SUBSTITUTED BICYCLES DERIVATIVES AS PESTICIDES Syngenta Participations AG (CH) 2019-05-29 EP disclosed
US-10300058-B2 Tyrosine kinase inhibitor and uses thereof Xuanzhu Pharma Co., Ltd. (CN) 2019-05-28 US disclosed
US-10301284-B2 Therapeutic inhibitory compounds LIFESCI PHARMACEUTICALS, INC. (BB) 2019-05-28 US disclosed
US-10300069-B2 Carbon monoxide-releasing molecules for therapeutic applications and methods of making and using thereof GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2019-05-28 US disclosed
US-10301317-B2 Inhibitors of ERK and methods of use KURA ONCOLOGY, INC. (US) 2019-05-28 US disclosed
US-20190151318-A1 FATTY LIVER DISEASE TREATMENT USING GLUCOCORTICOID AND MINERALOCORTICOID RECEPTOR ANTAGONISTS CORCEPT THERAPEUTICS, INC. 2019-05-23 US disclosed
US-20190152972-A1 MULTI-KINASE INHIBITOR COMPOUND, AND CRYSTAL FORM AND USE THEREOF TRANSTHERA SCIENCES (NANJING), INC. (CN) 2019-05-23 US disclosed
US-20190152913-A1 1,4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON LLC 2019-05-23 US disclosed
US-20190151289-A1 Identification of Small Molecule Inhibitors of Jumonji AT-Rich Interactive Domain 1A (JARID1A) Histone Demethylase UNIV YALE (US) 2019-05-23 US disclosed
US-20190152993-A1 Reversibly Switchable Surfactants and Methods of Use WARNER BABCOCK INSTITUTE FOR GREEN CHEMISTRY, LLC (US) 2019-05-23 US disclosed
US-20190153306-A1 Photochromic Water Harvesting Platform WARNER BABCOCK INSTITUTE FOR GREEN CHEMISTRY, LLC (US) 2019-05-23 US disclosed
US-20190152965-A1 AMINOPYRIDINE DERIVATIVES AS TAM FAMILY KINASE INHIBITORS SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2019-05-23 US disclosed
US-20190151324-A1 NON-CATALYTIC SUBSTRATE-SELECTIVE P38alpha-SPECIFIC MAPK INHIBITORS WITH ENDOTHELIAL-STABILIZING AND ANTI-INFLAMMATORY ACTIVITY, AND METHODS OF USE THEREOF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2019-05-23 US disclosed
EP-3484887-A1 WEE-1 INHIBITING PYRAZOLOPYRIMIDINONE COMPOUNDS Almac Discovery Limited (GB) 2019-05-22 EP disclosed
EP-3183254-B1 NEW SPIRO[3H-INDOLE-3,2´-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2019-05-22 EP disclosed
CN-109790112-A Cyanopyrrolidine derivatives having activity as USP30 inhibitors 特殊治疗有限公司 2019-05-21 CN disclosed
CN-109790169-A With the Cyanopyrolidine derivatives as USP30 inhibitor activity 特殊治疗有限公司 2019-05-21 CN disclosed
US-10294228-B2 Breathing control modulating compounds, and methods of making and using same NEURAD LTD. (IL) 2019-05-21 US disclosed
US-10294312-B2 Olefin polymerization catalyst system comprising mesoporous organosilica support EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2019-05-21 US disclosed
CN-109790146-A Medical compounds 阿尔麦克探索有限公司 2019-05-21 CN disclosed
CN-109776517-A Heterocyclic indole amine 2,3-dioxygenase inhibitor 南京药捷安康生物科技有限公司 2019-05-21 CN disclosed
US-20190144442-A1 ASH1L INHIBITORS AND METHODS OF TREATMENT THEREWITH THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2019-05-16 US disclosed
US-20190144578-A1 Polymerization Processes EXXONMOBIL CHEMICAL PATENTS INC. 2019-05-16 US disclosed
US-20190142788-A1 USE OF TOPICAL FORMULATIONS OF CANNABINOIDS IN THE TREATMENT OF EPIDERMOLYSIS BULLOSA AND RELATED CONNECTIVE TISSUE DISORDERS INMED PHARMACEUTICALS INC. (CA) 2019-05-16 US disclosed
US-20190144601-A1 PHOTOACTIVE MACROMOLECULES AND USES THEREOF BECKMAN COULTER, INC. 2019-05-16 US disclosed
US-20190144579-A1 Polymerization Processes EXXONMOBIL CHEMICAL PATENTS INC. 2019-05-16 US disclosed
US-20190144575-A1 Polyethylene Compositions and Articles Made Therefrom EXXONMOBIL CHEMICAL PATENTS INC. 2019-05-16 US disclosed
US-20190144576-A1 Polyethylene Compositions and Articles Made Therefrom EXXONMOBIL CHEMICAL PATENTS INC. 2019-05-16 US disclosed
US-20190144580-A1 Polymerization Processes EXXONMOBIL CHEMICAL PATENTS INC. 2019-05-16 US disclosed
US-20190142812-A1 5-SUBSTITUTED 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-05-16 US disclosed
US-20190142853-A1 Inhibition of Galectin 3 Binding to the Airway Epithelial Surface to Treat or Prevent Septic Shock Resulting From Influenza and Subsequent Pneumococcal Pneumonia Infection NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-05-16 US disclosed
US-20190144451-A1 PURINONE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS LLC 2019-05-16 US disclosed
US-20190142799-A1 ASH1L INHIBITORS AND METHODS OF TREATMENT THEREWITH THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2019-05-16 US disclosed
US-20190144424-A1 Macrophage Migration Inhibitory Factor Inhibitors, and Methods of Making and Using Same YALE UNIVERSITY 2019-05-16 US disclosed
US-20190142961-A1 ASH1L DEGRADERS AND METHODS OF TREATMENT THEREWITH THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2019-05-16 US disclosed
EP-3481391-A1 THERAPEUTIC INHIBITORY COMPOUNDS Lifesci Pharmaceuticals, Inc. (BB) 2019-05-15 EP disclosed
EP-2456842-B1 IONIC LIQUID FLAME RETARDANTS INOVIA MAT LLC (US) 2019-05-15 EP disclosed
EP-3043784-B1 ARYL ETHERS AND USES THEREOF PELOTON THERAPEUTICS INC (US) 2019-05-15 EP disclosed
US-10287286-B2 Compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2019-05-14 US disclosed
US-20190136184-A1 METHOD OF INHIBITING TAU PHOSPHORYLATION CASSAVA SCIENCES, INC. 2019-05-09 US disclosed
US-20190136281-A1 CONVERSION OF SUGARS TO IONIC LIQUIDS NATIONAL TECHNOLOGY & ENGINEERING SOLUTIONS OF SANDIA, LLC 2019-05-09 US disclosed
US-20190134028-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2019-05-09 US disclosed
US-20190135833-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2019-05-09 US disclosed
EP-3480204-A1 ORGANIC MAGNESIUM PHOSPHIDE AND METHOD FOR PRODUCING SAME, ORGANIC MAGNESIUM PHOSPHIDE COMPLEX AND METHOD FOR PRODUCING SAME, AND METHOD FOR PRODUCING ORGANIC PHOSPHORUS-CONTAINING COMPOUND USING SAID PHOSPHIDE Hokko Chemical Industry Co., Ltd. (JP) 2019-05-08 EP disclosed
EP-3480207-A1 ORPHAN NUCLEAR RECEPTOR NUR77 LIGAND AND APPLICATION THEREOF Xiamen University (CN) 2019-05-08 EP disclosed
EP-3478288-A1 METHOD OF TREATING IMMUNOGLOBULIN LIGHT CHAIN AMYLOIDOSIS Prana Biotechnology Ltd (AU) 2019-05-08 EP disclosed
EP-2970205-B1 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE TOLERO PHARMACEUTICALS INC (US) 2019-05-08 EP disclosed
EP-2969007-B1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2019-05-08 EP disclosed
EP-2970122-B1 SHIP1 MODULATORS AQUINOX PHARMACEUTICALS CANADA INC (CA) 2019-05-08 EP disclosed
US-10278942-B2 Compositions for use in treating pulmonary arterial hypertension PELOTON THERAPEUTICS, INC. (US) 2019-05-07 US disclosed
US-10280172-B2 Inhibitors of KRAS G12C mutant proteins ARAXES PHARMA LLC (US) 2019-05-07 US disclosed
US-10280190-B2 Nicotinic acid riboside or nicotinamide riboside compositions, reduced derivatives thereof, and the use thereof to enhance skin permeation in treating skin conditions CHROMADEX, INC. (US) 2019-05-07 US disclosed
CN-109721620-A HPK1 inhibitors and uses thereof 南京药捷安康生物科技有限公司 2019-05-07 CN disclosed
CN-109715598-A Process for preparing carotenoid monoesters 巴斯夫欧洲公司 2019-05-03 CN disclosed
CN-109715605-A Process for preparing carotenoid monoesters 巴斯夫欧洲公司 2019-05-03 CN disclosed
CN-109715638-A The method for preparing the structural unit phosphonium salt ester as carotenoid 巴斯夫欧洲公司 2019-05-03 CN disclosed
US-20190127336-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS AND METHODS OF USE ARAXES PHARMA, LLC 2019-05-02 US disclosed
US-20190126260-A1 Catalysts for Selective Coupling of Olefins, and Methods of Making and Using Same RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2019-05-02 US disclosed
US-20190127366-A1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS, INC. 2019-05-02 US disclosed
EP-3475387-A1 PHOTOCHROMIC WATER HARVESTING PLATFORM The Warner-Babcock Institute For Green Chemistry LLC (US) 2019-05-01 EP disclosed
EP-3474835-A1 NON-CATALYTIC SUBSTRATE-SELECTIVE P38 -SPECIFIC MAPK INHIBITORS WITH ENDOTHELIAL-STABILIZING AND ANTI-INFLAMMATORY ACTIVITY, AND METHODS OF USE THEREOF University of Maryland, Baltimore (US) 2019-05-01 EP disclosed
EP-3474975-A1 REVERSIBLY SWITCHABLE SURFACTANTS AND METHODS OF USE The Warner-Babcock Institute For Green Chemistry LLC (US) 2019-05-01 EP disclosed
EP-3475324-A1 BISPHENOL A-FREE CROSSLINKED POLYMER COMPOSITIONS The Warner-Babcock Institute For Green Chemistry LLC (US) 2019-05-01 EP disclosed
EP-2427195-B1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE LLC (US) 2019-05-01 EP disclosed
US-10272083-B2 Methods of treating chronic lymphocytic leukemia and small lymphocytic leukemia using a BTK inhibitor ACERTA PHARMA B.V. (NL) 2019-04-30 US disclosed
US-10273207-B2 Covalent inhibitors of kras G12C ARAXES PHARMA LLC (US) 2019-04-30 US disclosed
US-10272079-B2 NHE3-binding compounds and methods for inhibiting phosphate transport ARDELYX, INC. (US) 2019-04-30 US disclosed
US-10273242-B2 Compound inhibiting activities of BTK and/or JAK3 kinases Beijing Hanmi Pharmaceutical Co., Ltd. (CN) 2019-04-30 US disclosed
US-10273222-B2 Histone demethylase inhibitors CELGENE QUANTSCEL RESEARCH, INC. (US) 2019-04-30 US disclosed
US-10272081-B2 SHIP1 modulators and methods related thereto AQUINOX PHARMACEUTICALS (CANADA) INC. (CA) 2019-04-30 US disclosed
US-10272074-B2 Inhibitors of glucocorticoid receptor translocation Sanford Burnham Prebys Medical Discovery Institute (US) 2019-04-30 US disclosed
CN-109689610-A The method for preparing 12 '-apocarotenal esters of the structural unit as carotenoid 巴斯夫欧洲公司 2019-04-26 CN disclosed
CN-109689045-A Purposes of the topical formulations of cannboid in treatment epidermolysis bollosa and Related connective tissue illness 因美制药公司 2019-04-26 CN disclosed
US-20190119413-A1 Catalyst Systems and Polymerization Processes for Using the Same EXXONMOBIL CHEMICAL PATENTS INC. 2019-04-25 US disclosed
US-20190119417-A1 Polyethylene Compositions and Articles Made Therefrom EXXONMOBIL CHEMICAL PATENTS INC. 2019-04-25 US disclosed
US-20190119219-A1 PKM2 MODULATORS AND METHODS FOR THEIR USE SUMITOMO PHARMA ONCOLOGY, INC. 2019-04-25 US disclosed
US-20190119221-A1 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE SUMITOMO PHARMA AMERICA, INC. 2019-04-25 US disclosed
US-20190119214-A1 ARYL ETHERS AND USES THEREOF PELOTON THERAPEUTICS, INC. 2019-04-25 US disclosed
US-20190119277-A1 VINBLASTINE 20' AMIDES: SYNTHETIC ANALOGS THAT MAINTAIN OR IMPROVE POTENCY AND SIMULTANEOUSLY OVERCOME Pgp-DERIVED EFFLUX AND RESISTANCE THE SCRIPPS RESEARCH INSTITUTE 2019-04-25 US disclosed
US-20190119212-A1 A VERSATILE LIGAND FOR PALLADIUM-CATALYZED META-C-H FUNCTIONALIZATIONS THE SCRIPPS RESEARCH INSTITUTE 2019-04-25 US disclosed
US-20190117532-A1 ORAL CARE COMPOSITIONS FOR PROMOTING GUM HEALTH PROCTER & GAMBLE (US) 2019-04-25 US disclosed
EP-3471711-A1 ANTIMALARIAL COMPOSITIONS AND USES THEREOF The Scripps Research Institute (US) 2019-04-24 EP disclosed
US-10266622-B2 Olefin polymerization catalyst system comprising mesoporous organosilica support EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2019-04-23 US disclosed
US-10266515-B2 Therapeutic inhibitory compounds LIFESCI PHARMACEUTICALS, INC. (BB) 2019-04-23 US disclosed
US-10266497-B2 Pyrazole MAGL inhibitors ABIDE THERAPEUTICS, INC. (US) 2019-04-23 US disclosed
US-10266657-B2 Polyurethane/urea compositions COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2019-04-23 US disclosed
CN-109661229-A Compound and composition for treating cancer 加利福尼亚大学董事会 2019-04-19 CN disclosed
US-20190111056-A1 COMPOUND HAVING MUTANT IDH INHIBITORY ACTIVITY, PREPARATION METHOD AND USE THEREOF SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2019-04-18 US disclosed
US-20190112312-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC (US) 2019-04-18 US disclosed
WO-2019075367-A1 PKM2 ACTIVATORS IN COMBINATION WITH REACTIVE OXYGEN SPECIES FOR TREATMENT OF CANCER TOLERO PHARMACEUTICALS, INC. (US) 2019-04-18 WO disclosed
US-20190110476-A1 NOVEL ISOTHIAZOLAMIDES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS FUNGICIDES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2019-04-18 US disclosed
EP-3469601-A1 POLYMER-SILICA HYBRID PDOTS AND METHODS OF USE THEREOF University of Washington (US) 2019-04-17 EP disclosed
EP-3468915-A1 ORGANOSILICA MATERIALS, METHODS OF MAKING, AND USES THEREOF Exxonmobil Research And Engineering Company (US) 2019-04-17 EP disclosed
EP-3468712-A1 ORGANOSILICA POLYMER CATALYSTS AND METHODS OF MAKING THE SAME Exxonmobil Research And Engineering Company (US) 2019-04-17 EP disclosed
CN-109640984-A The purposes of nicotinic acid nucleoside or nicotinamide riboside derivative and its derivative of reduction as the precursor for increasing NAD+ 可劳迈戴斯有限公司 2019-04-16 CN disclosed
US-10259803-B2 Therapeutic inhibitory compounds LIFESCI PHARMACEUTICALS, INC. (BB) 2019-04-16 US disclosed
CN-106164047-B 1,2- substituted cyclopentane as orexin receptor antagonists 武田药品工业株式会社 2019-04-16 CN disclosed
US-20190105647-A1 CATALYSTS AND METHODS OF MAKING THE SAME EXXONMOBIL RES & ENG CO (US) 2019-04-11 US disclosed
WO-2019068613-A1 NEW [1,6]NAPHTHYRIDINE COMPOUNDS AND DERIVATIVES AS CDK8/CDK19 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2019-04-11 WO disclosed
WO-2019068772-A1 NOVEL COMPOUNDS INFLAZOME LIMITED (IE) 2019-04-11 WO disclosed
US-20190105643-A1 CINCHONIUM BETAINE CATALYSTS AND METHODS OF USING SAME BRANDEIS UNIVERSITY (US) 2019-04-11 US disclosed
US-20190105299-A1 LYMPH DIRECTING PRODRUGS MONASH UNIVERSITY (AU) 2019-04-11 US disclosed
US-20190106542-A1 CHROMOPHORIC POLYMER DOTS WITH NARROW-BAND EMISSION UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION 2019-04-11 US disclosed
EP-3230410-B1 AROMATICS HYDROGENATION CATALYST, ITS PREPARATION AND USE THEREOF EXXONMOBIL RES & ENG CO (US) 2019-04-10 EP disclosed
EP-3464267-A1 NEW PHENYLPYRAZOLYLACETAMIDE COMPOUNDS AND DERIVATIVES AS CDK8/CDK19 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2019-04-10 EP disclosed
EP-3463373-A1 COMBINATION THERAPIES WITH FARNESOID X RECEPTOR (FXR) MODULATORS Akarna Therapeutics, Ltd. (GB) 2019-04-10 EP disclosed
US-10253025-B2 Method of making tetrahydronaphthyridinyl nonanoic acid compounds SCIFLUOR LIFE SCIENCES, INC. (US) 2019-04-09 US disclosed
US-10253010-B2 C-glycoside derivative SIHUAN PHARMACEUTICAL HOLDINGS GROUP LTD. (CN) 2019-04-09 US disclosed
US-10253047-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2019-04-09 US disclosed
US-10253062-B2 Amino acid and peptide conjugates and uses thereof AUCKLAND UNISERVICES LIMITED (NZ) 2019-04-09 US disclosed
CN-109575016-A PDE9 inhibitors and uses thereof 南京药捷安康生物科技有限公司 2019-04-05 CN disclosed
WO-2019067974-A1 ANTI-INFLAMMATORY, ANTI-CANCER, AND ANTI-ANGIOGENIC COMPOUNDS, PHARMACEUTICALS COMPOSITIONS, AND METHODS OF MAKING AND USING THEREOF MEDICAL PHARMACEUTICALS, INC. (US) 2019-04-04 WO disclosed
US-20190100505-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC (US) 2019-04-04 US disclosed
US-20190099747-A1 NANO-TO-NANO FE/PPM Pd CATALYSIS OF CROSS-COUPLING REACTIONS IN WATER UNIV CALIFORNIA (US) 2019-04-04 US disclosed
US-10245259-B2 Methods of treating RBP4 related diseases with triazolopyridines BELITE BIO, INC (KY) 2019-04-02 US disclosed
US-10246424-B2 Substituted quinazoline compounds and methods of use thereof ARAXES PHARMA LLC (US) 2019-04-02 US disclosed
US-10246443-B2 Cyanoquinoline derivatives TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO., LTD. (CN) 2019-04-02 US disclosed
US-10246453-B2 Benzenesulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2019-04-02 US disclosed
US-10246464-B2 Thienopyrimidine and thienopyridine compounds and methods of use thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2019-04-02 US disclosed
US-10246467-B2 Spiro[3H-indole-3,2′-pyrrolidin]-2(1H)-one compounds and derivatives as MDM2-p53 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2019-04-02 US disclosed
US-20190092767-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC 2019-03-28 US disclosed
US-20190092787-A1 SUBSTITUTED 2,3,4,5,7,9,13,13A-OCTAHYDRO-1,5-METHANOPYRIDO[1',2':4,5]PYRAZINO[1,3]DIAZEPINES AND METHODS FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. 2019-03-28 US disclosed
US-20190092771-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2019-03-28 US disclosed
WO-2019056123-A1 TOPICAL FORMULATIONS OF CANNABINOIDS AND USE THEREOF IN THE TREATMENT OF PAIN INMED PHARMACEUTICALS INC. (CA) 2019-03-28 WO disclosed
EP-3458441-A1 PROCESS FOR THE MANUFACTURE OF 6-ALKYNYL-PYRIDINE DERIVATIVES Boehringer Ingelheim International GmbH (DE) 2019-03-27 EP disclosed
EP-3458449-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2019-03-27 EP disclosed
EP-3458459-A1 MACROCYCLIC INDOLE DERIVATIVES Bayer Aktiengesellschaft (DE) 2019-03-27 EP disclosed
US-10239967-B2 Olefin polymerization catalyst system comprising mesoporous organosilica support EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2019-03-26 US disclosed
US-10238659-B2 Fatty liver disease treatment using glucocorticoid and mineralocorticoid receptor antagonists CORCEPT THERAPEUTICS, INC. (US) 2019-03-26 US disclosed
CN-106164064-B Substituted cyclopentane, tetrahydrofuran and pyrrolidines as orexin receptor antagonists 武田药品工业株式会社 2019-03-22 CN disclosed
US-20190084962-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES TAKEDA PHARMACEUTICALS CO (JP) 2019-03-21 US disclosed
US-20190086757-A1 ELECTROCHROMIC POLYMER THIN FILMS HAVING REDUCED SELF-BLEACHING BEHAVIOR AND ENHANCED CYCLING STABILITY LANNRAY ADVANCED MATERIALS CO. LTD (CN) 2019-03-21 US disclosed
EP-3454945-A1 ASH1L INHIBITORS AND METHODS OF TREATMENT THEREWITH The Regents Of The University Of Michigan (US) 2019-03-20 EP disclosed
EP-3455226-A1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME Abide Therapeutics, Inc. (US) 2019-03-20 EP disclosed
EP-2983667-B1 NHE3-BINDING COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX INC (US) 2019-03-20 EP disclosed
EP-2900239-B1 DIHYDRO-6-AZAPHENALENE DERIVATIVES FOR THE TREATMENT OF CNS, OCULAR DISEASES AND RELATED DISORDERS WARNER BABCOCK INST FOR GREEN CHEMISTRY LLC (US) 2019-03-20 EP disclosed
US-10231957-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2019-03-19 US disclosed
US-10233176-B2 Aminopyridine derivatives as TAM family kinase inhibitors SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2019-03-19 US disclosed
CN-109475661-A Preparation method based on silicon-polycarbonate glycol polyurethane solutions 奥特克国际公开有限公司 2019-03-15 CN disclosed
US-20190077785-A1 INHIBITORS FOR SOLUBLE EPOXIDE HYDROLASE (SEH) AND FATTY ACID AMIDE HYDROLASE (FAAH) THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2019-03-14 US disclosed
US-20190077752-A1 PRODRUGS OF CYTOTOXIC ACTIVE AGENTS HAVING ENZYMATICALLY CLEAVABLE GROUPS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-03-14 US disclosed
US-20190077758-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2019-03-14 US disclosed
EP-3453710-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2019-03-13 EP disclosed
EP-3452036-A1 USE OF TOPICAL FORMULATIONS OF CANNABINOIDS IN THE TREATMENT OF EPIDERMOLYSIS BULLOSA AND RELATED CONNECTIVE TISSUE DISORDERS Inmed Pharmaceuticals Inc. (CA) 2019-03-13 EP disclosed
EP-3238722-B1 SOLID FORMS OF ISOQUINOLINONES INFINITY PHARMACEUTICALS INC (US) 2019-03-13 EP disclosed
US-10227342-B2 Heteroaryl compounds for kinase inhibition ARIAD PHARMACEUTICALS, INC. (US) 2019-03-12 US disclosed
WO-2019046330-A1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME ABIDE THERAPEUTICS, INC. (US) 2019-03-07 WO disclosed
WO-2019046318-A1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME ABIDE THERAPEUTICS, INC. (US) 2019-03-07 WO disclosed
WO-2019046711-A2 COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION OPTIKIRA LLC (US) 2019-03-07 WO disclosed
WO-2019046582-A1 TESTOSTERONE ESTER TRIGLYCERIDE FORMULATIONS ANTARES PHARMA, INC. (US) 2019-03-07 WO disclosed
US-20190069537-A1 Compositions and Methods for Reducing Ice Crystal Formation X-THERMA, INC. (US) 2019-03-07 US disclosed
US-20190070212-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF INFECTIONS SPRING BANK PHARMACEUTICALS, INC. 2019-03-07 US disclosed
US-10221135-B2 1,4-substituted piperidine derivatives 89BIO LTD (IL) 2019-03-05 US disclosed
US-10222368-B2 Alzheimer's disease assay in a living patient PAIN THERAPEUTICS, INC. (US) 2019-03-05 US disclosed
US-10221177-B2 Inhibiting the transient receptor potential A1 ion channel HYDRA BIOSCIENCES, INC. (US) 2019-03-05 US disclosed
CN-109414437-A The method for treating light chain immunoglobulin amyloidosis 普拉纳生物技术有限公司 2019-03-01 CN disclosed
CN-109415623-A Photosensitive macromolecules and uses thereof 拜克门寇尔特公司 2019-03-01 CN disclosed
WO-2019040467-A1 SELECTIVE α-CYANOACRYLAMIDE AND α-CYANOACRYLATE INHIBTORS OF THE MCL-1 ONCOPROTEIN AND METHODS OF USING THE SAME UNIVERSITY OF MARYLAND, BALTIMORE (US) 2019-02-28 WO disclosed
WO-2019040511-A1 DUAL INHIBITORS OF THE BCL-2 AND HDM2 FAMILIES THROUGH CO-MIMICRY OF THE BH3 AND P53-ALPHA-HELICES UNIVERSITY OF MARYLAND BATIMORE (US) 2019-02-28 WO disclosed
WO-2019040380-A1 BENZOSULFONYL COMPOUNDS VIVACE THERAPEUTICS, INC. (US) 2019-02-28 WO disclosed
CN-109384790-A Fibroblast growth factor acceptor inhibitor and application thereof 南京药捷安康生物科技有限公司 2019-02-26 CN disclosed
US-20190055279-A1 NOVEL POLYPEPTIDES WITH IMPROVED PROTEOLYTIC STABILITY, AND METHODS OF PREPARING AND USING SAME TUFTS UNIVERSITY (US) 2019-02-21 US disclosed
US-20190055211-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC 2019-02-21 US disclosed
US-20190055221-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2019-02-21 US disclosed
US-20190055242-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2019-02-21 US disclosed
US-20190055232-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LIMITED (GB) 2019-02-21 US disclosed
WO-2019035061-A1 NOVEL STEROIDS AND METHODS OF MANUFACTURE TRUSTEES OF DARTMOUTH COLLEGE (US) 2019-02-21 WO disclosed
WO-2019036008-A1 LIPIDS FOR USE IN LIPID NANOPARTICLE FORMULATIONS Acuitas Therapeutics, Inc. (CA) 2019-02-21 WO disclosed
WO-2019036030-A1 LIPIDS FOR USE IN LIPID NANOPARTICLE FORMULATIONS Acuitas Therapeutics, Inc. (CA) 2019-02-21 WO disclosed
WO-2019034693-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2019-02-21 WO disclosed
WO-2019034688-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LIMITED (IE) 2019-02-21 WO disclosed
WO-2019034686-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LIMITED (IE) 2019-02-21 WO disclosed
WO-2019034690-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2019-02-21 WO disclosed
WO-2019034696-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LIMITED (IE) 2019-02-21 WO disclosed
WO-2019034692-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2019-02-21 WO disclosed
WO-2019034697-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LIMITED (IE) 2019-02-21 WO disclosed
EP-3143015-B1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD PHARMA INC (US) 2019-02-20 EP disclosed
EP-3071204-B1 QUINAZOLINE DERIVATIVES AS TAM FAMILY KINASE INHIBITORS SIGNALCHEM LIFESCIENCES CORP (CA) 2019-02-20 EP disclosed
EP-3180318-B1 QUINAZOLINE-2,4(1H,3H)-DIONE DERIVATIVES AS TRCP5 MODULATORS FOR THE TREATMENT OF NEUROPSYCHIATRIC DISORDERS HYDRA BIOSCIENCES INC (US) 2019-02-20 EP disclosed
EP-3443049-A2 PHOTOACTIVE MACROMOLECULES AND USES THEREOF Beckman Coulter Inc. (US) 2019-02-20 EP disclosed
EP-3442996-A2 METHODS OF TREATMENT USING CHLOROTOXIN CONJUGATES Blaze Bioscience, Inc. (US) 2019-02-20 EP disclosed
EP-3442555-A1 METHODS OF TREATING BREAST CANCER Blaze Bioscience, Inc. (US) 2019-02-20 EP disclosed
US-10208039-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2019-02-19 US disclosed
US-10207999-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2019-02-19 US disclosed
US-10207249-B2 Organosilica materials and uses thereof EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2019-02-19 US disclosed
US-10208016-B2 1-sulfonyl piperidine derivatives as modulators of prokineticin receptors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2019-02-19 US disclosed
US-10208042-B1 Multi-kinase inhibitor compound, and crystal form and use thereof NANJING TRANSTHERA BIOSCIENCES CO. LTD. (CN) 2019-02-19 US disclosed
US-10208322-B2 In vivo and in vitro olefin cyclopropanation catalyzed by heme enzymes CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2019-02-19 US disclosed
US-10207996-B2 PKM2 modulators and methods for their use TOLERO PHARMACEUTICALS, INC. (US) 2019-02-19 US disclosed
CN-108218868-B Multi-kinase inhibitor compound, its crystal form and purposes 南京药捷安康生物科技有限公司 2019-02-19 CN disclosed
US-20190046526-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2019-02-14 US disclosed
US-20190048008-A1 SPIRO-CONDENSED PYRROLIDINE DERIVATIVES AS DEUBIQUITYLATING ENZYMES (DUB) INHIBITORS MISSION THERAPEUTICS LIMITED (GB) 2019-02-14 US disclosed
US-20190048421-A1 BIOMARKERS OF RESPONSE TO HIF-2-ALPHA INHIBITION IN CANCER AND METHODS FOR THE USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2019-02-14 US disclosed
EP-3441392-A1 A PHARMACEUTICAL COMPOSITION FOR ORAL ADMINISTRATION Intellikine, LLC (US) 2019-02-13 EP disclosed
EP-3440056-A2 PD(II)-CATALYZED ENANTIOSELECTIVE BETA-METHYLENE C(SP3)-H BOND ACTIVATION The Scripps Research Institute (US) 2019-02-13 EP disclosed
US-10202402-B2 Purification of rapamycin derivatives using temperature induced phase separation BIOSENSORS INTERNATIONAL GROUP, LTD. (BM) 2019-02-12 US disclosed
US-10202381-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2019-02-12 US disclosed
US-10201614-B2 Cytotoxic and anti-mitotic compounds, and methods of using the same ZYMEWORKS INC. 2019-02-12 US disclosed
US-10202356-B2 JAK2 and ALK2 inhibitors and methods for their use TOLERO PHARMACEUTICALS, INC. (US) 2019-02-12 US disclosed
US-10202334-B2 Pendant amines and derivatives as inhibitors of leukotriene A4 hydrolase CELTAXSYS, INC. (US) 2019-02-12 US disclosed
US-10202620-B2 Synthesis of olefinic alcohols via enzymatic terminal hydroxylation PROVIVI, INC. (US) 2019-02-12 US disclosed
US-10202360-B2 Therapeutic compounds CELGENE QUANTICEL RESEARCH, INC. (US) 2019-02-12 US disclosed
US-10201545-B2 Styrenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2019-02-12 US disclosed
US-10202362-B2 Inhibitors of leukotriene A4 hydrolase CELTAXSYS, INC. (US) 2019-02-12 US disclosed
US-10202602-B2 Oligonucleotide analogues having modified intersubunit linkages and/or terminal groups SAREPTA THERAPEUTICS, INC. (US) 2019-02-12 US disclosed
CN-103958508-B Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases 艾伯维公司 2019-02-12 CN disclosed
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WO-2019027905-A1 ORGANOPHOSPHATE DERIVATIVES JANUARY THERAPEUTICS, INC. (US) 2019-02-07 WO disclosed
WO-2019028164-A1 BENZOTHIAZOLE AND RELATED COMPOUNDS SPINOGENIX, INC. (US) 2019-02-07 WO disclosed
WO-2019025440-A1 COMBINATION OF ATR KINASE INHIBITORS AND PD-1/PD-L1 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-02-07 WO disclosed
WO-2019025562-A1 DIHYDROOXADIAZINONES BAYER AKTIENGESELLSCHAFT (DE) 2019-02-07 WO disclosed
WO-2019025554-A1 6-PHENYL-4,5-DIHYDROPYRIDAZIN-3(2H)-ONE DERIVATIVES AS PDE3A AND PDE3B INHIBITORS FOR TREATING CANCER BAYER AKTIENGESELLSCHAFT (DE) 2019-02-07 WO disclosed
US-20190037848-A1 Novel isothiazolamides, processes for their preparation and their use as herbicides and/or plant growth regulators BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2019-02-07 US disclosed
EP-3436445-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2019-02-06 EP disclosed
EP-3438106-A1 ANTI-VIRAL COMPOUNDS AbbVie Ireland Unlimited Company (IE) 2019-02-06 EP disclosed
US-10196405-B2 Ataxia telengiectasia and Rad3-related (ATR) protein kinase inhibitors Atrin Pharmaceuticals LLC (US) 2019-02-05 US disclosed
CN-109313954-A Polymer-silica hybrid PDOT and methods of use thereof 华盛顿大学 2019-02-05 CN disclosed
CN-109303918-A It can be used for the cyanoacrylate and combinations thereof of cutaneous penetration 中国人民解放军军事科学院军事医学研究院 2019-02-05 CN disclosed
US-10195600-B2 Catalysts and methods of making the same EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2019-02-05 US disclosed
US-10196365-B2 Quinazoline derivative, preparation method therefor, and pharmaceutical composition and application thereof ARROMAX PHARMATECH CO., LTD. (CN) 2019-02-05 US disclosed
CN-109293652-A A kind of substituted thiazole and application thereof 四川科伦博泰生物医药股份有限公司 2019-02-01 CN disclosed
WO-2019023634-A1 CYCLATIVE RELEASE OF PEPTIDIC COMPOUNDS CIRCLE PHARMA, INC. (US) 2019-01-31 WO disclosed
EP-3434674-A1 COMPOUND HAVING MUTANT IDH INHIBITORY ACTIVITY, PREPARATION METHOD AND USE THEREOF Shanghai Haihe Pharmaceutical Co., Ltd. (CN) 2019-01-30 EP disclosed
EP-3433246-A1 1-CYANO-PYRROLIDINE DERIVATIVES AS DBU INHIBITORS Mission Therapeutics Limited (GB) 2019-01-30 EP disclosed
EP-3432934-A1 PRODRUGS OF CYTOTOXIC ACTIVE AGENTS HAVING ENZYMATICALLY CLEAVABLE GROUPS Bayer Pharma Aktiengesellschaft (DE) 2019-01-30 EP disclosed
EP-3105210-B1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS Bayer Pharma AG (DE) 2019-01-30 EP disclosed
US-10189862-B2 Phenothiazine-pyridine compounds and uses thereof THE CHINESE UNIVERSITY OF HONG KONG (CN) 2019-01-29 US disclosed
US-10189812-B2 Bi-benzyl isoquinoline derivative, preparation method and use thereof in hepatopathy treatment and prevention THE KEY LABORATORY OF CHEMISTRY FOR NATURAL PRODUC (CN) 2019-01-29 US disclosed
US-10188615-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2019-01-29 US disclosed
US-10189016-B2 Nano-to-nano Fe/ppm Pd catalysis of cross-coupling reactions in water THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-01-29 US disclosed
US-20190023704-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2019-01-24 US disclosed
US-20190022092-A1 Therapeutic Combinations of a BTK Inhibitor and a GITR Binding Molecule, a 4-1BB Agonist, or an OX40 Agonist ACERTA PHARMA BV (NL) 2019-01-24 US disclosed
US-20190022247-A1 LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS Acuitas Therapeutics, Inc. (CA) 2019-01-24 US disclosed
US-20190023709-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO AQUINOX PHARMACEUTICALS CANADA INC (CA) 2019-01-24 US disclosed
US-20190023690-A1 INHIBITORS OF CELLULAR NECROSIS AND RELATED METHODS SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY (CN) 2019-01-24 US disclosed
EP-3229952-B1 ORGANOSILICA MATERIALS EXXONMOBIL RES & ENG CO (US) 2019-01-23 EP disclosed
EP-3429994-A1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER Mission Therapeutics Limited (GB) 2019-01-23 EP disclosed
EP-3429354-A1 B-VITAMIN AND AMINO ACID CONJUGATES OF NICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, DERIVATIVES THEREOF, AND METHODS OF PREPARATION THEREOF Chromadex Inc. (US) 2019-01-23 EP disclosed
EP-3430008-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2019-01-23 EP disclosed
EP-3430012-A1 4,6 DIHYDROPYRROLO [3,4-C]PYRAZOLE-5 (1H)-CARBONITRILE DERIVATES FOR TREATING CANCER Mission Therapeutics Limited (GB) 2019-01-23 EP disclosed
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US-10183036-B2 Use of nicotinic acid riboside or nicotinamide riboside derivatives, and reduced derivatives thereof, as NAD+ increasing precursors ChromaDex Inc. (US) 2019-01-22 US disclosed
CN-104487097-B Chromophoric polymer dots with narrow-band emission 华盛顿大学商业中心 2019-01-18 CN disclosed
WO-2019014370-A1 ELECTROCHROMIC POLYMER AND SYNTHESIS AND USES THEREOF Furcifer Inc. (US) 2019-01-17 WO disclosed
US-20190016852-A1 ELECTROCHROMIC POLYMER AND SYNTHESIS AND USES THEREOF LANNRAY ADVANCED MATERIALS CO. LTD (CN) 2019-01-17 US disclosed
US-20190015402-A1 Anti-Viral Compounds ABBVIE INC. (US) 2019-01-17 US disclosed
US-20190015377-A1 Compositions for Use in Treating Pulmonary Arterial Hypertension PELOTON THERAPEUTICS, INC. (US) 2019-01-17 US disclosed
EP-3426671-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF INFECTIONS Spring Bank Pharmaceuticals, Inc. (US) 2019-01-16 EP disclosed
EP-2882428-B1 A METHOD OF INHIBITING TAU PHOSPHORYLATION PAIN THERAPEUTICS INC (US) 2019-01-16 EP disclosed
US-10179839-B2 Sulfur terminated organosilica materials and uses thereof EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2019-01-15 US disclosed
CN-109207137-A Polyacrylamide particle oil displacement agent and preparation method thereof 中国石油化工股份有限公司胜利油田分公司勘探开发研究院 2019-01-15 CN disclosed
US-10179769-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2019-01-15 US disclosed
WO-2019008029-A1 SULFONYLUREAS AND SULFONYLTHIOUREAS AS NLRP3 INHIBITORS INFLAZOME LIMITED (IE) 2019-01-10 WO disclosed
WO-2019008025-A1 NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS INFLAZOME LIMITED (IE) 2019-01-10 WO disclosed
US-20190010133-A1 Novel Syringolin Analogues and Methods of Making and Using Same BROWN UNIVERSITY 2019-01-10 US disclosed
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US-20190008859-A1 Therapeutic Combinations of a MEK Inhibitor and a BTK Inhibitor ACERTA PHARMA BV (NL) 2019-01-10 US disclosed
US-20190010122-A1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER MISSION THERAPEUTICS LIMITED (GB) 2019-01-10 US disclosed
EP-3074414-B1 WITHANOLIDES USEFUL FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES IMSTAR THERAPEUTICS INC (CA) 2019-01-09 EP disclosed
EP-3423454-A1 SPIRO-CONDENSED PYRROLIDINE DERIVATIVES AS DEUBIQUITYLATING ENZYMES (DUB) INHIBITORS Mission Therapeutics Limited (GB) 2019-01-09 EP disclosed
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US-10174026-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2019-01-08 US disclosed
US-10172858-B2 Combination pharmaceutical compositions and uses thereof INTELLIKINE LLC (US) 2019-01-08 US disclosed
US-10172350-B2 Substituted 5-hydroxy-2-phenyl-3-heteroaryl pentanenitrile derivatives, method for the production thereof and use thereof as herbicides and/or plant growth regulators BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2019-01-08 US disclosed
US-10173996-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2019-01-08 US disclosed
US-10172837-B2 Insulin sensitisers and methods of treatment NAIA Metabolic, Inc. (US) 2019-01-08 US disclosed
US-10174005-B2 Fused pyrimidines as inhibitors of p97 complex CLEAVE BIOSCIENCES, INC. (US) 2019-01-08 US disclosed
US-10174046-B2 SHIP1 modulators and methods related thereto AQUINOX PHARMACEUTICALS (CANADA) INC. (CA) 2019-01-08 US disclosed
US-10174003-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2019-01-08 US disclosed
US-20190002437-A1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS, INC. 2019-01-03 US disclosed
WO-2019006445-A1 ANTI-THROMBOTIC AGENTS AND METHODS OF USE THEREOF TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2019-01-03 WO disclosed
US-20190002429-A1 Derivatives of Xanthone Compounds SINGAPORE HEALTH SERVICES PTE LTD (SG) 2019-01-03 US disclosed
US-20190002456-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2019-01-03 US disclosed
EP-3421473-A1 METHOD FOR PREPARING PYRROLOPYRIMIDINE COMPOUND AND APPLICATION THEREOF Cinkate Pharm Tech (Shanghai) Co., Ltd. (CN) 2019-01-02 EP disclosed
US-10167283-B2 β-lactamase inhibitors and uses thereof SUANZHU PHARMA CO., LTD. (CN) 2019-01-01 US disclosed
US-10166237-B2 Compounds and methods for inducing chondrogenesis THE SCRIPPS RESEARCH INSTITUTE (US) 2019-01-01 US disclosed
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US-10167267-B2 Conversion and purification of biomass AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2019-01-01 US disclosed
US-10167273-B2 Sulfonyl piperidine derivatives and their use for treating prokineticin mediated diseases TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2019-01-01 US disclosed
US-10166216-B2 Substituted triazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2019-01-01 US disclosed
WO-2018236879-A1 MICROTUBULE POLYMERIZATION INHIBITOR PRODRUGS AND METHODS OF USING THE SAME UNIVERSITY OF MARYLAND, BALTIMORE (US) 2018-12-27 WO disclosed
WO-2018236856-A1 CAR ACTIVATOR AGENTS FOR CYCLOPHOSPHAMIDE-BASED TREATMENTS OF CANCER UNIVERSITY OF MARYLAND, BALTIMORE (US) 2018-12-27 WO disclosed
US-20180369244-A1 BTK Inhibitors to Treat Solid Tumors Through Modulation of the Tumor Microenvironment ACERTA PHARMA BV (NL) 2018-12-27 US disclosed
US-20180371430-A1 Heme Protein Catalysts for Carbon-Silicon Bond Formation In Vitro and In Vivo CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-12-27 US disclosed
US-20180370911-A1 PHOTOCATALYST-FREE, LIGHT-INDUCED CARBON-SULFUR CROSS-COUPLING METHODS U.S. DEPARTMENT OF ENERGY 2018-12-27 US disclosed
WO-2018237268-A1 NOVEL ANTIBACTERIAL COMPOUNDS AND METHODS OF MAKING AND USING SAME BROWN UNIVERSITY (US) 2018-12-27 WO disclosed
EP-3417852-A1 ARYL ETHERS AND USES THEREOF Peloton Therapeutics, Inc. (US) 2018-12-26 EP disclosed
EP-3417851-A1 ARYL ETHERS AND USES THEREOF Peloton Therapeutics, Inc. (US) 2018-12-26 EP disclosed
EP-3416960-A1 NOVEL COMPOUNDS Mission Therapeutics Limited (GB) 2018-12-26 EP disclosed
EP-3164401-B1 NEW SPIRO[3H-INDOLE-3,2´-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2018-12-26 EP disclosed
US-10160745-B2 Piperidine and azepine derivatives as prokineticin receptor modulators TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-12-25 US disclosed
US-10160756-B2 Antiviral compounds and methods using same THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-12-25 US disclosed
US-20180364253-A1 IL-17F AND IL-17A-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING REGENERON PHARMACEUTICALS, INC. 2018-12-20 US disclosed
US-20180360828-A9 SHIP1 MODULATORS AND METHODS RELATED THERETO NEOLEUKIN THERAPEUTICS, INC. 2018-12-20 US disclosed
WO-2018232160-A1 METHODS OF TREATING METABOLIC DISEASES WITH PHENOXYETHYLAMIDES BELITE BIO, INC (KY) 2018-12-20 WO disclosed
WO-2018232158-A1 METHODS OF TREATING METABOLIC DISEASES WITH FUSED BICYCLIC PYRROLES BELITE BIO, INC. (KY) 2018-12-20 WO disclosed
WO-2018229543-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2018-12-20 WO disclosed
WO-2018232150-A1 METHODS OF TREATING RBP4 RELATED DISEASES WITH TRIAZOLOPYRIDINES BELITE BIO, INC (KY) 2018-12-20 WO disclosed
WO-2018232154-A1 METHODS OF TREATING METABOLIC DISEASES WITH FUSED BICYCLIC PYRAZOLES BELITE BIO, INC (KY) 2018-12-20 WO disclosed
US-20180362460-A1 CYANOPYRROLIDINE DERIVATIVES AS INHIBITORS FOR DUBS MISSION THERAPEUTICS LIMITED (GB) 2018-12-20 US disclosed
US-20180360818-A1 METHODS OF TREATING RBP4 RELATED DISEASES WITH TRIAZOLOPYRIDINES THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2018-12-20 US disclosed
US-10155826-B2 Olefin polymerization catalyst system comprising mesoporous organosilica support EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2018-12-18 US disclosed
US-10155726-B2 Substituted pyridines and uses thereof PELOTON THERAPEUTICS, INC. (US) 2018-12-18 US disclosed
CN-109020887-A Amides compound as prevention and treatment mental disorder 绍兴从零医药科技有限公司 2018-12-18 CN disclosed
US-20180358654-A1 SODIUM-ION ELECTROLYTE COMPOSITION MONASH UNIVERSITY (AU) 2018-12-13 US disclosed
US-20180355392-A1 AMMONIUM BASED IONIC LIQUIDS USEFUL FOR LIGNOCELLULOSIC PROCESSING UNITED STATES DEPARTMENT OF ENERGY 2018-12-13 US disclosed
US-20180354989-A1 ANTIMICROBIAL PEPTIDOMIMETICS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2018-12-13 US disclosed
EP-3157916-B1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD PHARMA INC (US) 2018-12-12 EP disclosed
US-10150754-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-12-11 US disclosed
US-10150841-B2 Chromophoric polymer dots with narrow-band emission UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2018-12-11 US disclosed
US-20180346938-A1 HIGH GRAVITY, FED-BATCH IONIC LIQUID BASED PROCESS FOR DECONSTRUCTING BIOMASS UNITED STATES DEPARTMENT OF ENERGY 2018-12-06 US disclosed
US-20180346407-A1 Methods for the Treatment of Diabetic Retinopathy and other Ophthalmic Diseases ACUCELA INC. 2018-12-06 US disclosed
US-20180344738-A1 6-6 Fused Bicyclic Heteroaryl Compounds and their Use as LATS Inhibitors NOVARTIS AG (CH) 2018-12-06 US disclosed
US-20180346626-A1 A POLYMERIC COMPOSITION AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2018-12-06 US disclosed
US-20180346654-A1 POLYURETHANE/UREA MATERIALS FOLDAX, INC. 2018-12-06 US disclosed
US-20180344729-A1 TRIAZOLE DAGLAlpha INHIBITORS THE SCRIPPS RESEARCH INSTITUTE 2018-12-06 US disclosed
US-20180344763-A1 METHODS FOR ADVERSELY AFFECTING BIOFILMS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2018-12-06 US disclosed
EP-2340271-B1 POLYMER-BIOACTIVE AGENT CONJUGATES POLYACTIVA PTY LTD (AU) 2018-12-05 EP disclosed
EP-2838902-B1 ASYMMETRIC SYNTHESES FOR SPIRO-OXINDOLE COMPOUNDS USEFUL AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2018-12-05 EP disclosed
EP-3180339-B1 6-ALKYNYL-PYRIDINE DERIVATIVES AS SMAC MIMETICS BOEHRINGER INGELHEIM INT (DE) 2018-12-05 EP disclosed
EP-3408258-A1 ORGANIC REACTIONS CARRIED OUT IN AQUEOUS SOLUTION IN THE PRESENCE OF A HYDROXYALKYL(ALKYL)CELLULOSE OR AN ALKYLCELLULOSE Abbvie Deutschland GmbH & Co. KG (DE) 2018-12-05 EP disclosed
EP-3407974-A1 AMLEXANOX ANALOGS The Regents Of The University Of Michigan (US) 2018-12-05 EP disclosed
EP-3408272-A1 SURFACE PRIMER COMPOSITIONS AND METHODS OF USE Acatechol, Inc. (US) 2018-12-05 EP disclosed
EP-3408253-A1 PHOTO-CLEAVABLE PRIMER COMPOSITIONS AND METHODS OF USE Acatechol, Inc. (US) 2018-12-05 EP disclosed
EP-3409669-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD Pharmaceuticals, Inc. (US) 2018-12-05 EP disclosed
US-10144739-B2 Spiro[3H-indole-3,2′-pyrrolidin]-2(1H)-one compounds and derivatives as MDM2-P53 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-12-04 US disclosed
US-10144711-B2 Aryl ethers and uses thereof PELOTON THERAPEUTICS, INC. (US) 2018-12-04 US disclosed
US-10144724-B2 Substituted quinazoline compounds and methods of use thereof ARAXES PHARMA LLC (US) 2018-12-04 US disclosed
US-10143638-B2 Method of treating skin with ingenol mebutate LEO LABORATORIES LIMITED (IE) 2018-12-04 US disclosed
WO-2018215818-A1 NOVEL COMPOUNDS AND USES THE UNIVERSITY OF QUEENSLAND (AU) 2018-11-29 WO disclosed
WO-2018218071-A1 COMPOUNDS AND METHODS OF USE THEREOF FOR TREATMENT OF CANCER ARAXES PHARMA LLC (US) 2018-11-29 WO disclosed
WO-2018218069-A1 QUINAZOLINE DERIVATIVES AS MODULATORS OF MUTANT KRAS, HRAS OR NRAS ARAXES PHARMA LLC (US) 2018-11-29 WO disclosed
WO-2018218070-A2 COVALENT INHIBITORS OF KRAS ARAXES PHARMA LLC (US) 2018-11-29 WO disclosed
WO-2018217809-A1 PYRAZOLE MAGL INHIBITORS ABIDE THERAPEUTICS, INC. (US) 2018-11-29 WO disclosed
WO-2018218154-A1 PENICILLIN-BINDING PROTEIN INHIBITORS VenatoRx Pharmaceuticals, Inc. (US) 2018-11-29 WO disclosed
WO-2018217567-A1 COMPOSITIONS AND METHODS OF MAKING EXPANDED HEMATOPOIETIC STEM CELLS USING PTEN INHIBITORS TRANSFUSION HEALTH, LLC (US) 2018-11-29 WO disclosed
WO-2018217805-A1 PYRAZOLE MAGL INHIBITORS ABIDE THERAPEUTICS, INC. (US) 2018-11-29 WO disclosed
WO-2018218190-A1 PENICILLIN-BINDING PROTEIN INHIBITORS VenatoRx Pharmaceuticals, Inc. (US) 2018-11-29 WO disclosed
US-20180339970-A1 PYRAZOLE MAGL INHIBITORS H. LUNDBECK A/S (DK) 2018-11-29 US disclosed
EP-3406606-A1 NITROGENOUS HETEROCYCLIC AMIDE DERIVATIVE, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL APPLICATION Sichuan Haisco Pharmaceutical Co., Ltd. (CN) 2018-11-28 EP disclosed
EP-3129380-B1 SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE DERIVATIVES AND THEIR USE AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2018-11-28 EP disclosed
US-10138251-B2 Spiro[3H-indole-3,2′-pyrrolidin]-2(1H)-one compounds and derivatives as MDM2-P53 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-11-27 US disclosed
US-10138226-B2 Benzimidazol-2-amines as MIDH1 inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-11-27 US disclosed
US-10137110-B2 1-cyclohexyl-2-phenylaminobenzimidazoles as mIDH1 inhibitors for the treatment of tumors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-11-27 US disclosed
CN-108884068-A 1- cyano-pyrolidin derivative as DUB inhibitor 特殊治疗有限公司 2018-11-23 CN disclosed
CN-107501279-B Furanoquinoline dione compound and medical application thereof 东莞市真兴贝特医药技术有限公司 2018-11-23 CN disclosed
WO-2018213236-A1 BIO-BASED, MULTI-AROMATIC COMPOUNDS, AND METHODS OF MAKING AND USING SAME ROWAN UNIVERSITY (US) 2018-11-22 WO disclosed
WO-2018213632-A1 KINASE INHIBITORS AND USES THEREOF DENALI THERAPEUTICS INC. (US) 2018-11-22 WO disclosed
US-20180334496-A1 COMPLEMENT FACTOR D ANTAGONIST ANTIBODIES AND CONJUGATES THEREOF KODIAK SCIENCES INC. 2018-11-22 US disclosed
EP-3402795-A1 5-SUBSTITUTED 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES Bayer Pharma Aktiengesellschaft (DE) 2018-11-21 EP disclosed
EP-3402503-A1 THERAPEUTIC COMBINATIONS OF AN ANTIFOLATE AND A BTK INHIBITOR Acerta Pharma B.V. (NL) 2018-11-21 EP disclosed
US-10130633-B2 Compounds BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-11-20 US disclosed
US-10131664-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2018-11-20 US disclosed
US-20180327519-A1 AMPHIPHILIC RAFT AGENT COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANIZATION (AU) 2018-11-15 US disclosed
US-20180327414-A1 METHODS AND COMPOSITIONS FOR INHIBITING THE INTERACTION OF MENIN WITH MLL PROTEINS WELLSPRING BIOSCIENCES LLC 2018-11-15 US disclosed
US-20180327391-A1 COMPOUND, COMPOSITIONS, AND METHODS DENALI THERAPEUTICS INC. 2018-11-15 US disclosed
US-20180327793-A1 METHODS AND ENZYME CATALYSTS FOR THE SYNTHESIS OF NON-CANONICAL AMINO ACIDS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-11-15 US disclosed
US-20180325887-A1 N-[2-(1-BENZYLPIPERIDIN-4-YL)ETHYL]-4-(PYRAZIN-2-YL)-PIPERAZINE-1-CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS MUSCARINIC RECEPTOR 4 (M4) ANTAGONISTS FOR TREATING NEUROLOGICAL DISEASES NEUROCRINE BIOSCIENCES, INC. 2018-11-15 US disclosed
US-20180325900-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 QUANTIEL PHARMACEUTICALS, INC. 2018-11-15 US disclosed
US-20180327416-A1 PYRAZOLE COMPOUNDS AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2018-11-15 US disclosed
US-20180325833-A1 NANOPARTICLES BASED ON OPTIONALLY ALKOXYLATED POLY(ALKYL CYANOACRYLATES) HAVING A DEFINED DEGREE OF POLYMERIZATION AbbVie Deutschland GmbH & Co. KG (DE) 2018-11-15 US disclosed
US-20180327407-A1 COMPOUNDS AND METHODS FOR TREATING SYNOVIAL SARCOMAS HOWARD HUGHES MEDICAL INSTITUTE 2018-11-15 US disclosed
WO-2018208985-A2 ANTIBACTERIAL COMPOUNDS FORGE THERAPEUTICS, INC. (US) 2018-11-15 WO disclosed
US-20180327410-A1 PYRAZOLE COMPOUNDS AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2018-11-15 US disclosed
WO-2018208987-A2 ANTIBACTERIAL COMPOUNDS FORGE THERAPEUTICS, INC. (US) 2018-11-15 WO disclosed
WO-2018206547-A1 COMBINATION OF BUB1 AND ATR INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-11-15 WO disclosed
EP-3401314-A1 COVALENT INHIBITORS OF KRAS G12C Araxes Pharma LLC (US) 2018-11-14 EP disclosed
EP-2363419-B1 Polymer product formed using raft agent UNIV SYDNEY (AU) 2018-11-14 EP disclosed
US-10124007-B2 Combination of PI3K-inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-11-13 US disclosed
CN-108779138-A Design and synthesis of nucleotides based on novel disulfide linkers for use as reversible terminators for DNA sequencing by synthesis 哥伦比亚大学董事会 2018-11-09 CN disclosed
CN-108778270-A A kind of bactericidal composition and application thereof 山东轩竹医药科技有限公司 2018-11-09 CN disclosed
WO-2018204691-A1 METHODS AND ENZYME CATALYSTS FOR THE SYNTHESIS OF NON-CANONICAL AMINO ACIDS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-11-08 WO disclosed
WO-2018204532-A1 NON-FUSED TRICYCLIC COMPOUNDS VIVACE THERAPEUTICS, INC. (US) 2018-11-08 WO disclosed
US-20180318438-A1 ANTIBODY DRUG CONJUGATES OF KINESIN SPINDEL PROTEIN (KSP) INHIBITORS WITH ANTI-TWEAKR-ANTIBODIES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-11-08 US disclosed
US-20180319793-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-11-08 US disclosed
WO-2018204370-A1 CX3CR1 SMALL MOLECULE ANTAGONISTS, AND METHODS USING SAME DREXEL UNIVERSITY (US) 2018-11-08 WO disclosed
US-20180319775-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC 2018-11-08 US disclosed
US-20180318437-A1 ANTIBODY DRUG CONJUGATES OF KINESIN SPINDEL PROTEIN (KSP) INHIBITORS WITH ANTI-CD123-ANTIBODIES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-11-08 US disclosed
US-20180318304-A1 Methods of Using BTK Inhibitors to Treat Dermatoses ACERTA PHARMA BV (NL) 2018-11-08 US disclosed
US-20180318790-A1 AROMATIC HYDROGENATION CATALYSTS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2018-11-08 US disclosed
US-20180319769-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-11-08 US disclosed
EP-3399038-A2 OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA Sarepta Therapeutics, Inc. (US) 2018-11-07 EP disclosed
EP-3030252-B1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX INC (US) 2018-11-07 EP disclosed
EP-3397613-A1 LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS Acuitas Therapeutics Inc. (CA) 2018-11-07 EP disclosed
EP-3397276-A1 ANTIBODIES AND CONJUGATES THEREOF Kodiak Sciences Inc. (US) 2018-11-07 EP disclosed
EP-3397617-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2018-11-07 EP disclosed
CN-108727361-A Indole amine 2,3-dioxygenase inhibitor and application 南京药捷安康生物科技有限公司 2018-11-02 CN disclosed
US-20180311210-A1 METHOD FOR INHIBITING GROWTH OF CANCER CELLS PAIN THERAPEUTICS 2018-11-01 US disclosed
WO-2018200571-A1 SUBSTITUTED 2,3-DIHYDRO-1H-INDENE ANALOGS AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2018-11-01 WO disclosed
WO-2018200812-A1 ANTIBODY CONJUGATES COMPRISING STING AGONIST NOVARTIS AG (CH) 2018-11-01 WO disclosed
WO-2018200943-A1 NOVEL CARBONYL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS Acuitas Therapeutics, Inc. (CA) 2018-11-01 WO disclosed
WO-2018200517-A1 METHODS OF MANUFACTURING OF NIRAPARIB TESARO, INC. (US) 2018-11-01 WO disclosed
WO-2018198077-A2 6-6 FUSED BICYCLIC HETEROARYL COMPOUNDS AND THEIR USE AS LATS INHIBITORS NOVARTIS AG (CH) 2018-11-01 WO disclosed
EP-3394079-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR Oric Pharmaceuticals, Inc. (US) 2018-10-31 EP disclosed
EP-3394049-A1 CYANOPYRROLIDINE DERIVATIVES AS INHIBITORS FOR DUBS Mission Therapeutics Limited (GB) 2018-10-31 EP disclosed
EP-2836487-B1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS INC (US) 2018-10-31 EP disclosed
EP-3395818-A1 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES Bayer Pharma Aktiengesellschaft (DE) 2018-10-31 EP disclosed
EP-2467141-B1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE LLC (US) 2018-10-31 EP disclosed
EP-3394078-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR Oric Pharmaceuticals, Inc. (US) 2018-10-31 EP disclosed
US-10111883-B1 Selective P2X3 modulators BELLUS HEALTH COUGH INC. (CA) 2018-10-30 US disclosed
US-10111874-B2 Combination therapies for treatment of cancer ARAXES PHARMA LLC (US) 2018-10-30 US disclosed
US-10112940-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-10-30 US disclosed
US-20180305348-A1 INHIBITORS OF BRUTONS TYROSINE KINASE PHARMACYCLICS LLC 2018-10-25 US disclosed
US-20180305721-A1 Biocatalytic Synthesis of Strained Carbocycles CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-10-25 US disclosed
US-20180305305-A1 2-BETA-NAPHTHYL-ACETIC ACID ANALOGS AS AKR1C3 INHIBITORS AND METHODS OF USING SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2018-10-25 US disclosed
US-20180305368-A1 ARTIFICIAL METALLOENZYMES CONTAINING NOBLE METAL-PORPHYRINS U.S. DEPARTMENT OF ENERGY 2018-10-25 US disclosed
WO-2018191789-A1 THERAPEUTIC COMPOUNDS AND METHODS UNIVERSITY OF TASMANIA (AU) 2018-10-25 WO disclosed
WO-2018193428-A1 MODIFIED OLIGOMERIC COMPOUNDS COMPRISING TRICYCLO-DNA NUCLEOSIDES AND USES THEREOF SYNTHENA AG (CH) 2018-10-25 WO disclosed
WO-2018195121-A1 VMAT2 INHIBITOR COMPOUNDS AND COMPOSITIONS THEREOF NEUROCRINE BIOSCIENCES, INC. (US) 2018-10-25 WO disclosed
WO-2018195155-A1 THERAPEUTIC COMPOUNDS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-10-25 WO disclosed
US-20180305336-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-10-25 US disclosed
US-20180303925-A1 Nucleoside-Modified RNA For Inducing an Adaptive Immune Response Acuitas Therapeutics, Inc. (CA) 2018-10-25 US disclosed
EP-3390391-A1 NOVEL COMPOUNDS Mission Therapeutics Limited (GB) 2018-10-24 EP disclosed
EP-2920175-B1 TRIAZOLOPYRIDAZINE DERIVATIVES AS BROMODOMAIN INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2018-10-24 EP disclosed
EP-2828395-B1 BORONIC ACID CONJUGATES OF OLIGONUCLEOTIDE ANALOGUES SAREPTA THERAPEUTICS INC (US) 2018-10-24 EP disclosed
CN-106488919-B 3-substituted 2-aminoindole derivatives 武田药品工业株式会社 2018-10-23 CN disclosed
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CN-108699035-A Noval chemical compound 特殊治疗有限公司 2018-10-23 CN disclosed
WO-2018191657-A1 LIPIDS FOR DELIVERY OF ACTIVE AGENTS Acuitas Therapeutics, Inc. (CA) 2018-10-18 WO disclosed
WO-2018191270-A1 CATALYSTS FOR OLEFIN ISOMERIZATION BRANDEIS UNIVERSITY (US) 2018-10-18 WO disclosed
WO-2018191719-A1 LIPID DELIVERY OF THERAPEUTIC AGENTS TO ADIPOSE TISSUE Acuitas Therapeutics, Inc. (CA) 2018-10-18 WO disclosed
US-20180297984-A1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS, INC. 2018-10-18 US disclosed
US-20180297999-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-10-18 US disclosed
US-20180296543-A1 THERAPEUTIC COMPOUNDS CELGENE QUANTICEL RESEARCH, INC. 2018-10-18 US disclosed
US-20180298383-A1 Peptide Oligonucleotide Conjugates JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2018-10-18 US disclosed
WO-2018191548-A2 COMPLEMENT FACTOR D ANTAGONIST ANTIBODIES AND CONJUGATES THEREOF KODIAK SCIENCES INC. (US) 2018-10-18 WO disclosed
WO-2018191283-A1 GLUCOCORTICOID RECEPTOR MODULATORS ORIC PHARMACEUTICALS, INC. (US) 2018-10-18 WO disclosed
EP-3386504-A2 THERAPEUTIC INHIBITORY COMPOUNDS Lifesci Pharmaceuticals, Inc. (BB) 2018-10-17 EP disclosed
US-10100311-B2 Fibrotic treatment MONASH UNIVERSITY (AU) 2018-10-16 US disclosed
US-10100046-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2018-10-16 US disclosed
US-10098878-B2 HIF-2α inhibitors for treating iron overload disorders THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2018-10-16 US disclosed
US-10100018-B2 Amide derivatives as lysophosphatidic acid receptor antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-10-16 US disclosed
US-10100056-B2 SHIP1 modulators and methods related thereto AQUINOX PHARMACEUTICALS (CANADA) INC. (CA) 2018-10-16 US disclosed
US-10100305-B2 Methods and compositions for manipulating translation of protein isoforms from alternative initiation of start sites SAREPTA THERAPEUTICS, INC. (US) 2018-10-16 US disclosed
US-20180290967-A1 Novel Antibacterial Compounds and Methods of Making and Using Same BRYANT UNIVERSITY 2018-10-11 US disclosed
US-20180291030-A1 NEW SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2018-10-11 US disclosed
US-20180291039-A1 BETA-LACTAMASE INHIBITORS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2018-10-11 US disclosed
EP-3383859-A1 1-CYANO-PYRROLIDINE DERIVATIVES AS INHIBITORS OF USP30. Mission Therapeutics Limited (GB) 2018-10-10 EP disclosed
EP-3180345-B1 THIENO- AND FURO[2,3-D]PYRIMIDINE-2,4[1H,3H]-DIONE DERIVATIVES AS TRPC5 MODULATORS FOR THE TREATMENT OF NEUROPSYCHIATRIC DISORDERS HYDRA BIOSCIENCES INC (US) 2018-10-10 EP disclosed
EP-3384549-A1 SODIUM-ION ELECTROLYTE COMPOSITION Deakin University (AU) 2018-10-10 EP disclosed
EP-3180337-B1 PYRIDO[3,4-D]PYRIMIDINE-2,4(1H,3H)-DIONE DERIVATIVES HYDRA BIOSCIENCES INC (US) 2018-10-10 EP disclosed
EP-3180340-B1 PYRIDO[2,3-D]PYRIMIDINE-2,4(1H,3H)-DIONE DERIVATIVES HYDRA BIOSCIENCES INC (US) 2018-10-10 EP disclosed
US-10093630-B2 Pyrazole compounds and methods of making and using same ABIDE THERAPEUTICS, INC. (US) 2018-10-09 US disclosed
US-10093624-B2 NAMPT and ROCK inhibitors ABBVIE INC. (US) 2018-10-09 US disclosed
US-10093906-B2 Cytochrome C protein variants for catalyzing carbon-silicon bond formation CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-10-09 US disclosed
US-10093635-B2 MAGL inhibitors ABIDE THERAPEUTICS, INC. (US) 2018-10-09 US disclosed
WO-2018183936-A1 COMPOUNDS AND METHODS USEFUL FOR TREATING OR PREVENTING CANCERS THE BROAD INSTITUTE, INC. (US) 2018-10-04 WO disclosed
WO-2018183635-A1 CD73 INHIBITORS AND USES THEREOF PELOTON THERAPEUTICS, INC. (US) 2018-10-04 WO disclosed
WO-2018183795-A1 METHOD OF MAKING TETRAHYDRONAPHTHYRIDINYL NONANOIC ACID COMPOUNDS SCIFLUOR LIFE SCIENCES, INC. (US) 2018-10-04 WO disclosed
WO-2018183654-A1 AGENTS FOR DIFFERENTIATING STEM CELLS AND TREATING CANCER MINERVA BIOTECHNOLOGIES CORPORATION (US) 2018-10-04 WO disclosed
WO-2018183328-A1 CROSS-COUPLING REACTION CATALYSTS, AND METHODS OF MAKING AND USING SAME YALE UNIVERSITY (US) 2018-10-04 WO disclosed
US-20180280367-A1 USE OF ANTHELMINTIC AGENTS AGAINST DIROFILARIA IMMITIS INTERVET INC. (US) 2018-10-04 US disclosed
US-20180282374-A1 ANTIMICROBIAL POLYMYXIN DERIVATIVE COMPOUNDS MONASH UNIVERSITY (AU) 2018-10-04 US disclosed
US-20180282947-A1 COATING FOR RECYCLABLE PAPER JL DARLING, LLC 2018-10-04 US disclosed
US-20180282327-A1 METHOD OF MAKING TETRAHYDRONAPHTHYRIDINYL NONANOIC ACID COMPOUNDS FELIQS CORPORATION (JP) 2018-10-04 US disclosed
US-20180282309-A1 1,2-SUBSTITUTED CYCLOPENTANES AS OREXIN RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-10-04 US disclosed
US-20180282288-A1 LP-PLA2 INHIBITORS H. LUNDBECK A/S (DK) 2018-10-04 US disclosed
US-20180282818-A1 Therapeutic Cancer Treatments Based on TP53 Gene Mutations WISTAR INST (US) 2018-10-04 US disclosed
US-20180282307-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC 2018-10-04 US disclosed
US-20180282308-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC 2018-10-04 US disclosed
EP-3380536-A1 A POLYMERIC COMPOSITION Agency For Science, Technology And Research (SG) 2018-10-03 EP disclosed
US-10087320-B2 Conductive polymer-matrix compositions and uses thereof POLYDROP, LLC (US) 2018-10-02 US disclosed
US-10085452-B2 Synergistic benzoxaborole-containing anti-fungicidal composition THE PENN STATE RESEARCH FOUNDATION (US) 2018-10-02 US disclosed
CN-108601832-A The medical usage of anti-C-met antibodies-cytotoxic drug conjugate 苏州盛迪亚生物医药有限公司 2018-09-28 CN disclosed
WO-2018172250-A1 2-METHYL-QUINAZOLINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-09-27 WO disclosed
WO-2018172852-A1 SUBSTITUTED DIHYDROINDENE-4-CARBOXAMIDES AND ANALOGS THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA CORPORATION (CA) 2018-09-27 WO disclosed
WO-2018175628-A1 BIOCATALYTIC SYNTHESIS OF STRAINED CARBOCYCLES CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-09-27 WO disclosed
US-20180273541-A1 NEW SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-09-27 US disclosed
US-20180271893-A1 METHODS FOR TREATING PROGEROID LAMINOPATHIES USING OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA SAREPTA THERAPEUTICS, INC. 2018-09-27 US disclosed
US-20180273580-A1 NOVEL 7-DEHYDROCHOLESTEROL DERIVATIVES AND METHODS USING SAME UNIVERSITY OF ROCHESTER 2018-09-27 US disclosed
US-20180273515-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC 2018-09-27 US disclosed
US-20180273535-A1 PROCESSES FOR PREPARING ISOQUINOLINONES AND SOLID FORMS OF ISOQUINOLINONES HCR COLLATERAL MANAGEMENT, LLC 2018-09-27 US disclosed
US-20180271843-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-09-27 US disclosed
US-20180273505-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2018-09-27 US disclosed
US-20180273547-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RES INC (US) 2018-09-27 US disclosed
US-20180273533-A1 [9,10-DIMETHOXY-3-(2-METHYLPROPYL)-1H,2H,3H,4H,6H,7H,11BH-PYRIDO-[2,1-A]ISOQUINOLIN-2-YL]METHANOL AND COMPOUNDS, COMPOSITIONS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES, INC. 2018-09-27 US disclosed
US-20180273523-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC 2018-09-27 US disclosed
US-20180273917-A1 HEME PROTEIN CATALYSTS FOR CARBON-BORON BOND FORMATION IN VITRO AND IN VIVO CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-09-27 US disclosed
EP-3377499-A1 COMPOUNDS AND METHODS FOR TREATING SYNOVIAL SARCOMAS Kadoch, Cigall (US) 2018-09-26 EP disclosed
EP-3377060-A1 PYRAZOLE COMPOUNDS AND METHODS OF MAKING AND USING SAME Abide Therapeutics, Inc. (US) 2018-09-26 EP disclosed
EP-3377487-A1 COMPOUNDS FOR MEDICINAL APPLICATIONS Australian Biomedical Co. Pty Ltd (AU) 2018-09-26 EP disclosed
EP-3377481-A1 2-SUBSTITUTED QUINAZOLINE COMPOUNDS COMPRISING A SUBSTITUTED HETEROCYCLIC GROUP AND METHODS OF USE THEREOF Araxes Pharma LLC (US) 2018-09-26 EP disclosed
EP-2686296-B1 SUBSTITUTED 4-CYAN-3-(2,6-DIFLUOROPHENYL)-4-PHENYLBUTANOATES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2018-09-26 EP disclosed
US-20180263964-A1 METHOD OF SCREENING FOR AGENTS FOR DIFFERENTIATING STEM CELLS MINERVA BIOTECHNOLOGIES CORPORATION (US) 2018-09-20 US disclosed
US-20180264128-A1 COMPOUNDS FOR MEDICINAL APPLICATIONS Australian Biomedical Co. Pty Ltd. (AU) 2018-09-20 US disclosed
US-20180265491-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2018-09-20 US disclosed
WO-2018169880-A1 DUAL MAGL AND FAAH INHIBITORS ABIDE THERAPEUTICS, INC. (US) 2018-09-20 WO disclosed
US-20180263970-A1 COMPOUNDS AND METHODS USEFUL FOR TREATING OR PREVENTING HEMATOLOGICAL CANCERS THE BROAD INSTITUTE, INC. (US) 2018-09-20 US disclosed
WO-2018167019-A1 TOSYLACETATE BASED COMPOUNDS AND DERIVATIVES THEREOF AS PHGDH INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-09-20 WO disclosed
EP-3375781-A1 BENZO RING DERIVATIVE WITH B2 RECEPTOR AGONIST AND M3 RECEPTOR ANTAGONIST ACTIVITIES AND USE THEREOF IN MEDICINE Sichuan Haisco Pharmaceutical Co., Ltd. (CN) 2018-09-19 EP disclosed
CN-105263855-B The system and method analyzed using polymer point 华盛顿大学商业中心 2018-09-18 CN disclosed
US-10076536-B2 Oligonucleotide analogues targeting human LMNA SAREPTA THERAPEUTICS, INC. (US) 2018-09-18 US disclosed
US-10077271-B2 Methods and compositions for inhibiting the interaction of menin with MLL proteins KURA ONCOLOGY, INC. (US) 2018-09-18 US disclosed
WO-2018165325-A1 HEME PROTEIN CATALYSTS FOR CARBON-BORON BOND FORMATION IN VITRO AND IN VIVO CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-09-13 WO disclosed
US-20180258111-A1 Acene-based transmitter molecules for photon upconversion THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2018-09-13 US disclosed
US-20180256591-A1 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-09-13 US disclosed
US-20180258103-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE, INC. 2018-09-13 US disclosed
US-20180258127-A1 B-VITAMIN AND AMINO ACID CONJUGATES OF NICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, DERIVATIVES THEREOF, AND METHODS OF PREPARATION THEREOF ChromaDex Inc. (US) 2018-09-13 US disclosed
US-20180256566-A1 DUAL MAGL AND FAAH INHIBITORS LUNDBECK LA JOLLA RESEARCH CENTER, INC. 2018-09-13 US disclosed
EP-3150609-B1 PROCESS FOR PREPARING CERTAIN CHEMICAL ENTITIES INTELLIKINE LLC (US) 2018-09-12 EP disclosed
EP-3370523-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR COLORING EDIBLE MATERIALS The Penn State Research Foundation (US) 2018-09-12 EP disclosed
EP-3371164-A1 N-[2-(1 -BENZYLPIPERIDIN-4-YL)ETHYL]-4-(PYRAZIN-2-YL)-PIPERAZINE-1 -CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS MUSCARINIC RECEPTOR 4 (M4) ANTAGONISTS FOR TREATING NEUROLOGICAL DISEASES NEUROCRINE BIOSCIENCES, INC. (US) 2018-09-12 EP disclosed
EP-3370518-A2 COMPOSITIONS AND METHODS FOR REDUCING ICE CRYSTAL FORMATION X-Therma, Inc. (US) 2018-09-12 EP disclosed
US-10071101-B2 Use of cinnabarinic acid as a modulator of immune response in autoimmune disorders THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-09-11 US disclosed
US-10071984-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-09-11 US disclosed
CN-108513537-A Method for screening agent for differentiating stem cells 米纳瓦生物技术公司 2018-09-07 CN disclosed
US-20180250298-A1 Therapeutic Combinations of a BTK Inhibitor, a PI3K Inhibitor, a JAK-2 Inhibitor, and/or a BCL-2 Inhibitor ACERTA PHARMA BV (NL) 2018-09-06 US disclosed
US-20180251445-A1 1-SULFONYL PIPERIDINE DERIVATIVES AS MODULATORS OF PROKINETICIN RECEPTORS TAKEDA PHARMACEUTICALS CO (JP) 2018-09-06 US disclosed
US-20180250313-A1 COMPOUNDS AND FORMULATIONS FOR TREATING OPHTHALMIC DISEASES VIEWPOINT THERAPEUTICS, INC. 2018-09-06 US disclosed
US-20180251458-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-09-06 US disclosed
US-20180250400-A1 Therapeutic Combinations of a BTK Inhibitor, a PI3K Inhibitor, a JAK-2 Inhibitor, and/or a CDK4/6 Inhibitor ACERTA PHARMA BV (NL) 2018-09-06 US disclosed
EP-3367999-A1 FRAGRANCE COMPOSITIONS COMPRISING IONIC LIQUIDS The Procter and Gamble Company (US) 2018-09-05 EP disclosed
EP-3368507-A1 NOVEL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS Acuitas Therapeutics, Inc. (CA) 2018-09-05 EP disclosed
EP-3368582-A1 POLYURETHANE/UREA MATERIALS Commonwealth Scientific and Industrial Research Organisation (AU) 2018-09-05 EP disclosed
EP-3368556-A2 NOVEL POLYPEPTIDES WITH IMPROVED PROTEOLYTIC STABILITY, AND METHODS OF PREPARING AND USING SAME Tufts University (US) 2018-09-05 EP disclosed
US-10065926-B2 Use of substituted dihydrooxindolylsulfonamides, or the salts thereof, for increasing the stress tolerance of plants BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-09-04 US disclosed
CN-108473632-A Polymeric compositions 新加坡科技研究局 2018-08-31 CN disclosed
CN-108473483-A Compound for medical applications 澳大利亚生物医学公司 2018-08-31 CN disclosed
US-20180244839-A1 MULTICOLORED ELECTROCHROMIC POLYMER COMPOSITIONS AND METHODS OF MAKING AND USING THE SAME LANNRAY ADVANCED MATERIALS CO. LTD (CN) 2018-08-30 US disclosed
US-20180243314-A1 NO-DONORS FOR THE TREATMENT OF CEREBROVASCULAR VASOSPASMS AFTER BRAIN HEMORRHAGE WESTFAELISCHE WILHELMS-UNIVERSITAET MUENSTER (DE) 2018-08-30 US disclosed
US-20180243303-A1 METHODS AND COMPOSITIONS FOR INHIBITING THE INTERACTION OF MENIN WITH MLL PROTEINS WELLSPRING BIOSCIENCES LLC 2018-08-30 US disclosed
US-20180244762-A1 DUAL PDGF/VEGF ANTAGONISTS KODIAK SCIENCES INC. (US) 2018-08-30 US disclosed
US-20180243425-A1 LYMPH DIRECTING PRODRUGS MONASH UNIVERSITY (AU) 2018-08-30 US disclosed
US-20180245011-A1 A BASE OIL ADDITIVE AGENCY FOR SCIENCE, TECHOLOGY AND RESEARCH (SG) 2018-08-30 US disclosed
US-20180246102-A1 METHOD FOR SCREENING INHIBITORS OF RAS ARAXES PHARMA LLC 2018-08-30 US disclosed
US-20180243239-A1 2,4,6-TRIALKOXYSTRYL ARYL SULFONES, SULFONAMIDES AND CARBOXAMIDES, AND METHODS OF PREPARATION AND USE TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2018-08-30 US disclosed
US-20180244674-A1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-08-30 US disclosed
WO-2018153972-A1 COMBINATION OF ATR KINASE INHIBITORS AND ANTIANDROGENS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-08-30 WO disclosed
WO-2018153973-A1 COMBINATION OF ATR KINASE INHIBITORS WITH PARP INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-08-30 WO disclosed
WO-2018153971-A1 COMBINATION OF ATR KINASE INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-08-30 WO disclosed
WO-2018153969-A1 COMBINATION OF ATR KINASE INHIBITORS WITH RADIUM-223 SALT BAYER AKTIENGESELLSCHAFT (DE) 2018-08-30 WO disclosed
EP-3364977-A2 METHOD FOR SCREENING INHIBITORS OF RAS Araxes Pharma LLC (US) 2018-08-29 EP disclosed
EP-2768830-B1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2018-08-29 EP disclosed
US-10059687-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-08-28 US disclosed
US-10059796-B2 Conjugated polymers COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2018-08-28 US disclosed
US-10059713-B2 3-substituted 2-amino-indole derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-08-28 US disclosed
CN-105745196-B The conversion and purifying of biomass 新加坡科技研究局 2018-08-28 CN disclosed
US-20180237626-A1 CONDUCTIVE POLYMER-MATRIX COMPOSITIONS AND USES THEREOF POLYDROP, LLC 2018-08-23 US disclosed
US-20180237641-A1 PHENYLETHYNYLNAPHTHALENE DYES AND METHODS FOR THEIR USE SONY CORPORATION (JP) 2018-08-23 US disclosed
US-20180237396-A1 Processes For Preparing AG-10, Its Intermediates, and Salts Thereof CALCILYTIX THERAPEUTICS INC. 2018-08-23 US disclosed
US-20180237444-A1 INHIBITORS OF ERK AND METHODS OF USE KURA ONCOLOGY, INC. 2018-08-23 US disclosed
WO-2018151837-A1 CONDUCTIVE POLYMER-MATRIX COMPOSITIONS AND USES THEREOF POLYDROP, LLC (US) 2018-08-23 WO disclosed
US-20180240565-A1 CONDUCTIVE POLYMER-MATRIX COMPOSITIONS AND USES THEREOF POLYDROP LLC (US) 2018-08-23 US disclosed
EP-1773768-B1 PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS EXELIXIS INC (US) 2018-08-22 EP disclosed
EP-3363800-A1 HETEROCYCLIC INHIBITORS OF ERK AND METHODS OF USE Kura Oncology, Inc. (US) 2018-08-22 EP disclosed
EP-2953940-B1 PIPERIDIN-1-YL AND AZEPIN-1-YL CARBOXYLATES AS MUSCARINIC M4 RECEPTOR AGONISTS HEPTARES THERAPEUTICS LTD (GB) 2018-08-22 EP disclosed
US-10053430-B2 RAF kinase modulator compounds and methods of use thereof AMBIT BIOSCIENCES CORP. (US) 2018-08-21 US disclosed
US-10053490-B2 Antimicrobial peptidomimetics AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2018-08-21 US disclosed
US-20180221406-A1 THERAPEUTIC COMBINATIONS OF ANTIVIRAL AND ANTI-INFLAMMATORY THERAPIES FORESIGHT BIOTHERAPEUTICS, INC. (US) 2018-08-09 US disclosed
US-20180221363-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2018-08-09 US disclosed
US-20180223278-A1 Functionally-Modified Oligonucleotides And Subunits Thereof JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2018-08-09 US disclosed
US-20180223287-A1 FIBROTIC TREATMENT MONASH UNIVERSITY (AU) 2018-08-09 US disclosed
EP-3356354-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS Araxes Pharma LLC (US) 2018-08-08 EP disclosed
EP-3356339-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS Araxes Pharma LLC (US) 2018-08-08 EP disclosed
EP-3356347-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS Araxes Pharma LLC (US) 2018-08-08 EP disclosed
EP-3356353-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS Araxes Pharma LLC (US) 2018-08-08 EP disclosed
EP-3356387-A1 ANTIMICROBIAL POLYMYXIN DERIVATIVE COMPOUNDS Monash University (AU) 2018-08-08 EP disclosed
EP-3356349-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS Araxes Pharma LLC (US) 2018-08-08 EP disclosed
EP-3356359-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS Araxes Pharma LLC (US) 2018-08-08 EP disclosed
EP-3356351-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS Araxes Pharma LLC (US) 2018-08-08 EP disclosed
US-10040767-B2 Benzimidazole derivatives and uses thereof PELOTON THERAPEUTICS, INC. (US) 2018-08-07 US disclosed
US-10039754-B2 Anti-viral compounds ABBVIE INC. (US) 2018-08-07 US disclosed
US-10040779-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-08-07 US disclosed
CN-108368089-A Novel Compounds 特殊治疗有限公司 2018-08-03 CN disclosed
US-20180215769-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2018-08-02 US disclosed
WO-2018140599-A1 BENZOTHIOPHENE AND BENZOTHIAZOLE COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC (US) 2018-08-02 WO disclosed
WO-2018140600-A1 FUSED HETERO-HETERO BICYCLIC COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC (US) 2018-08-02 WO disclosed
WO-2018140598-A1 FUSED N-HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC (US) 2018-08-02 WO disclosed
WO-2018140514-A1 1-(6-(3-HYDROXYNAPHTHALEN-1-YL)QUINAZOLIN-2-YL)AZETIDIN-1-YL)PROP-2-EN-1-ONE DERIVATIVES AND SIMILAR COMPOUNDS AS KRAS G12C INHIBITORS FOR THE TREATMENT OF CANCER ARAXES PHARMA LLC (US) 2018-08-02 WO disclosed
WO-2018140512-A1 FUSED BICYCLIC BENZOHETEROAROMATIC COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC (US) 2018-08-02 WO disclosed
WO-2018140513-A1 1-(3-(6-(3-HYDROXYNAPHTHALEN-1-YL)BENZOFURAN-2-YL)AZETIDIN-1YL)PROP-2-EN-1-ONE DERIVATIVES AND SIMILAR COMPOUNDS AS KRAS G12C MODULATORS FOR TREATING CANCER ARAXES PHARMA LLC (US) 2018-08-02 WO disclosed
EP-2367799-B1 2-AMINO-5-TRIFLUOROMETHYL-PYRIMIDINE DERIVATIVES AND THEIR USE AS PTK2 KINASE INHIBITORS IPHARMA H K LTD (HK) 2018-08-01 EP disclosed
EP-3352566-A2 METHOD OF SCREENING FOR AGENTS FOR DIFFERENTIATING STEM CELLS Minerva Biotechnologies Corporation (US) 2018-08-01 EP disclosed
EP-2970303-B3 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES INC (US) 2018-08-01 EP disclosed
US-10035809-B2 Substituted 2,3,4,5,7,9,13,13a-octahydro-1,5-methanopyrido[1′,2′:4,5]pyrazino[1,2-a][1,3]diazepines and methods for treating viral infections GILEAD SCIENCES, INC. (US) 2018-07-31 US disclosed
US-10036754-B2 Water soluble fluorescent or colored dyes and methods for their use SONY CORPORATION (JP) 2018-07-31 US disclosed
CN-108350034-A Antimicrobial polymyxin derived compounds 莫纳什大学 2018-07-31 CN disclosed
US-20180207140-A1 Pyrazolopyrimidines as Inhibitors of Glucocorticoid Receptor Translocation Sanford Burnham Prebys Medical Discovery Institute 2018-07-26 US disclosed
US-20180206495-A1 SUBSTITUTED ARYL AND HETEROARYL CARBOXYLIC ACID HYDRAZIDES OR SALTS THEREOF AND USE THEREOF TO INCREASE STRESS TOLERANCE IN PLANTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-07-26 US disclosed
US-20180208554-A1 Small Molecule Inhibitors of the MCL-1 Oncoprotein and Uses Thereof UNIVERSITY OF MARYLAND, BALTIMORE 2018-07-26 US disclosed
US-20180206491-A1 SUBSTITUTED CYCLIC ARYL AND HETEROARYL CARBOXYLIC ACID HYDRAZIDES OR SALTS THEREOF AND USE THEREOF TO INCREASE STRESS TOLERANCE IN PLANTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-07-26 US disclosed
US-20180206498-A1 SUBSTITUTED HETEROARYL CARBOXYLIC ACID HYDRAZIDES OR SALTS THEREOF AND USE THEREOF TO INCREASE STRESS TOLERANCE IN PLANTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-07-26 US disclosed
US-20180207154-A1 Therapeutic Combinations of a BTK Inhibitor, a PI3K Inhibitor and/or a JAK-2 Inhibitor ACERTA PHARMA BV (NL) 2018-07-26 US disclosed
WO-2018136650-A1 COMPOSITIONS AND METHODS FOR TREATING ANDROGEN-INDEPENDENT CANCER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-07-26 WO disclosed
WO-2018136546-A1 SUBSTITUTED 3-DIALKYLAMINOMETHYL-PIPERIDIN-4-YL-BENZAMIDES AND METHODS OF MAKING AND USING SAME MEBIAS DISCOVERY LLC (US) 2018-07-26 WO disclosed
WO-2018134335-A1 SUBSTITUTED IMIDAZOPYRIDINPYRIMIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-07-26 WO disclosed
WO-2018136014-A1 A FORMULATION, A METHOD OF FORMING THE SAME AND ITS USES THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2018-07-26 WO disclosed
WO-2018134148-A1 SUBSTITUTED DIHYDROIMIDAZOPYRIDINEDIONES AS MKNK1 AND MKNK2 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-07-26 WO disclosed
WO-2018134786-A1 COMPOSITIONS AND METHODS FOR THE ASSESSMENT OF DRUG TARGET OCCUPANCY FOR BRUTON'S TYROSINE KINASE ACERTA PHARMA B.V. (NL) 2018-07-26 WO disclosed
EP-3349747-A1 NO-DONORS FOR THE TREATMENT OF CEREBROVASCULAR VASOSPASMS AFTER BRAIN HEMORRHAGE Ehlert, Angelika (DE) 2018-07-25 EP disclosed
EP-3156387-B1 METHOD OF PREPARING INDENE DERIVATIVES AQUINOX PHARMACEUTICALS CANADA INC (CA) 2018-07-25 EP disclosed
EP-3351248-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS Ardelyx, Inc. (US) 2018-07-25 EP disclosed
US-10029207-B2 Composite gas separation membrane THE UNIVERSITY OF MELBOURNE (AU) 2018-07-24 US disclosed
US-10030017-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-07-24 US disclosed
US-10028937-B2 Anti-viral compounds ABBVIE INC. (US) 2018-07-24 US disclosed
US-10030020-B2 Spirocycle compounds and methods of making and using same ABIDE THERAPEUTICS, INC. (US) 2018-07-24 US disclosed
US-10030012-B2 Piperidin-1-yl and azepin-1-yl carboxylates as muscarinic M4 receptor agonists HEPTARES THERAPEUTICS LIMITED (GB) 2018-07-24 US disclosed
US-20180199575-A1 SUBSTITUTED OXOTETRAHYDROQUINOLINYLPHOSPHINIC ACID AND PHOSPHINIC ACID AMIDES OR SALTS THEREOF AND USE THEREOF TO INCREASE STRESS TOLERANCE IN PLANTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-07-19 US disclosed
US-20180201584-A1 ARYL SULFONAMIDE COMPOUNDS AS CARBONIC ANHYDRASE INHIBITORS AND THEIR THERAPEUTIC USE SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2018-07-19 US disclosed
EP-1463765-B1 AQUEOUS DISPERSIONS OF POLYMER PARTICLES UNIV SYDNEY (AU) 2018-07-18 EP disclosed
EP-3347368-A1 COMPOUNDS AND FORMULATIONS FOR TREATING OPHTHALMIC DISEASES Viewpoint Therapeutics, Inc. (US) 2018-07-18 EP disclosed
EP-3347340-A1 LYMPH DIRECTING PRODRUGS Monash University (AU) 2018-07-18 EP disclosed
EP-3004239-B1 SCRATCH RESISTANT POLYMERS TENASITECH PTY LTD (AU) 2018-07-18 EP disclosed
US-10022701-B2 Coating methods using organosilica materials and uses thereof EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2018-07-17 US disclosed
US-10023543-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2018-07-17 US disclosed
US-10023592-B2 Bromodomain inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-07-17 US disclosed
US-10021877-B2 Substituted 5-hydroxy-2,3-diphenylpentanonitrile derivatives, processes for their preparation and their use as herbicides and/or plant growth regulators BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-07-17 US disclosed
US-10022700-B2 Organosilica materials and uses thereof EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2018-07-17 US disclosed
US-10023557-B2 Therapeutic inhibitory compounds LIFESCI PHARMACEUTICALS, INC. (BB) 2018-07-17 US disclosed
CN-108290861-A 1- cyano-pyrolidin derivatives as USP30 inhibitor 特殊治疗有限公司 2018-07-17 CN disclosed
CN-108290893-A Dihydroperidinone derivatives, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2018-07-17 CN disclosed
CN-108290872-A Cyanopyrolidine derivatives as DUBs inhibitor 特殊治疗有限公司 2018-07-17 CN disclosed
WO-2018129552-A1 COMPOUNDS USEFUL FOR TREATING GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC. (US) 2018-07-12 WO disclosed
WO-2018129556-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC. (US) 2018-07-12 WO disclosed
WO-2018129533-A1 SELECTIVE HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF HUMAN DISEASE SHUTTLE PHARMACEUTICALS, LLC (US) 2018-07-12 WO disclosed
US-20180193337-A1 Methods of Blocking the CXCR-4/SDF-1 Signaling Pathway With Inhibitors of Bruton's Tyrosine Kinase ACERTA PHARMA BV (NL) 2018-07-12 US disclosed
WO-2018129557-A1 INHIBITORS OF NHE-MEDIATED ANTIPORT ARDELYX, INC. (US) 2018-07-12 WO disclosed
US-20180194748-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC 2018-07-12 US disclosed
US-20180193315-A1 SPIROCYCLIC HAT INHIBITORS AND METHODS FOR THEIR USE ABBVIE INC (US) 2018-07-12 US disclosed
US-20180194762-A1 PYRAZOLO[3,4-b]PYRIDINE AND PYRROLO[2,3-b]PYRIDINE INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC (US) 2018-07-12 US disclosed
US-20180194724-A1 CYANOPYRROLIDINES AS DUB INHIBITORS FOR THE TREATMENT OF CANCER MISSION THERAPEUTICS LIMITED (GB) 2018-07-12 US disclosed
EP-3169662-B1 SUBSTITUTED VINYL- AND ALKINYL-CYANOCYCLOALKANOLS AND VINYL- AND ALKINYL-CYANOHETEROCYCLOALKANOLS AS AGENTS TO COMBAT ABIOTIC PLANT STRESS BAYER CROPSCIENCE AG (DE) 2018-07-11 EP disclosed
EP-2964645-B1 PROCESS FOR IXABEPILONE, AND INTERMEDIATES THEREOF SCINOPHARM TAIWAN LTD (TW) 2018-07-11 EP disclosed
EP-2872899-B1 ALZHEIMER'S DISEASE ASSAY IN A LIVING PATIENT PAIN THERAPEUTICS INC (US) 2018-07-11 EP disclosed
US-10016401-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-07-10 US disclosed
US-10017736-B2 Method of inhibiting tau phosphorylation PAIN THERAPEUTICS, INC. (US) 2018-07-10 US disclosed
US-10017763-B2 dsRNA molecules comprising oligonucleotide analogs having modified intersubunit linkages and/or terminal groups SAREPTA THERAPEUTICS, INC. (US) 2018-07-10 US disclosed
WO-2018125901-A1 MODIFICATION OF SURFACE PROPERTIES OF MICROFLUIDIC DEVICES BIO-RAD LABORATORIES, INC. (US) 2018-07-05 WO disclosed
US-20180185516-A1 DELIVERY OF TARGET SPECIFIC NUCLEASES Acuitas Therapeutics, Inc. (CA) 2018-07-05 US disclosed
US-20180185510-A1 ANTIBODY DRUG CONJUGATES OF KINESIN SPINDEL PROTEIN (KSP) INHIBITORS WITH ANTI-B7H3-ANTIBODIES Bayer Pharma AG (DE) 2018-07-05 US disclosed
EP-3341421-A1 AMPHIPHILIC RAFT AGENT Commonwealth Scientific and Industrial Research Organisation (AU) 2018-07-04 EP disclosed
US-10011588-B2 1,2-substituted cyclopentanes as orexin receptor antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-07-03 US disclosed
US-10010538-B2 Use of anthelmintic agents against Dirofilaria immitis INTERVET INC. (US) 2018-07-03 US disclosed
US-10010554-B2 Fused pyrimidines as inhibitors of P97 complex CLEAVE BIOSCIENCES, INC. (US) 2018-07-03 US disclosed
US-10011600-B2 Methods and compositions for inhibition of Ras ARAXES PHARMA LLC (US) 2018-07-03 US disclosed
US-10011583-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2018-07-03 US disclosed
CN-108218868-A Multi-kinase inhibitor compound, its crystal form and purposes 南京药捷安康生物科技有限公司 2018-06-29 CN disclosed
CN-104955454-B Chemokine receptor anagonists 凯莫森特里克斯股份有限公司 2018-06-29 CN disclosed
US-20180179310-A1 Spray-Dried Olefin Polymerization Catalyst Compositions and Polymerization Processes for Using the Same EXXONMOBIL CHEMICAL PATENTS INC. 2018-06-28 US disclosed
US-20180179324-A1 SYNTHESIS OF POLYCARBONATE SILOXANE DIOLS AORTECH INTERNATIONAL PLC (GB) 2018-06-28 US disclosed
US-20180177746-A1 ALKOXY COMPOUNDS FOR DISEASE TREATMENT ACUCELA INC. 2018-06-28 US disclosed
US-20180179159-A1 1,4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON LLC 2018-06-28 US disclosed
US-20180179204-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2018-06-28 US disclosed
US-20180178213-A1 MODIFICATION OF SURFACE PROPERTIES OF MICROFLUIDIC DEVICES BIO-RAD LABORATORIES, INC. 2018-06-28 US disclosed
US-20180177754-A1 COMPOSITIONS FOR USE IN TREATING PULMONARY ARTERIAL HYPERTENSION PELOTON THERAPEUTICS, INC. 2018-06-28 US disclosed
US-20180177780-A1 PYRIDAZINONE COMPOUNDS AND THEIR USE AS DAAO INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-06-28 US disclosed
WO-2018118259-A1 SPRAY-DRIED OLEFIN POLYMERIZATION CATALYST COMPOSITIONS AND POLYMERIZATION PROCESSES FOR USING THE SAME EXXONMOBIL CHEMICAL PATENTS INC. (US) 2018-06-28 WO disclosed
WO-2018117974-A1 A CURABLE COATING COMPOSITION AND METHOD OF PREPARING A COATING FILM AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2018-06-28 WO disclosed
WO-2018114662-A1 SUBSTITUTED 1,2,4-THIADIAZOLYL PYRROLONES AND 1,2,4-THIADIAZOLYL HYDANTOINES AND SALTS THEREOF AND USE THEREOF AS HERBICIDES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-06-28 WO disclosed
WO-2018115380-A1 NOVEL BENZYLAMINO SUBSTITUTED QUINAZOLINES AND DERIVATIVES AS SOS1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-06-28 WO disclosed
WO-2018114798-A1 PRODRUGS OF CYTOTOXIC ACTIVE AGENTS HAVING ENZYMATICALLY CLEAVABLE GROUPS BAYER AKTIENGESELLSCHAFT (DE) 2018-06-28 WO disclosed
WO-2018112555-A1 AQUEOUS POLYMER COMPOSITION COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2018-06-28 WO disclosed
EP-2993165-B1 COMPOUNDS WITH (SUBSTITUTED PHENYL)-PROPENAL MOIETY, THEIR DERIVATIVES, BIOLOGICAL ACTIVITY, AND USE THEREOF ALLIANZ PHARMASCIENCE LTD (TW) 2018-06-27 EP disclosed
EP-2693878-B1 SUBSTITUTED (3R,4R)-4-CYAN-3,4-DIPHENYLBUTANOATES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER IP GMBH (DE) 2018-06-27 EP disclosed
US-20180170891-A1 4H-Pyran Compounds as Insulin-Regulated Aminopeptidase (IRAP) Inhibitors MONASH UNIVERSITY (AU) 2018-06-21 US disclosed
US-20180169256-A1 ANTIBODY DRUG CONJUGATES (ADCS) AND ANTIBODY PRODRUG CONJUGATES (APDCS) WITH ENZYMATICALLY CLEAVABLE GROUPS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-06-21 US disclosed
US-20180170906-A1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS, INC. 2018-06-21 US disclosed
WO-2018108704-A1 NEW 6-AMINO-QUINOLINONE COMPOUNDS AND DERIVATIVES AS BCL6 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-06-21 WO disclosed
WO-2018107226-A1 METHODS OF TREATING OCULAR DISORDERS Beta Therapeutics Pty. Ltd. (AU) 2018-06-21 WO disclosed
US-10000520-B2 B-vitamin and amino acid conjugates ofnicotinoyl ribosides and reduced nicotinoyl ribosides, derivatives thereof, and methods of preparation thereof ChromaDex Inc. (US) 2018-06-19 US disclosed
US-9999217-B2 Compositions for stabilizing DNA, RNA, and proteins in blood and other biological samples during shipping and storage at ambient temperatures BIOMATRICA, INC. (US) 2018-06-19 US disclosed
US-20180162868-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2018-06-14 US disclosed
US-20180162804-A1 PENDANT AMINES AND DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELLTAXIS, LLC 2018-06-14 US disclosed
US-20180162854-A1 Inhibitors of Leukotriene A4 Hydrolase CELLTAXIS, LLC 2018-06-14 US disclosed
US-20180162807-A1 AROMATIC COMPOUNDS AND USES THEREOF PELOTON THERAPEUTICS, INC. 2018-06-14 US disclosed
US-20180163052-A1 WATER SOLUBLE FLUORESCENT OR COLORED DYES AND METHODS FOR THEIR USE Sony Group Corporation (JP) 2018-06-14 US disclosed
US-20180162857-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-06-14 US disclosed
US-20180161324-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO AQUINOX PHARMACEUTICALS CANADA INC (CA) 2018-06-14 US disclosed
US-20180162852-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LIMITED 2018-06-14 US disclosed
US-20180162812-A1 COVALENT INHIBITORS OF KRAS G12C ARAXES PHARMA LLC 2018-06-14 US disclosed
US-20180162877-A1 PYRAZOLOPYRIDINAMINES AS MKNK1 AND MKNK2 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-06-14 US disclosed
US-20180161359-A1 METHODS AND COMPOUNDS FOR TREATMENT OF LYMPHOCYTE-RELATED DISEASES AND CONDITIONS JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2018-06-14 US disclosed
US-20180162836-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELLTAXIS, LLC 2018-06-14 US disclosed
US-20180162802-A1 MONAMINE AND MONOAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELLTAXIS, LLC 2018-06-14 US disclosed
WO-2018107167-A1 PENDANT AMINES AND DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS, INC. (US) 2018-06-14 WO disclosed
WO-2018107153-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS, INC. (US) 2018-06-14 WO disclosed
WO-2018107026-A1 DELIVERY OF TARGET SPECIFIC NUCLEASES SANGAMO THERAPEUTICS, INC. (US) 2018-06-14 WO disclosed
WO-2018107158-A1 MONAMINE AND MONOAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS, INC. (US) 2018-06-14 WO disclosed
WO-2018106284-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2018-06-14 WO disclosed
EP-3332645-A1 USE OF SUBSTITUTED PYRIMIDINE DIONES OR THEIR SALTS AS AGENTS TO COMBAT ABIOTIC PLANT STRESS Bayer Cropscience AG (DE) 2018-06-13 EP disclosed
EP-3203841-B1 SUBSTITUTED 5-HYDROXY-2-PHENYL-3-HETEROARYLPENTANONITRILE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND/OR PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2018-06-13 EP disclosed
EP-2001911-B1 POLYMER PRODUCT AND INTERFACIAL POLYMERISATION PROCESS USING RAFT AGENT UNIV SYDNEY (AU) 2018-06-13 EP disclosed
EP-3331894-A1 NICOTINAMIDE MONONUCLEOTIDE DERIVATIVES AND THEIR USES Metro International Biotech, LLC (US) 2018-06-13 EP disclosed
US-9994537-B2 Piperazine carbamates and methods of making and using same ABIDE THERAPEUTICS, INC. (US) 2018-06-12 US disclosed
US-9994561-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-06-12 US disclosed
US-9993484-B2 2-(morpholin-4-yl)-1,7-naphthyridines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-06-12 US disclosed
US-9994562-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-06-12 US disclosed
US-9994534-B2 Pain-relieving compositions and uses therefor THE UNIVERSITY OF QUEENSLAND (AU) 2018-06-12 US disclosed
US-9994518-B2 Alpha-7 nicotinic acetylcholine receptor modulators and uses thereof MERCK SHARP & DOHME CORP. (US) 2018-06-12 US disclosed
CN-108137482-A Lymphatic prodrugs 莫纳什大学 2018-06-08 CN disclosed
US-20180155279-A1 ARYL ETHERS AND USES THEREOF PELOTON THERAPEUTICS, INC. 2018-06-07 US disclosed
US-20180155359-A9 SHIP1 MODULATORS AND METHODS RELATED THERETO TARO PHARMACEUTICALS INC. (CA) 2018-06-07 US disclosed
US-20180155295-A1 CXCR4 CHEMOKINE RECEPTOR MODULATORS NORTHWESTERN UNIVERSITY 2018-06-07 US disclosed
US-20180153888-A1 COMBINATION THERAPY WITH AXL INHIBITOR AND IMMUNE CHECKPOINT MODULATOR OR ONCOLYTIC VIRUS BERGENBIO ASA (NO) 2018-06-07 US disclosed
US-20180153887-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES INC (US) 2018-06-07 US disclosed
US-20180155348-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC 2018-06-07 US disclosed
EP-3328384-A1 FIBROTIC TREATMENT Monash University (AU) 2018-06-06 EP disclosed
US-9988357-B2 Methods for preparation of quinazoline derivatives ARAXES PHARMA LLC (US) 2018-06-05 US disclosed
US-9988382-B2 [9,10-dimethoxy-3-(2-methylpropyl)-1H,2H,3H,4H,6H,7H,11bH-pyrido-[2,1-A]isoquinolin-2-yl]methanol and compounds, compositions and methods relating thereto NEUROCRINE BIOSCIENCES, INC. (US) 2018-06-05 US disclosed
US-9986733-B2 Compositions and methods for reducing ice crystal formation X-THERMA, INC. (US) 2018-06-05 US disclosed
CN-105308041-B Preparation method for ixabepilone and intermediate thereof 台湾神隆股份有限公司 2018-06-01 CN disclosed
US-20180147227-A1 NICOTINAMIDE MONONUCLEOTIDE DERIVATIVES AND THEIR USES METROBIOTECH, LLC 2018-05-31 US disclosed
US-20180148745-A1 HEMOPROTEIN CATALYSTS FOR IMPROVED ENANTIOSELECTIVE ENZYMATIC SYNTHESIS OF TICAGRELOR CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-05-31 US disclosed
US-20180148448-A1 ß-LACTAMASE INHIBITORS AND USES THEREOF Xuanzhu Pharma Co., Ltd. (CN) 2018-05-31 US disclosed
US-20180148413-A1 SUBSTITUTED PYRIDINES AND USES THEREOF PELOTON THERAPEUTICS, INC. 2018-05-31 US disclosed
EP-3325467-A1 SUBSTITUTED HETEROARYL CARBOXYLIC ACID HYDRAZIDES OR SALTS THEREOF AND USE THEREOF TO INCREASE STRESS TOLERANCE IN PLANTS Bayer CropScience Aktiengesellschaft (DE) 2018-05-30 EP disclosed
EP-3325466-A1 SUBSTITUTED CYCLIC ARYL AND HETEROARYL CARBOXYLIC ACID HYDRAZIDES OR SALTS THEREOF AND USE THEREOF TO INCREASE STRESS TOLERANCE IN PLANTS Bayer CropScience Aktiengesellschaft (DE) 2018-05-30 EP disclosed
EP-3325446-A1 SUBSTITUTED ARYL AND HETEROARYL CARBOXYLIC ACID HYDRAZIDES OR SALTS THEREOF AND USE THEREOF TO INCREASE STRESS TOLERANCE IN PLANTS Bayer CropScience Aktiengesellschaft (DE) 2018-05-30 EP disclosed
EP-3325447-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS AND THEIR USE AS INHIBITORS OF G12C MUTANT KRAS, HRAS AND/OR NRAS PROTEINS Araxes Pharma LLC (US) 2018-05-30 EP disclosed
US-9981989-B2 Ataxia telengiectasia and Rad3-related (ATR) protein kinase inhibitors Atrin Pharmaceuticals LLC (US) 2018-05-29 US disclosed
US-9981972-B2 N-hydroxy bicyclic hydantoin carbamates as tools for identification of serine hydrolase targets ABIDE THERAPEUTICS, INC. (US) 2018-05-29 US disclosed
US-9982010-B2 7-dehydrocholesterol derivatives and methods using same WOMEN & INFANTS HOSPITAL OF RHODE ISLAND (US) 2018-05-29 US disclosed
US-9981930-B1 MAGL inhibitors ABIDE THERAPEUTICS, INC. (US) 2018-05-29 US disclosed
US-20180140595-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2018-05-24 US disclosed
US-20180141898-A1 PESTICIDALLY ACTIVE OXIME AND HYDRAZONE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2018-05-24 US disclosed
US-20180141912-A1 VERSATILE RAFT AGENT COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2018-05-24 US disclosed
US-20180141953-A1 Novel Breathing Control Modulating Compounds, and Methods of Making and Using Same NEURAD LTD. (IL) 2018-05-24 US disclosed
US-20180141927-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC 2018-05-24 US disclosed
WO-2018094275-A1 ALVOCIDIB PRODRUGS AND THEIR USE AS PROTEIN KINASE INHIBITORS TOLERO PHARMACEUTICALS, INC. (US) 2018-05-24 WO disclosed
WO-2018093946-A1 MAGL INHIBITORS ABIDE THERAPEUTICS, INC. (US) 2018-05-24 WO disclosed
WO-2018093947-A1 MAGL INHIBITORS ABIDE THERAPEUTICS, INC. (US) 2018-05-24 WO disclosed
WO-2018093949-A1 MAGL INHIBITORS ABIDE THERAPEUTICS, INC. (US) 2018-05-24 WO disclosed
WO-2018093924-A1 CARBON MONOXIDE-RELEASING MOLECULES AND THERAPEUTIC APPLICATIONS THEREOF GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC. (US) 2018-05-24 WO disclosed
US-20180142066-A1 SULFUR TERMINATED ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2018-05-24 US disclosed
US-20180140569-A1 COMBINATION THERAPY OF A HIF-2-ALPHA INHIBITOR AND AN IMMUNOTHERAPEUTIC AGENT AND USES THEREOF PELOTON THERAPEUTICS, INC. (US) 2018-05-24 US disclosed
EP-3322702-A1 CYANOPYRROLIDINES AS DUB INHIBITORS FOR THE TREATMENT OF CANCER Mission Therapeutics Limited (GB) 2018-05-23 EP disclosed
EP-3322296-A1 SUBSTITUTED OXO-TETRAHYDROQUINOLINYL-PHOSPHINIC ACID AND PHOSPHINIC ACID AMIDES OR SALTS THEREOF AND USE THEREOF TO INCREASE STRESS TOLERANCE IN PLANTS Bayer CropScience Aktiengesellschaft (DE) 2018-05-23 EP disclosed
US-9975989-B2 Multicolored electrochromic polymer compositions and methods of making and using the same Furcifer Inc. (US) 2018-05-22 US disclosed
US-9975915-B1 Crystalline forms of nicotinoyl ribosides, modified derivatives thereof, and phosphorylated analogs thereof, and methods of preparation thereof THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2018-05-22 US disclosed
US-20180134742-A1 CRYSTALLINE FORMS OF NICOTINOYL RIBOSIDES, MODIFIED DERIVATIVES THEREOF, AND PHOSPHORYLATED ANALOGS THEREOF, AND METHODS OF PREPARATION THEREOF THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2018-05-17 US disclosed
US-20180134674-A1 MAGL INHIBITORS H. LUNDBECK A/S (DK) 2018-05-17 US disclosed
WO-2018089830-A1 EFFICIENT AND SCALABLE SYNTHESES OF NICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, MODIFIED DERIVATIVES THEREOF, PHOSPHORYLATED ANALOGS THEREOF, ADENYLYL DINUCLEOTIDE CONJUGATES THEREOF, AND NOVEL CRYSTALLINE FORMS THEREOF THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2018-05-17 WO disclosed
US-20180134675-A1 MAGL INHIBITORS H. LUNDBECK A/S (DK) 2018-05-17 US disclosed
US-20180134743-A1 EFFICIENT AND SCALABLE SYNTHESES OF NICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, MODIFIED DERIVATIVES THEREOF, PHOSPHORYLATED ANALOGS THEREOF, ADENYLYL DINUCLEOTIDE CONJUGATES THEREOF, AND NOVEL CRYSTALLINE FORMS THEREOF THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2018-05-17 US disclosed
US-20180134710-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-05-17 US disclosed
EP-2410987-B1 METHODS OF TREATMENT USING COMBINATION THERAPY AMBIT BIOSCIENCES CORP (US) 2018-05-16 EP disclosed
EP-3319938-A1 SMALL MOLECULE INHIBITORS OF THE MCL-1 ONCOPROTEIN AND USES THEREOF University of Maryland, Baltimore (US) 2018-05-16 EP disclosed
US-9969844-B2 Silicone ligands for quantum dots NANOSYS, INC. (US) 2018-05-15 US disclosed
US-9969736-B2 Substituted xanthines and methods of use thereof HYDRA BIOSCIENCES, INC. (US) 2018-05-15 US disclosed
US-9968684-B2 Polymer-NSAID conjugate POLYACTIVA PTY LTD (AU) 2018-05-15 US disclosed
US-9969689-B2 Aryl ethers and uses thereof PELOTON THERAPEUTICS, INC. (US) 2018-05-15 US disclosed
CN-108026142-A Ligands for orphan nuclear receptor Nur77 and uses thereof 厦门大学 2018-05-11 CN disclosed
CN-108026141-A Ligand of orphan nuclear receptor Nur77 and application thereof 厦门大学 2018-05-11 CN disclosed
US-20180127424-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELLTAXIS, LLC 2018-05-10 US disclosed
US-20180127408-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2018-05-10 US disclosed
US-20180125844-A1 TREATMENT OF RELAPSED AND/OR REFRACTORY SOLID TUMORS AND NON-HODGKIN'S LYMPHOMAS CELGENE CORPORATION (US) 2018-05-10 US disclosed
US-20180127464-A1 NOVEL EPHA4 INHIBITORS TARGETING ITS LIGAND BINDING DOMAIN SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE 2018-05-10 US disclosed
US-20180127396-A1 INHIBITORS OF RAS AND METHODS OF USE THEREOF ARAXES PHARMA LLC 2018-05-10 US disclosed
EP-3317255-A1 ARYL SULFONAMIDE COMPOUNDS AS CARBONIC ANHYDRASE INHIBITORS AND THEIR THERAPEUTIC USE SignalChem Lifesciences Corporation (CA) 2018-05-09 EP disclosed
EP-3317241-A2 THERAPEUTIC INHIBITORY COMPOUNDS Lifesci Pharmaceuticals, Inc. (BB) 2018-05-09 EP disclosed
EP-3317259-A2 THERAPEUTIC INHIBITORY COMPOUNDS Lifesci Pharmaceuticals, Inc. (BB) 2018-05-09 EP disclosed
EP-3316890-A1 NOVEL BREATHING CONTROL MODULATING COMPOUNDS, AND METHODS OF MAKING AND USING SAME Neurad Ltd. (IL) 2018-05-09 EP disclosed
EP-3316884-A1 THERAPEUTIC INHIBITORY COMPOUDS Lifesci Pharmaceuticals, Inc. (BB) 2018-05-09 EP disclosed
EP-2968282-B1 HISTONE DEMENTHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2018-05-09 EP disclosed
US-9963492-B2 High molecular weight, post-translationally modified protein brushes MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2018-05-08 US disclosed
US-9963441-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-05-08 US disclosed
CN-105189484-B Cxcr7 antagonists 凯莫森特里克斯股份有限公司 2018-05-04 CN disclosed
US-20180118757-A1 SUBSTITUTED QUINAZOLINES AS INHIBITORS OF KRAS G12C ARAXES PHARMA LLC 2018-05-03 US disclosed
WO-2018081638-A1 NUCLEOSIDE-MODIFIED RNA FOR INDUCING AN ADAPTIVE IMMUNE RESPONSE THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-05-03 WO disclosed
WO-2018081672-A1 BIARYL LIGANDS FOR TRANSITION METAL-CATALYZED REACTIONS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-05-03 WO disclosed
US-20180118720-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-05-03 US disclosed
WO-2018081480-A1 LIPID NANOPARTICLE FORMULATIONS Acuitas Therapeutics, Inc. (CA) 2018-05-03 WO disclosed
US-20180117163-A9 VAR2CSA-DRUG CONJUGATES ZYMEWORKS INC. (CA) 2018-05-03 US disclosed
US-20180117075-A1 THERAPY FOR MALIGNANT DISEASE WOMEN & INFANTS HOSPITAL OF RHODE ISLAND 2018-05-03 US disclosed
US-20180117574-A1 BIARYL LIGANDS FOR TRANSITION METAL-CATALYZED REACTIONS UNIV CALIFORNIA (US) 2018-05-03 US disclosed
US-20180118735-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE GRA VENTURE FUND, LLC 2018-05-03 US disclosed
EP-3313522-A1 ANTIBODY DRUG CONJUGATES OF KINESIN SPINDEL PROTEIN (KSP) INHIBITORS WITH ANTI-B7H3-ANTIBODIES Bayer Pharma Aktiengesellschaft (DE) 2018-05-02 EP disclosed
EP-3140304-B1 BENZIMIDAZOLE DERIVATIVES BOEHRINGER INGELHEIM INT (DE) 2018-05-02 EP disclosed
EP-3313525-A1 ANTIBODY DRUG CONJUGATES OF KINESIN SPINDEL PROTEIN (KSP) INHIBITORS WITH ANTI-B7H3-ANTIBODIES Bayer Pharma Aktiengesellschaft (DE) 2018-05-02 EP disclosed
EP-2095131-B1 TAGGED PETROLEUM PRODUCTS AND METHODS OF DETECTING THE SAME AUTHENTIX INC (US) 2018-05-02 EP disclosed
EP-3313521-A1 ANTIBODY DRUG CONJUGATES OF KINESIN SPINDEL PROTEIN (KSP) INHIBITORS WITH ANTI-TWEAKR-ANTIBODIES Bayer Pharma Aktiengesellschaft (DE) 2018-05-02 EP disclosed
US-9957235-B2 Benzimidazol-2-amines as mIDH1 inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-01 US disclosed
US-9956222-B2 Quinazoline derivative as tyrosine-kinase inhibitor, preparation method therefor and application thereof Xuanzhu Pharma Co., Ltd. (CN) 2018-05-01 US disclosed
US-9956541-B2 Methods of separating aromatic compounds from lube base stocks EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2018-05-01 US disclosed
US-9956551-B2 Nano-to-nano Fe/ppm Pd catalysis of cross-coupling reactions in water THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-05-01 US disclosed
US-9957248-B2 Substituted 5-hydroxy-2-heteroaryl-3-phenylpentanonitrile derivatives, processes for their preparation and their use as herbicides and/or plant growth regulators BAYER CROPSCIENCE AKTIENGESELLSHAFT (DE) 2018-05-01 US disclosed
US-9957224-B2 Methods for the treatment of diabetic retinopathy and other ophthalmic diseases ACUCELA INC (US) 2018-05-01 US disclosed
WO-2018075871-A1 NOVEL ANTIBIOTICS AND METHODS OF USING SAME THE BROAD INSTITUTE, INC. (US) 2018-04-26 WO disclosed
US-20180111910-A1 PAIN-RELIEVING COMPOSITIONS AND USES THEREFOR THE UNIVERSITY OF QUEENSLAND (AU) 2018-04-26 US disclosed
EP-3310440-A1 ANTIBODY DRUG CONJUGATES (ADCS) AND ANTIBODY PRODRUG CONJUGATES (APDCS) WITH ENZYMATICALLY CLEAVABLE GROUPS Bayer Pharma Aktiengesellschaft (DE) 2018-04-25 EP disclosed
EP-3177619-B1 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES Bayer Pharma AG (DE) 2018-04-25 EP disclosed
EP-3310773-A1 SUBSTITUTED 4-BENZYL AND 4-BENZOYL PIPERIDINE DERIVATIVES Cephalon, Inc. (US) 2018-04-25 EP disclosed
EP-3310776-A2 INHIBITORS OF BRUTON'S TYROSINE KINASE Pharmacyclics LLC (US) 2018-04-25 EP disclosed
US-9951027-B2 Benzimidazol-2-amines as MIDH1 inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-04-24 US disclosed
US-9949971-B2 Therapeutic combinations of a BTK inhibitor, a PI3K inhibitor and/or a JAK-2 inhibitor ACERTA PHARMA B.V. (NL) 2018-04-24 US disclosed
US-9951086-B2 Indazolecarboxamides, processes for their preparation, pharmaceutical preparations comprising them and their use for producing medicaments BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-04-24 US disclosed
US-9951078-B2 Inhibitors of ERK and methods of use KURA ONCOLOGY, INC. (US) 2018-04-24 US disclosed
US-20180105521-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-04-19 US disclosed
US-20180105531-A1 METHODS AND COMPOSITIONS FOR INHIBITING THE INTERACTION OF MENIN WITH MLL PROTEINS WELLSPRING BIOSCIENCES LLC 2018-04-19 US disclosed
EP-3307716-A1 VERSATILE RAFT AGENT Commonwealth Scientific and Industrial Research Organisation (AU) 2018-04-18 EP disclosed
EP-2595987-B1 NEW AMINOPYRAZOLOQUINAZOLINES BOEHRINGER INGELHEIM INT (DE) 2018-04-18 EP disclosed
EP-2863921-B1 POLYMER-NSAID CONJUGATE POLYACTIVA PTY LTD (AU) 2018-04-18 EP disclosed
US-9944628-B2 Inhibitors of cellular necrosis and related methods PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2018-04-17 US disclosed
US-9944636-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2018-04-17 US disclosed
CN-107922344-A general RAFT agent 联邦科学与工业研究组织 2018-04-17 CN disclosed
US-20180099972-A1 Compounds Useful for Inhibiting Metastasis from Cancer and Methods Using Same UNIV DREXEL (US) 2018-04-12 US disclosed
WO-2018068017-A1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF RAS AND METHODS OF USE THEREOF ARAXES PHARMA LLC (US) 2018-04-12 WO disclosed
WO-2018068021-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. (US) 2018-04-12 WO disclosed
US-20180100861-A1 WATER SOLUBLE FLUORESCENT OR COLORED DYES AND METHODS FOR THEIR USE SONY CORPORATION (JP) 2018-04-12 US disclosed
US-20180098983-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE, INC. 2018-04-12 US disclosed
US-20180099019-A1 Compositions and Methods for Managing Weight UNIGEN, INC. (US) 2018-04-12 US disclosed
EP-2882439-B1 APOPTOSIS-INDUCING AGENTS ABBVIE INC (US) 2018-04-11 EP disclosed
EP-3302481-A1 COMBINATION THERAPY WITH AXL INHIBITOR AND IMMUNE CHECKPOINT MODULATOR OR ONCOLYTIC VIRUS BerGenBio ASA (NO) 2018-04-11 EP disclosed
EP-3303285-A1 PESTICIDALLY ACTIVE OXIME AND HYDRAZONE DERIVATIVES Syngenta Participations AG (CH) 2018-04-11 EP disclosed
EP-3003036-B1 SUBSTITUTED 5-HYDROXY-2,3-DIPHENYLPENTANONITRILE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND/OR PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2018-04-11 EP disclosed
EP-3303317-A1 METHODS AND COMPOSITIONS FOR INHIBITING THE INTERACTION OF MENIN WITH MLL PROTEINS Kura Oncology, Inc. (US) 2018-04-11 EP disclosed
EP-3302589-A1 PROCESS FOR THE PREPARATION OF POLYURETHANE SOLUTIONS BASED ON SILICON-POLYCARBONATE DIOLS Aortech International PLC (GB) 2018-04-11 EP disclosed
EP-3303267-A2 HEMOPROTEIN CATALYSTS FOR IMPROVED ENANTIOSELECTIVE ENZYMATIC SYNTHESIS OF TICAGRELOR California Institute of Technology (US) 2018-04-11 EP disclosed
EP-3302489-A1 METHODS AND COMPOUNDS FOR TREATMENT OF LYMPHOCYTE-RELATED DISEASES AND CONDITIONS Sarepta Therapeutics, Inc. (US) 2018-04-11 EP disclosed
EP-3302057-A1 METHODS AND COMPOSITIONS FOR INHIBITING THE INTERACTION OF MENIN WITH MLL PROTEINS Kura Oncology, Inc. (US) 2018-04-11 EP disclosed
US-9938261-B2 Heterocyclic compounds and methods of use thereof AMBIT BIOSCIENCES CORPORATION (US) 2018-04-10 US disclosed
US-9937171-B2 Methods of blocking the CXCR-4/SDF-1 signaling pathway with inhibitors of bruton's tyrosine kinase ACERTA PHARMA B.V. (NL) 2018-04-10 US disclosed
US-9937167-B2 SHIP1 modulators and methods related thereto AQUINOX PHARMACEUTICALS (CANADA) INC. (CA) 2018-04-10 US disclosed
WO-2018060742-A1 CYANOPYRROLIDINE DERIVATIVES WITH ACTIVITY AS INHIBITORS OF USP30 MISSION THERAPEUTICS LIMITED (GB) 2018-04-05 WO disclosed
WO-2018060691-A1 CYANO-SUBTITUTED HETEROCYCLES WITH ACTIVITY AS INHIBITORS OF USP30 MISSION THERAPEUTICS LIMITED (GB) 2018-04-05 WO disclosed
US-20180092938-A1 OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2018-04-05 US disclosed
WO-2018064510-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC (US) 2018-04-05 WO disclosed
WO-2018064465-A1 COMPOUNDS FOR INCREASING NEURAL PLASTICITY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-04-05 WO disclosed
EP-2918587-B1 Filamin A binding compounds and their use as anti-inflammatory and analgesic agents PAIN THERAPEUTICS INC (US) 2018-04-04 EP disclosed
EP-2788487-B1 OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA SAREPTA THERAPEUTICS INC (US) 2018-04-04 EP disclosed
EP-2919790-B1 GEMCITABINE PRODRUGS AND USES THEREOF BOYEN THERAPEUTICS INC (TW) 2018-04-04 EP disclosed
US-9931340-B2 Pyridazinone compounds and their use as DAAO inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-03 US disclosed
CN-104797257-B Polymer NSAID conjugates 波利艾克蒂瓦有限公司 2018-04-03 CN disclosed
CN-107872956-A Synergistic antifungal composition containing benzoxaborole 宾夕法尼亚州研究基金会 2018-04-03 CN disclosed
US-20180085348-A1 METHODS FOR TREATING CANCER WITH RORGAMMA INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-03-29 US disclosed
US-20180086753-A1 FUSED-TRICYCLIC INHIBITORS OF KRAS AND METHODS OF USE THEREOF ARAXES PHARMA LLC 2018-03-29 US disclosed
US-20180086708-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS MISSION THERAPEUTICS LIMITED (GB) 2018-03-29 US disclosed
WO-2018055577-A1 MIXED TRICYCLO-DNA, 2'-MODIFIED RNA OLIGONUCLEOTIDE COMPOSITIONS AND USES THEREOF SYNTHENA AG (CH) 2018-03-29 WO disclosed
US-20180087005-A1 Fragrance Compositions Comprising Ionic Liquids THE PROCTER & GAMBLE COMPANY 2018-03-29 US disclosed
EP-3297758-A1 NANO-TO-NANO FE/PPM PD CATALYSIS OF CROSS-COUPLING REACTIONS IN WATER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-03-28 EP disclosed
EP-2160192-B1 ANTIMICROBIAL MATERIALS AND COATINGS COVIDIEN LP (US) 2018-03-28 EP disclosed
EP-3297990-A1 SODIUM CHANNEL MODULATORS The Florey Institute Of Neuroscience And Mental Health (AU) 2018-03-28 EP disclosed
US-9926267-B2 Covalent inhibitors of K-Ras G12C ARAXES PHARMA LLC (US) 2018-03-27 US disclosed
US-9926307-B2 Compounds MISSION THERAPEUTICS LTD (GB) 2018-03-27 US disclosed
US-9926245-B2 Fuels and chemicals from lower alkanes Pioneer Energy (US) 2018-03-27 US disclosed
CN-107847765-A The piperidine derivative of 1,4 substitutions 赛福伦公司 2018-03-27 CN disclosed
CN-107846883-A The solvent-free phosphorylation of selectivity 可劳迈戴斯有限公司 2018-03-27 CN disclosed
CN-107849013-A It is used for the cyanopyrrole alkanes for the treatment of cancer as DUB inhibitor 特殊治疗有限公司 2018-03-27 CN disclosed
CN-107840842-A Alkynes is for heterocyclic compound, its preparation method and its in application pharmaceutically 北京天诚医药科技有限公司 2018-03-27 CN disclosed
CN-105473548-B Amide derivatives as lpa receptor antagonist 武田药品工业株式会社 2018-03-23 CN disclosed
WO-2018050794-A1 PROCESS FOR PREPARING OF CAROTENOID MONO-ESTERS BASF SE (DE) 2018-03-22 WO disclosed
WO-2018050792-A1 PROCESS FOR PREPARING ESTERS OF 12'-APOCAROTENALS AS BUILDING BLOCKS FOR CAROTENOIDS BASF SE (DE) 2018-03-22 WO disclosed
WO-2018050795-A1 PROCESS FOR PREPARING OF CAROTENOID MONO-ESTERS BASF SE (DE) 2018-03-22 WO disclosed
WO-2018052967-A1 SUBSTITUTED CHROMANE-8-CARBOXAMIDE COMPOUNDS AND ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA, INC. (US) 2018-03-22 WO disclosed
WO-2018053447-A1 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME ABIDE THERAPEUTICS, INC. (US) 2018-03-22 WO disclosed
WO-2018050793-A1 PROCESS FOR PREPARING PHOSPHONIUM SALT ESTERS AS BUILDING BLOCKS FOR CAROTENOIDES BASF SE (DE) 2018-03-22 WO disclosed
WO-2018053161-A1 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS NATIONAL TAIWAN UNIVERSITY (TW) 2018-03-22 WO disclosed
US-20180079909-A1 ULTRA BRIGHT DIMERIC OR POLYMERIC DYES SONY CORPORATION (JP) 2018-03-22 US disclosed
EP-3294811-A1 ULTRA BRIGHT DIMERIC OR POLYMERIC DYES Sony Corporation (JP) 2018-03-21 EP disclosed
EP-2701506-B1 FORMULATION COMPONENT SYNGENTA LTD (GB) 2018-03-21 EP disclosed
EP-3294721-A1 4H-PYRAN COMPOUNDS AS INSULIN-REGULATED AMINOPEPTIDASE (IRAP) INHIBITORS Monash University (AU) 2018-03-21 EP disclosed
EP-2788488-B1 METHODS FOR TREATING PROGEROID LAMINOPATHIES USING OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA SAREPTA THERAPEUTICS INC (US) 2018-03-21 EP disclosed
EP-3294712-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD Pharmaceuticals, Inc. (US) 2018-03-21 EP disclosed
US-9920085-B2 Boronic acid conjugates of oligonucleotide analogues SAREPTA THERAPEUTICS, INC. (US) 2018-03-20 US disclosed
US-9919288-B2 ZIF-containing adsorbent materials and uses thereof EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2018-03-20 US disclosed
US-9919006-B2 Compositions and methods for treating hyperkalemia ARDELYX, INC. (US) 2018-03-20 US disclosed
US-9919003-B2 Nicotinamide mononucleotide derivatives and their uses METRO INTERNATIONAL BIOTECH, LLC (US) 2018-03-20 US disclosed
CN-107814798-A 3 substitutional crylic acid class compounds and its production and use 四川科伦博泰生物医药股份有限公司 2018-03-20 CN disclosed
US-20180072772-A1 MUTANT AKT-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING CALIFORNIA INSTITUTE OF TECHNOLOGY 2018-03-15 US disclosed
US-20180071262-A1 SPIROCYCLIC HAT INHIBITORS AND METHODS FOR THEIR USE ABBVIE INC. (US) 2018-03-15 US disclosed
US-20180072714-A1 Novel Compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 US disclosed
US-20180072656-A1 Sodium Channel Modulators THE UNIVERSITY OF MELBOURNE (AU) 2018-03-15 US disclosed
EP-2934136-B1 SUBSTITUTED 4-CYAN-3-(PYRIDYL)-4-PHENYLBUTANOATES, METHOD FOR THE PRODUCTION THEREOF AND USES AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2018-03-14 EP disclosed
US-9917328-B2 Halogenated organosilicon electrolytes, methods of using them, and electrochemical devices containing them SILATRONIX, INC. (US) 2018-03-13 US disclosed
US-9913875-B2 Botulinum neurotoxin-specific capture agents, compositions, and methods of using and making CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2018-03-13 US disclosed
CN-107793395-A Fibroblast growth factor acceptor inhibitor and application thereof 南京药捷安康生物科技有限公司 2018-03-13 CN disclosed
WO-2018045229-A1 SUBSTITUTED UREAS AND METHODS OF MAKING AND USING SAME MEBIAS DISCOVERY LLC (US) 2018-03-08 WO disclosed
US-20180064779-A1 Compositions and Methods for Managing or Improving Bone Disorders, Joint Disorders, Cartilage Disorders, or a Combination Thereof UNIGEN, INC. (US) 2018-03-08 US disclosed
US-20180064751-A1 COMPOSITIONS AND METHODS FOR TREATING HYPERKALEMIA ARDELYX, INC. 2018-03-08 US disclosed
US-20180065998-A1 WATER SOLUBLE FLUORESCENT OR COLORED DYES COMPRISING CONJUGATING GROUPS Sony Group Corporation (JP) 2018-03-08 US disclosed
EP-3290407-A1 BROMODOMAIN INHIBITORS Celgene Quanticel Research, Inc (US) 2018-03-07 EP disclosed
EP-3288932-A1 NOVEL EPHA4 INHIBITORS TARGETING ITS LIGAND BINDING DOMAIN Sanford-Burnham Medical Research Institute (US) 2018-03-07 EP disclosed
EP-3288589-A1 THERAPEUTIC COMBINATIONS OF ANTIVIRAL AND ANTI-INFLAMMATORY THERAPIES Foresight Biotherapeutics, Inc. (US) 2018-03-07 EP disclosed
EP-2855449-B1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES TAKEDA PHARMACEUTICALS CO (JP) 2018-03-07 EP disclosed
EP-2074115-B1 N3-HETEROARYL SUBSTITUTED TRIAZOLES AND N5-HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS INC (US) 2018-03-07 EP disclosed
EP-2970764-B1 METHOD FOR SOLVENTLESS QUANTUM DOT EXCHANGE NANOSYS INC (US) 2018-03-07 EP disclosed
EP-3289083-A1 NUCLEOSIDE-MODIFIED RNA FOR INDUCING AN ADAPTIVE IMMUNE RESPONSE The Trustees Of The University Of Pennsylvania (US) 2018-03-07 EP disclosed
US-9908865-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-03-06 US disclosed
US-9908885-B2 Bromodomain inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2018-03-06 US disclosed
US-9908845-B2 Aryl ethers and uses thereof PELOTON THERAPEUTICS, INC. (US) 2018-03-06 US disclosed
CN-105324372-B 1-sulfonylpiperidine derivatives as prokineticin receptor modulators 武田药品工业株式会社 2018-03-06 CN disclosed
US-20180055852-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2018-03-01 US disclosed
WO-2018039331-A1 NETWORK POLYMERS AND METHODS OF MAKING AND USING SAME THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2018-03-01 WO disclosed
US-20180055899-A1 Compositions and Methods for Managing or Improving Bone Disorders, Cartilage Disorders, or Both UNIGEN, INC. (US) 2018-03-01 US disclosed
EP-3041840-B1 RILYAZINE DERIVATIVES AND COMPOSITIONS FOR THE TREATMENT OF CANCER THE WARNER-BABCOCK INST FOR GREEN CHEMISTRY LLC (US) 2018-02-28 EP disclosed
EP-2268623-B9 QUINAZOLINE DERIVATIVES AS RAF KINASE MODULATORS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORP (US) 2018-02-28 EP disclosed
EP-2367800-B1 SUBSTITUTED PYRIMIDINES FOR THE TREATMENT OF DISEASES SUCH AS CANCER BOEHRINGER INGELHEIM INT (DE) 2018-02-28 EP disclosed
US-9902696-B2 1,4-substituted piperidine derivatives CEPHALON, INC. (US) 2018-02-27 US disclosed
US-9902738-B2 Compounds and methods for preventing, treating and/or protecting against sensory hair cell death UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2018-02-27 US disclosed
US-9902719-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2018-02-27 US disclosed
US-9902727-B2 Aminoalcohol substituted 2,3-dihydroimidazo[1,2-C]quinazoline derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis BAYER INTELLECTUAL PROPERTY GMBH (DE) 2018-02-27 US disclosed
CN-104902898-B Diazole lactams 凯莫森特里克斯股份有限公司 2018-02-23 CN disclosed
US-20180051036-A1 COMPOUND INHIBITING ACTIVITIES OF BTK AND/OR JAK3 KINASES Beijing Hanmi Pharmaceutical Co., Ltd. (CN) 2018-02-22 US disclosed
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EP-2847163-B1 IRON CHELATORS AS HIV-1 INHIBITORS UNIV HOWARD (US) 2018-02-21 EP disclosed
EP-2925760-B1 C20'-SUBSTITITED UREA DERIVATIVES OF VINCA ALKALOIDS SCRIPPS RESEARCH INST (US) 2018-02-21 EP disclosed
EP-3283462-A1 FUSED-TRICYCLIC INHIBITORS OF KRAS AND METHODS OF USE THEREOF Araxes Pharma LLC (US) 2018-02-21 EP disclosed
EP-3283076-A1 METHODS OF TREATING HEPATITIS B VIRUS Gilead Sciences, Inc. (US) 2018-02-21 EP disclosed
EP-3283077-A2 BROMODOMAIN INHIBITOR Celgene Quanticel Research, Inc. (US) 2018-02-21 EP disclosed
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US-9895334-B2 Treatment of virally induced lesions LEO LABORATORIES LIMITED (IE) 2018-02-20 US disclosed
US-9896418-B2 Aryl ethers and uses thereof PELOTON THERAPEUTICS, INC. (US) 2018-02-20 US disclosed
CN-107708757-A Method for negatively affecting biomembrane 联邦科学和工业研究组织 2018-02-16 CN disclosed
CN-107708701-A Novel respiratory control modulating compounds and methods of making and using the same 纽拉德有限公司 2018-02-16 CN disclosed
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US-20180042902-A1 Heterocyclic Compounds and Uses Thereof INTELLIKINE, LLC 2018-02-15 US disclosed
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US-20180044334-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-02-15 US disclosed
US-20180042931-A1 N-PHENYL-(MORPHOLIN-4-YL OR PIPERAZINYL)ACETAMIDE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE WNT SIGNALLING PATHWAYS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-02-15 US disclosed
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-02-15 US disclosed
WO-2018031658-A1 TREATMENT OF RELAPSED AND/OR REFRACTORY SOLID TUMORS AND NON-HODGKIN'S LYMPHOMAS CELGENE CORPORATION (US) 2018-02-15 WO disclosed
US-20180044296-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-02-15 US disclosed
US-20180044325-A1 FUSED PYRIMIDINES AS INHIBITORS OF P97 COMPLEX CLEAVE BIOSCIENCES, INC. 2018-02-15 US disclosed
US-20180044324-A1 Quinolinones as Inhibitors of Translation Initiation Complex Sanford Burnham Prebys Medical Discovery Institute 2018-02-15 US disclosed
US-20180042905-A1 METHODS OF TREATING HEPATITIS B VIRUS GILEAD SCIENCES, INC. 2018-02-15 US disclosed
EP-3280708-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS AND METHODS OF USE THEREOF Araxes Pharma LLC (US) 2018-02-14 EP disclosed
EP-2875018-B1 FUSED PYRIMIDINES AS INHIBITORS OF p97 COMPLEX CLEAVE BIOSCIENCES INC (US) 2018-02-14 EP disclosed
EP-3281942-A1 B-LACTAMASE INHIBITOR AND APPLICATION THEREOF Xuanzhu Pharma Co., Ltd. (CN) 2018-02-14 EP disclosed
EP-3280262-A1 SYNERGISTIC BENZOXABOROLE-CONTAINING ANTI-FUNGICIDAL COMPOSITION The Penn State Research Foundation (US) 2018-02-14 EP disclosed
US-9890189-B2 Gemcitabine prodrugs and uses thereof BoYen Therapeutics, Inc. (TW) 2018-02-13 US disclosed
US-20180037583-A1 PURINONE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS LLC (US) 2018-02-08 US disclosed
WO-2018026441-A1 METHODS FOR PREVENTING OR TREATING FIBROTIC DISEASES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-02-08 WO disclosed
EP-3277677-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS Mission Therapeutics Limited (GB) 2018-02-07 EP disclosed
US-9884843-B2 Cyclic sulfone and sulfoximine analogs and uses thereof PELOTON THERAPEUTICS, INC. (US) 2018-02-06 US disclosed
US-20180030090-A1 NON-MEMBRANE DISRUPTIVE P53 ACTIVATING STAPLED PEPTIDES AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2018-02-01 US disclosed
US-20180030027-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC (US) 2018-02-01 US disclosed
US-20180028507-A1 3-CARBAMOYLPHENYL-4-CARBOXAMIDE AND ISOPHTALAMIDE DERIVATIVES AS INHIBITORS OF THE WNT SIGNALLING PATHWAY BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-02-01 US disclosed
WO-2018022624-A1 INHIBITION OF GALECTIN 3 BINDING TO THE AIRWAY EPITHELIAL SURFACE TO TREAT OR PREVENT SEPTIC SHOCK RESULTING FROM INFLUENZA AND SUBSEQUENT PNEUMOCOCCAL PNEUMONIA INFECTION UNIVERSITY OF MARYLAND, BALTIMORE (US) 2018-02-01 WO disclosed
US-20180028508-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RES INC (US) 2018-02-01 US disclosed
EP-3273974-A1 THERAPY FOR MALIGNANT DISEASE Women and Infants Hospital of Rhode Island Inc. (US) 2018-01-31 EP disclosed
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US-9879025-B2 Transfer hydrogenation of cyclopamine analogs INFINITY PHARMACEUTICALS, INC. (US) 2018-01-30 US disclosed
US-9879200-B2 Lubricating compositions and methods for the use thereof INGEVITY SOUTH CAROLINA, LLC (US) 2018-01-30 US disclosed
WO-2018015328-A1 UREA AND THIOUREA SUBSTITUTED BICYCLES DERIVATIVES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2018-01-25 WO disclosed
WO-2018015818-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2018-01-25 WO disclosed
US-20180022756-A1 COMPOUNDS AND METHODS FOR PREVENTING OR TREATING SENSORY HAIR CELL DEATH FRED HUTCHINSON CANCER CENTER 2018-01-25 US disclosed
US-20180020662-A1 Substituted 1-cycloalkyl-2-oxotetrahydroquinolin-6-ylsulfonamides or salts thereof and use thereof to increase stress tolerance in plants BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-01-25 US disclosed
US-20180022757-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES, INC. 2018-01-25 US disclosed
EP-3270951-A1 BOTULINUM NEUROTOXIN-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING California Institute of Technology (US) 2018-01-24 EP disclosed
EP-3271352-A2 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME Abide Therapeutics, Inc. (US) 2018-01-24 EP disclosed
US-9873697-B2 Histone demethylase inhibitors Celgene Quantical Research, Inc. (US) 2018-01-23 US disclosed
CN-107614062-A Methods of treating cancer with ROR gamma inhibitors 加利福尼亚大学董事会 2018-01-19 CN disclosed
WO-2018011569-A1 WEE-1 INHIBITING PYRAZOLOPYRIMIDINONE COMPOUNDS ALMAC DISCOVERY LIMITED (GB) 2018-01-18 WO disclosed
US-20180015093-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS INFINITY PHARMACEUTICALS, INC. 2018-01-18 US disclosed
US-20180015087-A1 CONJUGATES OF CEREBLON BINDING COMPOUNDS AND G12C MUTANT KRAS, HRAS OR NRAS PROTEIN MODULATING COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC 2018-01-18 US disclosed
WO-2018011628-A1 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2018-01-18 WO disclosed
US-20180015082-A1 6-Alkynyl-pyridine Derivatives BOEHRINGER INGELHEIM INT (DE) 2018-01-18 US disclosed
EP-3052096-B1 INHIBITORS OF ERK AND METHODS OF USE KURA ONCOLOGY INC (US) 2018-01-17 EP disclosed
EP-3267792-A1 COMPOSITIONS FOR USE IN TREATING PULMONARY ARTERIAL HYPERTENSION Peloton Therapeutics, Inc. (US) 2018-01-17 EP disclosed
EP-3268362-A1 SUBSTITUTED PYRIDINES AND USES THEREOF Peloton Therapeutics, Inc. (US) 2018-01-17 EP disclosed
EP-3268087-A1 METHODS FOR TREATING CANCER WITH RORgamma INHIBITORS The Regents of the University of California (US) 2018-01-17 EP disclosed
US-9868722-B2 Monocyclic pyrimidine/pyridine compounds as inhibitors of P97 complex CLEAVE BIOSCIENCES, INC. (US) 2018-01-16 US disclosed
US-9867848-B2 Compositions and methods for treating hyperkalemia ARDELYX, INC. (US) 2018-01-16 US disclosed
WO-2018009891-A1 CONDUCTIVE CONFORMAL COATINGS POLYDROP, LLC (US) 2018-01-11 WO disclosed
US-20180009739-A1 Ligand-Enabled meta-C-H Activation Using a Transient Mediator THE SCRIPPS RESEARCH INSTITUTE 2018-01-11 US disclosed
US-20180009780-A1 PIPERIDINE AND AZEPINE DERIVATIVES AS PROKINETICIN RECEPTOR MODULATORS TAKEDA PHARMACEUTICALS CO (JP) 2018-01-11 US disclosed
EP-3265453-A1 NEW PYRIDINONES AND ISOQUINOLINONES AS INHIBITORS OF THE BROMODOMAIN BRD9 Boehringer Ingelheim International GmbH (DE) 2018-01-10 EP disclosed
EP-3266776-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES AbbVie Inc. (US) 2018-01-10 EP disclosed
EP-2858993-B1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES BAYER IP GMBH (DE) 2018-01-10 EP disclosed
EP-3265143-A1 METHODS FOR ADVERSELY AFFECTING BIOFILMS Commonwealth Scientific & Industrial Research Organisation ( C.S.I.R.O. ) (AU) 2018-01-10 EP disclosed
US-9862701-B2 Inhibitors of KRAS G12C mutant proteins ARAXES PHARMA LLC (US) 2018-01-09 US disclosed
US-9862946-B2 Peptide oligonucleotide conjugates SAREPTA THERAPEUTICS, INC. (US) 2018-01-09 US disclosed
WO-2018005430-A1 BISPHENOL A-FREE CROSSLINKED POLYMER COMPOSITIONS WARNER BABCOCK INSTITUTE FOR GREEN CHEMISTRY, LLC (US) 2018-01-04 WO disclosed
WO-2018000047-A1 METHOD OF TREATING IMMUNOGLOBULIN LIGHT CHAIN AMYLOIDOSIS PRANA BIOTECHNOLOGY LIMITED (AU) 2018-01-04 WO disclosed
US-20180002373-A1 Amino Acid and Peptide Conjugates and Uses Thereof AUCKLAND UNISERVICES LIMITED (NZ) 2018-01-04 US disclosed
US-20180002335-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS INFINITY PHARMACEUTICALS, INC. 2018-01-04 US disclosed
US-20180002348-A1 PHENOTHIAZINE-PYRIDINE COMPOUNDS AND USES THEREOF THE CHINESE UNIVERSITY OF HONG KONG, OFFICE OF RESEARCH AND KNOWLEDGE TRANSFER SERVICES (CN) 2018-01-04 US disclosed
EP-3262055-A1 WATER SOLUBLE FLUORESCENT OR COLORED DYES COMPRISING CONJUGATING GROUPS Sony Corporation (JP) 2018-01-03 EP disclosed
EP-3262022-A1 PHENYLETHYNYLNAPHTHALENE DYES AND METHODS FOR THEIR USE Sony Corporation (JP) 2018-01-03 EP disclosed
EP-3057957-B1 CYCLOPENTYLBENZAMIDE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF PSYCHOTIC AND COGNITIVE DISORDERS TAKEDA PHARMACEUTICALS CO (JP) 2018-01-03 EP disclosed
EP-3030553-B1 PIPERIDINE AND AZEPINE DERIVATIVES AS PROKINETICIN RECEPTOR MODULATORS TAKEDA PHARMACEUTICALS CO (JP) 2018-01-03 EP disclosed
EP-2738156-B1 9-AMINOMETHYL SUBSTITUTED TETRACYCLINE COMPOUNDS KBP BIOSCIENCES USA INC (US) 2018-01-03 EP disclosed
EP-3010900-B1 1-SULFONYL PIPERIDINE DERIVATIVES AS MODULATORS OF PROKINETICIN RECEPTORS TAKEDA PHARMACEUTICALS CO (JP) 2018-01-03 EP disclosed
US-9856249-B2 Inhibitors of leukotriene A4 hydrolase CELTAXSYS, INC. (US) 2018-01-02 US disclosed
US-9856260-B2 Compounds useful for inhibiting metastasis from cancer and methods using same DREXEL UNIVERSITY (US) 2018-01-02 US disclosed
US-9855289-B2 Nicotinamide mononucleotide derivatives and their uses METRO INTERNATIONAL BIOTECH, LLC (US) 2018-01-02 US disclosed
CN-107531759-A Non-film destructiveness p53 activation bookbinding peptides 新加坡科技研究局 2018-01-02 CN disclosed
CN-107531738-A Niacinetoside or nicotinamide riboside compositions, reduced derivatives thereof and uses thereof 可劳迈戴斯有限公司 2018-01-02 CN disclosed
CN-107531698-A With the active fused bicyclic heteroaryl group derivative as PHD inhibitor 武田药品工业株式会社 2018-01-02 CN disclosed
CN-107531709-A Beta lactamase restrainer and application thereof 山东轩竹医药科技有限公司 2018-01-02 CN disclosed
US-20170369474-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE AQUINNAH PHARMACEUTICALS INC (US) 2017-12-28 US disclosed
US-20170369492-A1 1,3-SUBSTITUTED 2-AMINO-INDOLE DERIVATIVES AND ANALOGUES USEFUL IN THE TREATMENT OR PREVENTION OF DIABETES MELLITUS, OBESITY, AND INFLAMMATORY BOWEL DISEASE TAKEDA PHARMACEUTICALS CO (JP) 2017-12-28 US disclosed
US-20170369511-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2017-12-28 US disclosed
WO-2017223413-A1 REVERSIBLY SWITCHABLE SURFACTANTS AND METHODS OF USE WARNER BABCOCK INSTITUTE FOR GREEN CHEMISTRY, LLC (US) 2017-12-28 WO disclosed
WO-2017223284-A1 NON-CATALYTIC SUBSTRATE-SELECTIVE P38α-SPECIFIC MAPK INHIBITORS WITH ENDOTHELIAL-STABILIZING AND ANTI-INFLAMMATORY ACTIVITY, AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2017-12-28 WO disclosed
WO-2017222996-A1 ANTIMALARIAL COMPOSITIONS AND USES THEREOF THE CALIFORNIA INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2017-12-28 WO disclosed
US-20170368028-A1 N-BENZOATE GROUP SUBSTITUTED BENZOPYRROLINE-2-ONE DERIVATIVE AND USE THEREOF Beijing Hanmi Pharmaceutical Co., Ltd. (CN) 2017-12-28 US disclosed
US-20170368004-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC. 2017-12-28 US disclosed
WO-2017223397-A1 PHOTOCHROMIC WATER HARVESTING PLATFORM WARNER BABCOCK INSTITUTE FOR GREEN CHEMISTRY, LLC (US) 2017-12-28 WO disclosed
EP-3259268-A1 1,3,4-THIADIAZOL-2-YL-BENZAMIDE DERIVATIVES AS INHIBITORSOF THE WNT SIGNALLING PATHWAY Bayer Pharma Aktiengesellschaft (DE) 2017-12-27 EP disclosed
EP-3259251-A1 N-PHENYL-(MORPHOLIN-4-YL OR PIPERAZINYL)ACETAMIDE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE WNT SIGNALLING PATHWAYS Bayer Pharma Aktiengesellschaft (DE) 2017-12-27 EP disclosed
EP-3259263-A1 3-CARBAMOYLPHENYL-4-CARBOXAMIDE AND ISOPHTALAMIDE DERIVATIVES AS INHIBITORS OF THE WNT SIGNALLING PATHWAY Bayer Pharma Aktiengesellschaft (DE) 2017-12-27 EP disclosed
US-9850247-B2 Pyrimidopyrimidinones useful as Wee-1 kinase inhibitors ALMAC HOUSE (GB) 2017-12-26 US disclosed
CN-107501297-A Phenothiazine-pyridine compounds and uses thereof 香港中文大学 2017-12-22 CN disclosed
CN-107501279-A Furanoquinoline dione compound and medical application thereof 东莞市真兴贝特医药技术有限公司 2017-12-22 CN disclosed
US-20170362263-A1 PHOSPHORUS LIGANDS AND METHODS OF USE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-12-21 US disclosed
US-20170360726-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE AQUINNAH PHARMACEUTICALS INC (US) 2017-12-21 US disclosed
US-20170360795-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS INFINITY PHARMACEUTICALS, INC. (US) 2017-12-21 US disclosed
US-20170360791-A1 PHARMACEUTICAL COMPOSITIONS FOR INCREASING THE BIOAVAILABILITY OF POORLY SOLUBLE DRUGS ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA 2017-12-21 US disclosed
US-20170362250-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO AQUINOX PHARMACEUTICALS (CANADA) INC (CA) 2017-12-21 US disclosed
WO-2017218516-A1 COMPOSITIONS COMPRISING CONJUGATED POLYMERS AND USES THEREOF POLYDROP, LLC (US) 2017-12-21 WO disclosed
EP-2776475-B1 CLEAN POLYCARBONATE MATERIAL FOR USE IN HARD DISK DRIVE AND SEMICONDUCTOR APPLICATIONS SABIC GLOBAL TECHNOLOGIES BV (NL) 2017-12-20 EP disclosed
EP-2560967-B1 Heterocyclic carboxylic acid amides as PDK1 inihibitors BOEHRINGER INGELHEIM INT (DE) 2017-12-20 EP disclosed
EP-2776393-B1 NAMPT INHIBITORS ABBVIE INC (US) 2017-12-20 EP disclosed
EP-3256484-A1 NON-MEMBRANE DISRUPTIVE p53 ACTIVATING STAPLED PEPTIDES Agency For Science, Technology And Research (SG) 2017-12-20 EP disclosed
US-9844547-B2 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases ABBVIE INC. (US) 2017-12-19 US disclosed
US-9844576-B2 Compositions and methods for managing weight UNIGEN, INC. (US) 2017-12-19 US disclosed
US-9845489-B2 Compositions for stabilizing DNA, RNA and proteins in saliva and other biological samples during shipping and storage at ambient temperatures BIOMATRICA, INC. (US) 2017-12-19 US disclosed
CN-107484415-A 1-cyanopyrrolidine compounds as USP30 inhibitors 特殊治疗有限公司 2017-12-15 CN disclosed
US-20170355823-A1 METHODS OF PRODUCING ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2017-12-14 US disclosed
US-20170355822-A1 ORGANOSILICA MATERIALS, METHODS OF MAKING, AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2017-12-14 US disclosed
US-20170354961-A1 CATALYSTS AND METHODS OF MAKING THE SAME EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2017-12-14 US disclosed
WO-2017214332-A1 CONVERSION OF SUGARS TO IONIC LIQUIDS NATIONAL TECHNOLOGY & ENGINEERING SOLUTIONS OF SANDIA, LLC (US) 2017-12-14 WO disclosed
WO-2017214334-A1 CONVERSION OF LIGNIN TO IONIC LIQUIDS NATIONAL TECHNOLOGY & ENGINEERING SOLUTIONS OF SANDIA, LLC (US) 2017-12-14 WO disclosed
WO-2017214269-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2017-12-14 WO disclosed
US-9840680-B2 Fragrance compositions comprising ionic liquids THE PROCTER & GAMBLE COMPANY (US) 2017-12-12 US disclosed
US-9840505-B2 Solid forms of (S)-3-(1-(9H-purin-6-ylamino)ethyl)-8-chloro-2-phenylisoquinolin-1 (2H)-one and methods of use thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-12-12 US disclosed
US-9840553-B2 Dual PDGF/VEGF antagonists KODIAK SCIENCES INC. (US) 2017-12-12 US disclosed
US-9840516-B2 Substituted quinazolines as inhibitors of KRAS G12C ARAXES PHARMA LLC (US) 2017-12-12 US disclosed
US-9840517-B2 Compound inhibiting activities of BTK and/or JAK3 kinases Beijing Hanmi Pharmaceutical Co., Ltd. (CN) 2017-12-12 US disclosed
CN-105452233-B Piperidine and azepane derivatives as prokineticin receptor modulators 武田药品工业株式会社 2017-12-08 CN disclosed
US-20170349586-A1 [9,10-DIMETHOXY-3-(2-METHYLPROPYL)-1H,2H,3H,4H,6H,7H,11BH-PYRIDO-[2,1-A]ISOQUINOLIN-2-YL]METHANOL AND COMPOUNDS, COMPOSITIONS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES, INC. 2017-12-07 US disclosed
US-20170349556-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 QUANTIEL PHARMACEUTICALS, INC. 2017-12-07 US disclosed
US-20170348320-A1 IMIDAZOLOTHIAZOLE COMPOUNDS FOR THE TREATMENT OF DISEASE AMBIT BIOSCIENCES CORP (US) 2017-12-07 US disclosed
US-20170349555-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2017-12-07 US disclosed
EP-3251675-A1 PREVENTION OR TREATMENT OF URIC ACID OR GOUT DISEASE Shanton Pharma Co., Ltd. (CN) 2017-12-06 EP disclosed
EP-3252058-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF HIV INFECTIONS Gilead Sciences, Inc. (US) 2017-12-06 EP disclosed
EP-3252038-A1 N-BENZOATE GROUP SUBSTITUTED BENZOPYRROLINE-2-ONE DERIVATIVE AND USE THEREOF Beijing Hanmi Pharmaceutical Co., Ltd. (CN) 2017-12-06 EP disclosed
EP-2106260-B1 INSULIN SENSITISERS AND METHODS OF TREATMENT VERVA PHARMACEUTICALS LTD (AU) 2017-12-06 EP disclosed
EP-3066104-B1 TRIAZOLOPYRAZINE DERIVATIVES AS BRD4 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2017-12-06 EP disclosed
EP-3252053-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF HIV INFECTIONS Gilead Sciences, Inc. (US) 2017-12-06 EP disclosed
US-9833468-B2 Methods for treating progeroid laminopathies using oligonucleotide analogues targeting human LMNA SAREPTA THERAPEUTICS, INC. (US) 2017-12-05 US disclosed
US-RE46621-E1 Processes for preparing isoquinolinones and solid forms of isoquinolinones INFINITY PHARMACEUTICALS, INC. (US) 2017-12-05 US disclosed
CN-107428824-A PDGF/VEGF dual antagonists 科达制药 2017-12-01 CN disclosed
WO-2017205766-A1 INHIBITORS OF INTERLEUKIN-1 RECEPTOR-ASSOCIATED KINASE PHARMACYCLICS LLC (US) 2017-11-30 WO disclosed
WO-2017205762-A1 INHIBITORS OF INTERLEUKIN-1 RECEPTOR-ASSOCIATED KINASE PHARMACYCLICS LLC (US) 2017-11-30 WO disclosed
WO-2017205769-A1 INHIBITORS OF INTERLEUKIN-1 RECEPTOR-ASSOCIATED KINASE PHARMACYCLICS LLC (US) 2017-11-30 WO disclosed
US-20170341069-A1 NANO-TO-NANO FE/PPM Pd CATALYSIS OF CROSS-COUPLING REACTIONS IN WATER UNIV CALIFORNIA (US) 2017-11-30 US disclosed
US-20170340621-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED GASTROINTESTINAL DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-11-30 US disclosed
WO-2017205684-A1 COMBINATION THERAPIES WITH FARNESOID X RECEPTOR (FXR) MODULATORS AKARNA THERAPEUTICS, LTD. (GB) 2017-11-30 WO disclosed
US-20170340623-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC. 2017-11-30 US disclosed
WO-2017202719-A1 NEW PHENYLPYRAZOLYLACETAMIDE COMPOUNDS AND DERIVATIVES AS CDK8/CDK19 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-11-30 WO disclosed
EP-3051946-B1 USE OF SUBSTITUTED DIHYDROOXINDOLYLSULFONAMIDES OR THEIR SALTS FOR INCREASING STRESS TOLERANCE IN PLANTS BAYER CROPSCIENCE AG (DE) 2017-11-29 EP disclosed
US-9828377-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-11-28 US disclosed
US-9828379-B2 Pyrrolo-pyrrole carbamate and related organic compounds, pharmaceutical compositions, and medical uses thereof ABIDE THERAPEUTICS, INC. (US) 2017-11-28 US disclosed
US-9828363-B2 Fused pyrimidines as inhibitors of P97 complex CLEAVE BIOSCIENCES, INC. (US) 2017-11-28 US disclosed
US-9828378-B2 Kinase inhibitors and methods of use INTELLIKINE LLC (US) 2017-11-28 US disclosed
US-9828351-B2 Enzyme interacting agents MONASH UNIVERSITY (AU) 2017-11-28 US disclosed
US-9828343-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-11-28 US disclosed
WO-2017198341-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2017-11-23 WO disclosed
WO-2017198734-A1 PROCESS FOR THE MANUFACTURE OF 6-ALKYNYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-11-23 WO disclosed
US-20170333942-A1 POLYMERISATION PROCESS AND POLYMER PRODUCT THE UNIVERSITY OF SYDNEY (AU) 2017-11-23 US disclosed
WO-2017201468-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2017-11-23 WO disclosed
US-20170334899-A1 AMINO-SUBSTITUTED ISOTHIAZOLES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-11-23 US disclosed
US-20170334928-A1 Purification of Rapamycin Derivatives Using Temperature Induced Phase Separation JOHNSON MATTHEY PHARMACEUTICAL MATERIALS, INC. D/B/A JOHNSON MATTHEY PHARMA SERVICES 2017-11-23 US disclosed
US-20170334879-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2017-11-23 US disclosed
US-20170334902-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2017-11-23 US disclosed
US-20170334874-A1 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2017-11-23 US disclosed
US-9822131-B2 Certain chemical entities, compositions and methods INTELLIKINE LLC (US) 2017-11-21 US disclosed
US-9822106-B2 Inhibitors of leukotriene A4 hydrolase CELTAXSYS, INC. (US) 2017-11-21 US disclosed
US-9822119-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2017-11-21 US disclosed
WO-2017197192-A1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME ABIDE THERAPEUTICS, INC. (US) 2017-11-16 WO disclosed
US-20170326103-A1 LYMPH DIRECTING PRODRUGS MONASH UNIVERSITY (AU) 2017-11-16 US disclosed
WO-2017197210-A1 IDENTIFICATION OF SMALL MOLECULE INHIBITORS OF JUMONJI AT-RICH INTERACTIVE DOMAIN 1A (JARID1A) HISTONE DEMETHYLASE YALE UNIVERSITY (US) 2017-11-16 WO disclosed
US-20170327500-A1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2017-11-16 US disclosed
US-20170326148-A1 PREVENTION OR TREATMENT OF URIC ACID OR GOUT DISEASE Shanton Pharma Pte. Ltd. (SG) 2017-11-16 US disclosed
US-20170327693-A1 IN VACUO COATING COMPOSITIONS CAMVAC LIMITED (GB) 2017-11-16 US disclosed
US-20170326116-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2017-11-16 US disclosed
WO-2017196261-A1 JAK AND HDAC DUAL-INHIBITOR COMPOUNDS NATIONAL UNIVERSITY OF SINGAPORE (SG) 2017-11-16 WO disclosed
US-20170327813-A1 3D Printable Hydrogel Materials UNIVERSITY OF WASHINGTON 2017-11-16 US disclosed
WO-2017197240-A1 ASH1L INHIBITORS AND METHODS OF TREATMENT THEREWITH THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2017-11-16 WO disclosed
US-20170327604-A1 OLEFIN POLYMERIZATION CATALYST SYSTEM COMPRISING MESOPOROUS ORGANOSILICA SUPPORT EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2017-11-16 US disclosed
EP-2748149-B9 PYRIDAZINONE COMPOUNDS AND THEIR USE AS DAAO INHIBITORS TAKEDA PHARMACEUTICALS CO (JP) 2017-11-15 EP disclosed
EP-2590656-B1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX INC (US) 2017-11-15 EP disclosed
EP-2934145-B1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2017-11-15 EP disclosed
EP-2384318-B1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX INC (US) 2017-11-15 EP disclosed
US-9815828-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-11-14 US disclosed
US-9815746-B2 Stereodynamic chemosensors GEORGETOWN UNIVERSITY (US) 2017-11-14 US disclosed
US-20170321002-A1 MULTICOLORED ELECTROCHROMIC POLYMER COMPOSITIONS AND METHODS OF MAKING AND USING THE SAME LANNRAY ADVANCED MATERIALS CO. LTD (CN) 2017-11-09 US disclosed
US-20170321101-A1 Refrigeration System With Dual Refrigerants and Liquid Working Fluids JEFF YANJIE (US) 2017-11-09 US disclosed
WO-2017190249-A1 USE OF TOPICAL FORMULATIONS OF CANNABINOIDS IN THE TREATMENT OF EPIDERMOLYSIS BULLOSA AND RELATED CONNECTIVE TISSUE DISORDERS INMED PHARMACEUTICALS INC. (CA) 2017-11-09 WO disclosed
US-20170320971-A1 OLEFIN POLYMERIZATION CATALYST SYSTEM COMPRISING MESOPOROUS ORGANOSILICA SUPPORT EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2017-11-09 US disclosed
US-20170320977-A1 OLEFIN POLYMERIZATION CATALYST SYSTEM COMPRISING MESOPOROUS ORGANOSILICA SUPPORT EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2017-11-09 US disclosed
US-20170320861-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-11-09 US disclosed
US-20170319549-A1 1-CYCLOHEXYL-2-PHENYLAMINOBENZIMIDAZOLES AS MIDH1 INHIBITORS FOR THE TREATMENT OF TUMORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-11-09 US disclosed
EP-2970316-B1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES INC (US) 2017-11-08 EP disclosed
EP-3241834-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2017-11-08 EP disclosed
US-9810690-B2 Method for screening inhibitors of Ras ARAXES PHARMA LLC (US) 2017-11-07 US disclosed
US-20170313702-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2017-11-02 US disclosed
US-20170313669-A1 LACTONE COMPOUNDS AND METHODS OF MAKING AND USING SAME THE SCRIPPS RESEARCH INSTITUTE 2017-11-02 US disclosed
EP-3236752-A2 NOVEL ISOTHIAZOLAMIDES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS FUNGICIDES Bayer CropScience Aktiengesellschaft (DE) 2017-11-01 EP disclosed
EP-3238722-A1 SOLID FORMS OF ISOQUINOLINONES Infinity Pharmaceuticals, Inc. (US) 2017-11-01 EP disclosed
EP-3237374-A1 AMINO ACID AND PEPTIDE CONJUGATES AND USES THEREOF Brimble, Margaret, Anne (NZ) 2017-11-01 EP disclosed
EP-3236940-A1 COMPOSITIONS AND METHODS FOR TREATING HYPERKALEMIA Ardelyx, Inc. (US) 2017-11-01 EP disclosed
EP-3083625-B1 PYRIMIDOPYRIMIDINONES USEFUL AS WEE-1 KINASE INHIBITORS ALMAC DISCOVERY LTD (GB) 2017-11-01 EP disclosed
US-9801871-B2 6-alkynyl-pyridine derivatives BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-10-31 US disclosed
WO-2017184589-A1 A VERSATILE LIGAND FOR PALLADIUM-CATALYZED META-C-H FUNCTIONALIZATIONS THE SCRIPPS RESEARCH INSTITUTE (US) 2017-10-26 WO disclosed
US-20170304300-A1 HIF-2alpha INHIBITORS FOR TREATING IRON OVERLOAD DISORDERS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-10-26 US disclosed
WO-2017184462-A1 THERAPEUTIC COMPOUNDS CELGENE QUANTICEL RESEARCH, INC. (US) 2017-10-26 WO disclosed
US-20170306068-A1 OLEFIN POLYMERIZATION CATALYST SYSTEM COMPRISING MESOPOROUS ORGANOSILICA SUPPORT EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2017-10-26 US disclosed
US-20170305910-A1 Substituted Xanthines and Methods of Use Thereof BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-10-26 US disclosed
WO-2017184491-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2017-10-26 WO disclosed
US-20170304338-A1 USE OF NICOTINIC ACID RIBOSIDE OR NICOTINAMIDE RIBOSIDE DERIVATIVES, AND REDUCED DERIVATIVES THEREOF, AS NAD+ INCREASING PRECURSORS ChromaDex Inc. (US) 2017-10-26 US disclosed
US-20170303542-A1 SYNERGISTIC BENZOXABOROLE-CONTAINING ANTI-FUNGICIDAL COMPOSITION THE PENN STATE RESEARCH FOUNDATION 2017-10-26 US disclosed
US-20170305948-A1 NOVEL PRECATALYST SCAFFOLDS FOR CROSS-COUPLING REACTIONS, AND METHODS OF MAKING AND USING SAME UNIV YALE (US) 2017-10-26 US disclosed
EP-3234094-A1 IONIC LIQUID SYSTEMS The Procter and Gamble Company (US) 2017-10-25 EP disclosed
EP-3233866-A1 PYRAZOLOPYRIDINAMINES AS MKNK1 AND MKNK2 INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2017-10-25 EP disclosed
US-9796712-B2 Heteroaryl compounds for kinase inhibition ARIAD PHARMACEUTICALS, INC. (US) 2017-10-24 US disclosed
US-9796697-B2 Tricyclic inhibitors of HIF-2-alpha and uses thereof PELOTON THERAPEUTICS, INC. (US) 2017-10-24 US disclosed
CN-105247010-B Solvent-free quantum dot exchange method 纳米系统公司 2017-10-24 CN disclosed
WO-2017180789-A2 METHODS OF TREATMENT USING CHLOROTOXIN CONJUGATES Blaze Bioscience, Inc. (US) 2017-10-19 WO disclosed
US-20170295777-A1 Compositions and Methods for Reducing Ice Crystal Formation X-THERMA, INC. (US) 2017-10-19 US disclosed
US-20170298044-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2017-10-19 US disclosed
US-20170296531-A9 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2017-10-19 US disclosed
WO-2017181012-A1 CINCHONIUM BETAINE CATALYSTS AND METHODS OF USING SAME BRANDEIS UNIVERSITY (US) 2017-10-19 WO disclosed
US-20170298026-A1 ALL PURPOSE RAFT AGENT COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2017-10-19 US disclosed
US-20170298029-A1 RAF KINASE MODULATOR COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2017-10-19 US disclosed
US-20170298040-A1 THERAPEUTIC COMPOUNDS CELGENE QUANTICEL RESEARCH, INC. 2017-10-19 US disclosed
WO-2017181149-A1 METHODS OF TREATING BREAST CANCER Blaze Bioscience, Inc. (US) 2017-10-19 WO disclosed
WO-2017180998-A2 PHOTOACTIVE MACROMOLECULES AND USES THEREOF BECKMAN COULTER, INC. (US) 2017-10-19 WO disclosed
US-20170298025-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2017-10-19 US disclosed
EP-3230325-A1 METHODS OF SEPARATING AROMATIC COMPOUNDS FROM LUBE BASE STOCKES ExxonMobil Research and Engineering Company (US) 2017-10-18 EP disclosed
EP-3229807-A1 INHIBITORS OF CELLULAR NECROSIS AND RELATED METHODS President and Fellows of Harvard College (US) 2017-10-18 EP disclosed
EP-3230296-A1 PHOSPHORUS LIGANDS AND METHODS OF USE The Regents of The University of California (US) 2017-10-18 EP disclosed
EP-3229593-A1 HETEROCYCLIC COMPOUNDS AS ANTIBIOTIC POTENTIATORS Synereca Pharmaceuticals, Inc. (US) 2017-10-18 EP disclosed
EP-2729449-B1 5- OR 6 - SUBSTITUTED 3 - HYDROXY - 2 ( 1H) - PYRIDINONES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS IN THERAPY OF DISEASES SUCH AS SCHIZOPHRENIA, COGNITIVE DISORDER AND PAIN TAKEDA PHARMACEUTICALS CO (JP) 2017-10-18 EP disclosed
EP-3230409-A1 ORGANOSILICA MATERIALS AND USES THEREOF ExxonMobil Research and Engineering Company (US) 2017-10-18 EP disclosed
EP-3229952-A1 ORGANOSILICA MATERIALS ExxonMobil Research and Engineering Company (US) 2017-10-18 EP disclosed
EP-3229944-A1 MEMBRANE FABRICATION METHODS USING ORGANOSILICA MATERIALS AND USES THEREOF ExxonMobil Research and Engineering Company (US) 2017-10-18 EP disclosed
EP-3230410-A1 AROMATIC HYDROGENATION CATALYSTS AND USES THEREOF Exxonmobil Research And Engineering Company (US) 2017-10-18 EP disclosed
EP-2079736-B1 SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS INC (US) 2017-10-18 EP disclosed
EP-3229953-A1 COATING METHODS USING ORGANOSILICA MATERIALS AND USES THEREOF ExxonMobil Research and Engineering Company (US) 2017-10-18 EP disclosed
US-9790201-B2 Piperidine and azepine derivatives as prokineticin receptor modulators TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-10-17 US disclosed
US-9790499-B2 Functionally-modified oligonucleotides and subunits thereof SAREPTA THERAPEUTICS, INC. (US) 2017-10-17 US disclosed
US-9790173-B2 Alpha-7 nicotinic acetylcholine receptor modulators and uses thereof-I MERCK SHARP & DOHME CORP. (US) 2017-10-17 US disclosed
US-9790220-B2 Substituted cyclopentanes, tetrahydrofuranes and pyrrolidines as orexin receptor antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-10-17 US disclosed
US-9790228-B2 Heterocyclic kinase inhibitors INTELLIKINE LLC (US) 2017-10-17 US disclosed
US-9790218-B2 Small molecule activators of calcium-activated chloride channels and methods of use THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-10-17 US disclosed
US-20170290330-A1 SUBSTITUTED 5-HYDROXY-2-PHENYL-3-HETEROARYL PENTANENITRILE DERIVATES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND/OR PLANT GROWH REGULATORS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2017-10-12 US disclosed
US-20170290850-A1 NICOTINAMIDE MONONUCLEOTIDE DERIVATIVES AND THEIR USES METRO INTERNATIONAL BIOTECH, LLC 2017-10-12 US disclosed
EP-2752415-B1 Fluorinated ligands for targeting peripheral benzodiazepine receptors AUSTRALIAN NUCLEAR SCIENCE & TECH ORGANISATION (AU) 2017-10-11 EP disclosed
US-9783543-B2 Aminoimidazopyridazines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-10-10 US disclosed
US-20170281614-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE LLC 2017-10-05 US disclosed
WO-2017172979-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS AND METHODS OF USE ARAXES PHARMA LLC (US) 2017-10-05 WO disclosed
EP-2951175-B1 SUBSTITUTED PYRAZOLOPYRIMIDINYLAMINO-INDAZOLES Bayer Pharma AG (DE) 2017-10-04 EP disclosed
US-9776974-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2017-10-03 US disclosed
US-9777006-B2 Inhibitors of leukotriene A4 hydrolase CELTAXSYS, INC. (US) 2017-10-03 US disclosed
US-9777004-B2 Amino-substituted imidazopyridazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-10-03 US disclosed
US-9775844-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-10-03 US disclosed
CN-107216312-A A kind of compound with saltant type IDH inhibitory activity, preparation method and the usage 上海海和药物研究开发有限公司 2017-09-29 CN disclosed
WO-2017163078-A1 1-CYANO-PYRROLIDINE DERIVATIVES AS DBU INHIBITORS MISSION THERAPEUTICS LIMITED (GB) 2017-09-28 WO disclosed
WO-2017162510-A1 SUBSTITUTED QUINAZOLINONE COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISEASES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-09-28 WO disclosed
WO-2017162663-A1 PRODRUGS OF CYTOTOXIC ACTIVE AGENTS HAVING ENZYMATICALLY CLEAVABLE GROUPS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-09-28 WO disclosed
US-20170273964-A1 FATTY ACID SYNTHASE INHIBITOR FOR USE IN THE TREATMENT OF DRUG RESISTANT CANCER SAGIMET BIOSCIENCES INC. 2017-09-28 US disclosed
WO-2017165304-A2 Pd(II)-CATALYZED ENANTIOSELECTIVE BETA-METHYLENE C(sp3)-H BOND ACTIVATION THE SCRIPPS RESEARCH INSTITUTE (US) 2017-09-28 WO disclosed
US-20170275285-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL ELI LILLY AND COMPANY 2017-09-28 US disclosed
US-20170275266-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2017-09-28 US disclosed
EP-3222620-A1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO., LTD. (CN) 2017-09-27 EP disclosed
EP-2598661-B1 COMPOSITIONS FOR STABILIZING DNA, RNA AND PROTEINS IN SALIVA AND OTHER BIOLOGICAL SAMPLES DURING SHIPPING AND STORAGE AT AMBIENT TEMPERATURES BIOMATRICA INC (US) 2017-09-27 EP disclosed
US-9771341-B2 Piperazine carbamates and methods of making and using same ABIDE THERAPEUTICS, INC. (US) 2017-09-26 US disclosed
US-9771333-B2 Quinazoline derivatives as TAM family kinase inhibitors SIGNALCHEM LIFESCIENCES CORP. (CA) 2017-09-26 US disclosed
US-9771329-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2017-09-26 US disclosed
CN-107208076-A Butyrylcholine esterase amphoteric ion polymer conjugate 科达制药 2017-09-26 CN disclosed
CN-107207735-A Organic silica material 埃克森美孚研究工程公司 2017-09-26 CN disclosed
WO-2017161165-A1 B-VITAMIN AND AMINO ACID CONJUGATES OF NICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, DERIVATIVES THEREOF, AND METHODS OF PREPARATION THEREOF ChromaDex Inc. (US) 2017-09-21 WO disclosed
WO-2017161033-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2017-09-21 WO disclosed
WO-2017157418-A1 COMBINATION OF MKNK1-INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-09-21 WO disclosed
US-20170266191-A1 Therapeutic Combination of PI3K Inhibitor and a BTK Inhibitor ACERTA PHARMA BV (NL) 2017-09-21 US disclosed
WO-2017160861-A1 INHIBITORS FOR SOLUBLE EPOXIDE HYDROLASE (SEH) AND FATTY ACID AMIDE HYDROLASE (FAAH) THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-09-21 WO disclosed
WO-2017158388-A1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER MISSION THERAPEUTICS LIMITED (GB) 2017-09-21 WO disclosed
US-20170267709-A1 B-VITAMIN AND AMINO ACID CONJUGATES OFNICOTINOYL RIBOSIDES AND REDUCED NICOTINOYL RIBOSIDES, DERIVATIVES THEREOF, AND METHODS OF PREPARATION THEREOF ChromaDex Inc. (US) 2017-09-21 US disclosed
WO-2017158381-A1 4,6 DIHYDROPYRROLO [3,4-C] PYRAZOLE-5 (1H)-CARBONITRILE DERIVATES FOR TRATING CANCER MISSION THERAPEUTICS LIMITED (GB) 2017-09-21 WO disclosed
WO-2017161116-A1 ISOTOPOLOGUES OF ISOQUINOLINONE AND QUINAZOLINONE COMPOUNDS AND USES THEREOF AS PI3K KINASE INHIBITORS INFINITY PHARMACEUTICALS, INC. (US) 2017-09-21 WO disclosed
WO-2017161012-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2017-09-21 WO disclosed
US-20170267679-A1 TRICYCLIC FUSED PYRIMIDINE COMPOUNDS AS INHIBITORS OF p97 COMPLEX CLEAVE BIOSCIENCES INC (US) 2017-09-21 US disclosed
EP-2970303-B9 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES INC (US) 2017-09-20 EP disclosed
EP-3218363-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED GASTROINTESTINAL DISORDERS Takeda Pharmaceutical Company Limited (JP) 2017-09-20 EP disclosed
US-9765220-B2 Water soluble fluorescent or colored dyes and methods for their use SONY CORPORATION (JP) 2017-09-19 US disclosed
US-9765085-B2 SHIP1 modulators and methods related thereto AQUINOX PHARMACEUTICALS (CANADA) INC. (CA) 2017-09-19 US disclosed
US-20170260204-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2017-09-14 US disclosed
US-20170258795-A1 FUSED PYRIMIDINES AS INHIBITORS OF P97 COMPLEX CLEAVE THERAPEUTICS, INC. 2017-09-14 US disclosed
US-20170260163-A1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS, INC. 2017-09-14 US disclosed
US-20170260161-A1 BI-BENZYL ISOQUINOLINE DERIVATIVE, PREPARATION METHOD AND USE THEREOF IN HEPATOPATHY TREATMENT AND PREVENTION VERSITECH LIMITED (CN) 2017-09-14 US disclosed
WO-2017156391-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF INFECTIONS SPRING BANK PHARMACEUTICALS, INC. (US) 2017-09-14 WO disclosed
EP-2920176-B1 AMINOIMIDAZOPYRIDAZINES AS MKNK1 KINASE INHIBITORS Bayer Pharma AG (DE) 2017-09-13 EP disclosed
EP-3003381-B1 PHARMACEUTICAL COMPOSITIONS Bayer Pharma AG (DE) 2017-09-13 EP disclosed
EP-2785688-B1 A PROCESS FOR THE MANUFACTURE OF CHIRAL CATALYSTS AND THEIR SALTS SCINOPHARM TAIWAN LTD (TW) 2017-09-13 EP disclosed
US-9758517-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-09-12 US disclosed
US-9758511-B2 NAMPT inhibitors ABBVIE INC. (US) 2017-09-12 US disclosed
CN-104684850-B Melamine-aldehyde polymers 新加坡科技研究局 2017-09-08 CN disclosed
US-20170253562-A1 Nampt Inhibitors ABBVIE INC (US) 2017-09-07 US disclosed
US-20170253596-A2 SHIP1 MODULATORS AND METHODS RELATED THERETO TARO PHARMACEUTICALS INC. (CA) 2017-09-07 US disclosed
US-20170253594-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-09-07 US disclosed
EP-1844020-B1 HETEROCYCLIC CARBOXAMIDE COMPOUNDS AS STEROID NUCLEAR RECEPTOR LIGANDS EXELIXIS INC (US) 2017-09-06 EP disclosed
EP-2804864-B1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES BAYER IP GMBH (DE) 2017-09-06 EP disclosed
US-9751888-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-09-05 US disclosed
US-20170246310-A1 VAR2CSA-DRUG CONJUGATES ZYMEWORKS INC. (CA) 2017-08-31 US disclosed
US-20170247339-A1 QUINAZOLINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF ARROMAX PHARMATECH CO., LTD. (CN) 2017-08-31 US disclosed
US-20170247725-A1 IN VIVO AND IN VITRO OLEFIN CYCLOPROPANATION CATALYZED BY HEME ENZYMES CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2017-08-31 US disclosed
US-20170247394-A1 SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-08-31 US disclosed
US-20170247729-A1 SWITCHABLE IONIC LIQUIDS FOR BIOMASS PRETREATMENT AND ENZYMATIC HYDROLYSIS UNITED STATES DEPARTMENT OF ENERGY 2017-08-31 US disclosed
US-20170247365-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2017-08-31 US disclosed
US-20170247391-A1 THIENOPYRIMIDINE AND THIENOPYRIDINE COMPOUNDS AND METHODS OF USE THEREOF WELLSPRING BIOSCIENCES LLC 2017-08-31 US disclosed
US-20170247376-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF RAS ARAXES PHARMA LLC (US) 2017-08-31 US disclosed
US-20170247389-A2 SHIP1 MODULATORS AND METHODS RELATED THERETO TARO PHARMACEUTICALS INC. (CA) 2017-08-31 US disclosed
EP-3210469-A1 USE OF SUBSTITUTED THIO-1,2,4-TRIAZOLES FOR INCREASING STRESS TOLERANCE IN PLANTS Bayer Cropscience AG (DE) 2017-08-30 EP disclosed
EP-2638044-B1 ALKOXY-SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINES BAYER IP GMBH (DE) 2017-08-30 EP disclosed
EP-3209660-A1 1-CYCLOHEXYL-2-PHENYLAMINOBENZIMIDAZOLES AS MIDH1 INHIBITORS FOR THE TREATMENT OF TUMORS Bayer Pharma Aktiengesellschaft (DE) 2017-08-30 EP disclosed
EP-3210966-A1 ALKOXYPHENYLPROPYLAMINES FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION Acucela, Inc. (US) 2017-08-30 EP disclosed
EP-3209646-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2017-08-30 EP disclosed
US-9745304-B2 Amidoimidazopyridazines as MKNK-1 kinase inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-08-29 US disclosed
US-9745272-B2 Quinazoline-2,4(1 H,3H)-dione derivatives HYDRA BIOSCIENCES, INC. (US) 2017-08-29 US disclosed
CN-107108489-A general RAFT agent 联邦科学与工业研究组织 2017-08-29 CN disclosed
US-20170240546-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2017-08-24 US disclosed
US-20170240529-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2017-08-24 US disclosed
WO-2017141036-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LIMITED (GB) 2017-08-24 WO disclosed
US-20170238544-A1 MOLECULES THAT INDUCE DISEASE RESISTANCE IN PLANTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2017-08-24 US disclosed
US-20170239351-A1 Therapeutic Combinations of a BTK Inhibitor, a PI3K Inhibitor, a JAK-2 Inhibitor, a PD-1 Inhibitor, and/or a PD-L1 Inhibitor ACERTA PHARMA BV (NL) 2017-08-24 US disclosed
EP-3208270-A1 FUSED PYRIMIDINES AS INHIBITORS OF P97 COMPLEX Cleave Biosciences, Inc. (US) 2017-08-23 EP disclosed
EP-3207128-A2 BUTYRYLCHOLINESTERASE ZWITTERIONIC POLYMER CONJUGATES Kodiak Sciences Inc. (US) 2017-08-23 EP disclosed
EP-3207031-A1 ATAXIA TELENGIECTASIA AND RAD3-RELATED (ATR) PROTEIN KINASE INHIBITORS Atrin Pharmaceuticals LLC (US) 2017-08-23 EP disclosed
EP-3206692-A1 FATTY LIVER DISEASE TREATMENT USING GLUCOCORTICOID AND MINERALOCORTICOID RECEPTOR ANTAGONISTS Corcept Therapeutics, Inc. (US) 2017-08-23 EP disclosed
EP-2512462-B1 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC (US) 2017-08-23 EP disclosed
US-9737075-B2 Synergistic benzoxaborole-containing anti-fungicidal composition THE PENN STATE RESEARCH FOUNDATION (US) 2017-08-22 US disclosed
US-9738644-B2 Chemical compounds, compositions and methods for kinase modulation INFINITY PHARMACEUTICALS, INC. (US) 2017-08-22 US disclosed
US-9737496-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2017-08-22 US disclosed
US-9738637-B2 Histone demethylase inhibitors Celgene Quantical Research, Inc. (US) 2017-08-22 US disclosed
US-20170231995-A1 BTK Inhibitors to Treat Solid Tumors Through Modulation of the Tumor Microenvironment LUCID TRUSTEE SERVICES LIMITED (GB) 2017-08-17 US disclosed
US-20170231986-A1 Therapeutic Combinations of a BTK Inhibitor, a PI3K Inhibitor, a JAK-2 Inhibitor, and/or a BCL-2 Inhibitor ACERTA PHARMA B.V. (NL) 2017-08-17 US disclosed
EP-3205644-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Celtaxsys Inc. (US) 2017-08-16 EP disclosed
EP-3204353-A1 ALL PURPOSE RAFT AGENT Commonwealth Scientific and Industrial Research Organisation (AU) 2017-08-16 EP disclosed
EP-3203991-A1 HIF-2 INHIBITORS FOR TREATING IRON OVERLOAD DISORDERS The Board of Regents of The University of Texas System (US) 2017-08-16 EP disclosed
EP-2668179-B1 NEW 5-ALKYNYL-PYRIDINES BOEHRINGER INGELHEIM INT (DE) 2017-08-16 EP disclosed
EP-3204395-A1 NOVEL PRECATALYST SCAFFOLDS FOR CROSS-COUPLING REACTIONS, AND METHODS OF MAKING AND USING SAME Yale University (US) 2017-08-16 EP disclosed
US-9730937-B2 RAF kinase modulator compounds and methods of use thereof AMBIT BIOSCIENCES CORPORATION (US) 2017-08-15 US disclosed
US-9730943-B2 Alkoxy-substituted 2,3-dihydroimidazo[1,2-C]quinazolines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-08-15 US disclosed
US-9730929-B2 Substituted aminoimidazopyridazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-08-15 US disclosed
US-9731321-B2 Polymerisation process and polymer product THE UNIVERSITY OF SYDNEY (AU) 2017-08-15 US disclosed
US-9732092-B2 Substituted 2,3,4,5,7,9,13,13a-octahydropyrido[1′,2′:4,5]pyrazino[2,1-b][1,3]OXAZEPINES and methods for treating viral infections GILEAD SCIENCES, INC. (US) 2017-08-15 US disclosed
US-20170226093-A1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO., LTD. (CN) 2017-08-10 US disclosed
US-20170226081-A1 GLUCOSE TRANSPORT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-08-10 US disclosed
US-20170226130-A1 Ataxia Telengiectasia And Rad3-Related (ATR) Protein Kinase Inhibitors Atrin Pharmaceuticals LLC (US) 2017-08-10 US disclosed
US-20170224688-A1 Methods of Using BTK Inhibitors to Treat Dermatoses ACERTA PHARMA BV (NL) 2017-08-10 US disclosed
US-20170226110-A1 INHIBITORS OF ERK AND METHODS OF USE KURA ONCOLOGY, INC. 2017-08-10 US disclosed
US-20170224819-A1 Therapeutic Combinations of a BTK Inhibitor, a PI3K Inhibitor, a JAK-2 Inhibitor, and/or a CDK 4/6 Inhibitor ACERTA PHARMA BV (NL) 2017-08-10 US disclosed
US-20170224682-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO NEOLEUKIN THERAPEUTICS, INC. 2017-08-10 US disclosed
WO-2017136466-A1 HEME PROTEIN CATALYSTS FOR CARBON-SILICON BOND FORMATION IN VITRO AND IN VIVO CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2017-08-10 WO disclosed
EP-2240451-B1 Isoquinolinone derivatives substituted with a purine useful as PI3K inhibitors INTELLIKINE LLC (US) 2017-08-09 EP disclosed
EP-2909181-B1 PKM2 MODULATORS AND METHODS FOR THEIR USE TOLERO PHARMACEUTICALS INC (US) 2017-08-09 EP disclosed
US-9725441-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-08-08 US disclosed
US-9725465-B2 Biaryl acetamide compounds and methods of use thereof AMBIT BIOSCIENCES CORPORATION (US) 2017-08-08 US disclosed
WO-2017129796-A1 ORGANIC REACTIONS CARRIED OUT IN AQUEOUS SOLUTION IN THE PRESENCE OF A HYDROXYALKYL(ALKYL)CELLULOSE OR AN ALKYLCELLULOSE AbbVie Deutschland GmbH & Co. KG (DE) 2017-08-03 WO disclosed
US-20170217946-A1 AMINO-SUBSTITUTED ISOXAZOLES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-08-03 US disclosed
WO-2017132463-A1 SURFACE PRIMER COMPOSITIONS AND METHODS OF USE ACatechol, Inc. (US) 2017-08-03 WO disclosed
US-20170218346-A1 Heme Protein Catalysts for Carbon-Silicon Bond Formation In Vitro and In Vivo CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2017-08-03 US disclosed
WO-2017132538-A1 AMLEXANOX ANALOGS THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2017-08-03 WO disclosed
US-20170216765-A1 COMPOSITE GAS SEPARATION MEMBRANE THE UNIVERSITY OF MELBOURNE (AU) 2017-08-03 US disclosed
WO-2017132484-A1 PHOTO-CLEAVABLE PRIMER COMPOSITIONS AND METHODS OF USE ACatechol, Inc. (US) 2017-08-03 WO disclosed
US-20170217997-A1 PHOTO-CLEAVABLE PRIMER COMPOSITIONS AND METHODS OF USE ORMCO CORPORATION 2017-08-03 US disclosed
US-20170217999-A1 SURFACE PRIMER COMPOSITIONS AND METHODS OF USE ORMCO CORPORATION 2017-08-03 US disclosed
US-20170218021-A1 BOTULINUM NEUROTOXIN-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING REGENERON PHARMACEUTICALS, INC. 2017-08-03 US disclosed
US-20170216304-A1 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-08-03 US disclosed
US-20170217980-A1 AMLEXANOX ANALOGS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2017-08-03 US disclosed
US-20170217850-A1 ORGANIC REACTIONS CARRIED OUT IN AQUEOUS SOLUTION IN THE PRESENCE OF A HYDROXYALKYL(ALKYL)CELLULOSE OR AN ALKYLCELLULOSE ABBVIE INC. 2017-08-03 US disclosed
US-20170217892-A1 ARYL ETHERS AND USES THEREOF PELOTON THERAPEUTICS, INC. 2017-08-03 US disclosed
US-20170217891-A1 ARYL ETHERS AND USES THEREOF PELOTON THERAPEUTICS, INC. 2017-08-03 US disclosed
EP-3197562-A1 FRAGRANCE COMPOSITIONS COMPRISING IONIC LIQUIDS The Procter and Gamble Company (US) 2017-08-02 EP disclosed
EP-3197989-A1 IONIC LIQUIDS The Procter and Gamble Company (US) 2017-08-02 EP disclosed
EP-3197883-A1 NOVEL COMPOUNDS Mission Therapeutics Limited (GB) 2017-08-02 EP disclosed
US-9718815-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-08-01 US disclosed
US-9718821-B2 Pyridopyrimidinone inhibitors of kinases ABBVIE INC. (US) 2017-08-01 US disclosed
US-9717770-B2 Compositions and methods for managing or improving bone disorders, cartilage disorders, or both UNIGEN, INC. (US) 2017-08-01 US disclosed
CN-106999481-A Processes and intermediates for preparing C5aR antagonists 凯莫森特里克斯股份有限公司 2017-08-01 CN disclosed
CN-107001339-A Novel compounds 特殊治疗有限公司 2017-08-01 CN disclosed
WO-2017127442-A1 METHODS FOR TREATING CANCER WITH RORGAMMA INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-07-27 WO disclosed
US-20170210738-A1 GLUCOSE TRANSPORT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-07-27 US disclosed
US-20170209448-A1 TREATMENT REGIMENS USING MULTIPLE PHARMACEUTICAL AGENTS INTELLIKINE LLC 2017-07-27 US disclosed
US-20170210701-A1 SUBSTITUTED CYANO CYCLOALKYL PENTA-2,4-DIENES, CYANO CYCLOALKYL PENT-2-EN-4-YNES, CYANO HETEROCYCLYL PENTA-2,4-DIENES AND CYANO HETEROCYCLYL PENT-2-EN-4-YNES AS ACTIVE SUBSTANCES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2017-07-27 US disclosed
EP-3193851-A1 COMBINATION THERAPIES FOR TREATMENT OF CANCER Araxes Pharma LLC (US) 2017-07-26 EP disclosed
EP-3193880-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL Hydra Biosciences, Inc. (US) 2017-07-26 EP disclosed
EP-2886540-B1 BICYCLIC SUBSTITUTED PYRIMIDINE COMPOUNDS XUANZHU PHARMA CO LTD (CN) 2017-07-26 EP disclosed
EP-3194387-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2017-07-26 EP disclosed
EP-3193601-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2017-07-26 EP disclosed
EP-2970211-B1 HISTONE DEMETHYLASE INHIBITORS QUANTICEL PHARMACEUTICALS INC (US) 2017-07-26 EP disclosed
EP-3193881-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2017-07-26 EP disclosed
US-9714230-B2 Histone demethylase inhibitors Celgene Quantical Research, Inc. (US) 2017-07-25 US disclosed
US-9714246-B2 [9,10-dimethoxy-3-(2-methylpropyl)-1H,2H,3H,4H,6H,7H,11bH-pyrido-[2,1-a]isoquinolin-2-yl]methanol and compounds, compositions and methods relating thereto NEUROCRINE BIOSCIENCES, INC. (US) 2017-07-25 US disclosed
US-9714244-B2 Substituted pyrido[4,3-d]pyrimidines as Wee-1 inhibitors ALMAC DISCOVERY LIMITED (GB) 2017-07-25 US disclosed
CN-106967257-A Form polythiophene:The method of polysulfonate complex compound 新加坡科技研究局 2017-07-21 CN disclosed
US-20170202816-A1 USE OF ANTHELMINTIC AGENTS AGAINST DIROFILARIA IMMITIS INTERVET INC. (US) 2017-07-20 US disclosed
US-20170204032-A1 PROCESS FOR PREPARING BRANCHED ALLYL COMPOUNDS SOUTH UNIVERSITY OF SCIENCE AND TECHNOLOGY OF CHINA (CN) 2017-07-20 US disclosed
WO-2017122175-A1 THERAPEUTIC COMBINATIONS OF AN ANTIFOLATE AND A BTK INHIBITOR ACERTA PHARMA B.V. (NL) 2017-07-20 WO disclosed
WO-2017121684-A1 5-SUBSTITUTED 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-07-20 WO disclosed
WO-2017123766-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF DISEASE SPEROVIE BIOSCIENCES, INC. (US) 2017-07-20 WO disclosed
EP-2887963-B1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX INC (US) 2017-07-19 EP disclosed
EP-2948460-B1 LOW TEMPERATURE SYNTHESIS OF RAPAMYCIN DERIVATIVES BIOSENSORS INT GROUP LTD (BM) 2017-07-19 EP disclosed
US-9707205-B2 S1P receptors modulators and their use thereof AKAAL PHARMA PTY LTD. (AU) 2017-07-18 US disclosed
US-9709571-B2 Method of drug design VAST BIOSCIENCE PTY LIMITED (AU) 2017-07-18 US disclosed
US-9708326-B2 Inhibitors of bruton's tyrosine kinase PHARMACYCLICS LLC (US) 2017-07-18 US disclosed
US-9708348-B2 Trisubstituted bicyclic heterocyclic compounds with kinase activities and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-07-18 US disclosed
US-20170197982-A1 THIOPHENE DERIVATIVES GANZHOU HEMAY PHARMACEUTICAL CO., LTD. (CN) 2017-07-13 US disclosed
US-20170198287-A1 OLIGONUCLEOTIDE ANALOGUES HAVING MODIFIED INTERSUBUNIT LINKAGES AND/OR TERMINAL GROUPS JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2017-07-13 US disclosed
US-20170197910-A1 SUBSTITUTED VINYL AND ALKYNYL CYANOCYCLOALKANOLS AND VINYL AND ALKYNYL CYANOHETEROCYCLOALKANOLS AS ACTIVE AGENTS AGAINST ABIOTIC PLANT STRESS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2017-07-13 US disclosed
US-20170197962-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD PHARMACEUTICALS, INC. 2017-07-13 US disclosed
US-20170196854-A1 USE OF ANTHELMINTIC AGENTS AGAINST DIROFILARIA IMMITIS INTERVET INC. (US) 2017-07-13 US disclosed
US-20170197945-A1 2-SUBSTITUTED QUINAZOLINE COMPOUNDS COMPRISING A SUBSTITUTED HETEROCYCLIC GROUP AND METHODS OF USE THEREOF ARAXES PHARMA LLC 2017-07-13 US disclosed
US-20170196903-A1 COMPOSITIONS AND METHODS FOR TREATING HYPERKALEMIA ARDELYX, INC. 2017-07-13 US disclosed
US-20170197922-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS DEUTSCHES KREBSFORSCHUNGSZENTRUM, STIFTUNG DES ÖFFENTLICHEN RECHTS (DE) 2017-07-13 US disclosed
US-20170197921-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS DEUTSCHES KREBSFORSCHUNGSZENTRUM, STIFTUNG DES ÖFFENTLICHEN RECHTS (DE) 2017-07-13 US disclosed
US-20170197979-A1 BENZOTHIADIAZOLAMINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-07-13 US disclosed
EP-3189038-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Celgene Quanticel Research, Inc. (US) 2017-07-12 EP disclosed
EP-2134723-B1 2,6 DIAMINO-9H-PURINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF PROLIFERATIVE DISEASES BOEHRINGER INGELHEIM INT (DE) 2017-07-12 EP disclosed
US-9701657-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-07-11 US disclosed
US-9700554-B2 Polycyclic-carbamoylpyridone compounds and their pharmaceutical use GILEAD SCIENCES, INC. (US) 2017-07-11 US disclosed
US-9701792-B2 Composite compositions and methods of preparing and using same THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2017-07-11 US disclosed
US-9702870-B2 Fluorescent dyes and related methods UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2017-07-11 US disclosed
US-20170189434-A1 NICOTINAMIDE MONONUCLEOTIDE DERIVATIVES AND THEIR USES METRO INTERNATIONAL BIOTECH, LLC 2017-07-06 US disclosed
US-20170190672-A1 METHODS FOR PREPARATION OF QUINAZOLINE DERIVATIVES ARAXES PHARMA LLC 2017-07-06 US disclosed
US-20170190669-A1 PYRAZOLE COMPOUNDS AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2017-07-06 US disclosed
US-20170190766-A1 ANTIBODIES AND CONJUGATES THEREOF KODIAK SCIENCES INC. 2017-07-06 US disclosed
US-20170190698-A1 ENZYME INTERACTING AGENTS CENTRAL ADELAIDE LOCAL HEALTH NETWORK INCORPORATED (AU) 2017-07-06 US disclosed
WO-2017117464-A1 ANTIBODIES AND CONJUGATES THEREOF KODIAK SCIENCES INC. (US) 2017-07-06 WO disclosed
WO-2017117154-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2017-07-06 WO disclosed
WO-2017117528-A1 LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS Acuitas Therapeutics, Inc. (CA) 2017-07-06 WO disclosed
EP-2925761-B1 TRIAZOLOPYRAZINES AS BRD4 INHIBITORS FOR USE IN THE TREATMENT OF CANCER BOEHRINGER INGELHEIM INT (DE) 2017-07-05 EP disclosed
WO-2017109488-A1 CYANOPYRROLIDINE DERVIVATIVES AS INHIBITORS FOR DUBS MISSION THERAPEUTICS LIMITED (GB) 2017-06-29 WO disclosed
WO-2017112902-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. (US) 2017-06-29 WO disclosed
WO-2017112909-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. (US) 2017-06-29 WO disclosed
US-20170183325-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2017-06-29 US disclosed
US-20170183353-A1 N-HYDROXY BICYCLIC HYDANTOIN CARBAMATES AS TOOLS FOR INDETIFICATION OF SERINE HYDROLASE TARGETS H. LUNDBECK A/S (DK) 2017-06-29 US disclosed
WO-2017112904-A1 INHIBITORS OF GLUCOCORTICOID RECEPTOR ORIC PHARMACEUTICALS, INC. (US) 2017-06-29 WO disclosed
US-20170183338-A1 PIPERIDIN-1 -YL AND AZEPIN-1 -YL CARBOXYLATES AS MUSCARINIC M4 RECEPTOR AGONISTS NXERA PHARMA UK LIMITED (GB) 2017-06-29 US disclosed
US-20170183356-A1 New Imaging Agents and Methods of Identifying Same THR TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2017-06-29 US disclosed
EP-3183254-A1 NEW SPIRO[3H-INDOLE-3,2´-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2017-06-28 EP disclosed
US-9689877-B2 Water soluble fluorescent or colored dyes and methods for their use SONY CORPORATION (JP) 2017-06-27 US disclosed
US-9688711-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2017-06-27 US disclosed
US-20170173072-A1 COMPOSITIONS AND METHODS FOR TREATING HYPERKALEMIA ARDELYX, INC. 2017-06-22 US disclosed
US-20170174695-A1 NEW SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-06-22 US disclosed
US-20170173569-A1 Fe-ppm Pd, Cu and/or Ni Nanoparticle-Catalyzed Reactions in Water LIPSHUTZ BRUCE H (US) 2017-06-22 US disclosed
US-20170176475-A1 NOVEL METHODS AND KITS FOR DETECTING A RIFAMYCIN, OR DERIVATIVE OR ANALOGUE THEREOF UNIV DREXEL (US) 2017-06-22 US disclosed
US-20170174678-A1 NOVEL ANTIVIRAL COMPOUNDS AND METHODS USING SAME Rhe Trustees of The University of Pennsylvania 2017-06-22 US disclosed
US-20170173007-A1 PYRIDAZINONE COMPOUNDS AND THEIR USE AS DAAO INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-06-22 US disclosed
US-20170174656-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2017-06-22 US disclosed
WO-2017106426-A1 FE NANOPARTICLES WITH PPM CONTENTS OF PD, CU AND/OR NI, REACTIONS IN WATER CATALYZED BY THEM THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-06-22 WO disclosed
WO-2017103614-A1 Novel Compounds MISSION THERAPEUTICS LIMITED (GB) 2017-06-22 WO disclosed
WO-2017105439-A1 CINCHONINE-DERIVED CATALYSTS AND METHODS OF USING SAME BRANDEIS UNIVERSITY (US) 2017-06-22 WO disclosed
EP-3179992-A1 THERAPEUTIC COMBINATIONS OF A BTK INHIBITOR, A PI3K INHIBITOR, A JAK-2 INHIBITOR, A PD-1 INHIBITOR AND/OR A PD-L1 INHIBITOR Acerta Pharma B.V. (NL) 2017-06-21 EP disclosed
EP-3181553-A1 QUINAZOLINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Arromax Pharmatech Co., Ltd. (CN) 2017-06-21 EP disclosed
EP-3180337-A1 PYRIDO[3,4-D]PYRIMIDINE-2,4(1H,3H)-DIONE DERIVATIVES Hydra Biosciences, Inc. (US) 2017-06-21 EP disclosed
EP-3180345-A1 THIENO- AND FURO[2,3-D]PYRIMIDINE-2,4[1H,3H]-DIONE DERIVATIVES AS TRPC5 MODULATORS FOR THE TREATMENT OF NEUROPSYCHIATRIC DISORDERS Hydra Biosciences, Inc. (US) 2017-06-21 EP disclosed
EP-3180318-A1 QUINAZOLINE-2,4(1H,3H)-DIONE DERIVATIVES AS TRCP5 MODULATORS FOR THE TREATMENT OF NEUROPSYCHIATRY DISORDERS Hydra Biosciences, Inc. (US) 2017-06-21 EP disclosed
EP-3180342-A1 PYRROLO[3,2-D]PYRIMIDINE-2,4(3H,5H)-DIONE DERIVATIVES Hydra Biosciences, Inc. (US) 2017-06-21 EP disclosed
EP-3179991-A1 THERAPEUTIC COMBINATIONS OF A BTK INHIBITOR, A PI3K INHIBITOR, A JAK-2 INHIBITOR, AND/OR A BCL-2 INHIBITOR Acerta Pharma B.V. (NL) 2017-06-21 EP disclosed
EP-3180340-A1 PYRIDO[2,3-D]PYRIMIDINE-2,4(1H,3H)-DIONE DERIVATIVES Hydra Biosciences, Inc. (US) 2017-06-21 EP disclosed
EP-2395993-B1 SKIN TREATMENT LEO LABORATORIES LTD (IE) 2017-06-21 EP disclosed
EP-2976327-B1 3-ACETYLAMINO-1-(PHENYL-HETEROARYL-AMINOCARBONYL OR PHENYL-HETEROARYL-CARBONYLAMINO)BENZENE DERIVATIVES FOR THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS Bayer Pharma AG (DE) 2017-06-21 EP disclosed
EP-3179990-A1 FATTY ACID SYNTHASE INHIBITOR FOR USE IN THE TREATMENT OF DRUG RESISTANT CANCER 3-V Biosciences, Inc. (US) 2017-06-21 EP disclosed
US-9682141-B2 Combination of kinase inhibitors and uses thereof INTELLIKINE LLC (US) 2017-06-20 US disclosed
US-9682097-B2 Oligonucleotide analogues targeting human LMNA SAREPTA THERAPEUTICS, INC. (US) 2017-06-20 US disclosed
US-20170166867-A1 2,4,5-TRI-SUBSTITUTED AZOLE-BASED CASEIN KINASE 1 INHIBITORS AS INDUCERS FOR CARDIOMYOGENESIS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2017-06-15 US disclosed
US-20170166549-A1 Substituted 5-hydroxy-2-heteroaryl-3-phenylpentanonitrile derivatives, processes for their preparation and their use as herbicides and/or plant growth regulators BAYER CROPSCIENCE AKTIENGESELLSHAFT (DE) 2017-06-15 US disclosed
US-20170166553-A1 Piperidine Derivatives for Use in the Treatment or Prevention of Psychiatric and Neurological Conditions TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-06-15 US disclosed
US-20170168073-A1 CHALCONE-UREA DERIVATIVES AS INSULIN SENSORS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2017-06-15 US disclosed
US-20170166598-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD PHARMACEUTICALS, INC. 2017-06-15 US disclosed
US-20170166555-A1 FUNCTIONALISED AND SUBSTITUTED INDOLES AS ANTI-CANCER AGENTS NOVOGEN LIMITED (AU) 2017-06-15 US disclosed
WO-2017100546-A1 METHODS FOR PREPARATION OF QUINAZOLINE DERIVATIVES ARAXES PHARMA LLC (US) 2017-06-15 WO disclosed
WO-2017100537-A1 BETA-LACTAMASE INHIBITORS VenatoRx Pharmaceuticals, Inc. (US) 2017-06-15 WO disclosed
WO-2017098328-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHAMACEUTICALS, INC. (BB) 2017-06-15 WO disclosed
EP-2556058-B1 RADIOPROTECTOR COMPOUNDS AND METHODS PETER MACCALLUM CANCER INST (AU) 2017-06-14 EP disclosed
EP-3177619-A1 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES Bayer Pharma Aktiengesellschaft (DE) 2017-06-14 EP disclosed
US-9675616-B2 Arylaminoalcohol-substituted 2,3-dihydroimidazo[1,2-C]quinolines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-06-13 US disclosed
US-9675612-B2 Substituted thiazolopyrimidines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-06-13 US disclosed
US-9676762-B2 Pyrimidine compounds containing seven-membered fused ring systems BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-06-13 US disclosed
US-9676766-B2 Triazolopyridines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-06-13 US disclosed
US-9675694-B2 Polycyclic agents for the treatment of respiratory syncytial virus infections BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2017-06-13 US disclosed
US-9676724-B2 Cyanoquinoline derivatives TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO., LTD. (CN) 2017-06-13 US disclosed
US-9676770-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-06-13 US disclosed
CN-104684906-B Nampt inhibitor 艾伯维公司 2017-06-09 CN disclosed
WO-2017096315-A1 TRIAZOLE DAGL(α) INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2017-06-08 WO disclosed
US-20170157105-A1 Anti-Viral Compounds ABBVIE INC. (US) 2017-06-08 US disclosed
US-20170158681-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2017-06-08 US disclosed
US-20170158628-A1 ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS AND USES THEREOF-I MERCK SHARP & DOHME CORP. (US) 2017-06-08 US disclosed
US-20170158636-A1 FUNCTIONALISED AND SUBSTITUTED CARBAZOLES AS ANTI-CANCER AGENTS Novogen ltd (AU) 2017-06-08 US disclosed
US-20170158664-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2017-06-08 US disclosed
US-20170157104-A1 Anti-Viral Compounds ABBVIE INC. (US) 2017-06-08 US disclosed
WO-2017096025-A1 NORPREGNANE DERIVATIVES FOR THE RISK REDUCTION OF BREAST CANCER Helix Twelve Pharmaceuticals Corporation, Inc. (US) 2017-06-08 WO disclosed
WO-2017091854-A1 SODIUM-ION ELECTROLYTE COMPOSITION DEAKIN UNIVERSITY (AU) 2017-06-08 WO disclosed
US-20170157143-A1 NORPREGNANE DERIVATIVES FOR THE RISK REDUCTION OF BREAST CANCER Helix Twelve Pharmaceuticals Corporation, Inc. (US) 2017-06-08 US disclosed
US-20170158709-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RES INC (US) 2017-06-08 US disclosed
US-20170157135-A1 FUNCTIONALISED AND SUBSTITUTED INDOLES AS ANTI-CANCER AGENTS NOVOGEN LIMITED (AU) 2017-06-08 US disclosed
WO-2017093718-A1 1-CYANO-PYRROLIDINE DERIVATIVES AS INHIBITORS OF USP30. MISSION THERAPEUTICS LIMITED (GB) 2017-06-08 WO disclosed
US-20170158700-A1 3-SUBSTITUTED 2-AMINO-INDOLE DERIVATIVES TAKEDA CAMBRIDGE LIMITED (GB) 2017-06-08 US disclosed
US-20170158685-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2017-06-08 US disclosed
EP-3174539-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE Pharmacyclics, LLC (US) 2017-06-07 EP disclosed
EP-2581372-B1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO LTD (CN) 2017-06-07 EP disclosed
EP-2638043-B1 ARYLAMINOALCOHOL-SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINOLINES BAYER IP GMBH (DE) 2017-06-07 EP disclosed
US-9670202-B2 Substituted triazolopyridines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-06-06 US disclosed
US-9669038-B1 Heterocyclic compounds and uses thereof GLOBAVIR BIOSCIENCES, INC. (US) 2017-06-06 US disclosed
US-9669032-B2 Enhanced treatment regimens using mTOR inhibitors INTELLIKINE LLC (US) 2017-06-06 US disclosed
WO-2017091150-A1 A POLYMERIC COMPOSITION AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2017-06-01 WO disclosed
WO-2017091781-A1 AMMONIUM BASED IONIC LIQUIDS USEFUL FOR LIGNOCELLULOSIC PROCESSING SANDIA CORPORATION (US) 2017-06-01 WO disclosed
US-20170152221-A1 ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS AND USES THEREOF MERCK SHARP & DOHME CORP. (US) 2017-06-01 US disclosed
US-20170152226-A1 FUNCTIONALISED AND SUBSTITUTED INDOLES AS ANTI-CANCER AGENTS Novogen ltd (AU) 2017-06-01 US disclosed
EP-2900674-B1 COMPOUNDS AND METHODS FOR PREVENTING, TREATING AND/OR PROTECTING AGAINST SENSORY HAIR CELL DEATH UNIV WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2017-05-31 EP disclosed
EP-3172204-A1 AMINO-SUBSTITUTED ISOXAZOLES Bayer Pharma Aktiengesellschaft (DE) 2017-05-31 EP disclosed
EP-2758401-B1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES BAYER IP GMBH (DE) 2017-05-31 EP disclosed
EP-3172192-A1 GLUCOSE TRANSPORT INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2017-05-31 EP disclosed
EP-3172194-A1 GLUCOSE TRANSPORT INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2017-05-31 EP disclosed
EP-2984090-B1 2-AMINOPYRIDO[4,3-D]PYRIMIDIN-5-ONE DERIVATIVES AND THEIR USE AS WEE-1 INHIBITORS ALMAC DISCOVERY LTD (GB) 2017-05-31 EP disclosed
CN-106727587-A A kind of pharmaceutical composition for treating arrhythmia cordis 李娜 2017-05-31 CN disclosed
CN-105102463-B Low Temperature Synthesis of Rapamycin Derivatives 生物传感器国际集团有限公司 2017-05-31 CN disclosed
US-9663528-B2 Substituted 1,2,3,4,6,8,12,12a-octahydro-1,4-methanodipyrido[1,2-a:1',2'-d]pyrazines and methods for treating viral infections GILEAD SCIENCES, INC. (US) 2017-05-30 US disclosed
US-9663510-B2 Substituted triazolopyridines and their use as TTK inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-05-30 US disclosed
US-9663634-B2 Scratch resistant polymers TENASITECH PTY LTD (AU) 2017-05-30 US disclosed
US-9663535-B2 Ataxia telengiectasia and Rad3-related (ATR) protein kinase inhibitors Atrin Pharmaceuticals LLC (US) 2017-05-30 US disclosed
US-9661848-B2 Substituted 4-cyan-3-(pyridyl)-4-phenylbutanoates, method for the production thereof and uses as herbicides and plant growth regulators BAYER CROPSCIENCE AG (DE) 2017-05-30 US disclosed
US-20170143727-A1 USE OF CINNABARINIC ACID AS A MODULATOR OF IMMUNE RESPONSE IN AUTOIMMUNE DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2017-05-25 US disclosed
US-20170143841-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS KODIAK SCIENCES INC. 2017-05-25 US disclosed
US-20170143712-A1 Methods of Treating Cancers, Immune and Autoimmune Diseases, and Inflammatory Diseases Based on BTK Occupancy and BTK Resynthesis Rate ACERTA PHARMA BV (NL) 2017-05-25 US disclosed
EP-3169325-A1 THERAPEUTIC INHIBITORY COMPOUNDS Lifesci Pharmaceuticals, Inc. (BB) 2017-05-24 EP disclosed
CN-106715456-A Lymphatic prodrugs 莫纳什大学 2017-05-24 CN disclosed
US-9656932-B2 Preparation of pentanol with ethanol derived from fermentation Pioneer Energy (US) 2017-05-23 US disclosed
US-9655921-B2 Compositions and methods for treating hyperkalemia ARDELYX, INC. (US) 2017-05-23 US disclosed
US-9656988-B2 Inhibitors of Bruton's tyrosine kinase PHARMACYCLICS LLC (US) 2017-05-23 US disclosed
US-9655892-B2 Certain chemical entities, compositions and methods INTELLIKINE LLC (US) 2017-05-23 US disclosed
US-20170137402-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Quanticel Pharmaceuticals, Inc. 2017-05-18 US disclosed
US-20170135343-A1 AGRICULTURAL PHEROMONE COMPOSITIONS COMPRISING POSITIONAL ISOMERS PROVIVI, INC. 2017-05-18 US disclosed
US-20170137407-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. 2017-05-18 US disclosed
WO-2017081003-A1 SUBSTITUTED PYRAZOLOPYRIDINAMINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-05-18 WO disclosed
US-20170135994-A9 NAMPT INHIBITORS ABBVIE INC. (US) 2017-05-18 US disclosed
US-20170136023-A1 QUINAZOLINE DERIVATIVE AS TYROSINE-KINASE INHIBITOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Xuanzhu Pharma Co., Ltd. (CN) 2017-05-18 US disclosed
US-20170137469-A1 POLYMYXIN DERIVATIVES AS ANTIMICROBIAL COMPOUNDS MONASH UNIVERSITY (AU) 2017-05-18 US disclosed
US-20170136014-A1 Therapeutic Combinations of a BTK Inhibitor, a PI3K Inhibitor and/or a JAK-2 Inhibitor ACERTA PHARMA BV (NL) 2017-05-18 US disclosed
EP-2716633-B1 QUINAZOLINE DERIVATIVE AS TYROSINE-KINASE INHIBITOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF XUANZHU PHARMA CO LTD (CN) 2017-05-17 EP disclosed
EP-2350083-B1 PYRIMIDO[5,4-D]PYRIMIDINES AS CELL PROLIFERATION INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2017-05-17 EP disclosed
EP-3166605-A1 USE OF ANTHELMINTIC AGENTS AGAINST DIROFILARIA IMMITIS Intervet International B.V. (NL) 2017-05-17 EP disclosed
US-9650450-B2 RAFT polymers COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2017-05-16 US disclosed
US-9650391-B2 N3-heteroaryl substituted triazoles and N5-heteroaryl substituted triazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS INC. (US) 2017-05-16 US disclosed
US-9650358-B2 Pyridine CDK9 kinase inhibitors ABBVIE INC. (US) 2017-05-16 US disclosed
US-20170128443-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2017-05-11 US disclosed
US-20170131278-A1 METHOD FOR SCREENING INHIBITORS OF RAS ARAXES PHARMA LLC 2017-05-11 US disclosed
WO-2017079564-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR COLORING EDIBLE MATERIALS THE PENN STATE RESEARCH FOUNDATION (US) 2017-05-11 WO disclosed
WO-2017079641-A1 N-[2-(1 -BENZYLPIPERIDIN-4-YL)ETHYL]-4-(PYRAZIN-2-YL)-PIPERAZINE-1 -CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS MUSCARINIC RECEPTOR 4 (M4) ANTAGONISTS FOR TREATING NEUROLOGICAL DISEASES NEUROCRINE BIOSCIENCES, INC. (US) 2017-05-11 WO disclosed
US-20170128444-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2017-05-11 US disclosed
US-20170129882-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2017-05-11 US disclosed
US-20170128456-A1 CARBON MONOXIDE-RELEASING MOLECULES FOR THERAPEUTIC APPLICATIONS AND METHODS OF MAKING AND USING THEREOF GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC, (US) 2017-05-11 US disclosed
EP-3164380-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Celgene Quanticel Research, Inc. (US) 2017-05-10 EP disclosed
EP-2970303-B1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES INC (US) 2017-05-10 EP disclosed
EP-3164401-A1 NEW SPIRO[3H-INDOLE-3,2´-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2017-05-10 EP disclosed
EP-3164509-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Celgene Quanticel Research, Inc. (US) 2017-05-10 EP disclosed
CN-106661032-A 1,3-substituted 2-aminoindole derivatives and analogues useful in the treatment or prevention of diabetes mellitus, obesity and inflammatory bowel disease 武田药品工业株式会社 2017-05-10 CN disclosed
CN-106661229-A Silicone ligands for quantum dots 纳米系统公司 2017-05-10 CN disclosed
CN-106661005-A Functionalized and substituted indoles as anticancer agents 诺沃根公司 2017-05-10 CN disclosed
CN-104105718-B RAFT polymers 联邦科学和工业研究组织 2017-05-10 CN disclosed
US-9643974-B2 Amino-substituted imidazopyridazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-05-09 US disclosed
US-9643971-B2 Breathing control modulating compounds, and methods of using same GALLEON PHARMACEUTICALS, INC. (US) 2017-05-09 US disclosed
US-9643965-B2 Histone demethylase inhibitors Celgene Quantical Research, Inc. (US) 2017-05-09 US disclosed
US-20170121363-A1 Compounds, Compositions and Methods for Coloring Edible Materials THE PENN STATE RESEARCH FOUNDATION 2017-05-04 US disclosed
WO-2017070743-A1 POLYURETHANE/UREA MATERIALS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2017-05-04 WO disclosed
WO-2017075531-A1 NOVEL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS Acuitas Therapeutics, Inc. (CA) 2017-05-04 WO disclosed
US-20170121633-A1 Fragrance Compositions Comprising Ionic Liquids THE PROCTER & GAMBLE COMPANY 2017-05-04 US disclosed
US-20170119923-A1 POLYURETHANE/UREA COMPOSITIONS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION 2017-05-04 US disclosed
WO-2017075522-A2 GLP-2 POLYPEPTIDES WITH IMPROVED PROTEOLYTIC STABILITY, AND METHODS OF PREPARING AND USING SAME TUFTS UNIVERSITY (US) 2017-05-04 WO disclosed
WO-2017075299-A1 FRAGRANCE COMPOSITIONS COMPRISING IONIC LIQUIDS THE PROCTER & GAMBLE COMPANY (US) 2017-05-04 WO disclosed
WO-2017075505-A2 NOVEL POLYPEPTIDES WITH IMPROVED PROTEOLYTIC STABILITY, AND METHODS OF PREPARING AND USING SAME TUFTS UNIVERSITY (US) 2017-05-04 WO disclosed
US-20170121338-A1 AMINO PRYAN RING DERIVATIVE AND COMPOSITION AND USE THEREOF SICHUAN HAISCO PHARMACEUTICAL CO., LTD (CN) 2017-05-04 US disclosed
US-20170119904-A1 NOVEL LIPIDS AND LIPID NANOPARTICLE FORMULATIONS FOR DELIVERY OF NUCLEIC ACIDS Acuitas Therapeutics, Inc. (CA) 2017-05-04 US disclosed
US-20170121752-A1 DETECTION OF ACRYLIC ACID AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2017-05-04 US disclosed
EP-3160965-A1 3-SUBSTITUTED 2-AMINO-INDOLE DERIVATIVES Takeda Pharmaceutical Company Limited (JP) 2017-05-03 EP disclosed
EP-3161000-A2 DUAL PDGF/VEGF ANTAGONISTS Kodiak Sciences Inc. (US) 2017-05-03 EP disclosed
EP-3160949-A1 ENZYME INTERACTING AGENTS Monash University (AU) 2017-05-03 EP disclosed
EP-3160955-A1 1,3-SUBSTITUTED 2-AMINOINDOLE DERIVATIVES AND ANALOGUES USEFUL IN THE TREATMENT OR PREVENTION OF DIABETES MELLITUS, OBESITY AND INFLAMMATORY BOWEL DISEASE Takeda Pharmaceutical Company Limited (JP) 2017-05-03 EP disclosed
EP-3160956-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Celgene Quanticel Research, Inc. (US) 2017-05-03 EP disclosed
US-9637487-B2 Purinone compounds as kinase inhibitors PHARMACYCLICS LLC (US) 2017-05-02 US disclosed
US-9637478-B2 Antiviral compounds and uses thereof ABBVIE INC. (US) 2017-05-02 US disclosed
US-20170114075-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2017-04-27 US disclosed
US-20170112833-A1 Tyrosine Kinase Inhibitor And Uses Thereof Xuanzhu Pharma Co., Ltd. (CN) 2017-04-27 US disclosed
US-20170114060-A1 NOVEL EFFECTIVE ANTIVIRAL COMPOUNDS AND METHODS USING SAME NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2017-04-27 US disclosed
US-20170114055-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. 2017-04-27 US disclosed
US-20170114024-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 QUANTIEL PHARMACEUTICALS, INC. 2017-04-27 US disclosed
US-20170114070-A1 INHIBITORS OF THE WNT SIGNALLING PATHWAYS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-04-27 US disclosed
US-20170112843-A1 COMPOUNDS AND METHODS FOR INDUCING CHONDROGENESIS THE SCRIPPS RESEARCH INSTITUTE 2017-04-27 US disclosed
US-20170114074-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2017-04-27 US disclosed
WO-2017070256-A2 METHOD FOR SCREENING INHIBITORS OF RAS ARAXES PHARMA LLC (US) 2017-04-27 WO disclosed
WO-2017070448-A1 2-BETA-NAPHTHYL-ACETIC ACID ANALOGS AS AKR1C3 INHIBITORS AND METHODS OF USING SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2017-04-27 WO disclosed
EP-3157933-A2 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS Gilead Sciences, Inc. (US) 2017-04-26 EP disclosed
EP-3157916-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD Pharmaceuticals, Inc. (US) 2017-04-26 EP disclosed
EP-3159344-A1 AMINO PYRANOID RING DERIVATIVE AND COMPOSITION AND USE THEREOF Sichuan Haisco Pharmaceutical Co., Ltd. (CN) 2017-04-26 EP disclosed
US-9630975-B2 Thiophene derivatives TIANJIN HEMAY BIO-TECH CO., LTD. (CN) 2017-04-25 US disclosed
US-9630979-B2 Inhibitors of monoacylglycerol lipase and methods of their use INFINITY PHARMACEUTICALS, INC. (US) 2017-04-25 US disclosed
WO-2017066454-A2 COMPOSITIONS AND METHODS FOR REDUCING ICE CRYSTAL FORMATION X-THERMA, INC. (US) 2017-04-20 WO disclosed
US-20170107245-A1 GEMCITABINE PRODRUGS AND USES THEREOF BoYen Therapeutics, Inc. (TW) 2017-04-20 US disclosed
US-20170107229-A1 SUBSTITUTED TETRAHYDROPYRIDOTHIENOPYRIMIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-04-20 US disclosed
US-20170107212-A1 NOVEL COMPOUNDS Bayer Pharma AG (DE) 2017-04-20 US disclosed
US-20170107440-A1 LUBRICATING COMPOSITIONS AND METHODS FOR THE USE THEREOF JPMORGAN CHASE BANK, N.A. 2017-04-20 US disclosed
EP-3154537-A1 ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS AND USES THEREOF Merck Sharp & Dohme Corp. (US) 2017-04-19 EP disclosed
EP-3036228-B1 NEW 6-ALKYNYL PYRIDINE COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2017-04-19 EP disclosed
EP-3036235-B1 NEW BIS-AMIDO PYRIDINES BOEHRINGER INGELHEIM INT (DE) 2017-04-19 EP disclosed
EP-2791184-B1 PROCESS FOR REMOVING THIOCARBONYLTHIO GROUPS FROM RAFT POLYMERS COMMW SCIENT IND RES ORG (AU) 2017-04-19 EP disclosed
EP-3156387-A1 INDENE DERIVATIVES AS PHARMACEUTICAL AGENTS Aquinox Pharmaceuticals (Canada) Inc. (CA) 2017-04-19 EP disclosed
US-9624229-B2 Pyrimidine-2-amine compounds and their use as inhibitors of JAK kinases RIGEL PHARMACEUTICALS, INC. (US) 2017-04-18 US disclosed
US-9622472-B2 Molecules that induce disease resistance in plants THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-04-18 US disclosed
US-9624228-B2 Inhibitors of ERK and methods of use KURA ONCOLOGY, INC. (US) 2017-04-18 US disclosed
US-9624224-B2 Inhibitors of Bruton's tyrosine kinase PHARMACYCLICS LLC (US) 2017-04-18 US disclosed
US-20170101388-A1 C-GLYCOSIDE DERIVATIVE Xuanzhu Pharma Co., Ltd. (CN) 2017-04-13 US disclosed
WO-2017062823-A1 THERAPEUTIC CANCER TREATMENTS BASED ON TP53 GENE MUTATIONS THE WISTAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2017-04-13 WO disclosed
WO-2017060431-A1 SPIRO[3H-INDOLE-3,2´-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-04-13 WO disclosed
EP-3153023-A1 BENZOXAZOLE KINASE INHIBITORS AND METHODS OF USE Intellikine, LLC (US) 2017-04-12 EP disclosed
US-9617277-B2 Polymeric materials COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2017-04-11 US disclosed
US-9617242-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-04-11 US disclosed
US-20170096391-A1 NOVEL LACTAMS BIOSIGNAL LIMITED (AU) 2017-04-06 US disclosed
US-20170095471-A1 Methods of Treating Chronic Lymphocytic Leukemia and Small Lymphocytic Leukemia Using a BTK Inhibitor ACERTA PHARMA B.V. (NL) 2017-04-06 US disclosed
US-20170095554-A1 AMINO ACID AND PEPTIDE CONJUGATES AND CONJUGATION PROCESS AUCKLAND UNISERVICES LIMITED (NZ) 2017-04-06 US disclosed
EP-3149003-A1 BENZOTHIADIAZOLAMINES Bayer Pharma Aktiengesellschaft (DE) 2017-04-05 EP disclosed
EP-3150203-A1 COMPOUNDS WITH (1E,6E)-1,7-BIS-(3,4- DIMETHOXYPHENYL)-4,4-DISSTITUTED-HEPA-1,6-DIENE-3,5-DI-ONE STRUCTURAL SCAFFOLD,THEIR BIOLOGICAL ACTIVITY, AND USES THEREOF Allianz Pharmascience Ltd (TW) 2017-04-05 EP disclosed
EP-3008062-B1 PRODRUG DERIVATIVES OF SUBSTITUTED TRIAZOLOPYRIDINES Bayer Pharma AG (DE) 2017-04-05 EP disclosed
EP-2766359-B9 HETEROCYCLIC COMPOUNDS AND USE THEREOF AS MODULATORS OF TYPE III RECEPTOR TYROSINE KINASES AMBIT BIOSCIENCES CORP (US) 2017-04-05 EP disclosed
EP-3150609-A1 PROCESS FOR PREPARING CERTAIN CHEMICAL ENTITIES Intellikine, LLC (US) 2017-04-05 EP disclosed
EP-2809708-B1 HALOGENATED ORGANOSILICON ELECTROLYTES, METHODS OF USING THEM, AND ELECTROCHEMICAL DEVICES CONTAINING THEM SILATRONIX INC (US) 2017-04-05 EP disclosed
EP-3150617-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS Achaogen, Inc. (US) 2017-04-05 EP disclosed
US-9611252-B2 Therapeutic inhibitory compounds LIFESCI PHARMACEUTICALS, INC. (BB) 2017-04-04 US disclosed
US-9611186-B2 Synthesis of high caloric fuels and chemicals via ketene and diketene intermediates Pioneer Energy (US) 2017-04-04 US disclosed
US-9611271-B2 C20′ urea derivatives of vinca alkaloids SCRIPPS RESEARCH INSTITUTE (US) 2017-04-04 US disclosed
US-9611221-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-04-04 US disclosed
WO-2017053886-A2 METHOD OF SCREENING FOR AGENTS FOR DIFFERENTIATING STEM CELLS MINERVA BIOTECHNOLOGIES CORPORATION (US) 2017-03-30 WO disclosed
WO-2017053192-A1 BIOMARKERS OF RESPONSE TO HIF-2-ALPHA INHIBITION IN CANCER AND METHODS FOR THE USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-03-30 WO disclosed
US-20170088523-A1 BENZIMIDAZOLE DERIVATIVES AND USES THEREOF PELOTON THERAPEUTICS, INC. 2017-03-30 US disclosed
EP-2389395-B1 RAFT POLYMERISATION COMMW SCIENT IND RES ORG (AU) 2017-03-29 EP disclosed
EP-2621923-B1 N-HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT FOR THE TREATMENT OF PARASITIC DISEASES INTERVET INT BV (NL) 2017-03-29 EP disclosed
EP-3147285-A2 PURINONE COMPOUNDS AS KINASE INHIBITORS Pharmacyclics, Inc. (US) 2017-03-29 EP disclosed
EP-3147281-A1 QUINAZOLINE DERIVATIVES AS RAF KINASE MODULATORS AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2017-03-29 EP disclosed
US-9604989-B2 Imidazopyridazines as Akt kinase inhibitors BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-03-28 US disclosed
US-9606440-B2 Lithographically produced features THE UNIVERSITY OF QUEENSLAND (AU) 2017-03-28 US disclosed
US-9604961-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-03-28 US disclosed
US-9605003-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-03-28 US disclosed
WO-2017046304-A1 NO-DONORS FOR THE TREATMENT OF CEREBROVASCULAR VASOSPASMS AFTER BRAIN HEMORRHAGE EHLERT ANGELIKA (DE) 2017-03-23 WO disclosed
WO-2017046746-A1 THERAPEUTIC COMBINATIONS OF A BTK INHIBITOR AND A GITR BINDING MOLECULE, A 4-1BB AGONIST, OR AN OX40 AGONIST ACERTA PHARMA B.V. (NL) 2017-03-23 WO disclosed
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EP-3143015-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD Pharmaceuticals, Inc. (US) 2017-03-22 EP disclosed
EP-2678334-B1 ANTI-VIRAL COMPOUNDS ABBVIE BAHAMAS LTD (BS) 2017-03-22 EP disclosed
EP-3004092-B1 SUBSTITUTED TRIAZOLOPYRIDINES Bayer Pharma AG (DE) 2017-03-22 EP disclosed
EP-2714692-B1 SUBSTITUTED AMINOIMIDAZOPYRIDAZINES BAYER IP GMBH (DE) 2017-03-22 EP disclosed
CN-106537124-A Detection of acrylic acid 新加坡科技研究局 2017-03-22 CN disclosed
CN-106536503-A Tyrosine kinase inhibitor and uses thereof 山东轩竹医药科技有限公司 2017-03-22 CN disclosed
US-9598439-B2 Purification of rapamycin derivatives using temperature induced phase separation BIOSENSORS INTERNATIONAL GROUP, LTD. (BM) 2017-03-21 US disclosed
US-9598372-B2 Bromodomain inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-03-21 US disclosed
US-20170073340-A1 SUBSTITUTED CYCLOPENTANES, TETRAHYDROFURANES AND PYRROLIDINES AS OREXIN RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-03-16 US disclosed
WO-2017044659-A1 COMPOUNDS AND FORMULATIONS FOR TREATING OPHTHALMIC DISEASES VIEWPOINT THERAPEUTICS, INC. (US) 2017-03-16 WO disclosed
WO-2017041139-A1 LYMPH DIRECTING PRODRUGS MONASH UNIVERSITY (AU) 2017-03-16 WO disclosed
US-20170071962-A1 Therapeutic Combinations of a Proteasome Inhibitor and a BTK Inhibitor ACERTA PHARMA BV (NL) 2017-03-16 US disclosed
WO-2017044043-A1 PROCESS FOR DIRECT AMIDATION OF AMINES VIA RH(I)-CATALYZED ADDITION OF BOROXINES AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2017-03-16 WO disclosed
EP-3140304-A1 BENZIMIDAZOLE DERIVATIVES Boehringer Ingelheim International GmbH (DE) 2017-03-15 EP disclosed
EP-2598660-B1 COMPOSITIONS FOR STABILIZING DNA, RNA AND PROTEINS IN BLOOD AND OTHER BIOLOGICAL SAMPLES DURING SHIPPING AND STORAGE AT AMBIENT TEMPERATURES BIOMATRICA INC (US) 2017-03-15 EP disclosed
EP-2663309-B1 PROCESSES FOR PREPARING ISOQUINOLINONES AND SOLID FORMS OF ISOQUINOLINONES INFINITY PHARMACEUTICALS INC (US) 2017-03-15 EP disclosed
US-9593096-B2 α7 nicotinic acetylcholine receptor modulators and uses thereof-III MERCK SHARP & DOHME CORP. (US) 2017-03-14 US disclosed
US-9593106-B2 Piperidin-1-yl and azepin-1-yl carboxylates as muscarinic M4 receptor agonists HEPTARES THERAPEUTICS LIMITED (GB) 2017-03-14 US disclosed
US-20170066744-A1 1,2-SUBSTITUTED CYCLOPENTANES AS OREXIN RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-03-09 US disclosed
US-20170066739-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE PHARMACEUTICALS INC (US) 2017-03-09 US disclosed
US-20170065575-A1 NAMPT INHIBITORS ABBVIE INC (US) 2017-03-09 US disclosed
US-20170066777-A1 ASYMMETRIC SYNTHESES FOR SPIRO-OXINDOLE COMPOUNDS USEFUL AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2017-03-09 US disclosed
WO-2017035570-A1 AMPHIPHILIC RAFT AGENT COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2017-03-09 WO disclosed
EP-3137169-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Celgene Quanticel Research, Inc. (US) 2017-03-08 EP disclosed
CN-106488919-A 3-substituted 2-aminoindole derivatives 武田药品工业株式会社 2017-03-08 CN disclosed
US-9586978-B2 Anti-viral compounds ABBVIE INC. (US) 2017-03-07 US disclosed
US-9586939-B2 Quinazoline derivative as tyrosine-kinase inhibitor, preparation method therefor and application thereof Xuanzhu Pharma Co., Ltd. (CN) 2017-03-07 US disclosed
US-9587104-B2 Release media THE UNIVERSITY OF QUEENSLAND (AU) 2017-03-07 US disclosed
US-9586958-B2 Prodrug derivatives of substituted triazolopyridines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-03-07 US disclosed
US-9586902-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-03-07 US disclosed
US-9586901-B2 Lactams UNILEVER PLC (GB) 2017-03-07 US disclosed
WO-2017033113-A1 THERAPEUTIC COMBINATIONS OF A MEK INHIBITOR AND A BTK INHIBITOR ACERTA PHARMA B.V. (NL) 2017-03-02 WO disclosed
US-20170057976-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2017-03-02 US disclosed
EP-2621903-B1 N-HETEROARYL COMPOUNDS INTERVET INT BV (NL) 2017-03-01 EP disclosed
EP-3134410-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL Hydra Biosciences, Inc. (US) 2017-03-01 EP disclosed
CN-104168768-B The method of preparation Cgrp receptor antagonist 默沙东公司 2017-03-01 CN disclosed
US-9580416-B2 Inhibitors of Bruton's tyrosine kinase PHARMACYCLICS LLC (US) 2017-02-28 US disclosed
US-20170050966-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL MERCK & CO., INC. 2017-02-23 US disclosed
US-20170049722-A1 ALKOXY COMPOUNDS FOR DISEASE TREATMENT ACUCELA INC. 2017-02-23 US disclosed
US-20170050970-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS, INC. 2017-02-23 US disclosed
US-20170051278-A1 METHODS FOR TREATING PROGEROID LAMINOPATHIES USING OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA SAREPTA THERAPEUTICS, INC. 2017-02-23 US disclosed
US-20170050968-A1 BROMODOMAIN INHIBITOR CELGENE QUANTICEL RESEARCH, INC. 2017-02-23 US disclosed
CN-106432557-A HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS 科迪亚科学企业公司 2017-02-22 CN disclosed
CN-104508049-B Silicone ligands for stabilizing quantum dot films 纳米系统公司 2017-02-22 CN disclosed
US-9573930-B2 Inhibitors of lysine specific demethylase-1 CELGENE QUANTICEL RESEARCH, INC. (US) 2017-02-21 US disclosed
US-20170042891-A1 AXL INHIBITORS FOR USE IN COMBINATION THERAPY FOR PREVENTING, TREATING OR MANAGING METASTATIC CANCER RIGEL PHARMACEUTICALS, INC. 2017-02-16 US disclosed
WO-2017025493-A1 QUINOLINE EZH2 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-02-16 WO disclosed
WO-2017025814-A1 METHODS OF TREATING CANCERS, IMMUNE AND AUTOIMMUNE DISEASES, AND INFLAMMATORY DISEASES BASED ON BTK OCCUPANCY AND BTK RESYNTHESIS RATE ACERTA PHARMA B.V. (NL) 2017-02-16 WO disclosed
EP-3128996-A1 Novel 7-Dehydrocholesterol Derivatives and Methods Using Same Women and Infants Hospital of Rhode Island Inc. (US) 2017-02-15 EP disclosed
EP-3129380-A1 SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE DERIVATIVES AND THEIR USE AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-02-15 EP disclosed
CN-106414480-A POLYMYXIN DERIVATIVES AS ANTIMICROBIAL COMPOUNDS 莫纳什大学 2017-02-15 CN disclosed
CN-104109168-B Tetra-cyclo-kinase inhibitor 山东轩竹医药科技有限公司 2017-02-15 CN disclosed
US-20170035881-A1 Therapeutic Combinations of an IRAK4 Inhibitor and a BTK Inhibitor ACERTA PHARMA BV (NL) 2017-02-09 US disclosed
WO-2017023912-A1 2,4,6-TRIALKOXYSTRYL ARYL SULFONES, SULFONAMIDES AND CARBOXAMIDES, AND METHODS OF PREPARATION AND USE TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2017-02-09 WO disclosed
US-20170035756-A1 METHODS OF BLOCKING THE CXCR-4/SDF-1 SIGNALING PATHWAY WITH INHIBITORS OF BRUTON'S TYROSINE KINASE ACERTA PHARMA B.V. (NL) 2017-02-09 US disclosed
US-20170037028-A1 GLUCOSE TRANSPORT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-02-09 US disclosed
WO-2017024255-A1 NICOTINAMIDE MONONUCLEOTIDE DERIVATIVES AND THEIR USES METROBIOTECH, LLC (US) 2017-02-09 WO disclosed
US-20170037010-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. 2017-02-09 US disclosed
EP-3126376-A1 POLYMYXIN DERIVATIVES AS ANTIMICROBIAL COMPOUNDS Monash University (AU) 2017-02-08 EP disclosed
EP-2978758-B1 DIHYDROQUINAZOLINONE ANALOGUES AS BRD4 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2017-02-08 EP disclosed
EP-3126005-A1 NOVEL ANTIVIRAL COMPOUNDS AND METHODS USING SAME The Trustees Of The University Of Pennsylvania (US) 2017-02-08 EP disclosed
EP-2978757-B1 INDOLINONE ANALOGUES AS BRD4 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2017-02-08 EP disclosed
US-9562029-B2 C-glycoside derivatives Xuanzhu Pharma Co., Ltd. (CN) 2017-02-07 US disclosed
US-9562025-B2 Compounds with (1E, 6E)-1,7-Bis-(3,4-dimethoxyphenyl)-4-4-distributed-hepta-1,6-diene-3,5-dione structural scaffold, their biological activity, and uses thereof ALLIANZ PHARMASCIENCE LTD. (TW) 2017-02-07 US disclosed
US-20170029433-A1 TRANSFER HYDROGENATION OF CYCLOPAMINE ANALOGS ROYALTY SECURITY, LLC 2017-02-02 US disclosed
US-20170029459-A1 Novel 7-Dehydrocholesterol Derivatives and Methods Using Same WOMEN & INFANTS HOSPITAL OF RHODE ISLAND 2017-02-02 US disclosed
WO-2017015720-A1 FIBROTIC TREATMENT MONASH UNIVERSITY (AU) 2017-02-02 WO disclosed
US-20170029490-A1 SULFONAMIDE-CONTAINING LINKAGE SYSTEMS FOR DRUG CONJUGATES ZYMEWORKS INC. (CA) 2017-02-02 US disclosed
US-20170027172-A1 USE OF SUBSTITUTE OXO TETRAHYDROQUINOLINE SULFONAMIDES OR SALTS THEREOF FOR RAISING STRESS TOLERANCE OF PLANTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2017-02-02 US disclosed
US-20170029478-A1 High Molecular Weight, Post-Translationally Modified Protein Brushes MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2017-02-02 US disclosed
US-20170029441-A1 AMIDO-SUBSTITUTED IMIDAZOPYRIDAZINES USEFUL IN THE TREATMENT OF HYPER-PROLIFERATIVE AND/OR ANGIOGENESIS DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-02-02 US disclosed
US-20170029406-A1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS, INC. 2017-02-02 US disclosed
US-9556181-B2 Substituted pyrazolopyrimidinylamino-indazoles BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-01-31 US disclosed
US-9555022-B2 Substituted triazolopyridines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-01-31 US disclosed
US-20170022189-A1 AMINOPYRIDINE DERIVATIVES AS TAM FAMILY KINASE INHIBITORS SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2017-01-26 US disclosed
WO-2017015562-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS AND THEIR USE AS INHIBITORS OF G12C MUTANT KRAS, HRAS AND/OR NRAS PROTEINS ARAXES PHARMA LLC (US) 2017-01-26 WO disclosed
US-20170022247-A1 WITHANOLIDES USEFUL FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES IMSTAR THERAPEUTICS INC. (CA) 2017-01-26 US disclosed
US-20170022184-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC 2017-01-26 US disclosed
US-20170020859-A1 6-ALKYNYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM INT (DE) 2017-01-26 US disclosed
US-20170022180-A1 SUBSTITUTED 3-PHENYLPROPYLAMINE DERIVATIVES FOR THE TREATMENT OF OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. 2017-01-26 US disclosed
EP-3119397-A1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF PI3K-GAMMA MEDIATED DISORDERS Infinity Pharmaceuticals, Inc. (US) 2017-01-25 EP disclosed
EP-2212328-B1 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF CHOONGWAE PHARMA CORP (KR) 2017-01-25 EP disclosed
EP-3121208-A1 POLYMERIC MATERIALS Commonwealth Scientific and Industrial Research Organisation (AU) 2017-01-25 EP disclosed
EP-3119759-A1 NOVEL COMPOUNDS Bayer Pharma Aktiengesellschaft (DE) 2017-01-25 EP disclosed
EP-3119787-A1 INHIBITORS OF THE WNT SIGNALLING PATHWAYS Bayer Pharma Aktiengesellschaft (DE) 2017-01-25 EP disclosed
US-9549947-B2 Pharmaceutical compositions for treating hyperkalemia ARDELYX, INC. (US) 2017-01-24 US disclosed
US-9549932-B2 2-(morpholin-4-yl)-1,7-naphthyridines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-01-24 US disclosed
US-20170015671-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC 2017-01-19 US disclosed
US-20170015631-A1 PKM2 MODULATORS AND METHODS FOR THEIR USE SUMITOMO PHARMA ONCOLOGY, INC. 2017-01-19 US disclosed
WO-2017009650-A1 CYANOPYRROLIDINES AS DUB INHIBITORS FOR THE TREATMENT OF CANCER MISSION THERAPEUTICS LIMITED (GB) 2017-01-19 WO disclosed
WO-2017011323-A1 SMALL MOLECULE INHIBITORS OF THE MCL-1 ONCOPROTEIN AND USES THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2017-01-19 WO disclosed
EP-2411352-B1 ANTIVIRAL COMPOUNDS AND USES THEREOF ABBVIE INC (US) 2017-01-18 EP disclosed
US-9546180-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-01-17 US disclosed
US-9545425-B2 Pharmaceutical compositions for treating hyperkalemia ARDELYX, INC. (US) 2017-01-17 US disclosed
US-20170007710-A1 TARGETED DRUG PHOSPHORYLCHOLINE POLYMER CONJUGATES KODIAK SCIENCES INC. 2017-01-12 US disclosed
EP-1689706-B1 ALPHA, BETA-UNSATURATED SULFOXIDES FOR TREATING PROLIFERATIVE DISORDERS TEMPLE UNIV - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2017-01-11 EP disclosed
US-9540410-B2 Gemcitabine prodrugs and uses thereof BoYen Therapeutics, Inc. (TW) 2017-01-10 US disclosed
US-9540353-B2 SHIP1 modulators and methods related thereto AQUINOX PHARMACEUTICALS (CANADA) INC. (CA) 2017-01-10 US disclosed
US-9540385-B2 Pyrrolopyrimidine compounds as kinase inhibitors PHARMACYCLICS LLC (US) 2017-01-10 US disclosed
US-9540392-B2 Thienopyrimidines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-01-10 US disclosed
WO-2017001924-A1 THERAPEUTIC INHIBITORY COMPOUDS LIFESCI PHARMACEUTICALS, INC. (BB) 2017-01-05 WO disclosed
WO-2017003822-A1 NOVEL BREATHING CONTROL MODULATING COMPOUNDS, AND METHODS OF MAKING AND USING SAME GALLEON PHARMACEUTICALS, INC. (US) 2017-01-05 WO disclosed
WO-2017001926-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC (BB) 2017-01-05 WO disclosed
WO-2017004543-A1 ARYL SULFONAMIDE COMPOUNDS AS CARBONIC ANHYDRASE INHIBITORS AND THEIR THERAPEUTIC USE SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2017-01-05 WO disclosed
WO-2017001936-A2 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2017-01-05 WO disclosed
US-20170003293-A1 ENCODED CHROMOPHORIC POLYMER PARTICLES AND METHODS OF USE THEREOF UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION 2017-01-05 US disclosed
EP-2819996-B1 6-ALKYNYL PYRIDINES AS SMAC MIMETICS BOEHRINGER INGELHEIM INT (DE) 2017-01-04 EP disclosed
US-9533991-B2 Inhibitors of Bruton's tyrosine kinase PHARMACYCLICS LLC (US) 2017-01-03 US disclosed
US-9533999-B2 Fused thiazin-3-ones as KCA3.1 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-01-03 US disclosed
WO-2016207104-A1 ANTIBODY DRUG CONJUGATES OF KINESIN SPINDEL PROTEIN (KSP) INHIBITORS WITH ANTI-B7H3-ANTIBODIES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-12-29 WO disclosed
WO-2016207103-A1 ANTIBODY DRUG CONJUGATES OF KINESIN SPINDEL PROTEIN (KSP) INHIBITORS WITH ANTI-B7H3-ANTIBODIES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-12-29 WO disclosed
US-20160376522-A1 IONIC LIQUID SYSTEMS THE PROCTER & GAMBLE COMPANY 2016-12-29 US disclosed
WO-2016207089-A1 ANTIBODY DRUG CONJUGATES (ADCS) AND ANTIBODY PRODRUG CONJUGATES (APDCS) WITH ENZYMATICALLY CLEAVABLE GROUPS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-12-29 WO disclosed
US-20160375026-A1 PYRROLOPYRIMIDINE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS, INC. 2016-12-29 US disclosed
WO-2016210352-A2 SYNTHESIS OF PHEROMONES AND OTHER OXY-FUNCTIONALIZED PRODUCTS VIA ENZYMATIC HYDROXYLATION OF CARBOXYLIC ACIDS PROVIVI, INC. (US) 2016-12-29 WO disclosed
US-20160376256-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-12-29 US disclosed
US-20160376587-A1 FUNCTIONALLY-MODIFIED OLIGONUCLEOTIDES AND SUBUNITS THEREOF JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2016-12-29 US disclosed
WO-2016207094-A1 ANTIBODY DRUG CONJUGATES OF KINESIN SPINDEL PROTEIN (KSP) INHIBITORS WITH ANTI-TWEAKR-ANTIBODIES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-12-29 WO disclosed
US-9527847-B2 Treatment of lupus, fibrotic conditions, and inflammatory myopathies and other disorders using PI3 kinase inhibitors INFINITY PHARMACEUTICALS, INC. (US) 2016-12-27 US disclosed
US-9527829-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2016-12-27 US disclosed
US-20160368905-A1 ANTIVIRAL COMPOUNDS AND USES THEREOF ABBOTT LABORATORIES 2016-12-22 US disclosed
US-20160368924-A1 PURINONE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS, INC. 2016-12-22 US disclosed
US-20160368942-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS Cipla USA, Inc. 2016-12-22 US disclosed
US-20160367962-A1 ZIF-CONTAINING ADSORBENT MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2016-12-22 US disclosed
US-20160368874-A1 1,4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON LLC 2016-12-22 US disclosed
WO-2016202898-A1 GLUCOSE TRANSPORT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-12-22 WO disclosed
WO-2016205590-A1 SUBSTITUTED 4-BENZYL AND 4-BENZOYL PIPERIDINE DERIVATIVES CEPHALON, INC. (US) 2016-12-22 WO disclosed
WO-2016202935-A1 GLUCOSE TRANSPORT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-12-22 WO disclosed
US-20160368893-A1 CYCLIC SULFONE AND SULFOXIMINE ANALOGS AND USES THEREOF Peloton Therapeutics ,Inc. 2016-12-22 US disclosed
EP-3105209-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2016-12-21 EP disclosed
EP-1976828-B1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS INC (US) 2016-12-21 EP disclosed
EP-2705181-B1 COMBINATION PHARMACEUTICAL COMPOSITIONS AND USES THEREOF INTELLIKINE LLC (US) 2016-12-21 EP disclosed
EP-3105210-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2016-12-21 EP disclosed
US-9522146-B2 Substituted Isoquinolin-1(2H)-one compounds, compositions, and methods thereof INTELLIKINE LLC (US) 2016-12-20 US disclosed
US-9522876-B2 Cytotoxic and anti-mitotic compounds, and methods of using the same ZYMEWORKS INC. 2016-12-20 US disclosed
WO-2016197187-A1 VERSATILE RAFT AGENT COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2016-12-15 WO disclosed
WO-2016200840-A1 MONO AND BICYCLIC RING BORONIC ACID, ESTER AND SALT COMPOUNDS AS INHIBITORS OF P97 COMPLEX CLEAVE BIOSCIENCES, INC. (US) 2016-12-15 WO disclosed
WO-2016200956-A1 PROCESS FOR THE PREPARATION OF POLYURETHANE SOLUTIONS BASED ON SILICON-POLYCARBONATE DIOLS MAGUIRE FRANCIS P (US) 2016-12-15 WO disclosed
US-20160362390-A1 TRICYCLIC INHIBITORS OF HIF-2-ALPHA AND USES THEREOF PELOTON THERAPEUTICS, INC. 2016-12-15 US disclosed
US-20160362405-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORP (US) 2016-12-15 US disclosed
US-20160362404-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-12-15 US disclosed
EP-3102207-A1 2,4,5-TRI-SUBSTITUTED AZOLE-BASED CASEIN KINASE 1 INHIBITORS AS INDUCERS FOR CARDIOMYOGENESIS Agency For Science, Technology And Research (SG) 2016-12-14 EP disclosed
EP-2265607-B1 PYRIMIDINE-2-AMINE COMPOUNDS AND THEIR USE AS INHIBITORS OF JAK KINASES RIGEL PHARMACEUTICALS INC (US) 2016-12-14 EP disclosed
US-20160355503-A1 NITROGEN HEXACYCLE COMPOUNDS AS INHIBITORS OF p97 COMPLEX CLEAVE BIOSCIENCES, INC. 2016-12-08 US disclosed
WO-2016196776-A2 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC. (US) 2016-12-08 WO disclosed
WO-2016197027-A1 METHODS AND COMPOSITIONS FOR INHIBITING THE INTERACTION OF MENIN WITH MLL PROTEINS KURA ONCOLOGY, INC. (US) 2016-12-08 WO disclosed
WO-2016195776-A1 METHODS AND COMPOSITIONS FOR INHIBITING THE INTERACTION OF MENIN WITH MLL PROTEINS KURA ONCOLOGY, INC. (US) 2016-12-08 WO disclosed
WO-2016193284-A1 PESTICIDALLY ACTIVE OXIME AND HYDRAZONE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2016-12-08 WO disclosed
US-20160355498-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS, INC. 2016-12-08 US disclosed
WO-2016193680-A1 COMBINATION THERAPY WITH AXL INHIBITOR AND IMMUNE CHECKPOINT MODULATOR OR ONCOLYTIC VIRUS BERGENBIO AS (NO) 2016-12-08 WO disclosed
US-20160355539-A1 SELECTIVE SOLVENT FREE PHOSPHORYLATION CHROMADEX, INC. (US) 2016-12-08 US disclosed
WO-2016196897-A1 METHODS AND COMPOUNDS FOR TREATMENT OF LYMPHOCYTE-RELATED DISEASES AND CONDITIONS SAREPTA THERAPEUTICS, INC. (US) 2016-12-08 WO disclosed
EP-3099682-A1 AMINO-SUBSTITUTED ISOTHIAZOLES Bayer Pharma Aktiengesellschaft (DE) 2016-12-07 EP disclosed
EP-2355853-B1 BIODEGRADABLE POLYMER - BIOACTIVE MOIETY CONJUGATES POLYACTIVA PTY LTD (AU) 2016-12-07 EP disclosed
US-9512126-B2 Substituted imidazopyridazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-12-06 US disclosed
US-20160347714-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2016-12-01 US disclosed
US-20160346318-A1 COMPOSITIONS AND METHODS FOR TREATING HYPERKALEMIA ARDELYX, INC. 2016-12-01 US disclosed
US-20160347733-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2016-12-01 US disclosed
WO-2016191612-A2 HEMOPROTEIN CATALYSTS FOR IMPROVED ENANTIOSELECTIVE ENZYMATIC SYNTHESIS OF TICAGRELOR CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2016-12-01 WO disclosed
EP-2773614-B1 SUBSTITUTED 4.CYAN-3-(PHENYL-4-(PYRIDIN-3-YL) BUTANOATES, METHOD FOR THEIR PRODUCTION AND THEIR USE AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER IP GMBH (DE) 2016-11-30 EP disclosed
CN-104039762-B Nampt inhibitor ABBVIE INC. (US) 2016-11-30 CN disclosed
US-20160339418-A1 NANO-TO-NANO FE/PPM Pd CATALYSIS OF CROSS-COUPLING REACTIONS IN WATER LIPSHUTZ BRUCE H (US) 2016-11-24 US disclosed
US-20160341736-A1 WATER SOLUBLE FLUORESCENT OR COLORED DYES AND METHODS FOR THEIR USE SONY CORPORATION (JP) 2016-11-24 US disclosed
US-20160338342-A1 COMPOSITIONS FOR STABILIZING DNA, RNA AND PROTEINS IN BLOOD AND OTHER BIOLOGICAL SAMPLES DURING SHIPPING AND STORAGE AT AMBIENT TEMPERATURES EXACT SCIENCES CORPORATION 2016-11-24 US disclosed
EP-3094687-A2 WATER SOLUBLE FLUORESCENT OR COLORED DYES Sony Corporation (JP) 2016-11-23 EP disclosed
CN-106164064-A Substituted cyclopentane, oxolane and pyrrolidine as orexin receptor antagonists 武田药品工业株式会社 2016-11-23 CN disclosed
CN-106164047-A 1,2 substituted cyclopentanes as orexin receptor antagonists 武田药品工业株式会社 2016-11-23 CN disclosed
US-9499521-B2 Inhibitors of cellular necrosis and related methods PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2016-11-22 US disclosed
US-9500640-B2 Alzheimer's disease assay in a living patient PAIN THERAPEUTICS, INC. (US) 2016-11-22 US disclosed
US-9499693-B2 Clean polycarbonate material for use in hard disk drive and semiconductor applications SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2016-11-22 US disclosed
US-9499547-B2 Amino-substituted imidazopyridazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-11-22 US disclosed
US-20160332970-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. 2016-11-17 US disclosed
WO-2016183185-A1 ULTRA BRIGHT DIMERIC OR POLYMERIC DYES SONY CORPORATION (JP) 2016-11-17 WO disclosed
US-20160332990-A1 FUSED PYRIMIDINES AS INHIBITORS OF P97 COMPLEX CLEAVE BIOSCIENCES, INC. (US) 2016-11-17 US disclosed
WO-2016183278-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD PHARMACEUTICALS, INC. (US) 2016-11-17 WO disclosed
WO-2016179645-A1 4H-PYRAN COMPOUNDS AS INSULIN-REGULATED AMINOPEPTIDASE (IRAP) INHIBITORS MONASH UNIVERSITY (AU) 2016-11-17 WO disclosed
WO-2016183586-A1 HIGH MOLECULAR WEIGHT, POST-TRANSLATIONALLY MODIFIED PROTEIN BRUSHES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2016-11-17 WO disclosed
US-20160331800-A1 BOTULINUM NEUROTOXIN-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING REGENERON PHARMACEUTICALS, INC. 2016-11-17 US disclosed
US-20160333048-A1 Antimicrobial Peptidomimetics AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2016-11-17 US disclosed
EP-2665775-B1 UV STABILIZATION OF ISOSORBIDE POLYCARBONATES SABIC GLOBAL TECHNOLOGIES BV (NL) 2016-11-16 EP disclosed
EP-3092242-A1 AMIDO-SUBSTITUTED IMIDAZOPYRIDAZINES USEFUL IN THE TREATMENT OF HYPER-PROLIFERATIVE AND/OR ANGIOGENESIS DISORDERS Bayer Pharma Aktiengesellschaft (DE) 2016-11-16 EP disclosed
US-9493799-B2 In vivo and in vitro olefin cyclopropanation catalyzed by heme enzymes CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2016-11-15 US disclosed
US-9493419-B2 Quinoline derivatives as anti-cancer agents THE HONG KONG POLYTECHNIC UNIVERSITY (HK) 2016-11-15 US disclosed
US-9493432-B2 Cyclopentylbenzamide derivatives and their use for the treatment of psychotic and cognitive disorders TAKEDA PHARMACEUTICALS COMPANY LIMITED (JP) 2016-11-15 US disclosed
US-9493482-B2 Compounds and methods for preventing or treating sensory hair cell death UNIVERSITY OF WASHINGTON (US) 2016-11-15 US disclosed
WO-2016179349-A1 CXCR4 CHEMOKINE RECEPTOR MODULATORS NORTHWESTERN UNIVERSITY (US) 2016-11-10 WO disclosed
US-20160324160-A1 SYNERGISTIC BENZOXABOROLE-CONTAINING ANTI-FUNGICIDAL COMPOSITION THE PENN STATE RESEARCH FOUNDATION 2016-11-10 US disclosed
US-20160326186-A1 COMPOUNDS AND METHODS FOR PREVENTING, TREATING AND/OR PROTECTING AGAINST SENSORY HAIR CELL DEATH FRED HUTCHINSON CANCER CENTER 2016-11-10 US disclosed
EP-2947072-B1 1-(3-(6,7-DIMETHOXYQUINAZOLIN-4-YLOXY)PHENYL)-3-(5-(1,1,1-TRIFLUORO-2-METHYLPROPAN-2-YL)ISOXAZOL-3-YL)UREA AS RAF KINASE MODULATOR IN THE TREATMENT OF CANCER DISEASES AMBIT BIOSCIENCES CORP (US) 2016-11-09 EP disclosed
CN-106075466-A Multi-functional amphoteric ion polymer conjugate 科迪亚科学企业公司 2016-11-09 CN disclosed
US-9487523-B2 Process for making CGRP receptor antagonists MERCK SHARP & DOHME CORP. (US) 2016-11-08 US disclosed
US-9487471-B1 Synthesis of pyrethroids and pyrethroid-containing compositions PROVIVI, INC. (US) 2016-11-08 US disclosed
US-9487545-B2 Fused ring-containing oxazolidinones antibiotics Xuanzhu Pharma Co., Ltd. (CN) 2016-11-08 US disclosed
US-9487535-B2 Asymmetric syntheses for spiro-oxindole compounds useful as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2016-11-08 US disclosed
US-9486457-B2 Use of cinnabarinic acid as a modulator of immune responses in autoimmune disorders THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-11-08 US disclosed
US-20160317486-A1 METHOD FOR WOUND HEALING PEPLIN RESEARCH PTY LTD (AU) 2016-11-03 US disclosed
WO-2016176330-A1 NUCLEOSIDE-MODIFIED RNA FOR INDUCING AN ADAPTIVE IMMUNE RESPONSE THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2016-11-03 WO disclosed
US-20160318936-A1 PYRIMIDOPYRIMIDINONES USEFUL AS WEE-1 KINASE INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2016-11-03 US disclosed
WO-2016176562-A1 NOVEL EPHA4 INHIBITORS TARGETING ITS LIGAND BINDING DOMAIN SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2016-11-03 WO disclosed
WO-2016176396-A1 THERAPEUTIC COMBINATIONS OF ANTIVIRAL AND ANTI-INFLAMMATORY THERAPIES FORESIGHT BIOTHERAPEUTICS, INC. (US) 2016-11-03 WO disclosed
EP-3087091-A1 VAR2CSA-DRUG CONJUGATES Zymeworks Inc. (CA) 2016-11-02 EP disclosed
EP-2331556-B1 BISTABLE CARBAZOLE COMPOUNDS ST MICROELECTRONICS SRL (IT) 2016-11-02 EP disclosed
EP-2217610-B1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN INC (US) 2016-11-02 EP disclosed
EP-3086815-A1 SULFONAMIDE-CONTAINING LINKAGE SYSTEMS FOR DRUG CONJUGATES Zymeworks Inc. (CA) 2016-11-02 EP disclosed
EP-2918589-B1 ADENINE DERIVATIVE AS PI3K INHIBITOR INTELLIKINE LLC (US) 2016-11-02 EP disclosed
US-9481673-B2 6-alkynyl-pyridine derivatives BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-11-01 US disclosed
US-20160311833-A1 NOVEL INDAZOLECARBOXAMIDES, PROCESSES FOR THEIR PREPARATION, PHARMACEUTICAL PREPARATIONS COMPRISING THEM AND THEIR USE FOR PRODUCING MEDICAMENTS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-10-27 US disclosed
US-20160313312-A1 Fluorescent Dyes and Related Methods UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION 2016-10-27 US disclosed
EP-3083598-A1 GLUCOSE TRANSPORT INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2016-10-26 EP disclosed
EP-2897957-B1 SUBSTITUTED PYRROLOPYRIMIDINYLAMINO-BENZOTHIAZOLONES AS MKNK KINASE INHIBITORS Bayer Pharma AG (DE) 2016-10-26 EP disclosed
CN-106061980-A Thienopyrimidines as MKNK1 and MKNK2 Inhibitors 拜耳制药股份公司 2016-10-26 CN disclosed
US-9475795-B2 Sulfonyl piperidine derivatives and their use for treating prokineticin mediated diseases TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-10-25 US disclosed
US-9475824-B2 Fused pyrimidines as inhibitors of p97 complex CLEAVE BIOSCIENCES, INC. (US) 2016-10-25 US disclosed
WO-2016168349-A1 METHODS OF TREATING HEPATITIS B VIRUS GILEAD SCIENCES, INC. (US) 2016-10-20 WO disclosed
WO-2016168510-A1 COMBINATION THERAPY OF A HIF-2-ALPHA INHIBITOR AND AN IMMUNOTHERAPEUTIC AGENT AND USES THEREOF PELOTON THERAPEUTICS, INC. (US) 2016-10-20 WO disclosed
US-20160304516-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Quanticel Pharmaceuticals, Inc. 2016-10-20 US disclosed
US-20160304495-A1 MONOCYCLIC PYRIMIDINE/PYRIDINE COMPOUNDS AS INHIBITORS OF P97 COMPLEX CLEAVE BIOSCIENCES, INC. (US) 2016-10-20 US disclosed
WO-2016168540-A1 FUSED-TRICYCLIC INHIBITORS OF KRAS AND METHODS OF USE THEREOF ARAXES PHARMA LLC (US) 2016-10-20 WO disclosed
WO-2016168682-A2 BROMODOMAIN INHIBITOR CELGENE QUANTICEL RESEARCH, INC. (US) 2016-10-20 WO disclosed
US-20160304498-A1 INHIBITORS OF CELLULAR NECROSIS AND RELATED METHODS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2016-10-20 US disclosed
US-20160303095-A1 METHODS OF TREATING HEPATITIS B VIRUS GILEAD SCIENCES, INC. 2016-10-20 US disclosed
US-20160303134-A1 COMBINATION OF PI3K-INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-10-20 US disclosed
EP-2507280-B1 POLYMERIC MATERIALS COMMW SCIENT IND RES ORG (AU) 2016-10-19 EP disclosed
EP-3080100-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Celgene Quanticel Research, Inc. (US) 2016-10-19 EP disclosed
US-9469642-B2 Purinone compounds as kinase inhibitors PHARMACYCLICS LLC (US) 2016-10-18 US disclosed
US-9468635-B2 Fused ring compound for use as mineralocorticoid receptor antagonist KBP BIOSCIENCES CO., LTD. (CN) 2016-10-18 US disclosed
US-9468642-B2 Imidazopyrazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-10-18 US disclosed
US-9469664-B2 Oligonucleotide analogues having modified intersubunit linkages and/or terminal groups SAREPTA THERAPEUTICS, INC. (US) 2016-10-18 US disclosed
US-20160297775-A1 QUINAZOLINE DERIVATIVES AS TAM FAMILY KINASE INHIBITORS SIGNALCHEM LIFESCIENCES CORP (CA) 2016-10-13 US disclosed
US-20160297774-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC 2016-10-13 US disclosed
US-20160297820-A1 DIMERIZER COMPOUND AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2016-10-13 US disclosed
US-20160297811-A1 SUBSTITUTED TRIAZOLOPYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-10-13 US disclosed
WO-2016164675-A1 SUBSTITUTED QUINAZOLINE COMPOUNDS AND METHODS OF USE THEREOF ARAXES PHARMA LLC (US) 2016-10-13 WO disclosed
WO-2016164589-A1 SYNERGISTIC BENZOXABOROLE-CONTAINING ANTI-FUNGICIDAL COMPOSITION THE PENN STATE RESEARCH FOUNDATION (US) 2016-10-13 WO disclosed
US-20160297833-A1 THIENOPYRIMIDINES AS MKNK1 AND MKNK2 INHIBITORS Bayer Pharma AG (DE) 2016-10-13 US disclosed
EP-3077003-A1 COMBINATION OF PI3K-INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2016-10-12 EP disclosed
EP-3076974-A1 THERAPEUTIC COMBINATION OF A PI3K INHIBITOR AND A BTK INHIBITOR Acerta Pharma B.V. (NL) 2016-10-12 EP disclosed
EP-2488177-B1 FILAMIN A BINDING ANTI-INFLAMMATORY AND ANALGESIC PAIN THERAPEUTICS INC (US) 2016-10-12 EP disclosed
EP-3077388-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE Pharmacyclics, LLC (US) 2016-10-12 EP disclosed
EP-2723748-B1 HETEROCYCLYL AMINOIMIDAZOPYRIDAZINES BAYER IP GMBH (DE) 2016-10-12 EP disclosed
CN-104797582-B Substituted pyrrolo-pyrimidine radicals amino-benzothiazole ketone as MKNK inhibitors of kinases 拜耳药业股份公司 2016-10-12 CN disclosed
US-9464033-B2 Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2016-10-11 US disclosed
US-9464060-B2 Compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-10-11 US disclosed
US-9464065-B2 Compounds and methods for inducing chondrogenesis THE SCRIPPS RESEARCH INSTITUTE (US) 2016-10-11 US disclosed
WO-2016161248-A1 TARGETING PIM KINASES IN COMBINATION WITH BTK INHIBITION TOLERO PHARMACEUTICALS, INC. (US) 2016-10-06 WO disclosed
WO-2016156816-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS MISSION THERAPEUTICS LIMITED (GB) 2016-10-06 WO disclosed
US-20160287604-A1 2-(MORPHOLIN-4-YL)-1,7-NAPHTHYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-10-06 US disclosed
US-20160287601-A1 ENHANCED TREATMENT REGIMENS USING PI3K INHIBITORS MILLENNIUM PHARMACEUTICALS INC 2016-10-06 US disclosed
US-20160289191-A1 ORGANIC COMPOUNDS XENON PHARMACEUTICALS INC. (CA) 2016-10-06 US disclosed
US-20160289226-A1 [9,10-DIMETHOXY-3-(2-METHYLPROPYL)-1H,2H,3H,4H,6H,7H,11BH-PYRIDO-[2,1-A]ISOQUINOLIN-2-YL]METHANOL AND COMPOUNDS, COMPOSITIONS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES, INC. 2016-10-06 US disclosed
US-20160287597-A1 Treatment Regimens Using Multiple Pharmaceutical Agents INTELLIKINE LLC 2016-10-06 US disclosed
US-20160287595-A1 Combination Pharmaceutical Compositions and Uses Thereof CALITHERA BIOSCIENCES, INC. 2016-10-06 US disclosed
US-20160287715-A1 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC (US) 2016-10-06 US disclosed
US-20160287596-A1 Benzoxazole Kinase Inhibitors and Methods of Use FAETH THERAPEUTICS, INC. 2016-10-06 US disclosed
US-20160287589-A1 SUBSTITUTED-IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-10-06 US disclosed
EP-2552905-B1 B-Raf kinase inhibitors BOEHRINGER INGELHEIM INT (DE) 2016-10-05 EP disclosed
EP-3074390-A2 AMINOPYRIDINE DERIVATIVES AS TAM FAMILY KINASE INHIBITORS SignalChem Lifesciences Corporation (CA) 2016-10-05 EP disclosed
EP-3074385-A1 PIPERIDINE DERIVATIVES FOR USE IN THE TREATMENT OR PREVENTION OF PSYCHIATRIC AND NEUROLOGICAL CONDITIONS Takeda Pharmaceutical Company Limited (JP) 2016-10-05 EP disclosed
EP-3074414-A1 WITHANOLIDES USEFUL FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES Imstar Therapeutics Inc. (CA) 2016-10-05 EP disclosed
US-9458088-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2016-10-04 US disclosed
US-9458159-B2 Substituted pyrido[1′,2′:4,5]pyrazino[1,2-a]azepines for treating viral infections GILEAD SCIENCES, INC. (US) 2016-10-04 US disclosed
US-9458178-B2 Spiro-oxindole compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2016-10-04 US disclosed
US-9458129-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2016-10-04 US disclosed
WO-2016154629-A1 THERAPY FOR MALIGNANT DISEASE WOMAN & INFANTS' HOSPITAL OF RHODE ISLAND (US) 2016-09-29 WO disclosed
WO-2016149765-A1 SODIUM CHANNEL MODULATORS THE FLOREY INSTITUTE OF NEUROSCIENCE AND MENTAL HEALTH (AU) 2016-09-29 WO disclosed
EP-2484679-B1 N3-heteroaryl substituted triazoles and n5-heteroaryl substitued triazoles useful as axl inhibitors RIGEL PHARMACEUTICALS INC (US) 2016-09-28 EP disclosed
EP-2590510-B1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX INC (US) 2016-09-28 EP disclosed
EP-3071591-A2 ANTIMICROBIAL PEPTIDOMIMETICS Agency For Science, Technology And Research (SG) 2016-09-28 EP disclosed
EP-3071204-A1 QUINAZOLINE DERIVATIVES AS TAM FAMILY KINASE INHIBITORS SignalChem Lifesciences Corp. (CA) 2016-09-28 EP disclosed
US-9452148-B2 Insulin sensitisers and methods of treatment VERVA PHARMACEUTICALS LTD (AU) 2016-09-27 US disclosed
US-9452167-B2 Heterocyclic compounds and methods of use thereof AMBIT BIOSCIENCES CORPORATION (US) 2016-09-27 US disclosed
US-9452153-B2 Amine derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2016-09-27 US disclosed
WO-2016149404-A1 BOTULINUM NEUROTOXIN-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2016-09-22 WO disclosed
WO-2016149401-A2 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME ABIDE THERAPEUTICS, INC. (US) 2016-09-22 WO disclosed
US-20160272602-A1 PIPERAZINE CARBAMATES AND METHODS OF MAKING AND USING SAME H. LUNDBECK A/S (DK) 2016-09-22 US disclosed
US-20160272668-A1 NICOTINIC ACID RIBOSIDE OR NICOTINAMIDE RIBOSIDE COMPOSITIONS, REDUCED DERIVATIVES THEREOF, AND THE USE THEREOF TO ENHANCE SKIN PERMEATION IN TREATING SKIN CONDITIONS ChromaDex Inc. (US) 2016-09-22 US disclosed
US-20160271178-A1 NANOPARTICLE-CONTAINING HYDROGELS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2016-09-22 US disclosed
US-20160272649-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS INC (US) 2016-09-22 US disclosed
EP-3070110-A1 POLYMERS HAVING ORTHOGONAL REACTIVE GROUPS AND USES THEREOF NVS Technologies Inc. (US) 2016-09-21 EP disclosed
US-9447045-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2016-09-20 US disclosed
US-9447078-B2 Substituted heterocyclic compounds for disease treatment ACUCELA INC. (US) 2016-09-20 US disclosed
US-9447114-B2 Thieno- and furo[2,3-d]pyrimidine-2,4[1H,3H]-dione derivatives HYDRA BIOSCIENCES, INC. (US) 2016-09-20 US disclosed
US-9447046-B2 Histone demethylase inhibitors Celegene Quanticel Research, Inc. (US) 2016-09-20 US disclosed
WO-2016144825-A1 AROMATIC COMPOUNDS AND USES THEREOF PELOTON THERAPEUTICS, INC. (US) 2016-09-15 WO disclosed
US-20160263013-A1 Skin Care Compositions and Methods of Use Thereof UNIGEN, INC. (US) 2016-09-15 US disclosed
US-20160266149-A1 ALZHEIMER'S DISEASE ASSAY IN A LIVING PATIENT CASSAVA SCIENCES, INC. 2016-09-15 US disclosed
US-20160263122-A1 NOVEL COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-09-15 US disclosed
US-20160264587-A1 Compounds Useful for Inhibiting Metastasis from Cancer and Methods Using Same UNIV DREXEL (US) 2016-09-15 US disclosed
WO-2016145045-A1 COMPOSITIONS FOR USE IN TREATING GLIOBLASTOMA PELOTON THERAPEUTICS, INC. (US) 2016-09-15 WO disclosed
WO-2016145032-A1 COMPOSITIONS FOR USE IN TREATING PULMONARY ARTERIAL HYPERTENSION PELOTON THERAPEUTICS, INC. (US) 2016-09-15 WO disclosed
US-20160264539-A1 COMPOUNDS WITH (1E, 6E)-1,7-BIS-(3,4-DIMETHOXYPHENYL)-4-4-DISUBSTITUTED-HEPTA-1,6-DIENE-3,5-DIONE STRUCTURAL SCAFFOLD, THEIR BIOLOGICAL ACTIVITY, AND USES THEREOF Annji Pharmaceutical Co., Ltd. (TW) 2016-09-15 US disclosed
WO-2016145298-A1 METHODS FOR TREATING CANCER WITH RORgamma INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-09-15 WO disclosed
WO-2016144826-A1 SUBSTITUTED PYRIDINES AND USES THEREOF PELOTON THERAPEUTICS, INC. (US) 2016-09-15 WO disclosed
US-20160264568-A1 SUBSTITUTED TRIAZOLOPYRIDINES HAVING ACTIVITY AS MPS-1 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-09-15 US disclosed
EP-2734520-B1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS INC (US) 2016-09-14 EP disclosed
EP-2825540-B1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER IP GMBH (DE) 2016-09-14 EP disclosed
EP-3067358-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE Gilead Sciences, Inc. (US) 2016-09-14 EP disclosed
EP-2277848-B1 Indene derivatives as pharmaceutical agents AQUINOX PHARMACEUTICALS CANADA INC (CA) 2016-09-14 EP disclosed
EP-3066104-A1 TRIAZOLOPYRAZINE DERIVATIVES AS BRD4 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2016-09-14 EP disclosed
CN-104520292-B Sulphonylpiperidine derivant and they are for treating the purposes of disease of front dynein mediation 武田药品工业株式会社 2016-09-14 CN disclosed
CN-104144929-B Cinchona alkaloid double-quaternary salt as asymmetric phase transfer catalyst 默沙东公司 2016-09-14 CN disclosed
US-9440973-B2 Pyrido[3,4-d]pyrimidine-2,4(1H,3H)-dione derivatives HYDRA BIOSCIENCES, INC. (US) 2016-09-13 US disclosed
US-9440983-B2 Pyrrolo[3,2-d]pyrimidine-2,4(3H,5H)-dione derivatives HYDRA BIOSCIENCES, INC. (US) 2016-09-13 US disclosed
US-9440898-B2 Preparation of pentanol with ethanol derived from fermentation Pioneer Energy (US) 2016-09-13 US disclosed
US-9440972-B2 Pyrido[2,3-d]pyrimidine-2,4(1 H,3H)-dione derivatives HYDRA BIOSCIENCES, INC. (US) 2016-09-13 US disclosed
US-20160256463-A1 NOVEL COMPOUNDS AS RESPIRATORY STIMULANTS FOR TREATMENT OF BREATHING CONTROL DISORDERS OR DISEASES GALLEON PHARMACEUTICALS INC (US) 2016-09-08 US disclosed
US-20160257671-A2 SHIP1 MODULATORS AND METHODS RELATED THERETO NEOLEUKIN THERAPEUTICS, INC. 2016-09-08 US disclosed
EP-2817308-B1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES ABBVIE INC (US) 2016-09-07 EP disclosed
EP-2591354-B1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX INC (US) 2016-09-07 EP disclosed
EP-3062767-A1 SKIN CARE COMPOSITIONS AND METHODS OF USE THEREOF Unigen, Inc. (US) 2016-09-07 EP disclosed
CN-105934498-A Encoded chromophoric polymer particles 华盛顿大学商业中心 2016-09-07 CN disclosed
CN-105934440-A Antimicrobial Peptide Mimetics 新加坡科技研究局 2016-09-07 CN disclosed
CN-103965180-B Benzsulfamide azoles and thiazole inhibitors of kinases 通化济达医药有限公司 2016-09-07 CN disclosed
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US-9434720-B2 Pyrazolylbenzothiazole derivatives and their use as therapeutic agents DIRMIRA (CANADA), INC. (US) 2016-09-06 US disclosed
US-9434744-B2 Low temperature synthesis of rapamycin derivatives BIOSENSORS INTERNATIONAL GROUP, LTD. (BM) 2016-09-06 US disclosed
US-9433640-B2 Compositions and methods for treating hyperkalemia ARDELYX, INC. (US) 2016-09-06 US disclosed
WO-2016138457-A1 PHENYLETHYNYLNAPHTHALENE DYES AND METHODS FOR THEIR USE SONY CORPORATION (JP) 2016-09-01 WO disclosed
US-20160251307-A1 ARYL ETHERS AND USES THEREOF PELOTON THERAPEUTICS, INC. (US) 2016-09-01 US disclosed
US-20160251374-A1 FILAMIN A BINDING ANTI-INFLAMMATORY AND ANALGESIC BURNS BARBIER LINDSAY (US) 2016-09-01 US disclosed
WO-2016138461-A1 WATER SOLUBLE FLUORESCENT OR COLORED DYES COMPRISING CONJUGATING GROUPS SONY CORPORATION (JP) 2016-09-01 WO disclosed
EP-2639226-B1 Anti-infective pyrimidines and uses thereof ABBVIE BAHAMAS LTD (BS) 2016-08-31 EP disclosed
CN-105916841-A Functionalised and substituted indoles as anti-cancer agents 诺沃根公司 2016-08-31 CN disclosed
US-9428515-B2 Benzimidazole derivatives BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-08-30 US disclosed
US-9428513-B2 Triazolopyrazine BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-08-30 US disclosed
WO-2016131794-A1 3-CARBAMOYLPHENYL-4-CARBOXAMIDE AND ISOPHTALAMIDE DERIVATIVES AS INHIBITORS OF THE WNT SIGNALLING PATHWAY BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-08-25 WO disclosed
WO-2016131810-A1 N-PHENYL-(MORPHOLIN-4-YL OR PIPERAZINYL)ACETAMIDE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE WNT SIGNALLING PATHWAYS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-08-25 WO disclosed
WO-2016131808-A1 1,3,4-THIADIAZOL-2-YL-BENZAMIDE DERIVATIVES AS INHIBITORSOF THE WNT SIGNALLING PATHWAY BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-08-25 WO disclosed
US-20160243085-A1 SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS MIDCAP FINANCIAL TRUST 2016-08-25 US disclosed
EP-3057957-A1 CYCLOPENTYLBENZAMIDE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF PSYCHOTIC AND COGNITIVE DISORDERS Takeda Pharmaceutical Company Limited (JP) 2016-08-24 EP disclosed
EP-2346508-B1 HETEROCYCLIC KINASE INHIBITORS INTELLIKINE LLC (US) 2016-08-24 EP disclosed
EP-3057586-A1 BROMODOMAIN INHIBITORS Celgene Quanticel Research, Inc. (US) 2016-08-24 EP disclosed
CN-103987711-B 8-carbamoyl-2- (2, 3-disubstituted pyridin-6-yl) -1,2,3, 4-tetrahydroisoquinoline derivatives as apoptosis inducers for the treatment of cancer and immune and autoimmune diseases 艾伯维公司 2016-08-24 CN disclosed
CN-103857664-B The method being prepared 5 hydroxymethyl furfural by carbohydrate 新加坡科技研究局 2016-08-24 CN disclosed
US-9422290-B2 Triazolopyridazine BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-08-23 US disclosed
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US-20160235716-A1 SPIROCYCLIC HAT INHIBITORS AND METHODS FOR THEIR USE ABBVIE INC. (US) 2016-08-18 US disclosed
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US-20160237089-A1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES, INC. 2016-08-18 US disclosed
US-20160237426-A1 PEPTIDE OLIGONUCLEOTIDE CONJUGATES JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2016-08-18 US disclosed
US-20160237091-A1 INHIBITORS OF ERK AND METHODS OF USE KURA ONCOLOGY, INC. 2016-08-18 US disclosed
WO-2016130092-A1 NON-MEMBRANE DISRUPTIVE P53 ACTIVATING STAPLED PEPTIDES AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2016-08-18 WO disclosed
WO-2016128912-A1 THERAPEUTIC COMBINATIONS OF A BTK INHIBITOR, A PI3K INHIBITOR, A JAK-2 INHIBITOR, A PD-1 INHIBITOR, AND/OR A PD-L1 INHIBITOR ACERTA PHARMA B.V. (NL) 2016-08-18 WO disclosed
EP-3054956-A1 METHOD FOR INHIBITING GROWTH OF CANCER CELLS Pain Therapeutics, Inc. (US) 2016-08-17 EP disclosed
EP-3055290-A1 INHIBITORS OF KRAS G12C Araxes Pharma LLC (US) 2016-08-17 EP disclosed
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WO-2016127123-A2 COMPOUNDS AND METHODS FOR PREVENTING OR TREATING SENSORY HAIR CELL DEATH UNIVERSITY OF WASHINGTON (US) 2016-08-11 WO disclosed
WO-2016127133-A1 [9,10-DIMETHOXY-3-(2-METHYLPROPYL)-1H,2H,3H,4H,6H,7H,11BH-PYRIDO-[2,1-A]ISOQUINOLIN-2-YL]METHANOL AND COMPOUNDS, COMPOSITIONS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES, INC. (US) 2016-08-11 WO disclosed
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EP-2766361-B1 8-CARBAMOYL-2-(2,3-DISUBSTITUTED PYRID-6-YL)-1,2,3,4-TETRAHYDROISOQUINOLINE DERIVATIVES AS APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2016-08-10 EP disclosed
EP-3052493-A1 ENHANCED TREATMENT REGIMENS USING PI3K INHIBITORS Millennium Pharmaceuticals, Inc. (US) 2016-08-10 EP disclosed
EP-3052486-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE Pharmacyclics LLC (US) 2016-08-10 EP disclosed
EP-2678016-B1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE LLC (US) 2016-08-10 EP disclosed
EP-3052485-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Infinity Pharmaceuticals, Inc. (US) 2016-08-10 EP disclosed
CN-103936728-B Thiazole inhibitors of kinases 通化济达医药有限公司 2016-08-10 CN disclosed
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US-20160222030-A1 Cyclopentylbenzamide Derivatives and their Use for the Treatment of Psychotic and Cognitive Disorders TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-08-04 US disclosed
WO-2016123361-A1 LIGAND-ENABLED META-C-H ACTIVATION USING A TRANSIENT MEDIATOR THE SCRIPPS RESEARCH INSTITUTE (US) 2016-08-04 WO disclosed
WO-2016123392-A2 PYRAZOLOPYRIMIDINES AS INHIBITORS OF GLUCOCORTICOID RECEPTOR TRANSLOCATION SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2016-08-04 WO disclosed
EP-2725031-B1 C-GLYCOSIDE DERIVATIVES XUANZHU PHARMA CO LTD (CN) 2016-08-03 EP disclosed
CN-105828838-A NANOPARTICLE-CONTAINING HYDROGELS 新加坡科技研究局 2016-08-03 CN disclosed
US-20160213787-A1 POLYMER-FLAVONOID CONJUGATES AND HYDROGELS FOR BIOMEDICAL APPLICATIONS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2016-07-28 US disclosed
US-20160214944-A1 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE SUMITOMO PHARMA AMERICA, INC. 2016-07-28 US disclosed
WO-2016116777-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF CHRONIC LYMPHOCYTIC LEUKEMIA AND SMALL LYMPHOCYTIC LEUKEMIA USING A BTK INHIBITOR ACERTA PHARMA B.V. (NL) 2016-07-28 WO disclosed
EP-3046572-A1 CHLOROTOXIN CONJUGATES AND METHODS OF USE THEREOF Blaze Bioscience, Inc. (US) 2016-07-27 EP disclosed
EP-3046913-A1 CONVERSION AND PURIFICATION OF BIOMASS Agency For Science, Technology And Research (SG) 2016-07-27 EP disclosed
EP-3048098-A1 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS AbbVie Bahamas Limited (BS) 2016-07-27 EP disclosed
EP-3048105-A1 COMPOUND INHIBITING ACTIVITIES OF BTK AND/OR JAK3 KINASES Beijing Hanmi Pharmaceutical Co., Ltd. (CN) 2016-07-27 EP disclosed
EP-2504374-B1 WATER CURABLE RESIN FORMULATIONS PETROLIAM NASIONAL BERHAD PETRONAS (MY) 2016-07-27 EP disclosed
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US-20160207880-A1 AMIDE DERIVATIVES AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-07-21 US disclosed
US-20160207928-A1 NOVEL COMPOUNDS FOR THE TREATMENT OF CANCER BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-07-21 US disclosed
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CN-105793249-A Piperidine derivatives for the treatment or prevention of psychiatric and neurological disorders 武田药品工业株式会社 2016-07-20 CN disclosed
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US-9394299-B2 Rilyazine derivatives and compositions for the treatment of cancer WARNER BABCOCK INSTITUTE FOR GREEN CHEMISTRY, LLC (US) 2016-07-19 US disclosed
US-9394313-B2 Transfer hydrogenation of cyclopamine analogs INFINITY PHARMACEUTICALS, INC. (US) 2016-07-19 US disclosed
US-9394257-B2 PKM2 modulators and methods for their use TOLERO PHARMACEUTICALS, INC. (US) 2016-07-19 US disclosed
US-20160200704-A1 THERAPEUTIC INHIBITORY COMPOUNDS ATTUNE PHARMACEUTICALS, INC. 2016-07-14 US disclosed
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WO-2016111855-A1 COMPOSITIONS AND METHODS FOR TREATING HYPERKALEMIA ARDELYX, INC. (US) 2016-07-14 WO disclosed
US-20160199375-A1 RAF KINASE MODULATOR COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORP. 2016-07-14 US disclosed
US-20160200645-A1 Fuels and Chemicals from Lower Alkanes PIONEER ENERGY INC (US) 2016-07-14 US disclosed
EP-3042895-A1 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2016-07-13 EP disclosed
EP-3041830-A1 POLYMER-FLAVONOID CONJUGATES AND HYDROGELS FOR BIOMEDICAL APPLICATIONS Agency For Science, Technology And Research (SG) 2016-07-13 EP disclosed
EP-3041840-A1 RILYAZINE DERIVATIVES AND COMPOSITIONS FOR THE TREATMENT OF CANCER The Warner-Babcock Institute For Green Chemistry LLC (US) 2016-07-13 EP disclosed
US-9388183-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2016-07-12 US disclosed
US-9388177-B2 Method for preparing substituted triazolopyridines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-07-12 US disclosed
US-9388140-B2 Substituted benzimidazoles BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-07-12 US disclosed
US-20160193181-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. 2016-07-07 US disclosed
US-20160193160-A1 Styrenyl Derivative Compounds for Treating Ophthalmic Diseases and Disorders ACUCELA INC. 2016-07-07 US disclosed
US-20160193209-A1 NAMPT INHIBITORS ABBVIE INC. (US) 2016-07-07 US disclosed
US-20160194439-A1 CONJUGATED POLYMERS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2016-07-07 US disclosed
US-20160194315-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC 2016-07-07 US disclosed
US-20160194306-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. 2016-07-07 US disclosed
US-20160194323-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2016-07-07 US disclosed
US-20160194335-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2016-07-07 US disclosed
US-20160194299-A1 COMPOUNDS FOR TREATMENT OF DRUG RESISTANT AND PERSISTENT TUBERCULOSIS THE CALIFORNIA INSTITUTE FOR BIOMEDICAL RESEARCH 2016-07-07 US disclosed
EP-3039021-A1 BIARYL ACETAMIDE COMPOUNDS AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2016-07-06 EP disclosed
EP-2571357-B1 CHEMICAL COMPOUNDS, COMPOSITIONS AND METHODS FOR KINASE MODULATION INFINITY PHARMACEUTICALS INC (US) 2016-07-06 EP disclosed
EP-2697193-B1 SUBSTITUTED 5-(CYCLOHEX-2-EN-1-YL)-PENTA-2,4-DIENES AND 5-(CYCLOHEX-2-EN-1-YL)-PENT-2-EN-4-INES AS ACTIVE AGENTS AGAINST ABIOTIC STRESS IN PLANTS BAYER IP GMBH (DE) 2016-07-06 EP disclosed
CN-103270034-B The 2-pyridine carboxylic acid replaced and salt and acid derivative, and the purposes as herbicide 拜耳知识产权有限责任公司 2016-07-06 CN disclosed
CN-105742702-A Rechargeable lithium battery 三星SDI株式会社 2016-07-06 CN disclosed
CN-105745196-A Conversion and purification of biomass 新加坡科技研究局 2016-07-06 CN disclosed
US-9382255-B2 Substituted pyrrolopyrimidinylamino-benzothiazolones as MKNK kinase inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-07-05 US disclosed
US-9382246-B2 Inhibitors of Bruton's tyrosine kinase PHARMACYCLICS LLC (US) 2016-07-05 US disclosed
WO-2016102435-A2 NOVEL ISOTHIAZOLAMIDES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS FUNGICIDES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-06-30 WO disclosed
WO-2016102493-A1 IMIDAZOPYRIDINE EZH2 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-06-30 WO disclosed
WO-2016103192-A1 AMINO ACID AND PEPTIDE CONJUGATES AND USES THEREOF BRIMBLE MARGARET ANNE (NZ) 2016-06-30 WO disclosed
US-20160190644-A1 RECHARGEABLE LITHIUM BATTERY SAMSUNG SDI CO., LTD. (KR) 2016-06-30 US disclosed
US-20160185728-A1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY ONCOLOGY PHARMACEUTICAL CO., LTD. (CN) 2016-06-30 US disclosed
US-20160184281-A1 NAMPT INHIBITORS ABBVIE INC. (US) 2016-06-30 US disclosed
US-20160184445-A1 BUTYRYLCHOLINESTERASE ZWITTERIONIC POLYMER CONJUGATES OLIGASIS, LLC 2016-06-30 US disclosed
US-20160184282-A1 NAMPT INHIBITORS ABBVIE INC. (US) 2016-06-30 US disclosed
US-20160184387-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT CHARMOT DOMINIQUE (US) 2016-06-30 US disclosed
US-20160185800-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE, INC. 2016-06-30 US disclosed
US-20160185752-A1 PIPERIDINE AND AZEPINE DERIVATIVES AS PROKINETICIN RECEPTOR MODULATORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-30 US disclosed
EP-3036235-A1 NEW BIS-AMIDO PYRIDINES Boehringer Ingelheim International GmbH (DE) 2016-06-29 EP disclosed
EP-3038194-A1 RECHARGEABLE LITHIUM BATTERY Samsung SDI Co., Ltd. (KR) 2016-06-29 EP disclosed
EP-3036228-A1 NEW 6-ALKYNYL PYRIDINE Boehringer Ingelheim International GmbH (DE) 2016-06-29 EP disclosed
US-9376447-B2 Transfer hydrogenation of cyclopamine analogs INFINITY PHARMACEUTICALS, INC. (US) 2016-06-28 US disclosed
US-9375474-B2 Compounds useful for inhibiting metastasis from cancer and methods using same DREXEL UNIVERSITY (US) 2016-06-28 US disclosed
US-9376431-B2 Bis-quaternary cinchona alkaloid salts as asymmetric phase transfer catalysts MERCK SHARP & DOHME CORP. (US) 2016-06-28 US disclosed
US-9376709-B2 Compositions for stabilizing DNA and RNA in blood and other biological samples during shipping and storage at ambient temperatures BIOMATRICA, INC. (US) 2016-06-28 US disclosed
WO-2016100711-A1 MODULATORS OF HEPATIC LIPOPROTEIN METABOLISM THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed
WO-2016096721-A1 PYRAZOLOPYRIDINAMINES AS MKNK1 AND MKNK2 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-06-23 WO disclosed
US-20160176894-A1 TAXANE AND ABEO-TAXANE ANALOGS Arbor Therapeutics, LLC (US) 2016-06-23 US disclosed
WO-2016100123-A1 IONIC LIQUID SYSTEMS THE PROCTER & GAMBLE COMPANY (US) 2016-06-23 WO disclosed
US-20160175346-A1 PHARMACEUTICAL COMPOSITIONS FOR TREATING HYPERKALEMIA ARDELYX, INC. 2016-06-23 US disclosed
US-20160175345-A1 PHARMACEUTICAL COMPOSITIONS FOR TREATING HYPERKALEMIA ARDELYX, INC. 2016-06-23 US disclosed
US-20160176885-A1 SUBSTITUTED 1,2,3,4,6,8,12,12a-OCTAHYDRO-1,4-METHANODIPYRIDO[1,2-a:1',2'-d]PYRAZINES AND METHODS FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. 2016-06-23 US disclosed
US-20160175344-A1 COMPOSITIONS AND METHODS FOR TREATING HYPERKALEMIA ARDELYX, INC. 2016-06-23 US disclosed
US-20160177222-A1 IONIC LIQUID SYSTEMS THE PROCTER & GAMBLE COMPANY 2016-06-23 US disclosed
EP-3033335-A1 PYRIDINONES Boehringer Ingelheim International GmbH (DE) 2016-06-22 EP disclosed
EP-2852596-B1 THIENOPYRIMIDINES Bayer Pharma AG (DE) 2016-06-22 EP disclosed
EP-2575462-B1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE LLC (US) 2016-06-22 EP disclosed
EP-2852595-B1 SUBSTITUTED BENZOTHIENOPYRIMIDINES Bayer Pharma AG (DE) 2016-06-22 EP disclosed
CN-103596431-B Pyrimidine cyclohexyl glucocorticoid receptor modulators 科赛普特治疗公司 2016-06-22 CN disclosed
US-9370510-B2 Small molecule compounds to treat hearing loss FATE THERAPEUTICS, INC. (US) 2016-06-21 US disclosed
US-20160168149-A1 PURINONE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS LLC 2016-06-16 US disclosed
US-20160167015-A1 ADSORBENT FOR HETEROATOM SPECIES REMOVAL AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 US disclosed
US-20160168140-A1 HETEROCYCLIC COMPOUNDS AS ANTIBIOTIC POTENTIATORS SYNERECA PHARMACEUTICALS (US) 2016-06-16 US disclosed
US-20160166571-A1 COMBINATION THERAPIES FOR TREATMENT OF CANCER ARAXES PHARMA LLC 2016-06-16 US disclosed
US-20160168173-A1 ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 US disclosed
WO-2016094777-A1 ORGANOSILICA MATERIALS EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 WO disclosed
US-20160168171-A1 METHODS OF PRODUCING ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 US disclosed
WO-2016094773-A1 ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 WO disclosed
US-20160168477-A1 Synthesis of Drop-in Liquid Fuels and Chemicals from Methanol, Ethanol or Syngas Using Mixed Catalysts Pioneer Energy Inc. (US) 2016-06-16 US disclosed
WO-2016094730-A1 HETEROCYCLIC COMPOUNDS AS ANTIBIOTIC POTENTIATORS SYNERECA PHARMACEUTICALS, INC. (US) 2016-06-16 WO disclosed
WO-2016094784-A1 COATING METHODS USING ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 WO disclosed
WO-2016094866-A1 OLEFIN POLYMERIZATION CATALYST SYSTEM COMPRISING MESOPOROUS ORGANOSILICA SUPPORT EXXONMOBIL CHEMICAL PATENTS INC. (US) 2016-06-16 WO disclosed
US-20160168134-A1 NAMPT INHIBITORS ABBVIE INC. (US) 2016-06-16 US disclosed
US-20160168174-A1 ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 US disclosed
WO-2016094830-A1 METHODS OF SEPARATING AROMATIC COMPOUNDS FROM LUBE BASE STOCKES EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 WO disclosed
WO-2016094769-A1 AROMATIC HYDROGENATION CATALYSTS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 WO disclosed
US-20160168333-A1 ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 US disclosed
WO-2016094788-A1 ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 WO disclosed
WO-2016094489-A1 PHOSPHORUS LIGANDS AND METHODS OF USE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-06-16 WO disclosed
WO-2016094774-A2 METHODS OF PRODUCING ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 WO disclosed
US-20160168128-A1 INHIBITORS OF CELLULAR NECROSIS AND RELATED METHODS PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2016-06-16 US disclosed
WO-2016094820-A1 ADSORBENT FOR HETEROATOM SPECIES REMOVAL AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 WO disclosed
WO-2016094848-A1 ORGANOSILICA MATERIALS FOR USE AS ADSORBENTS FOR OXYGENATE REMOVAL EXXONMOBIL CHEMICAL PATENTS INC. (US) 2016-06-16 WO disclosed
US-20160168172-A1 ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 US disclosed
WO-2016094778-A1 ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 WO disclosed
US-20160167016-A1 COATING METHODS USING ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 US disclosed
WO-2016094770-A1 ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 WO disclosed
WO-2016094803-A1 MEMBRANE FABRICATION METHODS USING ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 WO disclosed
WO-2016094843-A2 OLEFIN POLYMERIZATION CATALYST SYSTEM COMPRISING MESOPOROUS ORGANOSILICA SUPPORT EXXONMOBIL CHEMICAL PATENTS INC. (US) 2016-06-16 WO disclosed
US-20160167032-A1 AROMATIC HYDROGENATION CATALYSTS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 US disclosed
WO-2016094846-A1 INHIBITORS OF CELLULAR NECROSIS AND RELATED METHODS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2016-06-16 WO disclosed
US-20160168484-A1 METHODS OF SEPARATING AROMATIC COMPOUNDS FROM LUBE BASE STOCKS EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 US disclosed
US-20160168157-A1 HETEROCYCLIC KINASE INHIBITORS INTELLIKINE LLC 2016-06-16 US disclosed
US-20160168485-A1 MEMBRANE FABRICATION METHODS USING ORGANOSILICA MATERIALS AND USES THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-06-16 US disclosed
EP-3030553-A1 PIPERIDINE AND AZEPINE DERIVATIVES AS PROKINETICIN RECEPTOR MODULATORS Takeda Pharmaceutical Company Limited (JP) 2016-06-15 EP disclosed
EP-3030252-A2 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT Ardelyx, Inc. (US) 2016-06-15 EP disclosed
US-9365499-B2 9-aminomethyl substituted tetracycline compounds KBP BIOSCIENCES CO., LTD. (CN) 2016-06-14 US disclosed
US-20160161475-A1 HYBRID SEMICONDUCTING POLYMER NANOPARTICLES AS POLARIZATION-SENSITIVE FLUORESCENT PROBES UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION 2016-06-09 US disclosed
US-20160159789-A1 SUBSTITUTED PYRAZOLOPYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-06-09 US disclosed
WO-2016087488-A1 ADMINISTRATION REGIME FOR AMINOALCOHOL SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-06-09 WO disclosed
WO-2016090313-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE AQUINNAH PHARMACEUTICALS, INC. (US) 2016-06-09 WO disclosed
WO-2016087994-A1 BTK INHIBITORS TO TREAT SOLID TUMORS THROUGH MODULATION OF THE TUMOR MICROENVIRONMENT ACERTA PHARMA B.V. (NL) 2016-06-09 WO disclosed
WO-2016090240-A1 PHARMACEUTICAL COMPOSITIONS FOR INCREASING THE BIOAVAILABILITY OF POORLY SOLUBLE DRUGS ASTEX PHARMACEUTICALS, INC. (US) 2016-06-09 WO disclosed
WO-2016087490-A1 COMBINATION OF PI3K-INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-06-09 WO disclosed
WO-2016090317-A1 SULFONAMIDE DERIVATIVES, COMPOSITIONS AND METHODS OF USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES AQUINNAH PHARMACEUTICALS, INC. (US) 2016-06-09 WO disclosed
US-20160159816-A1 SUBSTITUTED THIENOPYRIMIDINES AND PHARMACEUTICAL USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-06-09 US disclosed
US-20160159738-A1 COVALENT INHIBITORS OF KRAS G12C ARAXES PHARMA LLC 2016-06-09 US disclosed
US-20160158218-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2016-06-09 US disclosed
US-20160158239-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE, INC. 2016-06-09 US disclosed
CN-105658633-A Polymer-flavonoid conjugates and hydrogels for biomedical applications 新加坡科技研究局 2016-06-08 CN disclosed
US-9359344-B2 Biaryl heterocycle substituted oxazolidinone antibacterial agents Xuanzhu Pharma Co., Ltd. (CN) 2016-06-07 US disclosed
US-9362126-B2 Process for making a patterned metal oxide structure AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2016-06-07 US disclosed
US-9359371-B2 Bicyclic substituted pyrimidine compounds Xuanzhu Pharma Co., Ltd. (CN) 2016-06-07 US disclosed
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US-9359352-B2 Substituted benzimidazoles as PI3 kinase inhibitors INTELLIKINE LLC (US) 2016-06-07 US disclosed
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US-20160152595-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. 2016-06-02 US disclosed
US-20160151527-A1 Ionic Liquids THE PROCTER & GAMBLE COMPANY 2016-06-02 US disclosed
US-20160151369-A1 SUBSTITUTED 3-PHENYLPROPYLAMINE DERIVATIVES FOR THE TREATMENT OF OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. 2016-06-02 US disclosed
US-20160150782-A1 USE OF SELECTED PYRIDONE CARBOXAMIDES OR SALTS THEREOF AS ACTIVE SUBSTANCES AGAINST ABIOTIC PLANT STRESS BAYER CROPSCIENCE AG (DE) 2016-06-02 US disclosed
US-9353124-B2 Bridged bicyclic aryl and bridged bicyclic heteroaryl substituted triazoles useful as axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2016-05-31 US disclosed
US-9351972-B2 Compounds as respiratory stimulants for treatment of breathing control disorders or diseases GALLEON PHARMACEUTICALS, INC. (US) 2016-05-31 US disclosed
US-9353126-B2 Substituted triazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2016-05-31 US disclosed
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EP-2670731-B1 POSITIVE ALLOSTERIC MODULATORS OF THE ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR AND USES THEREOF. BIONOMICS LTD (AU) 2016-05-25 EP disclosed
US-9345706-B2 Benzoxazole kinase inhibitors and methods of use INTELLIKINE, LLC (US) 2016-05-24 US disclosed
US-9346813-B2 Substituted pyrrolo[2,3-d]pyrimindines as CDK9 kinase inhibitors ABBVIE INC. (US) 2016-05-24 US disclosed
US-9346785-B2 Process for making HCV protease inhibitors ABBVIE INC. (US) 2016-05-24 US disclosed
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WO-2016075457-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED GASTROINTESTINAL DISORDERS TAKEDA CAMBRIDGE LIMITED (GB) 2016-05-19 WO disclosed
EP-2681221-B1 TRICYCLIC INHIBITORS OF KINASES ABBVIE INC (US) 2016-05-18 EP disclosed
EP-3019559-A1 WATER SOLUBLE FLUORESCENT OR COLORED DYES AND METHODS FOR THEIR USE Sony Corporation (JP) 2016-05-18 EP disclosed
EP-3019503-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF HIV INFECTIONS Gilead Sciences, Inc. (US) 2016-05-18 EP disclosed
EP-3019443-A1 HYBRID SEMICONDUCTING POLYMER NANOPARTICLES AS POLARIZATION SENSITIVE FLUORESCENT PROBES University Of Washington Through Its Center For Commercialization (US) 2016-05-18 EP disclosed
EP-3019499-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF HIV INFECTIONS Gilead Sciences, Inc. (US) 2016-05-18 EP disclosed
EP-3019505-A1 SUBSTITUTED PYRAZOLO-PYRIDINAMINES Bayer Pharma Aktiengesellschaft (DE) 2016-05-18 EP disclosed
CN-105593320-A Coating layer, coating solution, method for forming the coating layer, and method for producing medical tool KANEKA CORP 2016-05-18 CN disclosed
US-9340528-B2 Substituted aminoquinoxalines as tyrosine threonine kinase inhibitors BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-05-17 US disclosed
US-9340558-B2 Filamin a binding anti-inflammatory and analgesic PAIN THERAPEUTICS INC. (US) 2016-05-17 US disclosed
US-9340498-B2 Raft polymerisation COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESERACH ORGANISATION (AU) 2016-05-17 US disclosed
US-9339781-B2 Polymer particles THE UNIVERSITY OF SYDNEY (AU) 2016-05-17 US disclosed
US-20160130247-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 QUANTIEL PHARMACEUTICALS, INC. 2016-05-12 US disclosed
US-20160129001-A1 SUBSTITUTED [1,2,4]TRIAZOLO[4,3-a]PYRAZINES AS BRD4 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2016-05-12 US disclosed
EP-3016653-A1 PYRROLO-PYRROLE CARBAMATE AND RELATED ORGANIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND MEDICAL USES THEREOF Abide Therapeutics, Inc. (US) 2016-05-11 EP disclosed
EP-3016953-A1 PURINONE COMPOUNDS AS KINASE INHIBITORS Pharmacyclics, LLC (US) 2016-05-11 EP disclosed
EP-3017013-A1 REFRIGERATION SYSTEM WITH DUAL REFRIGERANTS AND LIQUID WORKING FLUIDS Xu, Yanjie (US) 2016-05-11 EP disclosed
US-9334264-B2 NAMPT inhibitors ABBVIE INC. (US) 2016-05-10 US disclosed
WO-2016069542-A2 LACTONE COMPOUNDS AND METHODS OF MAKING AND USING SAME THE SCRIPPS RESEARCH INSTITUTE (US) 2016-05-06 WO disclosed
US-20160122365-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2016-05-05 US disclosed
US-20160122317-A1 1-SULFONYL PIPERIDINE DERIVATIVES AS MODULATORS OF PROKINETICIN RECEPTORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-05-05 US disclosed
US-20160122314-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC 2016-05-05 US disclosed
US-20160120854-A1 PHARMACEUTICAL COMPOSITIONS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-05-05 US disclosed
US-20160122514-A1 SCRATCH RESISTANT POLYMERS MILLER WASTE MILLS INC. DBA RTP COMPANY 2016-05-05 US disclosed
EP-3013789-A2 AMINO ACID AND PEPTIDE CONJUGATES AND CONJUGATION PROCESS Auckland Uniservices Limited (NZ) 2016-05-04 EP disclosed
EP-2781520-B1 THREE-RING PI3K AND/OR MTOR INHIBITOR XUANZHU PHARMA CO LTD (CN) 2016-05-04 EP disclosed
EP-2739626-B1 NOVEL SPIROINDOLINE COMPOUNDS INTERVET INT BV (NL) 2016-05-04 EP disclosed
US-9326992-B2 Methods for treating progeroid laminopathies using oligonucleotide analogues targeting human LMNA SAREPTA THERAPEUTICS, INC. (US) 2016-05-03 US disclosed
US-9328112-B2 Tetracyclic CDK9 kinase inhibitors ABBVIE INC. (US) 2016-05-03 US disclosed
US-9328100-B2 Process for the preparation of β-C-arylglucosides SCINOPHARM TAIWAN, LTD. (TW) 2016-05-03 US disclosed
US-20160115131-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC 2016-04-28 US disclosed
US-20160115134-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2016-04-28 US disclosed
US-20160113914-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2016-04-28 US disclosed
US-20160113277-A1 Substituted 5-Hydroxy-2,3-Diphenylpentanonitrile Derivatives, Processes For Their Preparation And Their Use As Herbicides And/Or Plant Growth Regulators BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-04-28 US disclosed
US-20160113932-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS INFINITY PHARMACEUTICALS, INC. (US) 2016-04-28 US disclosed
US-20160115424-A1 FRAGRANCE COMPOSITIONS COMPRISING IONIC LIQUIDS THE PROCTER & GAMBLE COMPANY 2016-04-28 US disclosed
EP-3010928-A1 COMPOSITIONS AND METHODS FOR JOINT HEALTH Unigen, Inc. (US) 2016-04-27 EP disclosed
EP-3010900-A1 1-SULFONYL PIPERIDINE DERIVATIVES AS MODULATORS OF PROKINETICIN RECEPTORS Takeda Pharmaceutical Company Limited (JP) 2016-04-27 EP disclosed
EP-3010550-A2 CYCLIC PEPTIDES AS PROTEIN TARGETING AGENTS California Institute of Technology (US) 2016-04-27 EP disclosed
CN-102304300-B The solid particulate materials of polymeric encapsulate and comprise its discrete particle UNIV. OF SYDNEY (AU) 2016-04-27 CN disclosed
CN-105530814-A Use of selected pyridone carboxamides or salts thereof as active substances against abiotic plant stress BAYER CROPSCIENCE AG 2016-04-27 CN disclosed
US-9320739-B2 RAF kinase modulator compounds and methods of use thereof AMBIT BIOSCIENCES CORPORATION (US) 2016-04-26 US disclosed
US-9321749-B1 Heterocyclic compounds and uses thereof GLOBAVIR BIOSCIENCES, INC. (US) 2016-04-26 US disclosed
US-9321730-B2 Method of making and administering quinoline derivatives as anti-cancer agents THE HONG KONG POLYTECHNIC UNIVERSITY (HK) 2016-04-26 US disclosed
US-9320737-B2 Substituted imidazopyridazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-04-26 US disclosed
US-9321736-B2 Pyrimidine cyclohexyl glucocorticoid receptor modulators CORCEPT THERAPEUTICS, INC. (US) 2016-04-26 US disclosed
US-9321724-B2 Heteroaryl compounds with A-cyclic bridging unit INTERVET INC. (US) 2016-04-26 US disclosed
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US-20160108033-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2016-04-21 US disclosed
US-20160108019-A1 INHIBITORS OF KRAS G12C MUTANT PROTEINS ARAXES PHARMA LLC 2016-04-21 US disclosed
US-20160106749-A1 FATTY LIVER DISEASE TREATMENT USING GLUCOCORTICOID AND MINERALOCORTICOID RECEPTOR ANTAGONISTS CORCEPT THERAPEUTICS, INC. 2016-04-21 US disclosed
US-20160108046-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. 2016-04-21 US disclosed
US-20160107995-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2016-04-21 US disclosed
US-20160108032-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2016-04-21 US disclosed
WO-2016061195-A1 FATTY LIVER DISEASE TREATMENT USING GLUCOCORTICOID AND MINERALOCORTICOID RECEPTOR ANTAGONISTS CORCEPT THERAPEUTICS, INC. (US) 2016-04-21 WO disclosed
WO-2016061562-A2 BUTYRYLCHOLINESTERASE ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC. (US) 2016-04-21 WO disclosed
WO-2016061097-A1 ATAXIA TELENGIECTASIA AND RAD3-RELATED (ATR) PROTEIN KINASE INHIBITORS Atrin Pharmaceuticals LLC (US) 2016-04-21 WO disclosed
US-20160108436-A1 SYNTHESIS OF OLEFINIC ALCOHOLS VIA ENZYMATIC TERMINAL HYDROXYLATION PROVIVI, INC. (US) 2016-04-21 US disclosed
EP-3008061-A1 NOVEL COMPOUNDS FOR THE TREATMENT OF CANCER Bayer Pharma Aktiengesellschaft (DE) 2016-04-20 EP disclosed
EP-3009436-A1 KINASE INHIBITORS AND METHODS OF USE Intellikine, LLC (US) 2016-04-20 EP disclosed
EP-2590965-B1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX INC (US) 2016-04-20 EP disclosed
CN-105517949-A Hybrid semiconducting polymer nanoparticles as polarization sensitive fluorescent probes UNIV OF WASHINGTON CENTER FOR COMMERCIALIZATION 2016-04-20 CN disclosed
CN-103228141-B Substituted fused pyrimidinones and dihydropyrimidinones BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-04-20 CN disclosed
US-9315505-B2 Heterocyclic compounds and uses thereof INTELLIKINE LLC (US) 2016-04-19 US disclosed
US-9314467-B2 Styrenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2016-04-19 US disclosed
US-9315509-B2 Diamine derivatives as inhibitors of leukotriene A4 hydrolase CELTAXSYS, INC. (US) 2016-04-19 US disclosed
WO-2016057242-A1 HIF-2α INHIBITORS FOR TREATING IRON OVERLOAD DISORDERS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2016-04-14 WO disclosed
WO-2016057600-A1 NOVEL PRECATALYST SCAFFOLDS FOR CROSS-COUPLING REACTIONS, AND METHODS OF MAKING AND USING SAME YALE UNIVERSITY (US) 2016-04-14 WO disclosed
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO disclosed
WO-2016054689-A1 ALL PURPOSE RAFT AGENT COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2016-04-14 WO disclosed
US-20160102307-A1 OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2016-04-14 US disclosed
US-20160102104-A1 Ataxia Telengiectasia And Rad3-Related (ATR) Protein Kinase Inhibitors Atrin Pharmaceuticals LLC (US) 2016-04-14 US disclosed
EP-3003309-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS Infinity Pharmaceuticals, Inc. (US) 2016-04-13 EP disclosed
EP-3004093-A1 SUBSTITUTED TRIAZOLOPYRIDINES HAVING ACTIVITY AS MPS-1 INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2016-04-13 EP disclosed
EP-3004239-A1 SCRATCH RESISTANT POLYMERS Tenasitech Pty Ltd. (AU) 2016-04-13 EP disclosed
EP-2766359-B1 HETEROCYCLIC COMPOUNDS AND USE THEREOF AS MODULATORS OF TYPE III RECEPTOR TYROSINE KINASES AMBIT BIOSCIENCES CORP (US) 2016-04-13 EP disclosed
EP-3003381-A1 PHARMACEUTICAL COMPOSITIONS Bayer Pharma Aktiengesellschaft (DE) 2016-04-13 EP disclosed
EP-3004083-A1 COMPOUNDS FOR TREATMENT OF DRUG RESISTANT AND PERSISTENT TUBERCULOSIS The California Institute for Biomedical Research (US) 2016-04-13 EP disclosed
US-9309508-B2 Boronic and borinic acid compound as inhibitors of sulfenic acid-containing proteins THE PENN STATE RESEARCH FOUNDATION (US) 2016-04-12 US disclosed
US-9308207-B2 JAK kinase modulating compounds and methods of use thereof AMBIT BIOSCIENCES CORP. (US) 2016-04-12 US disclosed
US-9309211-B2 Arylalkene derivatives and use thereof as selective estrogen receptor modulators CENTAURUS BIOPHARMA CO., LTD. (CN) 2016-04-12 US disclosed
US-9309259-B2 Process for ixabepilone, and intermediates thereof SCINOPHARM TAIWAN, LTD. (TW) 2016-04-12 US disclosed
WO-2016054491-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2016-04-07 WO disclosed
US-20160096869-A1 CHLOROTOXIN CONJUGATES AND METHODS OF USE THEREOF Blaze Bioscience, Inc. 2016-04-07 US disclosed
EP-2807166-B1 5,8-DIHYDRO-6H-PYRAZOLO[3,4-H]QUINAZOLINES AS IGF-1R/IR INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2016-04-06 EP disclosed
EP-2611300-B1 SUBSTITUTED ANNELATED DIHYDROPYRIMIDINONE COMPOUNDS BAYER IP GMBH (DE) 2016-04-06 EP disclosed
US-9302989-B2 NAMPT and rock inhibitors ABBVIE INC. (US) 2016-04-05 US disclosed
US-9301951-B2 Compounds and methods for inhibiting phosphate transport ARDELYX, INC. (US) 2016-04-05 US disclosed
US-9302993-B2 8-hydroxy quinoline derivatives PRANA BIOTECHNOLOGY LIMITED (AU) 2016-04-05 US disclosed
US-9303026-B2 Antiviral agents BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2016-04-05 US disclosed
WO-2016049568-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF RAS ARAXES PHARMA LLC (US) 2016-03-31 WO disclosed
WO-2016049565-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS ARAXES PHARMA LLC (US) 2016-03-31 WO disclosed
US-20160089371-A1 Combination of Kinase Inhibitors and Uses Thereof INTELLIKINE LLC 2016-03-31 US disclosed
WO-2016049390-A1 FRAGRANCE COMPOSITIONS COMPRISING IONIC LIQUIDS THE PROCTER & GAMBLE COMPANY (US) 2016-03-31 WO disclosed
WO-2016048982-A2 COMBINATION TREATMENT WITH PI3Kα INHIBITORS AND TAXANES MILLENNIUM PHARMACEUTICALS, INC. (US) 2016-03-31 WO disclosed
WO-2016046530-A1 NOVEL COMPOUNDS MISSION THERAPEUTICS LTD (GB) 2016-03-31 WO disclosed
WO-2016049391-A1 IONIC LIQUIDS THE PROCTER & GAMBLE COMPANY (US) 2016-03-31 WO disclosed
CN-105451553-A Substituted 5-hydroxy-2,3-diphenylpentanonitrile derivatives, processes for their preparation and their use as herbicides and/or plant growth regulators BAYER CROPSCIENCE AG 2016-03-30 CN disclosed
US-9296748-B2 Pyridinones BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-03-29 US disclosed
US-9296723-B2 NAMPT inhibitors ABBVIE INC. (US) 2016-03-29 US disclosed
US-9296742-B2 Heterocyclic kinase inhibitors INTELLIKINE LLC (US) 2016-03-29 US disclosed
US-9296757-B2 Substituted benzothienopyrimidines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-03-29 US disclosed
US-9295673-B2 Combination of mTOR inhibitors and P13-kinase inhibitors, and uses thereof INTELLIKINE LLC (US) 2016-03-29 US disclosed
US-9296665-B2 Synthesis of drop-in liquid fuels and chemicals from methanol, ethanol or syngas using mixed catalysts Pioneer Energy Inc. (US) 2016-03-29 US disclosed
US-9296722-B2 Azolyl urea compounds and methods of use thereof AMBIT BIOSCIENCES CORPORATION (US) 2016-03-29 US disclosed
WO-2016044770-A1 SPIROCYCLIC HAT INHIBITORS AND METHODS FOR THEIR USE ABBVIE INC. (US) 2016-03-24 WO disclosed
WO-2016044771-A1 HAT INHIBITORS AND METHODS FOR THEIR USE ABBVIE INC. (US) 2016-03-24 WO disclosed
US-20160083379-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2016-03-24 US disclosed
WO-2016044429-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2016-03-24 WO disclosed
WO-2016044777-A1 HAT INHIBITORS AND METHODS FOR THEIR USE ABBVIE INC. (US) 2016-03-24 WO disclosed
WO-2016044138-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2016-03-24 WO disclosed
WO-2016044342-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2016-03-24 WO disclosed
WO-2016044772-A1 COMBINATION THERAPIES FOR TREATMENT OF CANCER ARAXES PHARMA LLC (US) 2016-03-24 WO disclosed
WO-2016044792-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL HYDRA BIOSCIENCES, INC. (US) 2016-03-24 WO disclosed
US-20160083387-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO AQUINOX PHARMACEUTICALS CANADA INC (CA) 2016-03-24 US disclosed
EP-2794568-B1 SUBSTITUTED 4-CYANO-3-PHENYL-4-(PYRIDIN-3-YL) BUTANOATES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER IP GMBH (DE) 2016-03-23 EP disclosed
EP-2091527-B1 SULFIDE, SULFOXIDE AND SULFONE CHALCONE ANALOGUES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF UNIV TEMPLE (US) 2016-03-23 EP disclosed
EP-2367824-B1 Anti-viral derivatives of pyrimidine ABBVIE INC (US) 2016-03-23 EP disclosed
EP-2373648-B1 SUBSTITUTED 1-(THIAZOLYL)- AND 1-(ISOTHIAZOLYL)PYRAZOL-4-YL ACETIC ACIDS, METHOD FOR THEIR PRODUCTION AND THEIR USE AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER IP GMBH (DE) 2016-03-23 EP disclosed
US-9289429-B2 Compounds and methods for inhibiting phosphate transport ARDELYX, INC. (US) 2016-03-22 US disclosed
US-9289430-B2 Compounds and methods for inhibiting phosphate transport ARDELYX, INC. (US) 2016-03-22 US disclosed
US-9290507-B2 B-RAF kinase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-03-22 US disclosed
US-9290456-B2 Pyridazinone compounds and their use as DAAO inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-03-22 US disclosed
US-9290497-B2 Processes for preparing isoquinolinones and solid forms of isoquinolinones INFINITY PHARMACEUTICALS, INC. (US) 2016-03-22 US disclosed
US-9290482-B2 2016-03-22 US disclosed
WO-2016037221-A1 LIGHT ACTIVATED ELECTROCHEMISTRY NEWSOUTH INNOVATIONS PTY LIMITED (AU) 2016-03-17 WO disclosed
WO-2016040330-A1 THIENOPYRIMIDINE AND THIENOPYRIDINE COMPOUNDS AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2016-03-17 WO disclosed
US-20160075716-A1 POLYMERIC MATERIALS COMMONWEALTH SCIENTIFIC INDUSTRIAL AND RESEARCH ORGANISATION (AU) 2016-03-17 US disclosed
US-20160075684-A1 ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS AND USES THEREOF-III MERCK SHARP & DOHME CORP. (US) 2016-03-17 US disclosed
EP-2691375-B1 SUBSTITUTED BENZIMIDAZOLES AS MPS-1 KINASE INHIBITORS BAYER IP GMBH (DE) 2016-03-16 EP disclosed
EP-2619232-B1 CONTINUOUS FLOW POLYMERISATION PROCESS COMMW SCIENT IND RES ORG (AU) 2016-03-16 EP disclosed
US-9284319-B2 Heterocyclyl aminoimidazopyridazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-03-15 US disclosed
US-9284315-B2 Three-ring PI3K and/or mTOR inhibitor ZUANZHU PHARMA CO., LTD. (CN) 2016-03-15 US disclosed
US-9284317-B2 Substituted imidazo[1,2-a]pyrazines as MPS-1 inhibitors BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-03-15 US disclosed
WO-2016037005-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Quanticel Pharmaceuticals, Inc. (US) 2016-03-10 WO disclosed
US-20160067296-A1 Compositions and Methods for Joint Health UNIGEN, INC. (US) 2016-03-10 US disclosed
US-20160068524-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELLTAXIS, LLC 2016-03-10 US disclosed
US-20160068534-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELLTAXIS, LLC 2016-03-10 US disclosed
US-20160067242-A1 NHE3-BINDING COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. 2016-03-10 US disclosed
US-20160068522-A1 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELLTAXIS, LLC 2016-03-10 US disclosed
US-20160068507-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2016-03-10 US disclosed
EP-2993165-A2 COMPOUNDS WITH (SUBSTITUTED PHENYL)-PROPENAL MOIETY, THEIR DERIVATIVES, BIOLOGICAL ACTIVITY, AND USE THEREOF Allianz Pharmascience Ltd (TW) 2016-03-09 EP disclosed
EP-2822954-B1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES INC (US) 2016-03-09 EP disclosed
EP-1685119-B1 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS ABBVIE BAHAMAS LTD (BS) 2016-03-09 EP disclosed
CN-101605763-B Radioprotector compounds and methods involving PETER MACCALLUM CANCER INSTITUTE (AU) 2016-03-09 CN disclosed
US-9278102-B2 Compounds and methods for inhibiting phosphate transport ARDELYX, INC. (US) 2016-03-08 US disclosed
US-9278922-B2 Anti-viral compounds ABBVIE INC. (US) 2016-03-08 US disclosed
US-9278978-B2 6-Alkynyl Pyridine BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-03-08 US disclosed
US-9278987-B2 Functionally-modified oligonucleotides and subunits thereof SAREPTA THERAPEUTICS, INC. (US) 2016-03-08 US disclosed
US-20160060258-A1 2-AMINOPYRIDO[4,3-D]PYRIMIDIN-5-ONE DERIVATIVES AND THEIR USE AS WEE-1 INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2016-03-03 US disclosed
US-20160060257-A1 PYRROLO [2,3-B] PYRIDINE CDK9 KINASE INHIBITORS ABBVIE INC. (US) 2016-03-03 US disclosed
US-20160060247-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC 2016-03-03 US disclosed
EP-2498600-B1 FILAMIN A-BINDING ANTI-INFLAMMATORY ANALGESIC PAIN THERAPEUTICS INC (US) 2016-03-02 EP disclosed
US-20160050895-A1 TRANSGENIC NON-HUMAN ORGANISMS WITH NON-FUNCTIONAL TSPO GENES THE UNIVERSITY OF SYDNEY (AU) 2016-02-25 US disclosed
US-20160052938-A1 SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-02-25 US disclosed
WO-2016026937-A1 NEW SPIRO[3H-INDOLE-3,2´-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-02-25 WO disclosed
US-20160052898-A1 NOVEL COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-02-25 US disclosed
EP-2628481-B1 Trisubstituted heterocycles as replication inhibitors of hepatitis C virus HCV ABBVIE BAHAMAS LTD (BS) 2016-02-24 EP disclosed
EP-2307013-B1 PAIN-RELIEVING COMPOSITIONS OF FUROXAN NO DONORS AND USES THEREOF UNIV QUEENSLAND (AU) 2016-02-24 EP disclosed
CN-105358617-A Scratch resistant polymers TENASITECH PTY LTD 2016-02-24 CN disclosed
US-9266877-B2 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases ABBVIE INC. (US) 2016-02-23 US disclosed
US-9266919-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2016-02-23 US disclosed
US-9266891-B2 Substituted [1,2,4]triazolo[4,3-A]pyrazines that are BRD4 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-02-23 US disclosed
WO-2016023832-A1 THIENO- AND FURO[2,3-D]PYRIMIDINE-2,4[1H,3H]-DIONE DERIVATIVES AS TRPC5 MODULATORS FOR THE TREATMENT OF NEUROPSYCHIATRIC DISORDERS HYDRA BIOSCIENCES, INC. (US) 2016-02-18 WO disclosed
US-20160045559-A1 COMPOSITIONS AND METHODS FOR MANAGING OR IMPROVING BONE DISORDERS, CARTILAGE DISORDERS, OR BOTH UNIGEN, INC. (KR) 2016-02-18 US disclosed
WO-2016024232-A1 THERAPEUTIC COMBINATIONS OF A BTK INHIBITOR, A PI3K INHIBITOR, A JAK-2 INHIBITOR AND/OR A CDK 4/6 INHIBITOR ACERTA PHARMA B.V. (NL) 2016-02-18 WO disclosed
WO-2016023826-A1 QUINAZOLINE-2,4(1H,3H)-DIONE DERIVATIVES AS TRCP5 MODULATORS FOR THE TREATMENT OF NEUROPSYCHIATRY DISORDERS HYDRA BIOSCIENCES, INC. (US) 2016-02-18 WO disclosed
WO-2016024231-A1 THERAPEUTIC COMBINATIONS OF A BTK INHIBITOR, A PI3K INHIBITOR, A JAK-2 INHIBITOR, A PD-1 INHIBITOR AND/OR A PD-L1 INHIBITOR ACERTA PHARMA B.V. (NL) 2016-02-18 WO disclosed
WO-2016023830-A1 PYRIDO[2,3-D]PYRIMIDINE-2,4(1H,3H)-DIONE DERIVATIVES HYDRA BIOSCIENCES, INC. (US) 2016-02-18 WO disclosed
US-20160046635-A1 NOVEL BREATHING CONTROL MODULATING COMPOUNDS, AND METHODS OF USING SAME GALLEON PHARMACEUTICALS, INC. 2016-02-18 US disclosed
WO-2016024227-A1 BTK INHIBITORS TO TREAT SOLID TUMORS THROUGH MODULATION OF THE TUMOR MICROENVIRONMENT ACERTA PHARMA B.V. (NL) 2016-02-18 WO disclosed
WO-2016025816-A1 FATTY ACID SYNTHASE INHIBITOR FOR USE IN THE TREATMENT OF DRUG RESISTANT CANCER 3-V BIOSCIENCES, INC. (US) 2016-02-18 WO disclosed
WO-2016023825-A1 PYRIDO[3,4-D]PYRIMIDINE-2,4(1H,3H)-DIONE DERIVATIVES HYDRA BIOSCIENCES, INC. (US) 2016-02-18 WO disclosed
WO-2016024228-A1 THERAPEUTIC COMBINATIONS OF A BTK INHIBITOR, A PI3K INHIBITOR, A JAK-2 INHIBITOR, A PD-1 INHIBITOR AND/OR A PD-L1 INHIBITOR ACERTA PHARMA B.V. (NL) 2016-02-18 WO disclosed
WO-2016024230-A1 THERAPEUTIC COMBINATIONS OF A BTK INHIBITOR, A PI3K INHIBITOR, A JAK-2 INHIBITOR, AND/OR A BCL-2 INHIBITOR ACERTA PHARMA B.V. (NL) 2016-02-18 WO disclosed
WO-2016023831-A1 PYRROLO[3,2-D]PYRIMIDINE-2,4(3H,5H)-DIONE DERIVATIVES HYDRA BIOSCIENCES, INC. (US) 2016-02-18 WO disclosed
US-20160046624-A1 PYRIDO[2,3-d]PYRIMIDINE-2,4(1H,3H)-DIONE DERIVATIVES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-02-18 US disclosed
EP-1877481-B1 STABILISER COMPOSITION FOR HALIDE-CONTAINING POLYMERS SUN ACE KAKOH PTE LTD (SG) 2016-02-17 EP disclosed
US-9260441-B2 Heteroaryl compounds with cyclic bridging unit INTERVET INC. (US) 2016-02-16 US disclosed
US-9260655-B2 Alkyl-acid ligands for nanocrystals NANOSYS, INC. (US) 2016-02-16 US disclosed
US-9259402-B2 Compounds with (1 E, 6E)-1,7-bis-(3,4-dimethoxyphenyI)-4,4-disubstituted-hepta-1,6-diene-3,5-dione structural scaffold, their biological activity, and uses thereof ALLIANZ PHARMASCIENCE LTD. (TW) 2016-02-16 US disclosed
US-9260367-B2 Methods of converting polyols Univesity of Washington Through Its Center For Communication (US) 2016-02-16 US disclosed
US-20160039808-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC 2016-02-11 US disclosed
US-20160038606-A1 CYTOTOXIC AND ANTI-MITOTIC COMPOUNDS, AND METHODS OF USING THE SAME ZYMEWORKS BC INC. (CA) 2016-02-11 US disclosed
US-20160038455-A1 S1P RECEPTORS MODULATORS AND THEIR USE THEREOF AKAAL PHARMA PTY LTD. (AU) 2016-02-11 US disclosed
WO-2016020901-A1 METHODS OF TREATING CANCERS, IMMUNE AND AUTOIMMUNE DISEASES, AND INFLAMMATORY DISEASES BASED ON BTK OCCUPANCY AND BTK RESYNTHESIS RATE ACERTA PHARMA B.V. (NL) 2016-02-11 WO disclosed
US-20160039831-A1 PYRROLO[3,2-d]PYRIMIDINE-2,4(3H,5H)-DIONE DERIVATIVES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-02-11 US disclosed
WO-2016020320-A1 2-(MORPHOLIN-4-YL)-L,7-NAPHTHYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-02-11 WO disclosed
US-20160039772-A1 QUINAZOLINE-2,4(1H,3H)-DIONE DERIVATIVES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-02-11 US disclosed
US-20160039814-A1 6-ALKYNYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-02-11 US disclosed
US-20160040199-A1 ENZYMATIC METHODS FOR NITROGEN-ATOM TRANSFER CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2016-02-11 US disclosed
US-20160039723-A1 STEREODYNAMIC CHEMOSENSORS GEORGETOWN UNIVERSITY (US) 2016-02-11 US disclosed
US-20160039815-A1 PYRIDO[3,4-d]PYRIMIDINE-2,4(1H,3H)-DIONE DERIVATIVES HYDRA BIOSCIENCES, INC. 2016-02-11 US disclosed
US-20160039841-A1 THIENO- AND FURO[2,3-d]PYRIMIDINE-2,4[1H,3H]-DIONE DERIVATIVES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-02-11 US disclosed
US-20160038497-A1 Enhanced Treatment Regimens Using mTOR Inhibitors FAETH THERAPEUTICS, INC. 2016-02-11 US disclosed
CN-102858437-B For the substrate and preparation method thereof of fixed function material TEMASEK POLYTECHNIC (SG) 2016-02-10 CN disclosed
US-9255198-B2 Water swellable polymer materials comprising particulate core and water swellable R.A.F.T polymer shell THE UNIVERSITY OF SYDNEY (AU) 2016-02-09 US disclosed
US-9255097-B2 Inhibitors of lysine specific demethylase-1 Quanticel Pharmaceuticals, Inc. (US) 2016-02-09 US disclosed
US-9255108-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2016-02-09 US disclosed
US-9255100-B2 Substituted imidazopyridazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-02-09 US disclosed
US-20160031813-A1 Nampt Inhibitors ABBVIE INC. 2016-02-04 US disclosed
WO-2016019237-A2 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC (US) 2016-02-04 WO disclosed
WO-2016019233-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC (US) 2016-02-04 WO disclosed
US-20160031891-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC 2016-02-04 US disclosed
US-20160031776-A1 Preparation of Butanol from Ethanol Derived from Fermentation PIONEER ENERGY, INC. (US) 2016-02-04 US disclosed
US-20160031899-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO AQUINOX PHARMACEUTICALS CANADA INC (CA) 2016-02-04 US disclosed
US-20160032330-A1 P-450-CATALYZED ENANTIOSELECTIVE CYCLOPROPANATION OF ELECTRON-DEFICIENT OLEFINS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2016-02-04 US disclosed
US-20160031886-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE LLC 2016-02-04 US disclosed
US-20160031880-A1 Nampt and Rock Inhibitors ABBVIE INC. (US) 2016-02-04 US disclosed
EP-2978758-A1 DIHYDROQUINAZOLINONE ANALOGUES AS BRD4 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2016-02-03 EP disclosed
EP-2685827-B1 PYRIMIDINE CYCLOHEXYL GLUCOCORTICOID RECEPTOR MODULATORS CORCEPT THERAPEUTICS INC (US) 2016-02-03 EP disclosed
EP-2980088-A1 Amino-substituted isothiazoles Bayer Pharma Aktiengesellschaft (DE) 2016-02-03 EP disclosed
EP-2978757-A1 INDOLINONE ANALOGUES AS BRD4 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2016-02-03 EP disclosed
CN-105308041-A Preparation method for ixabepilone and intermediate thereof SCINOPHARM TAIWAN LTD 2016-02-03 CN disclosed
US-9249138-B2 Anti-viral compounds ABBVIE INC. (US) 2016-02-02 US disclosed
US-9248193-B2 Formulations of phenyl uracil compounds ABBVIE INC. (US) 2016-02-02 US disclosed
US-9249151-B2 Bis-amido pyridines BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-02-02 US disclosed
WO-2016012477-A1 AMINO-SUBSTITUTED ISOXAZOLES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-01-28 WO disclosed
US-20160024099-A1 KINASE INHIBITORS AND METHODS OF USE INTELLIKINE LLC 2016-01-28 US disclosed
WO-2016012481-A1 GLUCOSE TRANSPORT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-01-28 WO disclosed
US-20160022642-A1 Compounds Useful for Promoting Protein Degradation and Methods Using Same YALE UNIVERSITY 2016-01-28 US disclosed
US-20160022692-A1 TREATMENT OF RHEUMATOID ARTHRITIS AND ASTHMA USING PI3 KINASE INHIBITORS INFINITY PHARMACEUTICALS, INC. 2016-01-28 US disclosed
WO-2016012474-A1 GLUCOSE TRANSPORT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-01-28 WO disclosed
EP-2977376-A1 Amino-substituted isoxazoles Bayer Pharma Aktiengesellschaft (DE) 2016-01-27 EP disclosed
EP-2670749-B1 NEW AZAINDOLYLPHENYL SULFONAMIDES AS SERINE/THREONINE KINASE INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2016-01-27 EP disclosed
EP-2316827-B1 Piperazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC (CA) 2016-01-27 EP disclosed
EP-2977377-A1 Amino-substituted isoxazoles Bayer Pharma Aktiengesellschaft (DE) 2016-01-27 EP disclosed
EP-2976327-A2 3-ACETYLAMINO-1-(PHENYL-HETEROARYL-AMINOCARBONYL OR PHENYL-HETEROARYL-CARBONYLAMINO)BENZENE DERIVATIVES FOR THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS Bayer Pharma Aktiengesellschaft (DE) 2016-01-27 EP disclosed
EP-2976343-A2 SUBSTITUTED N-BIPHENYL-3-ACETYLAMINO-BENZAMIDES AND N-[3-(ACETYLAMINO)PHENYL]-BIPHENYL-CARBOXAMIDES AND THEIR USE AS INHIBITORS OF THE WNT SIGNALLING PATHWAY Bayer Pharma Aktiengesellschaft (DE) 2016-01-27 EP disclosed
US-9242968-B2 Histone demethylase inhibitors Quanticel Pharmaceuticals, Inc. (US) 2016-01-26 US disclosed
US-9242945-B2 Substituted 2-benzylidene-2H-benzo[b][1,4]thiazin-3(4H)-ones, derivatives thereof, and therapeutic uses thereof Temple University—Of the Commonwealth System of Higher Education (US) 2016-01-26 US disclosed
US-20160018395-A1 POLYMER DOT COMPOSITIONS AND RELATED METHODS UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION 2016-01-21 US disclosed
US-20160015786-A1 MOBILIZING AGENTS AND USES THEREFOR MATER MEDICAL RESEARCH INSTITUTE LIMITED (AU) 2016-01-21 US disclosed
WO-2016011209-A1 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2016-01-21 WO disclosed
US-20160018405-A1 METHODS AND SYSTEMS FOR ANALYSIS USING POLYMER DOTS University of Washington Through it's Center for Commercialization (US) 2016-01-21 US disclosed
US-20160017099-A1 Silicone Ligands for Quantum Dots SHOEI CHEMICAL INC. (JP) 2016-01-21 US disclosed
US-20160016957-A1 CHEMICAL COMPOUNDS, COMPOSITIONS AND METHODS FOR KINASE MODULATION INFINITY PHARMACEUTICALS, INC. 2016-01-21 US disclosed
EP-2972349-A1 POLYMER DOT COMPOSITIONS AND RELATED METHODS University Of Washington Through Its Center For Commercialization (US) 2016-01-20 EP disclosed
EP-2668178-B1 NEW 5-ALKYNYL-PYRIDINES BOEHRINGER INGELHEIM INT (DE) 2016-01-20 EP disclosed
EP-2971007-A1 TRANSGENIC NON-HUMAN ORGANISMS WITH NON-FUNCTIONAL TSPO GENES AUSTRALIAN NUCLEAR SCIENCE AND TECHNOLOGY ORGANISATION (AU) 2016-01-20 EP disclosed
EP-2969007-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals Inc (US) 2016-01-20 EP disclosed
EP-2972258-A1 PURIFICATION OF RAPAMYCIN DERIVATIVES Biosensors International Group, Ltd. (SG) 2016-01-20 EP disclosed
EP-2968329-A1 NOVEL BREATHING CONTROL MODULATING COMPOUNDS, AND METHODS OF USING SAME Galleon Pharmaceuticals, Inc. (US) 2016-01-20 EP disclosed
EP-2970316-A2 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF Hydra Biosciences, Inc. (US) 2016-01-20 EP disclosed
EP-2968265-A2 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Celtaxsys Inc. (US) 2016-01-20 EP disclosed
EP-2970100-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO Aquinox Pharmaceuticals (Canada) Inc. (CA) 2016-01-20 EP disclosed
EP-2970264-A1 PYRROLO[2,3-B]PYRIDINE CDK9 KINASE INHIBITORS AbbVie Inc. (US) 2016-01-20 EP disclosed
EP-2970299-A1 PYRROLOPYRIMINDINE CDK9 KINASE INHIBITORS Abbvie Inc. (US) 2016-01-20 EP disclosed
EP-2970122-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO Aquinox Pharmaceuticals (Canada) Inc. (CA) 2016-01-20 EP disclosed
EP-2968440-A1 CYTOTOXIC AND ANTI-MITOTIC COMPOUNDS, AND METHODS OF USING THE SAME Centre For Drug Research And Development (CA) 2016-01-20 EP disclosed
EP-2970211-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals Inc (US) 2016-01-20 EP disclosed
EP-2970205-A2 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE Tolero Pharmaceuticals, Inc. (US) 2016-01-20 EP disclosed
EP-2968264-A2 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Celtaxsys Inc. (US) 2016-01-20 EP disclosed
EP-2970309-A2 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Celtaxsys Inc. (US) 2016-01-20 EP disclosed
EP-2968340-A1 COMBINATION OF KINASE INHIBITORS AND USES THEREOF Intellikine, LLC (US) 2016-01-20 EP disclosed
EP-2970099-A1 SUBSTITUTED 3-PHENYLPROPYLAMINE DERIVATIVES FOR THE TREATMENT OF OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2016-01-20 EP disclosed
EP-2970200-A1 PYRIDINE CDK9 KINASE INHIBITORS Abbvie Inc. (US) 2016-01-20 EP disclosed
EP-2970121-A1 COVALENT INHIBITORS OF KRAS G12C Araxes Pharma LLC (US) 2016-01-20 EP disclosed
CN-105263855-A Western blot analysis using polymer dots UNIV WASHINGTON CT COMMERCIALIZATION 2016-01-20 CN disclosed
WO-2016005577-A1 USE OF ANTHELMINTIC AGENTS AGAINST DIROFILARIA IMMITIS INTERVET INTERNATIONAL B.V. (NL) 2016-01-14 WO disclosed
US-20160009734-A1 SUBSTITUTED THIAZOLOPYRIMIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-01-14 US disclosed
EP-2964645-A1 PROCESS FOR IXABEPILONE, AND INTERMEDIATES THEREOF Scinopharm Taiwan Ltd. (TW) 2016-01-13 EP disclosed
EP-2964656-A1 SUBSTITUTED THIAZOLOPYRIMIDINES Bayer Pharma Aktiengesellschaft (DE) 2016-01-13 EP disclosed
EP-2614063-B1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER IP GMBH (DE) 2016-01-13 EP disclosed
EP-2964565-A1 WESTERN BLOT ANALYSIS USING POLYMER DOTS University Of Washington Through Its Center For Commercialization (US) 2016-01-13 EP disclosed
CN-102612514-B Anti influenza agent GRIFFITH UNIVERSITY (AU) 2016-01-13 CN disclosed
CN-105247010-A Method for solventless quantum dot exchange NANOSYS INC 2016-01-13 CN disclosed
WO-2016004105-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Quanticel Pharmaceuticals, Inc. (US) 2016-01-07 WO disclosed
WO-2016003917-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Quanticel Pharmaceuticals, Inc. (US) 2016-01-07 WO disclosed
WO-2016004272-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC (US) 2016-01-07 WO disclosed
WO-2016004305-A2 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC (US) 2016-01-07 WO disclosed
US-20160002245-A1 SUBSTITUTED PYRAZOLOPYRIMIDINYLAMINO-INDAZOLES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2016-01-07 US disclosed
WO-2016001376-A1 NEW SPIRO[3H-INDOLE-3,2´-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-01-07 WO disclosed
US-20160002682-A1 IN VIVO AND IN VITRO OLEFIN CYCLOPROPANATION CATALYZED BY HEME ENZYMES UNITED STATES DEPARTMENT OF ENERGY 2016-01-07 US disclosed
US-20160004163-A1 LITHOGRAPHICALLY PRODUCED FEATURES THE UNIVERSITY OF QUEENSLAND (AU) 2016-01-07 US disclosed
US-20160000764-A1 NEW SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-01-07 US disclosed
US-20160002262-A1 PURIFICATION OF RAPAMYCIN DERIVATIVES USING TEMPERATURE INDUCED PHASE SEPARATION BIOSENSORS INTERNATIONAL GROUP, LTD. (BM) 2016-01-07 US disclosed
US-20160002225-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE SCHRODINGER, LLC 2016-01-07 US disclosed
US-20160002201-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2016-01-07 US disclosed
US-20160002241-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS, LLC. (US) 2016-01-07 US disclosed
EP-2802595-B1 PROCESSES FOR MAKING HCV PROTEASE INHIBITORS ABBVIE INC (US) 2016-01-06 EP disclosed
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US-9226505-B2 4-substituted 1-phenylpyrazole-3-carboxylic acid derivatives as agents against abiotic plant stress BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-01-05 US disclosed
US-9227983-B2 Taxane and abeo-taxane analogs Arbor Therapeutics, LLC (US) 2016-01-05 US disclosed
US-9227978-B2 Covalent inhibitors of Kras G12C ARAXES PHARMA LLC (US) 2016-01-05 US disclosed
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US-20150376189-A1 AMIDOIMIDAZOPYRIDAZINES AS MKNK-1 KINASE INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-12-31 US disclosed
US-20150376179-A1 PIPERIDIN-1 -YL AND AZEPIN-1 -YL CARBOXYLATES AS MUSCARINIC M4 RECEPTOR AGONISTS NXERA PHARMA UK LIMITED (GB) 2015-12-31 US disclosed
US-20150376141-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2015-12-31 US disclosed
US-20150376169-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2015-12-31 US disclosed
US-20150374706-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR TREATMENT OF BREATHING CONTROL DISORDERS OR DISEASES GALLEON PHARMACEUTICALS, INC. 2015-12-31 US disclosed
US-20150376271-A1 DUAL PDGF/VEGF ANTAGONISTS OLIGASIS, LLC (US) 2015-12-31 US disclosed
WO-2015200905-A2 DUAL PDGF/VEGF ANTAGONISTS OLIGASIS, LLC (US) 2015-12-30 WO disclosed
WO-2015198045-A1 3-SUBSTITUTED 2-AMINO-INDOLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-12-30 WO disclosed
WO-2015198046-A1 1,3-SUBSTITUTED 2-AMINOINDOLE DERIVATIVES AND ANALOGUES USEFUL IN THE TREATMENT OR PREVENTION OF DIABETES MELLITUS, OBESITY AND INFLAMMATORY BOWEL DISEASE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-12-30 WO disclosed
WO-2015200843-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Quanticel Pharmaceuticals, Inc. (US) 2015-12-30 WO disclosed
WO-2015196258-A1 ENZYME INTERACTING AGENTS MONASH UNIVERSITY (AU) 2015-12-30 WO disclosed
EP-2958920-A1 SUBSTITUTED-IMIDAZO[1,2-B]PYRIDAZINES AS MKNK1 INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2015-12-30 EP disclosed
CN-105209916-A Polymer dot compositions and related methods UNIV WASHINGTON CT COMMERCIALIZATION 2015-12-30 CN disclosed
US-20150368264-A1 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES, INC. 2015-12-24 US disclosed
US-20150368250-A1 IMIDAZOPYRIDAZINES AS AKT KINASE INHIBITORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-12-24 US disclosed
EP-2483249-B1 PYRIMIDINE DERIVATIVES AS PROTEIN TYROSINE KINASE 2 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2015-12-23 EP disclosed
WO-2015195656-A2 SYNTHESIS OF POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS GILEAD SCIENCES ,INC. (US) 2015-12-23 WO disclosed
WO-2015195228-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD PHARMACEUTICALS, INC. (US) 2015-12-23 WO disclosed
WO-2015192175-A1 POLYMER HYDROGEL THE UNIVERSITY OF QUEENSLAND (AU) 2015-12-23 WO disclosed
CN-105189584-A Alkyl-acid ligands for nanocrystals NANOSYS INC 2015-12-23 CN disclosed
CN-103502282-B Amine-functionalized polyolefine and preparation method thereof EXXONMOBIL CHEMICAL PATENTS INC. (US) 2015-12-23 CN disclosed
US-9216996-B2 Substituted 2,3,4,5,7,9,13,13a-octahydropyrido[1′,2′:4,5]pyrazino[2,1-b][1,3]oxazepines and methods for treating viral infections GILEAD SCIENCES, INC. (US) 2015-12-22 US disclosed
US-9216982-B2 Certain chemical entities, compositions and methods INTELLIKINE LLC (US) 2015-12-22 US disclosed
WO-2015191799-A1 ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS AND USES THEREOF MERCK SHARP & DOHME CORP. (US) 2015-12-17 WO disclosed
EP-2953940-A1 PIPERIDIN-1 -YL AND AZEPIN-1 -YL CARBOXYLATES AS MUSCARINIC M4 RECEPTOR AGONISTS Takeda Pharmaceutical Company Limited (JP) 2015-12-16 EP disclosed
US-9212192-B2 Bicyclic carboxamide inhibitors of kinases ABBVIE INC. (US) 2015-12-15 US disclosed
US-9212184-B2 6-thio-substituted imidazo[1,2-a]pyrazines as Mps-1 inhibitors BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-12-15 US disclosed
US-9212257-B2 Polymeric materials COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2015-12-15 US disclosed
US-20150353832-A1 PHOSPHINATE IONIC LIQUID COMPOSITIONS AND METHODS OF USE H & C Scientific Resources International, LLC (US) 2015-12-10 US disclosed
WO-2015187827-A1 NOVEL EFFECTIVE ANTIVIRAL COMPOUNDS AND METHODS USING SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2015-12-10 WO disclosed
US-20150353854-A1 SYNTHESIS OF FUELS AND CHEMICALS FROM SUGARS PIONEER ENERGY INC (US) 2015-12-10 US disclosed
EP-2951181-A1 AMIDOIMIDAZOPYRIDAZINES AS MKNK-1 KINASE INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2015-12-09 EP disclosed
EP-2951175-A1 SUBSTITUTED PYRAZOLOPYRIMIDINYLAMINO-INDAZOLES Bayer Pharma Aktiengesellschaft (DE) 2015-12-09 EP disclosed
CN-105143235-A Polyhedral oligomeric silsesquioxane nanocrystal stabilization ligands NANOSYS INC 2015-12-09 CN disclosed
US-9206185-B2 Imidazopyridazines as Akt kinase inhibitors BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-12-08 US disclosed
US-9205038-B2 Brightener-containing hair relaxer SHURNEY GLENN (US) 2015-12-08 US disclosed
US-9206182-B2 Substituted isoquinolin-1(2H)-one compounds, compositions, and methods thereof INTELLIKINE LLC (US) 2015-12-08 US disclosed
WO-2015181104-A1 BENZOTHIADIAZOLAMINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-12-03 WO disclosed
US-20150344436-A1 PKM2 MODULATORS AND METHODS FOR THEIR USE SUMITOMO PHARMA ONCOLOGY, INC. 2015-12-03 US disclosed
US-20150344523-A1 MUTANT AKT-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING CALIFORNIA INSTITUTE OF TECHNOLOGY 2015-12-03 US disclosed
EP-2692346-B1 An antiviral 1-phenyl-2,5-dibenzimidazol-5-yl-pyrrolidine derivative ABBVIE BAHAMAS LTD (BS) 2015-12-02 EP disclosed
US-9198420-B2 Rodenticidal norbormide analogues LANDCARE RESEARCH NEW ZEALAND LIMITED (NZ) 2015-12-01 US disclosed
US-9199988-B2 Dihydroquinazolinone analogues BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-12-01 US disclosed
US-9199999-B2 Substituted imidazopyrazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-12-01 US disclosed
US-20150335635-A1 8-HYDROXY QUINOLINE DERIVATIVES PRANA BIOTECHNOLOGY LIMITED (AU) 2015-11-26 US disclosed
WO-2015179563-A2 N-HYDROXY BICYCLIC HYDANTOIN CARBAMATES AS TOOLS FOR IDENTIFICATION OF SERINE HYDROLASE TARGETS ABIDE THERAPEUTICS, INC. (US) 2015-11-26 WO disclosed
US-20150337128-A1 RELEASE MEDIA THE UNIVERSITY OF QUEENSLAND (AU) 2015-11-26 US disclosed
US-20150336892-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC (US) 2015-11-26 US disclosed
US-20150336935-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO AQUINOX PHARMACEUTICALS CANADA INC (CA) 2015-11-26 US disclosed
EP-2947072-A1 1-(3-(6,7-DIMETHOXYQUINAZOLIN-4-YLOXY)PHENYL)-3-(5-(1,1,1-TRIFLUORO-2-METHYLPROPAN-2-YL)ISOXAZOL-3-YL)UREA AS RAF KINASE MODULATOR IN THE TREATMENT OF CANCER DISEASES Ambit Biosciences Corporation (US) 2015-11-25 EP disclosed
CN-105102463-A Low temperature synthesis of rapamycin derivatives BIOSENSORS INTERNANTIONAL GROUP LTD 2015-11-25 CN disclosed
CN-105102967-A Purification of rapamycin derivatives BIOSENSORS INTERNANTIONAL GROUP LTD 2015-11-25 CN disclosed
US-9193716-B2 S1P receptors modulators and their use thereof AKAAL PHARMA PTY LTD. (AU) 2015-11-24 US disclosed
US-9193669-B2 Compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2015-11-24 US disclosed
US-9193723-B2 NAMPT inhibitors ABBVIE INC. (US) 2015-11-24 US disclosed
WO-2015176020-A1 SYNTHESIS OF OLEFINIC ALCOHOLS VIA ENZYMATIC TERMINAL HYDROXYLATION PROVIVI, INC. (US) 2015-11-19 WO disclosed
WO-2015175845-A1 BENZIMIDAZOLE DERIVATIVES AND USES THEREOF PELOTON THERAPEUTICS, INC. (US) 2015-11-19 WO disclosed
WO-2015175632-A1 HETEROARYL COMPOUNDS FOR KINASE INHIBITION ARIAD PHARMACEUTICALS, INC. (US) 2015-11-19 WO disclosed
US-20150329473-A1 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. 2015-11-19 US disclosed
US-20150327546-A1 SUBSTITUTED 4-CYAN-3-(PYRIDYL)-4-PHENYLBUTANOATES, METHOD FOR THE PRODUCTION THEREOF AND USES AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2015-11-19 US disclosed
EP-2943470-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO Aquinox Pharmaceuticals (Canada) Inc. (CA) 2015-11-18 EP disclosed
CN-105072906-A Substituted 4-cyano-3- (pyridyl) -4-phenylbutyrates, method for the production thereof and use thereof as herbicides and plant growth regulators BAYER CROPSCIENCE AG 2015-11-18 CN disclosed
US-9187426-B2 Organic compounds NOVARTIS AG (CH) 2015-11-17 US disclosed
US-9185914-B2 Substituted 5-(cyclohex-2-en-1-yl)-penta-2,4-dienes and 5-(cyclohex-2-en-1-yl)-pent-2-en-4-ines as active agents against abiotic stress in plants BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-11-17 US disclosed
US-9187458-B2 Cyanoquinoline derivatives TIANJIN HEMAY BIO-TECH CO., LTD. (CN) 2015-11-17 US disclosed
US-9187472-B2 NAMPT inhibitors ABBVIE INC. (US) 2015-11-17 US disclosed
WO-2015169962-A1 BENZIMIDAZOLE DERIVATIVES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-11-12 WO disclosed
US-20150322094-A1 USE OF SUBSTITUTED 2,3-DIHYDRO-1-BENZOFURAN-4-CARBOXYLIC ACIDS OR SALTS THEREOF AS ACTIVE SUBSTANCES AGAINST ABIOTIC PLANT STRESS BAYER CROPSCIENCE AG (DE) 2015-11-12 US disclosed
WO-2015171543-A1 MUTANT AKT-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2015-11-12 WO disclosed
US-20150320727-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, LLC 2015-11-12 US disclosed
US-20150322064-A1 Heterocyclic Compounds and Uses Thereof MILLENNIUM PHARMACEUTICALS, INC. 2015-11-12 US disclosed
US-20150322086-A1 LOW TEMPERATURE SYNTHESIS OF RAPAMYCIN DERIVATIVES JOHNSON MATTHEY PHARMACEUTICAL MATERIALS, INC. D/B/A JOHNSON MATTHEY PHARMA SERVICES 2015-11-12 US disclosed
US-20150322073-A1 Benzimidazole Derivatives BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-11-12 US disclosed
EP-2942350-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2015-11-11 EP disclosed
CN-105051605-A Lithographically produced features UNIV QUEENSLAND 2015-11-11 CN disclosed
US-9181221-B2 Chemical compounds, compositions and methods for kinase modulation INFINITY PHARMACEUTICALS, INC. (US) 2015-11-10 US disclosed
US-9181244-B1 Substituted pyrido[2,3-c]pyridazin-4(1H)-ones as tumor necrosis factor alpha and phosphodiesterase 4 inhibitors Xuanzhu Pharma Co., Ltd. (CN) 2015-11-10 US disclosed
US-9181246-B2 Pyrrolopyridine inhibitors of kinases ABBVIE INC. (US) 2015-11-10 US disclosed
US-9182402-B2 Hepsin inhibitors FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2015-11-10 US disclosed
US-9181182-B2 S1P receptors modulators AKAAL PHARMA PTY LTD (AU) 2015-11-10 US disclosed
US-9181239-B2 Pyridopyrimidinone inhibitors of kinases ABBVIE INC. (US) 2015-11-10 US disclosed
US-9180122-B2 5- or 6-substituted 3-hydroxy-2 (1 H)-pyridinones as D-amino acid oxidase (DAAO) inhibitors in therapy of diseases such as schizophrenia, cognitive disorder and pain TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-11-10 US disclosed
WO-2015168466-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Quanticel Pharmaceuticals, Inc. (US) 2015-11-05 WO disclosed
WO-2015168079-A1 PYRIMIDINE OR PYRIDINE DERIVATIVES USEFUL AS PI3K INHIBITORS INFINITY PHARMACEUTICALS, INC. (US) 2015-11-05 WO disclosed
US-20150315187-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 CELGENE QUANTICEL RESEARCH, INC. 2015-11-05 US disclosed
US-20150315146-A1 USE OF SUBSTITUTED 1-(ARYL ETHYNYL)-, 1-(HETEROARYL ETHYNYL)-, 1-(HETEROCYCLYL ETHYNYL)- AND 1-(CYCLOALKENYLETHYNYL)-BICYCLOALKANOLS AS ACTIVE AGENTS AGAINST ABIOTIC PLANT STRESS BAYER CROPSCIENCE AG (DE) 2015-11-05 US disclosed
EP-2313414-B1 KINASE INHIBITORS AND METHODS OF USE INTELLIKINE LLC (US) 2015-11-04 EP disclosed
EP-2419404-B1 ANTI-VIRAL COMPOUNDS ABBVIE INC (US) 2015-11-04 EP disclosed
US-9174994-B2 Enhanced treatment regimens using mTor inhibitors INTELLIKINE, LLC (US) 2015-11-03 US disclosed
US-9173395-B2 Use of substituted isoquinolinones, isoquinolindiones, isoquinolintriones and dihydroisoquinolinones or in each case salts thereof as active agents against abiotic stress in plants BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-11-03 US disclosed
US-9173882-B2 Polycyclic heteroaryl substituted triazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2015-11-03 US disclosed
US-9173397-B2 Formulation component SYNGENTA LIMITED (GB) 2015-11-03 US disclosed
US-9176380-B2 Photoinduced alkyne-azide click reactions THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2015-11-03 US disclosed
US-9174949-B2 Hedgehog inhibitors SELEXAGEN THERAPEUTICS, INC. (US) 2015-11-03 US disclosed
WO-2015164419-A1 PUPILLOMETRIC ASSESSMENT OF RETINAL PHARMACODYNAMICS AND RESPONSES THEREFROM ACUCELA INC. (US) 2015-10-29 WO disclosed
US-20150306105-A1 BENZOXAZOLE KINASE INHIBITORS AND METHODS OF USE FAETH THERAPEUTICS, INC. 2015-10-29 US disclosed
US-20150307426-A9 INDENE DERIVATIVES AS PHARMACEUTICAL AGENTS AQUINOX PHARMACEUTICALS INC. (CA) 2015-10-29 US disclosed
US-20150305334-A1 USE OF SUBSTITUTED 1-(ARYL ETHYNYL)-, 1-(HETEROARYL ETHYNYL)-, 1-(HETEROCYCLYL ETHYNYL)- AND 1-(CYCLOALKENYL ETHYNYL)-CYCLOHEXANOLS AS ACTIVE AGENTS AGAINST ABIOTIC PLANT STRESS BAYER CROPSCIENCE AG (DE) 2015-10-29 US disclosed
WO-2015164643-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL HYDRA BIOSCIENCES, INC. (US) 2015-10-29 WO disclosed
EP-2934145-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals Inc (US) 2015-10-28 EP disclosed
EP-2935217-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals Inc (US) 2015-10-28 EP disclosed
US-9169211-B2 8-hydroxy quinoline derivatives PRANA BIOTECHNOLOGY LIMITED (AU) 2015-10-27 US disclosed
US-20150299131-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC (US) 2015-10-22 US disclosed
EP-2748149-B1 PYRIDAZINONE COMPOUNDS AND THEIR USE AS DAAO INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2015-10-21 EP disclosed
US-9161948-B2 Peptide oligonucleotide conjugates SAREPTA THERAPEUTICS, INC. (US) 2015-10-20 US disclosed
US-9161537-B2 Substituted 4-cyan-3-phenyl-4-(pyridine-3-yl)butanoates, processes for preparation thereof and use thereof as herbicides and plant growth regulators BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-10-20 US disclosed
US-9162992-B2 Compounds and compositions for treatment of breathing control disorders or diseases GALLEON PHARMACEUTICALS, INC. (US) 2015-10-20 US disclosed
US-9162939-B2 Carbon nanohoops and methods of making THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-10-20 US disclosed
US-9163017-B2 Anti-viral compounds ABBVIE INC. (US) 2015-10-20 US disclosed
US-9163018-B2 Method of treatment of age-related macular degeneration (AMD) PRANA BIOTECHNOLOGY INC. (AU) 2015-10-20 US disclosed
US-20150291599-A1 AMINOIMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-10-15 US disclosed
US-20150289511-A1 MOLECULES THAT INDUCE DISEASE RESISTANCE AND IMPROVE GROWTH IN PLANTS UNIV CALIFORNIA (US) 2015-10-15 US disclosed
WO-2015157262-A1 Novel 7-Dehydrocholesterol Derivatives and Methods Using Same WOMEN & INFANTS HOSPITAL OF RHODE ISLAND (US) 2015-10-15 WO disclosed
US-20150291597-A1 NOVEL ORALLY BIOAVAILABLE BREATHING CONTROL MODULATING COMPOUNDS, AND METHODS OF USING SAME GALLEON PHARMACEUTICALS, INC. 2015-10-15 US disclosed
WO-2015155332-A1 SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE DERIVATIVES AND THEIR USE AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-10-15 WO disclosed
US-20150290207-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2015-10-15 US disclosed
WO-2015155739-A1 PROCESS FOR THE PREPARATION OF BETA-C-ARYLGLUCOSIDES SCINOPHARM TAIWAN, LTD. (TW) 2015-10-15 WO disclosed
US-20150291569-A1 PROCESS FOR THE PREPARATION OF beta-C-ARYLGLUCOSIDES SCINOPHARM TAIWAN, LTD. (TW) 2015-10-15 US disclosed
WO-2015157512-A1 NOVEL METHODS AND KITS FOR DETECTING A RIFAMYCIN, OR DERIVATIVE OR ANALOGUE THEREOF DREXEL UNIVERSITY (US) 2015-10-15 WO disclosed
US-20150291611-A1 NEW SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-10-15 US disclosed
US-20150293080-A1 Fluorescent Dyes and Related Methods NATIONAL SCIENCE FOUNDATION 2015-10-15 US disclosed
US-20150291623-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2015-10-15 US disclosed
US-20150291610-A1 C20' Urea Derivatives of Vinca Alkaloids NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-10-15 US disclosed
US-20150291529-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2015-10-15 US disclosed
EP-2928471-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals Inc (US) 2015-10-14 EP disclosed
EP-2476679-B1 Substituted triazoles useful as AXL inhibitors RIGEL PHARMACEUTICALS INC (US) 2015-10-14 EP disclosed
EP-2694510-B1 IMIDAZOPYRIDAZINES AS AKT KINASE INHIBITORS BAYER IP GMBH (DE) 2015-10-14 EP disclosed
US-9156820-B2 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2015-10-13 US disclosed
US-9156853-B2 AKT inhibitor compounds for treatment of cancer ALMAC DISCOVERY LIMITED (GB) 2015-10-13 US disclosed
US-9156829-B2 Cycloalkyl and heterocycloalkyl compounds as orexin receptor antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-10-13 US disclosed
WO-2015149131-A1 POLYMYXIN DERIVATIVES AS ANTIMICROBIAL COMPOUNDS MONASH UNIVERSITY (AU) 2015-10-08 WO disclosed
WO-2015153554-A1 NOVEL ANTIVIRAL COMPOUNDS AND METHODS USING SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2015-10-08 WO disclosed
US-20150284420-A1 E-SELECTIN ANTAGONIST COMPOUNDS AND METHODS OF USE GLYCOMIMETICS, INC. (US) 2015-10-08 US disclosed
US-20150283142-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS INFINITY PHARMACEUTICALS, INC. (US) 2015-10-08 US disclosed
EP-2925761-A1 TRIAZOLOPYRAZINE Boehringer Ingelheim International GmbH (DE) 2015-10-07 EP disclosed
CN-104968353-A Gemcitabine prodrugs and uses thereof BOYEN THERAPEUTICS INC 2015-10-07 CN disclosed
US-9150578-B2 5,8-dihydro-6H-pyrazolo[3,4-h]quinazolines as IGF-1R/IR inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-10-06 US disclosed
US-9150608-B2 Neuro-protective compounds and their use Biotechnology Research Corp. Ltd. (CN) 2015-10-06 US disclosed
US-20150272939-A1 Identification of Small Molecule Inhibitors of Jumonji AT-Rich Interactive Domain 1A (JARID1A) and 1B (JARID1B) Histone Demethylase YALE UNIVERSITY (US) 2015-10-01 US disclosed
EP-2576560-B1 SUBSTITUTED IMIDAZOPYRAZINES BAYER IP GMBH (DE) 2015-09-30 EP disclosed
EP-2731933-B1 2,3-DIPHENYL-VALERONITRILE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER IP GMBH (DE) 2015-09-30 EP disclosed
US-20150270573-A1 HALOGENATED ORGANOSILICON ELECTROLYTES, METHODS OF USING THEM, AND ELECTROCHEMICAL DEVICES CONTAINING THEM SILATRONIX, INC. (US) 2015-09-24 US disclosed
WO-2015140195-A1 NOVEL COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-09-24 WO disclosed
WO-2015140196-A1 INHIBITORS OF THE WNT SIGNALLING PATHWAYS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-09-24 WO disclosed
WO-2015143012-A1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF PI3K-GAMMA MEDIATED DISORDERS INFINITY PHARMACEUTICALS, INC. (US) 2015-09-24 WO disclosed
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EP-2920155-A2 NOVEL ORALLY BIOAVAILABLE BREATHING CONTROL MODULATING COMPOUNDS, AND METHODS OF USING SAME Galleon Pharmaceuticals, Inc. (US) 2015-09-23 EP disclosed
EP-2920180-A1 PYRROLOPYRIMIDINE COMPOUNDS AS KINASE INHIBITORS Pharmacyclics, Inc. (US) 2015-09-23 EP disclosed
EP-2920176-A1 AMINOIMIDAZOPYRIDAZINES Bayer Pharma Aktiengesellschaft (DE) 2015-09-23 EP disclosed
EP-2651944-B1 SUBSTITUTED 6-IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER IP GMBH (DE) 2015-09-23 EP disclosed
EP-2919790-A1 GEMCITABINE PRODRUGS AND USES THEREOF Boyen Therapeutics, Inc. (TW) 2015-09-23 EP disclosed
EP-2920175-A1 TRIAZOLOPYRIDAZINE Boehringer Ingelheim International GmbH (DE) 2015-09-23 EP disclosed
US-9139536-B2 Anti-infective agents and uses thereof ABBVIE INC. (US) 2015-09-22 US disclosed
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EP-2918587-A2 Filamin a binding anti-inflammatory and analgesic Pain Therapeutics, Inc. (US) 2015-09-16 EP disclosed
EP-2918589-A1 ADENINE DERIVATIVE AS PI3K INHIBITOR Intellikine, LLC (US) 2015-09-16 EP disclosed
EP-2729454-B1 NOVEL TRIFLUOROMETHYL-OXADIAZOLE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2015-09-16 EP disclosed
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EP-2914295-A1 TREATMENT OF RHEUMATOID ARTHRITIS AND ASTHMA USING P13 KINASE INHIBITORS Infinity Pharmaceuticals, Inc. (US) 2015-09-09 EP disclosed
EP-2914296-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS Infinity Pharmaceuticals, Inc. (US) 2015-09-09 EP disclosed
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US-20150246029-A1 Positive Allosteric Modulators and Uses Thereof MERCK SHARP & DOHME CORP. 2015-09-03 US disclosed
US-20150246919-A1 PYRIDINONES BOEHRINGER INGELHEIM INT (DE) 2015-09-03 US disclosed
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US-20150246042-A1 RAF KINASE MODULATOR COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2015-09-03 US disclosed
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CN-104884432-A Alpha7 nicotinic acetylcholine receptor modulators and uses thereof-I MERCK SHARP & DOHME 2015-09-02 CN disclosed
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US-20150238497-A1 STYRENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. 2015-08-27 US disclosed
US-20150239836-A1 ALKOXY COMPOUNDS FOR DISEASE TREATMENT ACUCELA INC. 2015-08-27 US disclosed
US-20150239897-A1 PYRROLOPYRIMIDINE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS LLC 2015-08-27 US disclosed
US-20150239891-A1 SUBSTITUTED PYRROLOPYRIMIDINYLAMINO-BENZOTHIAZOLONES AS MKNK KINASE INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-08-27 US disclosed
US-20150239900-A1 INHIBITORS OF KRAS G12C ARAXES PHARMA LLC 2015-08-27 US disclosed
EP-2909181-A2 PKM2 MODULATORS AND METHODS FOR THEIR USE Tolero Pharmaceuticals, Inc. (US) 2015-08-26 EP disclosed
EP-2663553-B1 QUINOLINE AND ISOQUINOLINE DERIVATIVES FOR USE AS JAK MODULATORS AMBIT BIOSCIENCES CORP (US) 2015-08-26 EP disclosed
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US-9115056-B2 Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2015-08-25 US disclosed
US-9115141-B2 Substituted isoquinolinones and methods of treatment thereof INFINITY PHARMACEUTICALS, INC. (US) 2015-08-25 US disclosed
US-20150232476-A1 COMPOUNDS AND METHODS FOR PREVENTING, TREATING AND/OR PROTECTING AGAINST SENSORY HAIR CELL DEATH UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION 2015-08-20 US disclosed
WO-2015121210-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-08-20 WO disclosed
US-20150232460-A1 NOVEL COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-08-20 US disclosed
US-20150232484-A1 FUSED THIAZIN-3-ONES AS KCA3.1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-08-20 US disclosed
US-20150232474-A1 Bicyclic Substituted Pyrimidine Compounds Xuanzhu Biopharmaceutical Co., Ltd. (CN) 2015-08-20 US disclosed
WO-2015121209-A1 BENZIMIDAZOL-2-AMINES AS MIDH1 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-08-20 WO disclosed
US-20150232455-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. 2015-08-20 US disclosed
EP-2906607-A2 POLYMERS HAVING ORTHOGONAL REACTIVE GROUPS AND USES THEREOF NVS Technologies Inc. (US) 2015-08-19 EP disclosed
US-9107916-B2 Histone demethylase inhibitors Quanticel Pharmaceuticals, Inc. (US) 2015-08-18 US disclosed
WO-2015119712-A1 TETRACYCLIC CDK9 KINASE INHIBITORS ABBVIE INC. (US) 2015-08-13 WO disclosed
WO-2015119579-A1 2,4,5-TRI-SUBSTITUTED AZOLE-BASED CASEIN KINASE 1 INHIBITORS AS INDUCERS FOR CARDIOMYOGENESIS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-08-13 WO disclosed
US-20150225410-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2015-08-13 US disclosed
EP-2903988-A1 COMPOUNDS USEFUL FOR MAKING HCV PROTEASE INHIBITORS AbbVie Inc. (US) 2015-08-12 EP disclosed
EP-2904048-A1 SUSTAINABLE ISOSORBIDE - CONTAINING POLYCARBONATE - POLYLACTIDE BLENDS SABIC Global Technologies B.V. (NL) 2015-08-12 EP disclosed
EP-2408752-B1 SUBSTITUTED PYRIMIDINES FOR THE TREATMENT OF CANCER BOEHRINGER INGELHEIM INT (DE) 2015-08-12 EP disclosed
US-9102636-B2 Analgesic compounds, compositions, and uses thereof GALLEON PHARMACEUTICALS, INC. (US) 2015-08-11 US disclosed
US-9102684-B2 Indolinone analogues BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-08-11 US disclosed
WO-2015113920-A1 AMINO-SUBSTITUTED ISOTHIAZOLES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-08-06 WO disclosed
WO-2015113927-A1 AMINO-SUBSTITUTED ISOTHIAZOLES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-08-06 WO disclosed
US-20150216168-A1 USE OF SUBSTITUTED 2-AMIDOBENZIMIDAZOLES, 2-AMIDOBENZOXAZOLES AND 2-AMIDOBENZOTHIAZOLES OR SALTS THEREOF AS ACTIVE SUBSTANCES AGAINST ABIOTIC PLANT STRESS BAYER CROPSCIENCE AG (DE) 2015-08-06 US disclosed
US-20150219657-A1 PHOSPHORYLATED AKT-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING CALIFORNIA INSTITUTE OF TECHNOLOGY 2015-08-06 US disclosed
US-20150218194-A1 Anti-Viral Compounds ABBVIE INC. (US) 2015-08-06 US disclosed
US-20150216864-A1 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS MIDCAP FINANCIAL TRUST 2015-08-06 US disclosed
US-20150218173-A1 SUBSTITUTED INDAZOL-PYRROLOPYRIMIDINES USEFUL IN THE TREATMENT OF HYPERFOLIFERATIVE DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-08-06 US disclosed
US-20150218110-A1 USE OF SUBSTITUTED BENZODIAZEPINONES AND BENZAZEPINONES OR THE SALTS THEREOF AS ACTIVE SUBSTANCES AGAINST ABIOTIC PLANT STRESS BAYER CROPSCIENCE AG (DE) 2015-08-06 US disclosed
US-20150218165-A1 TETRACYCLIC CDK9 KINASE INHIBITORS ABBVIE INC. (US) 2015-08-06 US disclosed
EP-2547680-B1 IMIDAZOPYRAZINES BAYER IP GMBH (DE) 2015-08-05 EP disclosed
EP-2900239-A1 DIHYDRO-6-AZAPHENALENE DERIVATIVES FOR THE TREATMENT OF CNS, ONCOLOGICAL DISEASES AND RELATED DISORDERS The Warner-Babcock Institute For Green Chemistry LLC (US) 2015-08-05 EP disclosed
EP-2029516-B1 PROCESS FOR PREPARING FLUORINATED MOLECULES BAYER IP GMBH (DE) 2015-08-05 EP disclosed
EP-2900671-A1 SUBSTITUTED INDAZOL-PYRROLOPYRIMIDINES USEFUL IN THE TREATMENT OF HYPERPROLIFERATIVE DISEASES Bayer Pharma Aktiengesellschaft (DE) 2015-08-05 EP disclosed
EP-2900674-A1 COMPOUNDS AND METHODS FOR PREVENTING, TREATING AND/OR PROTECTING AGAINST SENSORY HAIR CELL DEATH University of Washington through its Center for Commercialization (US) 2015-08-05 EP disclosed
US-9096604-B2 Pyrrolopyrimidine compounds as kinase inhibitors PHARMACYCLICS, INC. (US) 2015-08-04 US disclosed
US-9096599-B2 Spiroindoline compounds INTERVET INC. (US) 2015-08-04 US disclosed
US-9095590-B2 Anti-infective agents and uses thereof ABBVIE INC. (US) 2015-08-04 US disclosed
US-9096590-B2 Substituted benzoxazoles as PI3 kinase inhibitors INTELLIKINE LLC (US) 2015-08-04 US disclosed
US-9096611-B2 Kinase inhibitors and methods of use INTELLIKINE LLC (US) 2015-08-04 US disclosed
US-9096524-B2 Anthelmintic agents and their use INTERVET INTERNATIONAL B.V. (NL) 2015-08-04 US disclosed
US-20150210683-A1 SUBSTITUTED TRIAZOLOPYRIDINES AND THEIR USE AS TTK INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-07-30 US disclosed
WO-2015110923-A2 METHODS OF TREATING CHRONIC LYMPHOCYTIC LEUKEMIA AND SMALL LYMPHOCYTIC LEUKEMIA USNG A BTK INHIBITOR ACERTA PHARMA B.V. (NL) 2015-07-30 WO disclosed
WO-2015112093-A2 ANTIMICROBIAL PEPTIDOMIMETICS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-07-30 WO disclosed
EP-2791136-B1 SUBSTITUTED TRIAZOLOPYRIDINES AND THEIR USE AS TTK INHIBITORS BAYER IP GMBH (DE) 2015-07-29 EP disclosed
EP-2104659-B1 COMPOUNDS WITH (SUBSTITUTED PHENYL)-PROPENAL MOIETY, THEIR DERIVATIVES, BIOLOGICAL ACTIVITY, AND USES THEREOF ANDROSCIENCE CORP (US) 2015-07-29 EP disclosed
WO-2015109136-A2 WATER SOLUBLE FLUORESCENT OR COLORED DYES AND METHODS FOR THEIR USE SONY CORPORATION (JP) 2015-07-23 WO disclosed
EP-2114896-B1 RADIOPROTECTOR COMPOUNDS AND RELATED METHODS PETER MACCALLUM CANCER INST (AU) 2015-07-22 EP disclosed
CN-104797257-A Polymer-NSAID conjugate POLYACTIVA PTY LTD 2015-07-22 CN disclosed
US-9085534-B2 Histone demethylase inhibitors Quanticel Pharmaceuticals, Inc. (US) 2015-07-21 US disclosed
US-9085511-B2 Atropisomeric 1,8-bisphenolnapthalenes and their use in enantioselective recognition and asymmetric synthesis GEORGETOWN UNIVERSITY (US) 2015-07-21 US disclosed
US-9084425-B2 2,3-diphenyl-valeronitrile derivatives, method for the production thereof and use thereof as herbicides and plant growth regulators BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-07-21 US disclosed
US-9085560-B2 Heterocyclic compounds and uses thereof INTELLIKINE, INC. (US) 2015-07-21 US disclosed
US-20150196566-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2015-07-16 US disclosed
WO-2015104254-A1 AMIDO-SUBSTITUTED IMIDAZOPYRIDAZINES USEFUL IN THE TREATMENT OF HYPER-PROLIFERATIVE AND/OR ANGIOGENESIS DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-07-16 WO disclosed
US-9079898-B2 Polycyclic heteroaryl substituted triazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2015-07-14 US disclosed
US-9079825-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2015-07-14 US disclosed
US-9078440-B2 6-(2-aminophenyl)picolinates and their use as herbicides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-07-14 US disclosed
US-9080119-B2 Synthesis of high caloric fuels and chemicals including pentanol from coal, natural gas, and biomass Pioneer Energy (US) 2015-07-14 US disclosed
US-20150192589-A1 METHOD USING FLUORESCENT TURN-ON PROBES FOR CELL-SPECIFIC DETECTION AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-07-09 US disclosed
US-20150190351-A1 Compounds with (1E, 6E)-1,7-bis-(3,4-dimethoxyphenyl)-4,4-disubstituted-hepta-1,6-diene-3,5-dione structural scaffold, their biological activity, and uses thereof Annji Pharmaceutical Co., Ltd. (TW) 2015-07-09 US disclosed
US-20150190389-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDER ARDELYX, INC. (US) 2015-07-09 US disclosed
EP-2424537-B1 SUBSTITUTED IMIDAZOQUINOXALINES BAYER IP GMBH (DE) 2015-07-08 EP disclosed
US-9073922-B2 Pyrrolo[2,3-B]pyridine CDK9 kinase inhibitors ABBVIE, INC. (US) 2015-07-07 US disclosed
WO-2015095953-A1 SULFONAMIDE-CONTAINING LINKAGE SYSTEMS FOR DRUG CONJUGATES THE CENTRE FOR DRUG RESEARCH AND DEVELOPMENT (CA) 2015-07-02 WO disclosed
WO-2015095952-A1 VAR2CSA-DRUG CONJUGATES THE CENTRE FOR DRUG RESEARCH AND DEVELOPMENT (CA) 2015-07-02 WO disclosed
US-20150183784-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2015-07-02 US disclosed
EP-2887963-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS Ardelyx, Inc. (US) 2015-07-01 EP disclosed
EP-2887964-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS Ardelyx, Inc. (US) 2015-07-01 EP disclosed
US-9066967-B2 Oligonucleotide analogues targeting human LMNA SAREPTA THERAPEUTICS, INC. (US) 2015-06-30 US disclosed
WO-2015091428-A1 GLUCOSE TRANSPORT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-06-25 WO disclosed
WO-2015091315-A1 SPIRO[INDOLIN-3,4'-PIPERIDINE] DERIVATIVES AS GNRH RECEPTOR ANTAGONISTS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-06-25 WO disclosed
US-20150173359-A1 SUBSTITUTED FUSED PYRIMIDINONES AND DIHYDROPYRIMIDINONES BAYER IP GMBH (DE) 2015-06-25 US disclosed
US-20150175534-A1 Alpha-7 NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS AND USES THEROF-I MERCK SHARP & DOHME CORP. 2015-06-25 US disclosed
EP-2886540-A1 BICYCLIC SUBSTITUTED PYRIMIDINE COMPOUNDS Xuanzhu Pharma Co., Ltd. (CN) 2015-06-24 EP disclosed
EP-2590655-B1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX INC (US) 2015-06-24 EP disclosed
CN-104736153-A Apoptosis-inducing agents ABBVIE INC 2015-06-24 CN disclosed
US-9062013-B2 Positive allosteric modulators of the α7 nicotinic acetylcholine receptor and uses thereof BIONOMICS LIMITED (AU) 2015-06-23 US disclosed
US-9062073-B2 Pyrimido-pyrrolo-oxazine-dione compound inhibitors of the cystic fibrosis transmembrane conductance regulator protein and uses therefor THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-06-23 US disclosed
US-9062058-B2 2015-06-23 US disclosed
US-9062026-B2 Fused pyrimidines and substituted quinazolines as inhibitors of p97 CLEAVE BIOSCIENCES, INC. (US) 2015-06-23 US disclosed
US-20150164876-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. 2015-06-18 US disclosed
US-20150166494-A1 Styrenyl Derivative Compounds for Treating Ophthalmic Diseases and Disorders ACUCELA INC. 2015-06-18 US disclosed
US-20150166495-A1 Styrenyl Derivative Compounds for Treating Ophthalmic Diseases and Disorders ACUCELA INC. 2015-06-18 US disclosed
US-20150164905-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. 2015-06-18 US disclosed
WO-2015089192-A1 INHIBITORS OF LYSINE SPECIFIC DEMETHYLASE-1 Quanticel Pharmaceuticals, Inc. (US) 2015-06-18 WO disclosed
US-20150164904-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. 2015-06-18 US disclosed
US-20150164872-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2015-06-18 US disclosed
US-20150166539-A1 THREE-RING PI3K AND/OR MTOR INHIBITOR Xuanzhu Pharma Co., Ltd. (CN) 2015-06-18 US disclosed
EP-2882439-A1 APOPTOSIS-INDUCING AGENTS AbbVie Inc. (US) 2015-06-17 EP disclosed
EP-2882428-A2 A METHOD OF INHIBITING TAU PHOSPHORYLATION Pain Therapeutics, Inc. (US) 2015-06-17 EP disclosed
CN-104718250-A Sustainable isosorbide-containing polycarbonate-polylactide blends SABIC INNOVATIVE PLASTICS IP 2015-06-17 CN disclosed
US-9056849-B2 Amine derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2015-06-16 US disclosed
US-9056843-B2 Trifluoromethyl-oxadiazole derivatives and their use in the treatment of disease NOVARTIS AG (CH) 2015-06-16 US disclosed
US-9056877-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2015-06-16 US disclosed
WO-2015083008-A1 THERAPEUTIC COMBINATION OF A PI3K INHIBITOR AND A BTK INHIBITOR ACERTA PHARMA B.V. (NL) 2015-06-11 WO disclosed
WO-2015082378-A1 COMBINATION OF PI3K-INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-06-11 WO disclosed
WO-2015082376-A2 USE OF PI3K-INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-06-11 WO disclosed
US-20150158880-A1 TAXANE AND ABEO-TAXANE ANALOGS Arbor Therapeutics, LLC (US) 2015-06-11 US disclosed
US-20150157637-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. 2015-06-11 US disclosed
WO-2015084998-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS, INC. (US) 2015-06-11 WO disclosed
US-20150158865-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC 2015-06-11 US disclosed
WO-2015082374-A1 SPIROINDOLINE-THIOPYRAN-IMINE-OXIDE DERIVATIVES AS GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS AND PHARMACEUTICAL COMPOSITIONS THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-06-11 WO disclosed
US-20150158909-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. 2015-06-11 US disclosed
US-20150158859-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE LLC (US) 2015-06-11 US disclosed
EP-2881391-A1 Spiroindoline carbocycle derivatives and pharmaceutical compositions thereof Bayer Pharma Aktiengesellschaft (DE) 2015-06-10 EP disclosed
EP-1973917-B1 PROTEIN KINASE INHIBITORS ABBVIE INC (US) 2015-06-10 EP disclosed
US-9049863-B2 Substituted (3R,4R)-4-cyan-3,4-diphenylbutanoates, method for the production thereof and use thereof as herbicides and plant growth regulators BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-06-09 US disclosed
US-9051327-B2 Pyridazino[4,5-D]pyrimidin-5(6H)-one inhibitors of kinases ABBVIE INC. (US) 2015-06-09 US disclosed
US-20150152121-A1 Substituted Benzothienopyrimidines BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-06-04 US disclosed
US-20150152022-A1 CARBON NANOHOOPS AND METHODS OF MAKING ENERGY, UNITED STATES DEPARTMENT OF 2015-06-04 US disclosed
US-20150152097-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2015-06-04 US disclosed
WO-2015081257-A2 AMINOPYRIDINE DERIVATIVES AS TAM FAMILY KINASE INHIBITORS SIGNALCHEM LIFESCIENCES CORPORATION (CA) 2015-06-04 WO disclosed
WO-2015080665-A1 CHALCONE-UREA DERIVATIVES AS INSULIN SENSORS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-06-04 WO disclosed
US-20150150999-A1 POLYMER-NSAID CONJUGATE POLYACTIVA PTY LTD (AU) 2015-06-04 US disclosed
US-20150150874-A1 JAK KINASE MODULATING COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORP. (US) 2015-06-04 US disclosed
WO-2015079224-A1 PIPERIDINE DERIVATIVES FOR USE IN THE TREATMENT OR PREVENTION OF PSYCHIATRIC AND NEUROLOGICAL CONDITIONS TAKEDA CAMBRIDGE LIMITED (GB) 2015-06-04 WO disclosed
EP-2350091-B1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2015-06-03 EP disclosed
EP-2350090-B1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2015-06-03 EP disclosed
CN-104684850-A Melamine-aldehyde polymers AGENCY SCIENCE TECH & RES 2015-06-03 CN disclosed
US-9045429-B2 Substituted phenoxypyridines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-06-02 US disclosed
US-9045444-B2 Apoptosis promoters ABBVIE INC. (US) 2015-06-02 US disclosed
US-20150148311-A1 NON-SYSTEMIC TGR5 AGONISTS ARDELYX INC (US) 2015-05-28 US disclosed
US-20150148318-A1 METHOD FOR INHIBITING GROWTH OF CANCER CELLS PAIN THERAPEUTICS, INC. 2015-05-28 US disclosed
WO-2015077780-A1 WITHANOLIDES USEFUL FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES IMSTAR THERAPEUTICS INC. (CA) 2015-05-28 WO disclosed
US-20150148542-A1 METHOD FOR PREPARING SUBSTITUTED TRIAZOLOPYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-05-28 US disclosed
WO-2015077375-A1 QUINAZOLINE DERIVATIVES AS TAM FAMILY KINASE INHIBITORS SIGNALCHEM LIFESCIENCES CORP. (CA) 2015-05-28 WO disclosed
EP-2651946-B1 2-SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER IP GMBH (DE) 2015-05-27 EP disclosed
EP-2694500-B1 SUBSTITUTED IMIDAZOPYRIDINES AND INTERMEDIATES THEREOF Bayer Pharma AG (DE) 2015-05-27 EP disclosed
EP-2875018-A1 FUSED PYRIMIDINES AS INHIBITORS OF p97 COMPLEX Cleave Biosciences, Inc. (US) 2015-05-27 EP disclosed
US-9040757-B2 Synthesis of high caloric fuels and chemicals Pioneer Energy (US) 2015-05-26 US disclosed
US-20150140635-A1 Boronic and Borinic Acid Compound as Inhibitors of Sulfenic Acid-Containing Proteins THE PENN STATE RESEARCH FOUNDATION 2015-05-21 US disclosed
US-20150141398-A1 NAMPT INHIBITORS ABBVIE INC. 2015-05-21 US disclosed
EP-2872506-A1 METHOD FOR PREPARING SUBSTITUTED TRIAZOLOPYRIDINES Bayer Pharma Aktiengesellschaft (DE) 2015-05-20 EP disclosed
EP-2872899-A1 ALZHEIMER'S DISEASE ASSAY IN A LIVING PATENT Pain Therapeutics, Inc. (US) 2015-05-20 EP disclosed
CN-104640972-A Release medium UNIV QUEENSLAND 2015-05-20 CN disclosed
US-9034900-B2 Bromodomain inhibitors Quanticel Pharmaceuticals, Inc. (US) 2015-05-19 US disclosed
US-20150133426-A1 SUBSTITUTED PYRROLOPYRIMIDINES Bayer Pharma AG (DE) 2015-05-14 US disclosed
WO-2015067770-A1 TRIAZOLOPYRAZINE DERIVATIVES AS BRD4 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-05-14 WO disclosed
US-20150132298-A1 GEMCITABINE PRODRUGS AND USES THEREOF BoYen Therapeutics, Inc. (TW) 2015-05-14 US disclosed
US-20150133425-A1 THIENOPYRIMIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-05-14 US disclosed
US-20150133447-A1 Triazolopyrazine BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-05-14 US disclosed
US-20150126501-A1 Fused Ring Compound For Use As Mineralocorticoid Receptor Antagonist NOVO NORDISK A/S (DK) 2015-05-07 US disclosed
US-20150126506-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. 2015-05-07 US disclosed
US-20150126507-A1 COMPOUNDS TO TREAT HEARING LOSS US ARMY, SECRETARY OF THE ARMY 2015-05-07 US disclosed
WO-2015066352-A1 SKIN CARE COMPOSITIONS AND METHODS OF USE THEREOF UNIGEN, INC. (US) 2015-05-07 WO disclosed
US-20150126747-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. 2015-05-07 US disclosed
US-20150126505-A1 IMIDAZOLOTHIAZOLE COMPOUNDS FOR THE TREATMENT OF DISEASE AMBIT BIOSCIENCES CORP (US) 2015-05-07 US disclosed
EP-2268623-B1 QUINAZOLINE DERIVATIVES AS RAF KINASE MODULATORS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORP (US) 2015-05-06 EP disclosed
US-9023957-B2 Compound for use in peptide synthesis NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2015-05-05 US disclosed
US-9023759-B2 Molecules that induce disease resistance and improve growth in plants THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-05-05 US disclosed
US-20150119397-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2015-04-30 US disclosed
US-20150119435-A1 COMPOUNDS USEFUL FOR PROMOTING PROTEIN DEGRADATION AND METHODS USING SAME YALE UNIVERSITY 2015-04-30 US disclosed
US-20150119429-A1 Iron Chelators as HIV-1 Inhibitors HOWARD UNIVERSITY (US) 2015-04-30 US disclosed
EP-2864420-A1 SILICONE LIGANDS FOR STABILIZING QUANTUM DOT FILMS Nanosys, Inc. (US) 2015-04-29 EP disclosed
EP-2863902-A1 TREATMENT OF LUPUS, FIBROTIC CONDITIONS, AND INFLAMMATORY MYOPATHIES AND OTHER DISORDERS USING PI3 KINASE INHIBITORS Infinity Pharmaceuticals, Inc. (US) 2015-04-29 EP disclosed
CN-104583194-A Pyridazine and pyridine derivatives as NAMPT inhibitors ABBVIE INC 2015-04-29 CN disclosed
WO-2015055994-A1 CYCLOPENTYLBENZAMIDE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF PSYCHOTIC AND COGNITIVE DISORDERS TAKEDA CAMBRIDGE LIMITED (GB) 2015-04-23 WO disclosed
US-20150111922-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-04-23 US disclosed
WO-2014205317-A9 CYCLIC PEPTIDES AS PROTEIN TARGETING AGENTS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2015-04-23 WO disclosed
US-20150111874-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2015-04-23 US disclosed
US-20150111885-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RESEARCH, INC. 2015-04-23 US disclosed
WO-2015058160-A1 BROMODOMAIN INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2015-04-23 WO disclosed
WO-2014152287-A9 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES, INC. (US) 2015-04-23 WO disclosed
WO-2015054572-A1 INHIBITORS OF KRAS G12C ARAXES PHARMA LLC (US) 2015-04-16 WO disclosed
US-20150105548-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. 2015-04-16 US disclosed
US-20150105385-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2015-04-16 US disclosed
US-20150104526-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-04-16 US disclosed
WO-2015054027-A1 METHOD FOR INHIBITING GROWTH OF CANCER CELLS PAIN THERAPEUTICS, INC. (US) 2015-04-16 WO disclosed
EP-2858993-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2015-04-15 EP disclosed
CN-104520279-A Novel 1,3-benzoxazol-2(3H)-ones and their use as medicaments and cosmetics WOLFF AUGUST GMBH & CO KG ARZNEIMITTEL DR 2015-04-15 CN disclosed
US-9005480-B2 Method for solventless quantum dot exchange NANOSYS, INC. (US) 2015-04-14 US disclosed
US-9006265-B2 Substituted fused pyrimidinones and dihydropyrimidinones BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-04-14 US disclosed
US-9006281-B2 Compounds and methods for inhibiting NHE-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders ARDELYX, INC. (US) 2015-04-14 US disclosed
US-9006387-B2 Anti-viral compounds ABBVIE INC. (US) 2015-04-14 US disclosed
WO-2015051193-A1 ENHANCED TREATMENT REGIMENS USING PI3Kα INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2015-04-09 WO disclosed
US-20150099128-A1 LINEAR GLYCIDYL CARBAMATE (GC) RESINS FOR HIGHLY FLEXIBLE COATINGS NDSU RESEARCH FOUNDATION 2015-04-09 US disclosed
WO-2015051241-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2015-04-09 WO disclosed
US-20150099658-A1 ANTI-GP41 ANTIBODY-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING CALIFORNIA INSTITUTE OF TECHNOLOGY 2015-04-09 US disclosed
WO-2015051244-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2015-04-09 WO disclosed
EP-2855438-A2 NOVEL COMPOUNDS AND COMPOSITIONS FOR TREATMENT OF BREATHING CONTROL DISORDERS OR DISEASES Galleon Pharmaceuticals, Inc. (US) 2015-04-08 EP disclosed
EP-2212330-B1 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF (3) CHOONGWAE PHARMA CORP (KR) 2015-04-08 EP disclosed
EP-2855449-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed
CN-104508049-A Silicone ligands for stabilizing quantum dot films NANOSYS INC 2015-04-08 CN disclosed
US-9000022-B2 Imidazole based LXR modulators EXELIXIS PATENT COMPANY LLC (US) 2015-04-07 US disclosed
US-9000222-B2 Compounds with (1E, 6E)-1,7-bis-(3,4-dimethoxyphenyl)-4,4-disubstituted-hepta-1,6-diene-3,5-dione structural scaffold, their biological activity, and uses thereof ANDROSCIENCE CORPORATION (US) 2015-04-07 US disclosed
WO-2015048689-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS, INC. (US) 2015-04-02 WO disclosed
US-20150094334-A1 8-HYDROXY QUINOLINE DERIVATIVES PRANA BIOTECHNOLOGY LIMITED (AU) 2015-04-02 US disclosed
US-20150094319-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS LLC 2015-04-02 US disclosed
US-20150094300-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-04-02 US disclosed
EP-2570441-B1 Bioabsorbable surgical composition COVIDIEN LP (US) 2015-04-01 EP disclosed
EP-2852596-A1 THIENOPYRIMIDINES Bayer Pharma Aktiengesellschaft (DE) 2015-04-01 EP disclosed
EP-2853531-A2 Antiviral compounds AbbVie Bahamas Ltd. (BS) 2015-04-01 EP disclosed
EP-2852595-A1 SUBSTITUTED BENZOTHIENOPYRIMIDINES Bayer Pharma Aktiengesellschaft (DE) 2015-04-01 EP disclosed
EP-2464354-B1 PYRIMIDO-PYRROLO-QUINOXALINEDIONE INHIBITORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR PROTEIN AND USES THEREFOR UNIV CALIFORNIA (US) 2015-04-01 EP disclosed
CN-104487097-A Chromophoric polymer dots with narrow-band emission UNIV WASHINGTON CT COMMERCIALIZATION 2015-04-01 CN disclosed
US-8993697-B2 Conducting and semiconducting organic materials Commonwealth Scientific and Industrial Research Institute Organisation (AU) 2015-03-31 US disclosed
US-8993807-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2015-03-31 US disclosed
US-8993262-B2 In vivo and in vitro olefin cyclopropanation catalyzed by heme enzymes CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2015-03-31 US disclosed
US-8993671-B2 Poly(aliphatic ester)-polycarbonate copolymer/polylactic acid blend Sabic Global Technolgies B.V. (NL) 2015-03-31 US disclosed
US-20150087618-A1 Anti-Viral Compounds ABBVIE INC. (US) 2015-03-26 US disclosed
WO-2015042202-A1 CHLOROTOXIN CONJUGATES AND METHODS OF USE THEREOF Blaze Bioscience, Inc. (US) 2015-03-26 WO disclosed
WO-2015041601-A1 CONVERSION AND PURIFICATION OF BIOMASS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-03-26 WO disclosed
US-20150087627-A1 COMBINATION OF KINASE INHIBITORS AND USES THEREOF INTELLIKINE LLC (US) 2015-03-26 US disclosed
US-20150087631-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-03-26 US disclosed
EP-2699575-B1 TRIAZOLOPYRIDINES BAYER IP GMBH (DE) 2015-03-25 EP disclosed
US-8986740-B2 Anti-infective agents and uses thereof ABBVIE INC. (US) 2015-03-24 US disclosed
US-8987538-B2 Carbon nanohoops and methods of making THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-03-24 US disclosed
US-8987493-B2 Process for synthesis of silane dipeptide analogs Temple University—Of the Commonwealth System of Higher Education (US) 2015-03-24 US disclosed
US-8987461-B2 Histone demethylase inhibitors Quanticel Pharmaceuticals, Inc. (US) 2015-03-24 US disclosed
WO-2015038904-A1 ANTI-GP41 ANTIBODY-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2015-03-19 WO disclosed
US-20150080374-A1 AMINOALCOHOL SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-03-19 US disclosed
WO-2015038933-A1 PHOSPHORYLATED AKT-SPECIFIC CAPTURE AGENTS, COMPOSITIONS, AND METHODS OF USING AND MAKING CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2015-03-19 WO disclosed
US-20150080340-A1 BORONIC ACID CONJUGATES OF OLIGONUCLEOTIDE ANALOGUES JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2015-03-19 US disclosed
US-20150080382-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE DOMAIN PARTNERS VIII, L.P. 2015-03-19 US disclosed
US-20150080365-A1 HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT INTERVET INC. 2015-03-19 US disclosed
US-20150078999-A1 CYCLIC PEPTIDES AS PROTEIN TARGETING AGENTS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-03-19 US disclosed
EP-2847163-A1 IRON CHELATORS AS HIV-1 INHIBITORS Howard University (US) 2015-03-18 EP disclosed
EP-2456444-B1 ADENINE DERIVATIVE AS PI3K INHIBITOR INTELLIKINE LLC (US) 2015-03-18 EP disclosed
EP-2846784-A1 COMPOUNDS USEFUL FOR PROMOTING PROTEIN DEGRADATION AND METHODS USING SAME Yale University (US) 2015-03-18 EP disclosed
EP-2655355-B1 NEW TRIAZOLYLPHENYL SULFONAMIDES AS SERINE/THREONINE KINASE INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2015-03-18 EP disclosed
US-8980544-B2 Boronic and borinic acid compounds as inhibitors of sulfenic acid-containing proteins THE PENN STATE RESEARCH FOUNDATION (US) 2015-03-17 US disclosed
US-8981153-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2015-03-17 US disclosed
US-20150072953-A1 COMPOSITIONS AND METHODS FOR JOINT HEALTH UNIGEN, INC. 2015-03-12 US disclosed
US-20150073140-A1 OLIGONUCLEOTIDE ANALOGUES HAVING MODIFIED INTERSUBUNIT LINKAGES AND/OR TERMINAL GROUPS SAREPTA THERAPEUTICS, INC. (US) 2015-03-12 US disclosed
WO-2015034440-A2 A Dimerizer Compound AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-03-12 WO disclosed
WO-2015034436-A1 POLYMER-FLAVONOID CONJUGATES AND HYDROGELS FOR BIOMEDICAL APPLICATIONS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-03-12 WO disclosed
US-20150072959-A1 SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS MIDCAP FINANCIAL TRUST 2015-03-12 US disclosed
US-20150072978-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2015-03-12 US disclosed
WO-2015034785-A1 RILYAZINE DERIVATIVES AND COMPOSITIONS FOR THE TREATMENT OF CANCER WARNER BABCOCK INSTITUTE FOR GREEN CHEMISTRY, LLC (US) 2015-03-12 WO disclosed
EP-2844636-A2 METHODS FOR THE TREATMENT OF DIABETIC RETINOPATHY AND OTHER OPHTHALMIC DISEASES Acucela, Inc. (US) 2015-03-11 EP disclosed
US-8975412-B2 Substituted 4-cyano-3-phenyl-4-(pyridin-3-yl)butanoates, processes for preparation thereof and use thereof as herbicides and plant growth regulators BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-03-10 US disclosed
US-8975278-B2 8-hydroxy quinoline derivatives PRANA BIOTECHNOLOGY LIMITED (AU) 2015-03-10 US disclosed
US-8975288-B2 F2 derivatives as antibacterial agents THE PENN STATE RESEARCH FOUNDATION (US) 2015-03-10 US disclosed
US-8975398-B2 NAMPT inhibitors ABBVIE INC. (US) 2015-03-10 US disclosed
US-20150065510-A1 Rilyazine Derivatives and Compositions for The Treatment of Cancer WARNER BABCOCK INSTITUTE FOR GREEN CHEMISTRY, LLC (US) 2015-03-05 US disclosed
US-20150065468-A1 BIARYL ACETAMIDE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORP (US) 2015-03-05 US disclosed
US-20150065542-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. 2015-03-05 US disclosed
WO-2015031613-A1 BIARYL ACETAMIDE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2015-03-05 WO disclosed
US-20150065532-A1 PYRIMIDINE CYCLOHEXYL GLUCOCORTICOID RECEPTOR MODULATORS CORCEPT THERAPEUTICS, INC. 2015-03-05 US disclosed
US-8969377-B2 Compounds and methods for inhibiting NHE-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders ARDELYX, INC. (US) 2015-03-03 US disclosed
US-8969587-B2 RAF kinase modulator compounds and methods of use thereof AMBIT BIOSCIENCES CORPORATION (US) 2015-03-03 US disclosed
US-8969343-B2 Histone demethylase inhibitors Quanticel Pharmaceuticals, Inc. (US) 2015-03-03 US disclosed
US-8969363-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2015-03-03 US disclosed
US-8969375-B2 CDK9 kinase inhibitors ABBVIE, INC. (US) 2015-03-03 US disclosed
WO-2015025019-A1 NEW 6-ALKYNYL PYRIDINE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-02-26 WO disclosed
WO-2015027176-A1 WATER SOLUBLE FLUORESCENT OR COLORED DYES AND METHODS FOR THEIR USE SONY CORPORATION (JP) 2015-02-26 WO disclosed
US-20150057298-A1 NOVEL COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED 2015-02-26 US disclosed
US-20150057286-A1 NEW BIS-AMIDO PYRIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-02-26 US disclosed
US-20150057295-A1 New 6-Alkynyl Pyridine BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-02-26 US disclosed
WO-2015025018-A1 NEW BIS-AMIDO PYRIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-02-26 WO disclosed
US-20150057279-A1 HETEROARYL COMPOUNDS WITH A-CYCLIC BRIDGING UNIT INTERVET INC. 2015-02-26 US disclosed
US-20150056164-A1 Antiviral Compounds and Uses Thereof ABBVIE INC. (US) 2015-02-26 US disclosed
EP-2838902-A1 ASYMMETRIC SYNTHESES FOR SPIRO-OXINDOLE COMPOUNDS USEFUL AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2015-02-25 EP disclosed
CN-103221435-B Continuous flow polymerisation process COMMW SCIENT IND RES ORG 2015-02-25 CN disclosed
US-8962606-B2 Substituted benzosulphonamides BAYER INTELLECTUAL PROPERTY GMBH (US) 2015-02-24 US disclosed
US-8962529-B2 Substituted picolinic acids, salts and acid derivatives thereof, and use thereof as herbicides BAYER CROPSCIENCE AG (DE) 2015-02-24 US disclosed
US-20150051404-A1 PAIN-RELIEVING COMPOSITIONS AND USES THEREFOR THE UNIVERSITY OF QUEENSLAND (AU) 2015-02-19 US disclosed
US-20150051208-A1 PYRIDINONES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-02-19 US disclosed
US-20150051207-A1 USE OF UNSATURATED SPHINGOSINE COMPOUNDS AS CHEMOTHERAPEUTIC AGENTS FOR THE TREATMENT OF CANCER NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-02-19 US disclosed
WO-2015022332-A1 PYRIDINONES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-02-19 WO disclosed
EP-2836487-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Infinity Pharmaceuticals, Inc. (US) 2015-02-18 EP disclosed
EP-2044938-B1 Radioprotectors PETER MACCALLUM CANCER INST (AU) 2015-02-18 EP disclosed
CN-102361556-B Pyrimindine-4-ylpropane dinitrile derivatives, method for the production thereof, and use thereof as herbicide and plant growth regulators BAYER CROPSCIENCE AG 2015-02-18 CN disclosed
US-8956613-B2 Gemcitabine prodrugs and uses thereof BoYen Therapeutics, Inc. (TW) 2015-02-17 US disclosed
WO-2015021358-A2 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT CHARMOT DOMINIQUE (US) 2015-02-12 WO disclosed
WO-2015019103-A1 PIPERIDINE AND AZEPINE DERIVATIVES AS PROKINETICIN RECEPTOR MODULATORS TAKEDA CAMBRIDGE LIMITED (GB) 2015-02-12 WO disclosed
US-20150045317-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS Cipla USA, Inc. 2015-02-12 US disclosed
US-20150045377-A1 PHARMACEUTICAL COMPOUNDS ALMAC DISCOVERY LIMITED (GB) 2015-02-12 US disclosed
US-20150045444-A1 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. 2015-02-12 US disclosed
EP-2106213-B1 SUBSTITUTED 1-(3-PYRIDINYL)PYRAZOL-4-YL-ACETIC ACIDS, PROCESS FOR THEIR PREPARATION AND THEIR USE AS HERBICIDE AND PLANT GROWTH REGULATORS BAYER IP GMBH (DE) 2015-02-11 EP disclosed
EP-2834245-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Pharma Aktiengesellschaft (DE) 2015-02-11 EP disclosed
US-8952151-B2 Histone demethylase inhibitors Quanticel Pharmaceuticals, Inc. (US) 2015-02-10 US disclosed
US-8952058-B2 Heterocyclic compounds and methods of use thereof AMBIT BIOSCIENCES CORPORATION (US) 2015-02-10 US disclosed
US-8952178-B2 Thiophene derivatives TIANJIN HEMAY BIO-TECH CO., LTD. (CN) 2015-02-10 US disclosed
US-20150037686-A1 HALOGENATED ORGANOSILICON ELECTROLYTES, METHODS OF USING THEM, AND ELECTROCHEMICAL DEVICES CONTAINING THEM ORBIA FLUOR & ENERGY MATERIALS USA, INC. 2015-02-05 US disclosed
US-20150038485-A1 HETEROCYCLYL AMINOIMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-02-05 US disclosed
US-8946360-B2 Continuous flow polymerisation process COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2015-02-03 US disclosed
US-8946279-B2 Fused ring compound for use as mineralocorticoid receptor antagonist KBP BIOSCIENCES CO., LTD. (CN) 2015-02-03 US disclosed
US-20150031891-A1 BIS-QUARTERNARY CINCHONA ALKALOID SALTS AS ASYMMETRIC PHASE TRANSFER CATALYSTS MERCK SHARP & DOHME CORP. (US) 2015-01-29 US disclosed
US-20150031884-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. (US) 2015-01-29 US disclosed
US-20150031672-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. 2015-01-29 US disclosed
US-20150030588-A1 COMBINATION OF KINASE INHIBITORS AND USES THEREOF INTELLIKINE LLC 2015-01-29 US disclosed
US-20150030704-A1 PYRIDAZINONE COMPOUNDS AND THEIR USE AS DAAO INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-01-29 US disclosed
US-8940742-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2015-01-27 US disclosed
US-8940737-B2 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases ABBVIE INC. (US) 2015-01-27 US disclosed
US-20150025266-A1 SYNTHESIS OF HIGH CALORIC FUELS AND CHEMICALS PIONEER ENERGY, INC. (US) 2015-01-22 US disclosed
US-20150025113-A1 RODENTICIDAL NORBORMIDE ANALOGUES ANIMAL CONTROL PRODUCTS LIMITED (NZ) 2015-01-22 US disclosed
US-20150025096-A1 SMALL MOLECULE COMPOUNDS TO TREAT HEARING LOSS FATE THERAPEUTICS, INC. 2015-01-22 US disclosed
US-20150025108-A1 8-HYDROXY QUINOLINE DERIVATIVES PRANA BIOTECHNOLOGY LIMITED (AU) 2015-01-22 US disclosed
US-20150024488-A1 NUCLEIC ACID COMPLEX COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2015-01-22 US disclosed
EP-2825540-A1 SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2015-01-21 EP disclosed
EP-2825536-A1 BIS-QUARTERNARY CINCHONA ALKALOID SALTS AS ASYMMETRIC PHASE TRANSFER CATALYSTS Merck Sharp & Dohme Corp. (US) 2015-01-21 EP disclosed
EP-2825044-A2 PROCESS FOR MAKING CGRP RECEPTOR ANTAGONISTS Merck Sharp & Dohme Corp. (US) 2015-01-21 EP disclosed
US-8937150-B2 Anti-viral compounds ABBVIE INC. (US) 2015-01-20 US disclosed
WO-2015006733-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF HIV INFECTIONS GILEAD SCIENCES, INC. (US) 2015-01-15 WO disclosed
WO-2015004024-A1 SUBSTITUTED PYRAZOLO-PYRIDINAMINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2015-01-15 WO disclosed
WO-2015006731-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF HIV INFECTIONS GILEAD SCIENCES, INC. (US) 2015-01-15 WO disclosed
EP-2822938-A1 RODENTICIDAL NORBORMIDE ANALOGUES Landcare Research New Zealand Limited (NZ) 2015-01-14 EP disclosed
CN-102884054-B Fluoroalkyl-substituted 2-amidobenzimidazoles and the use thereof for boosting stress tolerance in plants BAYER IP GMBH 2015-01-14 CN disclosed
CN-102099408-B Polymer microgel beads and method for producing same UNIV SYDNEY 2015-01-14 CN disclosed
WO-2015002894-A1 PURINONE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS, INC. (US) 2015-01-08 WO disclosed
WO-2015003002-A1 PYRROLO-PYRROLE CARBAMATE AND RELATED ORGANIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND MEDICAL USES THEREOF ABIDE THERAPEUTICS, INC. (US) 2015-01-08 WO disclosed
EP-2819996-A1 6 - ALKYNYL PYRIDINES AS SMAC MIMETICS Boehringer Ingelheim International GmbH (DE) 2015-01-07 EP disclosed
US-8927789-B1 Synthesis of high caloric fuels and chemicals Pioneer Energy (US) 2015-01-06 US disclosed
US-8927711-B2 JAK kinase modulating compounds and methods of use thereof AMBIT BIOSCIENCES CORP. (US) 2015-01-06 US disclosed
US-20150004128-A1 TARGETED DRUG PHOSPHORYLCHOLINE POLYMER CONJUGATES OLIGASIS, LLC (US) 2015-01-01 US disclosed
WO-2014151871-A9 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE TOLERO PHARMACEUTICALS, INC. (US) 2014-12-31 WO disclosed
WO-2014207708-A2 AMINO ACID AND PEPTIDE CONJUGATES AND CONJUGATION PROCESS AUCKLAND UNISERVICES LIMITED (NZ) 2014-12-31 WO disclosed
US-8921514-B2 Anti-viral compounds ABBVIE INC. (US) 2014-12-30 US disclosed
US-8921546-B2 Imidazolothiazole compounds for the treatment of disease AMBIT BIOSCIENCES CORPORATION (US) 2014-12-30 US disclosed
US-20140378446-A1 PURINONE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS, INC. (US) 2014-12-25 US disclosed
US-20140377258-A1 Treatment Of Cancers Using PI3 Kinase Isoform Modulators INFINITY PHARMACEUTICALS, INC. (US) 2014-12-25 US disclosed
US-20140378510-A1 SMALL MOLECULE ACTIVATORS OF CALCIUM-ACTIVATED CHLORIDE CHANNELS AND METHODS OF USE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-12-25 US disclosed
US-20140377285-A1 TREATMENT REGIMENS USING MULTIPLE PHARMACEUTICAL AGENTS INTELLIKINE LLC 2014-12-25 US disclosed
US-20140378490-A1 Formulations of Phenyl Uracil Compounds ABBVIE INC. (US) 2014-12-25 US disclosed
WO-2014204866-A1 COMPOSITIONS AND METHODS FOR JOINT HEALTH UNIGEN, INC. (US) 2014-12-24 WO disclosed
WO-2014205317-A2 CYCLIC PEPTIDES AS PROTEIN TARGETING AGENTS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2014-12-24 WO disclosed
WO-2014202999-A1 1-SULFONYL PIPERIDINE DERIVATIVES AS MODULATORS OF PROKINETICIN RECEPTORS TAKEDA CAMBRIDGE LIMITED (GB) 2014-12-24 WO disclosed
US-8916569-B2 Compounds and methods for inhibiting phosphate transport ARDELYX, INC. (US) 2014-12-23 US disclosed
US-8916270-B2 Glass filled copolymer products for thin wall and high surface gloss articles SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2014-12-23 US disclosed
US-8916580-B2 Spiro-oxindole compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2014-12-23 US disclosed
US-20140371493-A1 METHODS OF CONVERTING POLYOLS UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION 2014-12-18 US disclosed
WO-2014198594-A1 NOVEL COMPOUNDS FOR THE TREATMENT OF CANCER BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-12-18 WO disclosed
US-20140371224-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR TREATMENT OF BREATHING CONTROL DISORDERS OR DISEASES GALLEON PHARMACEUTICALS, INC. 2014-12-18 US disclosed
US-20140371252-A1 INDENE DERIVATIVES AS PHARMACEUTICAL AGENTS AQUINOX PHARMACEUTICALS INC. (CA) 2014-12-18 US disclosed
US-20140371450-A1 PROCESSES FOR PREPARING ISOQUINOLINONES AND SOLID FORMS OF ISOQUINOLINONES HCR COLLATERAL MANAGEMENT, LLC 2014-12-18 US disclosed
US-20140371205-A1 SUBSTITUTED PYRIMIDINES FOR THE TREATMENT OF DISEASES SUCH AS CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-12-18 US disclosed
EP-2507236-B1 Triazolopyridine derivates BAYER IP GMBH (DE) 2014-12-17 EP disclosed
US-8912124-B2 Use of derivatives of (1-cyanocyclopropyl)phenylphosphinic acid, esters thereof and/or salts thereof for enhancing tolerance in plants to abiotic stress BAYER CROPSCIENCE AG (DE) 2014-12-16 US disclosed
US-8912229-B2 Taxane and abeo-taxane analogs Arbor Therapeutics, LLC (US) 2014-12-16 US disclosed
US-20140364616-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. (IL) 2014-12-11 US disclosed
WO-2014194380-A1 SCRATCH RESISTANT POLYMERS TENASITECH PTY LTD (AU) 2014-12-11 WO disclosed
US-20140364435-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-12-11 US disclosed
WO-2014195408-A1 PHARMACEUTICAL COMPOSITIONS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-12-11 WO disclosed
WO-2014195276-A1 SUBSTITUTED TRIAZOLOPYRIDINES HAVING ACTIVITY AS MPS-1 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-12-11 WO disclosed
US-20140364617-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. 2014-12-11 US disclosed
US-20140364315-A1 SUBSTITUTED 4-CYAN-3-PHENYL-4-(PRYRIDINE-3-YL)BUTANOATES, PROCESSES FOR PREPARATION THEREOF AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-12-11 US disclosed
EP-1827438-B2 PIPERAZIN DERIVATIVES FOR INHIBITING HUMAN STEAROYL-COA-DESATURASE XENON PHARMACEUTICALS INC (CA) 2014-12-10 EP disclosed
EP-2651947-B1 6-THIO-SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER IP GMBH (DE) 2014-12-10 EP disclosed
EP-2809672-A1 PURINONE COMPOUNDS AS KINASE INHIBITORS Pharmacyclics, Inc. (US) 2014-12-10 EP disclosed
EP-2809708-A1 HALOGENATED ORGANOSILICON ELECTROLYTES, METHODS OF USING THEM, AND ELECTROCHEMICAL DEVICES CONTAINING THEM Silatronix, Inc. (US) 2014-12-10 EP disclosed
US-8906922-B2 Substituted triazoles useful as AXl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2014-12-09 US disclosed
US-8906917-B2 Pyrimidine cyclohexyl glucocorticoid receptor modulators CORCEPT THERAPEUTICS, INC. (US) 2014-12-09 US disclosed
WO-2014190398-A1 INHIBITION OF AMYLOID FIBRIL FORMATION THE UNIVERSITY OF MELBOURNE (AU) 2014-12-04 WO disclosed
WO-2014194254-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS INFINITY PHARMACEUTICALS, INC. (US) 2014-12-04 WO disclosed
US-20140357878-A1 METHOD OF PRODUCING 5-HYDROXYMETHYLFURFURAL FROM CARBOHYDRATES AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2014-12-04 US disclosed
US-20140357655-A1 SPIROINDOLINE DERIVATIVES AS GONADOTROPIN- RELEASING HORMONE RECEPTOR ANTAGONISTS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-12-04 US disclosed
US-20140352351-A1 REFRIGERATION SYSTEM WITH DUAL REFRIGERANTS AND LIQUID WORKING FLUIDS H & C Scientific Resources International, LLC (US) 2014-12-04 US disclosed
US-20140357616-A1 PYRROLOPYRIDINE INHIBITORS OF KINASES ABBVIE INC (US) 2014-12-04 US disclosed
US-20140357651-A1 COMBINATION PHARMACEUTICAL COMPOSITIONS AND USES THEREOF CALITHERA BIOSCIENCES, INC. 2014-12-04 US disclosed
WO-2014193857-A1 REFRIGERATION SYSTEM WITH DUAL REFRIGERANTS AND LIQUID WORKING FLUIDS XU YANJIE (US) 2014-12-04 WO disclosed
EP-2807166-A1 5, 8 -DIHYDRO- 6H- PYRAZOLO [3, 4 -H]QUINAZOLINES AS IGF-LR/LR INHIBITORS Boehringer Ingelheim International GmbH (DE) 2014-12-03 EP disclosed
CN-101606069-B Tagged petroleum products and methods of detecting the same AUTHENTIX INC 2014-12-03 CN disclosed
US-8901133-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2014-12-02 US disclosed
US-20140350183-A1 CHROMOPHORIC POLYMER DOTS WITH NARROW-BAND EMISSION UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION 2014-11-27 US disclosed
US-20140350182-A1 RAFT POLYMERS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2014-11-27 US disclosed
US-20140349918-A1 DERIVATIVES OF XANTHONE COMPOUNDS SINGAPORE HEALTH SERVICES PTE LTD. (SG) 2014-11-27 US disclosed
WO-2014190199-A1 COMPOUNDS FOR TREATMENT OF DRUG RESISTANT AND PERSISTENT TUBERCULOSIS THE CALIFORNIA INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2014-11-27 WO disclosed
US-20140350009-A1 PYRAZOLYLBENZOTHIAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS DERMIRA (CANADA), INC. (US) 2014-11-27 US disclosed
EP-2804605-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS FOR DISEASE TREATMENT Acucela, Inc. (US) 2014-11-26 EP disclosed
EP-2455376-B1 Heterocyclic compounds as inhibitors of hepatitis C virus (HCV) ABBVIE BAHAMAS LTD (BS) 2014-11-26 EP disclosed
EP-2804864-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2014-11-26 EP disclosed
EP-2804867-A1 SPIROINDOLINE DERIVATIVES AS GONADOTROPIN- RELEASING HORMONE RECEPTOR ANTAGONISTS Bayer Intellectual Property GmbH (DE) 2014-11-26 EP disclosed
US-8895549-B2 Aminoalcohol substituted 2,3-dihydroimidazo[1,2-c]quinazoline derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-11-25 US disclosed
US-8895581-B2 1H-imidazo[4,5-c]quinolines BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-11-25 US disclosed
US-8895782-B2 Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2014-11-25 US disclosed
US-20140343057-A1 TREATMENT OF LUPUS, FIBROTIC CONDITIONS, AND INFLAMMATORY MYOPATHIES AND OTHER DISORDERS USING PI3 KINASE INHIBITORS INFINITY PHARMACEUTICALS, INC. 2014-11-20 US disclosed
US-20140341894-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE, INC. 2014-11-20 US disclosed
US-20140343286-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. 2014-11-20 US disclosed
EP-2802595-A1 PROCESSES FOR MAKING HCV PROTEASE INHIBITORS AbbVie Inc. (US) 2014-11-19 EP disclosed
EP-2655358-B1 OXINDOLOPYRIMIDINE AS IGF1R RECEPTOR INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2014-11-19 EP disclosed
EP-2032583-B1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2014-11-19 EP disclosed
US-8889675-B2 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases ABBVIE INC. (US) 2014-11-18 US disclosed
US-8889696-B2 Substituted pyrido[2,3-d]pyrimidin-7(8H)-ones and therapeutic uses thereof Temple University—Of the Commonwealth System of Higher Education (US) 2014-11-18 US disclosed
US-8889665-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-11-18 US disclosed
US-8889684-B2 Azaindolylphenyl sulfonamides as serine/threonine kinase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-11-18 US disclosed
US-20140336168-A1 NAMPT INHIBITORS ABBVIE INC. 2014-11-13 US disclosed
US-20140336167-A1 NAMPT INHIBITORS ABBVIE INC. (US) 2014-11-13 US disclosed
US-8883791-B2 N-heteroaryl compounds with cyclic bridging unit for the treatment of parasitic diseases INTERVET INC. (US) 2014-11-11 US disclosed
US-8883784-B2 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases ABBVIE INC. (US) 2014-11-11 US disclosed
US-20140329684-A1 USE OF 4-SUBSTITUTED 1-PHENYLPYRAZOLE-3-CARBOXYLIC ACID DERIVATIVES AS AGENTS AGAINST ABIOTIC PLANT STRESS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-11-06 US disclosed
US-20140330006-A1 FUNCTIONALLY-MODIFIED OLIGONUCLEOTIDES AND SUBUNITS THEREOF SAREPTA THERAPEUTICS, INC. (US) 2014-11-06 US disclosed
US-20140329932-A1 POLYMER PARTICLES THE UNIVERSITY OF SYDNEY (AU) 2014-11-06 US disclosed
US-20140326672-A1 MELAMINE ALDEHYDE POLYMERS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2014-11-06 US disclosed
EP-2797889-A1 NOVEL ARYLALKENE DERIVATIVES AND USE THEREOF AS SELECTIVE ESTROGEN RECEPTOR MODULATORS Centaurus Biopharma Co., Ltd. (CN) 2014-11-05 EP disclosed
US-8877720-B2 Epirubicin derivatives TIANJIN HEMAY BIO-TECH CO., LTD. (CN) 2014-11-04 US disclosed
US-8877934-B2 N-heteroaryl compounds INTERVET INC. (US) 2014-11-04 US disclosed
US-20140323527-A1 ARYLOXY AMINE COMPOUNDS AND THEIR USE AS SODIUM CHANNEL MODULATORS HOWARD FLOREY INSTITUTE (AU) 2014-10-30 US disclosed
US-20140323490-A1 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2014-10-30 US disclosed
US-20140323530-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. (US) 2014-10-30 US disclosed
US-20140323721-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE LLC 2014-10-30 US disclosed
EP-2435411-B1 2,4-DIAMINOPYRIMIDINES FOR THE TREATMENT OF DISEASES CHARACTERISED BY EXCESSIVE OR ABNORMAL CELL PROLIFERATION BOEHRINGER INGELHEIM INT (DE) 2014-10-29 EP disclosed
EP-2793893-A2 ENHANCED TREATMENT REGIMENS USING MTOR INHIBITORS Intellikine, LLC (US) 2014-10-29 EP disclosed
CN-104125945-A Substituted 4-cyano-3-phenyl-4- (pyridin-3-yl) butanoic acid esters, process for their preparation and their use as herbicides and plant growth regulators BAYER IP GMBH 2014-10-29 CN disclosed
CN-102245214-B Biodegradable polymer-bioactive moiety conjugates POLYACTIVA PTY LTD. (AU) 2014-10-29 CN disclosed
US-8871718-B2 Transglutaminase inhibitors and methods of use thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2014-10-28 US disclosed
US-20140315954-A1 CYTOTOXIC AND ANTI-MITOTIC COMPOUNDS, AND METHODS OF USING THE SAME ZYMEWORKS BC INC. (CA) 2014-10-23 US disclosed
US-20140315792-A1 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES 2014-10-23 US disclosed
EP-2791136-A1 SUBSTITUTED TRIAZOLOPYRIDINES AND THEIR USE AS TTK INHIBITORS Bayer Intellectual Property GmbH (DE) 2014-10-22 EP disclosed
EP-2507235-B1 TRIAZOLOPYRIMIDINES BAYER IP GMBH (DE) 2014-10-22 EP disclosed
EP-2552907-B1 PYRIDYLTRIAZOLES BOEHRINGER INGELHEIM INT (DE) 2014-10-22 EP disclosed
CN-104114547-A Derivatives of xanthone compounds AGENCY SCIENCE TECH & RES 2014-10-22 CN disclosed
US-8865703-B2 Pyridyltriazoles BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-10-21 US disclosed
EP-2788488-A2 METHODS FOR TREATING PROGEROID LAMINOPATHIES USING OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA Sarepta Therapeutics, Inc. (US) 2014-10-15 EP disclosed
EP-2387395-B1 AXL INHIBITORS FOR USE IN COMBINATION THERAPY FOR PREVENTING, TREATING OR MANAGING METASTATIC CANCER RIGEL PHARMACEUTICALS INC (US) 2014-10-15 EP disclosed
EP-2788487-A2 OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA Sarepta Therapeutics, Inc. (US) 2014-10-15 EP disclosed
CN-104105718-A RAFT polymers COMMW SCIENT IND RES ORG 2014-10-15 CN disclosed
US-8859541-B2 6-alkynylpyridines BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-10-14 US disclosed
US-8859546-B2 Picolinamide inhibitors of kinases ABBVIE INC. (US) 2014-10-14 US disclosed
US-8859765-B2 Process for the manufacture of chiral catalysts and their salts SCINOPHARM TAIWAN, LTD. (TW) 2014-10-14 US disclosed
US-20140302010-A1 SUBSTITUTED BENZIMIDAZOLES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-10-09 US disclosed
US-20140302987-A1 USE OF SUBSTITUTED ISOQUINOLINONES, ISOQUINOLINDIONES, ISOQUINOLINTRIONES AND DIHYDROISOQUINOLINONES OR IN EACH CASE SALTS THEREOF AS ACTIVE AGENTS AGAINST ABIOTIC STRESS IN PLANTS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-10-09 US disclosed
WO-2014164905-A1 SUBSTITUTED 3-PHENYLPROPYLAMINE DERIVATIVES FOR THE TREATMENT OF OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. (US) 2014-10-09 WO disclosed
EP-2785650-A1 Melamine Aldehyde Polymers Agency For Science, Technology And Research (SG) 2014-10-08 EP disclosed
US-8853420-B2 Compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-10-07 US disclosed
US-8853330-B2 Hybrid polymers AGENCY FOR SCIENCE TECHNOLOGY AND RESEARCH (SG) 2014-10-07 US disclosed
US-8852641-B2 Polymer microgel beads and preparative method thereof THE UNIVERSITY OF SYDNEY (AU) 2014-10-07 US disclosed
US-20140294766-A1 Anti-Infective Agents and Uses Thereof ABBVIE INC (US) 2014-10-02 US disclosed
US-20140296073-A1 SUBSTITUTED 4-CYANO-3-PHENYL-4-(PYRIDIN-3-YL)BUTANOATES, PROCESSES FOR PREPARATION THEREOF AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-10-02 US disclosed
US-20140296230-A1 DIHYDROQUINAZOLINONE ANALOGUES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-10-02 US disclosed
US-20140296321-A1 METHODS AND COMPOSITIONS FOR MANIPULATING TRANSLATION OF PROTEIN ISOFORMS FROM ALTERNATIVE INITIATION OF START SITES SAREPTA THERAPEUTICS, INC. (US) 2014-10-02 US disclosed
WO-2014154762-A1 DIHYDROQUINAZOLINONE ANALOGUES AS BRD4 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-10-02 WO disclosed
WO-2014154760-A1 INDOLINONE ANALOGUES AS BRD4 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-10-02 WO disclosed
US-20140296220-A1 PYRIDAZINO[4,5-D]PYRIMIDIN-5(6H)-ONE INHIBITORS OF KINASES ABBVIE INC (US) 2014-10-02 US disclosed
WO-2014158654-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO AQUINOX PHARMACEUTICALS INC. (CA) 2014-10-02 WO disclosed
US-20140296231-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-10-02 US disclosed
WO-2014160017-A1 PYRIDINE CDK9 KINASE INHIBITORS ABBVIE INC. (US) 2014-10-02 WO disclosed
WO-2014160028-A1 PYRROLOPYRIMINDINE CDK9 KINASE INHIBITORS ABBVIE INC. (US) 2014-10-02 WO disclosed
US-20140296207-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, INC. 2014-10-02 US disclosed
US-20140296229-A1 INDOLINONE ANALOGUES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-10-02 US disclosed
EP-2782571-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Intellikine, LLC (US) 2014-10-01 EP disclosed
EP-2782962-A1 POLY(ALIPHATIC ESTER)-POLYCARBONATE COPOLYMER/POLYLACTIC ACID BLEND SABIC Innovative Plastics IP B.V. (NL) 2014-10-01 EP disclosed
US-8846689-B2 Substituted pyrimidines for the treatment of diseases such as cancer BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-09-30 US disclosed
US-20140288045-A1 COVALENT INHIBITORS OF KRAS G12C ARAXES PHARMA LLC 2014-09-25 US disclosed
US-20140288048-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. 2014-09-25 US disclosed
US-20140288069-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES AS MKNK1 KINASE INHIBITORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-09-25 US disclosed
US-20140287031-A1 ENHANCED TREATMENT REGIMENS USING MTOR INHIBITORS INTELLIKINE, LLC (US) 2014-09-25 US disclosed
WO-2014152287-A2 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES, INC. (US) 2014-09-25 WO disclosed
US-20140283438-A1 Synthesis of High Caloric Fuels and Chemicals Pioneer Energy (US) 2014-09-25 US disclosed
WO-2014151871-A2 JAK2 AND ALK2 INHIBITORS AND METHODS FOR THEIR USE TOLERO PHARMACEUTICALS, INC. (US) 2014-09-25 WO disclosed
WO-2014152229-A2 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS, INC. (US) 2014-09-25 WO disclosed
WO-2014151444-A1 PYRROLO[2,3-B]PYRIDINE CDK9 KINASE INHIBITORS ABBVIE INC. (US) 2014-09-25 WO disclosed
US-20140287945-A1 SURFACE OXIDATION FOR SEQUESTERING BIOMOLECULES AND RELATED METHODS NVS Technologies, Inc. (US) 2014-09-25 US disclosed
WO-2014151106-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2014-09-25 WO disclosed
WO-2014149837-A1 COMPOUNDS AND METHODS TO ENHANCE THE ORAL AVAILABILITY OF GLYCOMIMETICS GLYCOMIMETICS, INC. (US) 2014-09-25 WO disclosed
WO-2014152536-A2 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS, INC. (US) 2014-09-25 WO disclosed
WO-2014152518-A2 INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS, INC. (US) 2014-09-25 WO disclosed
WO-2014152588-A1 COVALENT INHIBITORS OF KRAS G12C ARAXES PHARMA LLC (US) 2014-09-25 WO disclosed
WO-2014151462-A1 NOVEL BREATHING CONTROL MODULATING COMPOUNDS, AND METHODS OF USING SAME GALLEON PHARMACEUTICALS, INC. (US) 2014-09-25 WO disclosed
WO-2014151945-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2014-09-25 WO disclosed
WO-2014147182-A2 NOVEL COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-09-25 WO disclosed
WO-2014147021-A2 NOVEL COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-09-25 WO disclosed
WO-2014151147-A1 COMBINATION OF KINASE INHIBITORS AND USES THEREOF INTELLIKINE, LLC (US) 2014-09-25 WO disclosed
WO-2014153051-A1 POLYMER DOT COMPOSITIONS AND RELATED METHODS UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2014-09-25 WO disclosed
EP-2780299-A1 FUNCTIONALLY-MODIFIED OLIGONUCLEOTIDES AND SUBUNITS THEREOF Sarepta Therapeutics, Inc. (US) 2014-09-24 EP disclosed
EP-2781520-A1 THREE-RING PI3K AND/OR MTOR INHIBITOR Xuanzhu Pharma Co., Ltd. (CN) 2014-09-24 EP disclosed
CN-101563331-B Substituted 2, 4-diamino-1, 3, 5-triazines, method for the production thereof and use thereof as herbicides and plant growth regulators BAYER CROPSCIENCE AG 2014-09-24 CN disclosed
US-8840339-B2 Soil remediation process THE UNIVERSITY OF QUEENSLAND (AU) 2014-09-23 US disclosed
US-20140275431-A1 ALKYL-ACID LIGANDS FOR NANOCRYSTALS NANOSYS, INC. (US) 2014-09-18 US disclosed
WO-2014138791-A1 TRANSGENIC NON-HUMAN ORGANISMS WITH NON-FUNCTIONAL TSPO GENES AUSTRALIAN NUCLEAR SCIENCE AND TECHNOLOGY ORGANISATION (AU) 2014-09-18 WO disclosed
US-20140275598-A1 POLYHEDRAL OLIGOMERIC SILSESQUIOXANE NANOCRYSTAL STABILIZATION LIGANDS NANOSYS, INC. (US) 2014-09-18 US disclosed
WO-2014144871-A1 CYTOTOXIC AND ANTI-MITOTIC COMPOUNDS, AND METHODS OF USING THE SAME THE CENTRE FOR DRUG RESEARCH AND DEVELOPMENT (CA) 2014-09-18 WO disclosed
US-20140274700-A1 MOLECULES THAT INDUCE DISEASE RESISTANCE AND IMPROVE GROWTH IN PLANTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-09-18 US disclosed
US-20140275004-A1 PYRROLOPYRIMINDINE CDK9 KINASE INHIBITORS ABBVIE INC. 2014-09-18 US disclosed
US-20140275027-A1 PYRROLO[2,3-B]PYRIDINE CDK9 KINASE INHIBITORS ABBVIE INC. 2014-09-18 US disclosed
WO-2014143561-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO AQUINOX PHARMACEUTICALS INC. (CA) 2014-09-18 WO disclosed
US-20140274699-A1 MOLECULES THAT INDUCE DISEASE RESISTANCE IN PLANTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-09-18 US disclosed
US-20140275011-A1 PYRIDINE CDK9 KINASE INHIBITORS ABBVIE INC. (US) 2014-09-18 US disclosed
US-20140275153-A1 CDK9 KINASE INHIBITORS ABBIVE INC. 2014-09-18 US disclosed
US-20140275528-A1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES, INC. (US) 2014-09-18 US disclosed
US-20140264189-A1 METHOD FOR SOLVENTLESS QUANTUM DOT EXCHANGE NANOSYS, INC. (US) 2014-09-18 US disclosed
US-20140275071-A1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES, INC. (US) 2014-09-18 US disclosed
US-20140275084-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2014-09-18 US disclosed
US-20140275043-A1 SUBSTITUTED 3-PHENYLPROPYLAMINE DERIVATIVES FOR THE TREATMENT OF OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. (US) 2014-09-18 US disclosed
US-20140275192-A1 F2 DERIVATIVES AS ANTIBACTERIAL AGENTS THE PENN STATE RESEARCH FOUNDATION 2014-09-18 US disclosed
WO-2014144197-A1 STEREODYNAMIC CHEMOSENSORS GEORGETOWN UNIVERSITY (US) 2014-09-18 WO disclosed
WO-2014145780-A1 PURIFICATION OF RAPAMYCIN DERIVATIVES BIOSENSORS INTERNATIONAL GROUP, LTD. (SG) 2014-09-18 WO disclosed
EP-2776434-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES Abbvie Inc. (US) 2014-09-17 EP disclosed
EP-2776475-A1 CLEAN POLYCARBONATE MATERIAL FOR USE IN HARD DISK DRIVE AND SEMICONDUCTOR APPLICATIONS SABIC Innovative Plastics IP B.V. (NL) 2014-09-17 EP disclosed
EP-2776837-A1 COMBINATION OF KINASE INHIBITORS AND USES THEREOF Intellikine, LLC (US) 2014-09-17 EP disclosed
EP-2428515-B9 Spiro-oxindole compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC (CA) 2014-09-17 EP disclosed
EP-2776393-A1 NAMPT INHIBITORS Abbvie Inc. (US) 2014-09-17 EP disclosed
EP-2776441-A1 TREATMENT REGIMENS USING MULTIPLE PHARMACEUTICAL AGENTS Intellikine, LLC (US) 2014-09-17 EP disclosed
CN-104053729-A Polymer particles UNIV SYDNEY 2014-09-17 CN disclosed
CN-102361889-B Raft polymerisation COMMW SCIENT IND RES ORG 2014-09-17 CN disclosed
US-8836218-B2 Methods of treatment using combination therapy AMBIT BIOSCIENCES CORPORATION (US) 2014-09-16 US disclosed
WO-2014135480-A1 SUBSTITUTED THIAZOLOPYRIMIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-09-12 WO disclosed
WO-2014138312-A1 WESTERN BLOT ANALYSIS USING POLYMER DOTS UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2014-09-12 WO disclosed
WO-2014136099-A1 PROCESS FOR IXABEPILONE, AND INTERMEDIATES THEREOF SCINOPHARM TAIWAN, LTD. (CN) 2014-09-12 WO disclosed
US-20140256992-A1 SYNTHESIS OF HIGH CALORIC FUELS AND CHEMICALS Pioneer Energy (US) 2014-09-11 US disclosed
US-20140255392-A1 SUBSTITUTED IMIDAZOPYRIDINES AND INTERMEDIATES THEREOF BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-09-11 US disclosed
US-20140256952-A1 PROCESS FOR IXABEPILONE, AND INTERMEDIATES THEREOF SCINOPHARM TAIWAN, LTD. (TW) 2014-09-11 US disclosed
US-20140255342-A1 THIOPHENE DERIVATIVES TIANJIN HEMAY BIO-TECH CO., LTD. (CN) 2014-09-11 US disclosed
EP-2542533-B1 FLUORALKYL-SUBSTITUTED 2-AMIDOBENZIMIDAZOLES AND THEIR USE FOR INCREASING STRESS TOLERANCE IN PLANTS BAYER IP GMBH (DE) 2014-09-10 EP disclosed
US-8828998-B2 Treatment of lupus, fibrotic conditions, and inflammatory myopathies and other disorders using PI3 kinase inhibitors INFINITY PHARMACEUTICALS, INC. (US) 2014-09-09 US disclosed
US-8829244-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2014-09-09 US disclosed
US-20140245658-A1 SYNTHESIS OF ETHANOL AND HIGHER ALCOHOLS BY HYDROGENATION OF KETENE PIONEER ENERGY INC (US) 2014-09-04 US disclosed
EP-2326641-B1 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS INC (US) 2014-09-03 EP disclosed
EP-1910308-B1 IMIDAZOLE BASED LXR MODULATORS EXELIXIS PATENT CO LLC (US) 2014-09-03 EP disclosed
EP-2408742-B1 ANTHELMINTIC AGENTS AND THEIR USE INTERVET INT BV (NL) 2014-09-03 EP disclosed
US-8822509-B2 Pain-relieving compositions and uses therefor THE UNIVERSITY OF QUEENSLAND (AU) 2014-09-02 US disclosed
US-8822424-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2014-09-02 US disclosed
US-8822446-B2 Pyrrolopyridine inhibitors of kinases ABBVIE INC. (US) 2014-09-02 US disclosed
US-20140243353-A1 5- OR 6-SUBSTITUTED 3-HYDROXY-2(1H)-PYRIDINONES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS IN THERAPY OF DISEASES SUCH AS SCHIZOPHRENIA, COGNITIVE DISORDER AND PAID TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2014-08-28 US disclosed
US-20140243288-A1 FUSED RING-CONTAINING OXAZOLIDINONES ANTIBIOTICS Xuanzhu Pharma Co., Ltd. (CN) 2014-08-28 US disclosed
US-20140243525-A1 IMIDAZOLOTHIAZOLE COMPOUNDS FOR THE TREATMENT OF DISEASE AMBIT BIOSCIENCES CORPORATION (US) 2014-08-28 US disclosed
US-20140242647-A1 IN VIVO AND IN VITRO OLEFIN CYCLOPROPANATION CATALYZED BY HEME ENZYMES CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2014-08-28 US disclosed
WO-2014130693-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE PHARMACYCLICS, INC. (US) 2014-08-28 WO disclosed
WO-2014128093-A1 SUBSTITUTED-IMIDAZO[1,2-B]PYRIDAZINES AS MKNK1 INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-08-28 WO disclosed
WO-2014127430-A1 LITHOGRAPHICALLY PRODUCED FEATURES THE UNIVERSITY OF QUEENSLAND (AU) 2014-08-28 WO disclosed
CN-102099407-B Polymer microgel beads UNIV SYDNEY 2014-08-27 CN disclosed
US-8815908-B2 Compounds and methods for inhibiting phosphate transport ARDELYX, INC. (US) 2014-08-26 US disclosed
US-8815910-B2 Compounds and methods for inhibiting phosphate transport ARDELYX, INC. (US) 2014-08-26 US disclosed
US-20140235638-A1 Anti-Infective Agents and Uses Thereof ABBVIE INC. (US) 2014-08-21 US disclosed
US-20140235548-A1 COMPOSITIONS AND METHODS FOR JAMM PROTEIN INHIBITION CLEAVE BIOSCIENCES, INC. (US) 2014-08-21 US disclosed
US-20140235584-A1 BIARYL HETEROCYCLE SUBSTITUTED OXAZOLIDINONE ANTIBACTERIAL AGENTS Xuanzhu Pharma Co., Ltd. (CN) 2014-08-21 US disclosed
US-20140235580-A1 INHIBITORS OF MONOACYLGLYCEROL LIPASE AND METHODS OF THEIR USE INFINITY PHARMACEUTICALS, INC. 2014-08-21 US disclosed
US-20140235446-A1 2,3-DIPHENYL-VALERONITRILE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-08-21 US disclosed
EP-2766359-A2 HETEROCYCLIC COMPOUNDS AND USE THEREOF AS MODULATORS OF TYPE III RECEPTOR TYROSINE KINASES Ambit Biosciences Corporation (US) 2014-08-20 EP disclosed
EP-2498599-B1 ANALGESIC THAT BINDS FILAMIN A PAIN THERAPEUTICS INC (US) 2014-08-20 EP disclosed
EP-2766361-A1 8 - CARBAMOYL - 2 - (2,3- DI SUBSTITUTED PYRID - 6 - YL) -1,2,3,4 -TETRAHYDROISOQUINOLINE DERIVATIVES AS APOPTOSIS - INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES AbbVie Inc. (US) 2014-08-20 EP disclosed
US-8809364-B2 Polycyclic aryl substituted triazoles and polycyclic heteroaryl substituted triazoles useful as axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2014-08-19 US disclosed
US-8809349-B2 Processes for preparing isoquinolinones and solid forms of isoquinolinones INFINITY PHARMACEUTICALS, INC. (US) 2014-08-19 US disclosed
US-8808702-B2 Sulfide, sulfoxide and sulfone chalcone analogues, derivatives thereof and therapeutic uses thereof TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2014-08-19 US disclosed
US-8809339-B2 Compounds and methods for inhibiting phosphate transport ARDELYX, INC. (US) 2014-08-19 US disclosed
US-8809347-B2 Bicyclic aryl and bicyclic heteroaryl substituted triazoles useful as AXL inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2014-08-19 US disclosed
US-20140228443-A1 COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. (US) 2014-08-14 US disclosed
WO-2014122474-A1 PIPERIDIN-1 -YL AND AZEPIN-1 -YL CARBOXYLATES AS MUSCARINIC M4 RECEPTOR AGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2014-08-14 WO disclosed
US-20140228370-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-08-14 US disclosed
US-20140227191-A1 L-GLUTAMIC ACID AND L-GLUTAMINE DERIVATIVE (III), USE THEREOF AND METHOD FOR OBTAINING THEM BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2014-08-14 US disclosed
EP-2350052-B1 ANTIPROLIFERATIVE COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2014-08-13 EP disclosed
EP-2368882-B1 ANTI-INFECTIVE PYRIMIDINES AND USES THEREOF ABBVIE BAHAMAS LTD (BS) 2014-08-13 EP disclosed
EP-2558469-B1 PYRROLOPYRAZINONE INHIBITORS OF KINASES ABBVIE INC (US) 2014-08-13 EP disclosed
US-20140221355-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2014-08-07 US disclosed
US-20140221356-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2014-08-07 US disclosed
WO-2014118135-A1 AMIDOIMIDAZOPYRIDAZINES AS MKNK-1 KINASE INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-08-07 WO disclosed
WO-2014120488-A1 PHOSPHINATE IONIC LIQUID COMPOSITIONS AND METHODS OF USE XU YANJIE (US) 2014-08-07 WO disclosed
WO-2014118226-A1 SUBSTITUTED PYRAZOLOPYRIMIDINYLAMINO-INDAZOLES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-08-07 WO disclosed
EP-2762480-A1 OXAZOLIDINONE ANTIBIOTICS CONTAINING FUSED RING Xuanzhu Pharma Co., Ltd. (CN) 2014-08-06 EP disclosed
EP-2762479-A1 BIARYL HETEROCYCLE SUBSTITUTED OXAZOLIDINON ANTIBACTERIAL DRUG Xuanzhu Pharma Co., Ltd. (CN) 2014-08-06 EP disclosed
CN-103974932-A Preparation method of chiral catalyst and salt thereof SCINOPHARM TAIWAN LTD 2014-08-06 CN disclosed
US-8796277-B2 Radioprotector compounds and related methods PETER MACCALLUM CANCER INSTITUTE (AU) 2014-08-05 US disclosed
US-8796359-B2 Polymer product and interfacial polymerisation process using raft agent THE UNIVERSITY OF SYDNEY (AU) 2014-08-05 US disclosed
US-8796289-B2 Pyridazino[4,5-D]pyrimidin-5(6H)-one inhibitors of kinases ABBVIE INC. (US) 2014-08-05 US disclosed
US-8796259-B2 N3-heteroaryl substituted triazoles and N5-heteroaryl substituted triazoles useful as axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2014-08-05 US disclosed
US-20140213617-A1 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. (US) 2014-07-31 US disclosed
US-20140213585-A1 PYRIMIDINE-2-AMINE COMPOUNDS AND THEIR USE AS INHIBITORS OF JAK KINASES RIGEL PHARMACEUTICALS, INC. (US) 2014-07-31 US disclosed
US-20140213591-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2014-07-31 US disclosed
US-20140213601-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. (US) 2014-07-31 US disclosed
US-20140213595-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. (US) 2014-07-31 US disclosed
EP-2758400-A1 SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2014-07-30 EP disclosed
EP-2758401-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2014-07-30 EP disclosed
EP-2212329-B1 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF (1) CHOONGWAE PHARMA CORP (KR) 2014-07-30 EP disclosed
US-20140206684-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE LLC (US) 2014-07-24 US disclosed
US-20140206685-A1 HETEROCYCLIC KINASE INHIBITORS INTELLIKINE LLC (US) 2014-07-24 US disclosed
EP-2337781-B1 ANTI-VIRAL COMPOUNDS TO TREAT HCV INFECTION ABBVIE BAHAMAS LTD (BS) 2014-07-23 EP disclosed
EP-2291175-B1 ADMINISTRABLE COMPOSITIONS UNIV SYDNEY (AU) 2014-07-23 EP disclosed
US-8785454-B2 Heterocyclic compounds and uses thereof INTELLIKINE LLC (US) 2014-07-22 US disclosed
US-8785470-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2014-07-22 US disclosed
US-8785464-B2 Pyrimidine derivatives that inhibit FAK/PTK2 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-07-22 US disclosed
US-8785456-B2 Substituted isoquinolin-1(2H)-ones, and methods of use thereof INTELLIKINE LLC (US) 2014-07-22 US disclosed
WO-2014110036-A1 SHIP1 MODULATORS AND METHODS RELATED THERETO AQUINOX PHARMACEUTICALS INC. (CA) 2014-07-17 WO disclosed
US-8779128-B2 Oligonucleotide analogues having modified intersubunit linkages and/or terminal groups SAREPTA THERAPEUTICS, INC. (US) 2014-07-15 US disclosed
US-8779029-B2 Polymer product and interfacial polymerisation process using raft agent THE UNIVERSITY OF SYDNEY (AU) 2014-07-15 US disclosed
US-8778929-B2 Substituted heteroaryl inhibitors of B-RAF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-07-15 US disclosed
US-20140194418-A1 BICYCLIC CARBOXAMIDE INHIBITORS OF KINASES ABBVIE INC. (US) 2014-07-10 US disclosed
US-20140194291-A1 SUBSTITUTED (3R,4R)-4-CYAN-3,4-DIPHENYLBUTANOATES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-07-10 US disclosed
US-20140194469-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2014-07-10 US disclosed
US-20140194430-A1 SUBSTITUTED AMINOIMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-07-10 US disclosed
EP-2751093-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Infinity Pharmaceuticals, Inc. (US) 2014-07-09 EP disclosed
EP-2752415-A1 Fluorinated ligands for targeting peripheral benzodiazepine receptors AUSTRALIAN NUCLEAR SCIENCE & TECHNOLOGY ORGANISATION (AU) 2014-07-09 EP disclosed
EP-2752417-A1 Spiro-oxindole compounds and their uses as therapeutic agents Xenon Pharmaceuticals Inc. (CA) 2014-07-09 EP disclosed
US-20140187531-A1 APOPTOSIS PROMOTERS ABBVIE INC. (US) 2014-07-03 US disclosed
US-20140187548-A1 6 SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-07-03 US disclosed
EP-2234973-B1 ANTHELMINTIC AGENTS AND THEIR USE INTERVET INT BV (NL) 2014-07-02 EP disclosed
EP-2035421-B1 2-Arylpyrazolo[l,5-alpha]pyrimidin-3-yl acetamide derivatives as ligands for translocator protein (18 kDa) UNIV SYDNEY (AU) 2014-07-02 EP disclosed
CN-103906747-A Preparation method of cabazitaxel and intermediate thereof SCINOPHARM TAIWAN LTD 2014-07-02 CN disclosed
US-8765183-B2 Polymer microgel beads THE UNIVERSITY OF SYDNEY (AU) 2014-07-01 US disclosed
US-8766006-B2 Use of nitroaniline derivatives for the production of nitric oxide STMICROELECTRONICS S.R.L. (IT) 2014-07-01 US disclosed
US-8765432-B2 Targeted drug phosphorylcholine polymer conjugates OLIGASIS, LLC (US) 2014-07-01 US disclosed
US-8765939-B2 Pyrimidline derivatives having immune modulating properties that act via TLR7 for the treatment of viral or allergic diseases and cancers ASTRAZENECA AB (SE) 2014-07-01 US disclosed
US-8766007-B2 Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC (US) 2014-07-01 US disclosed
US-20140178322-A1 BRIGHTENER-CONTAINING HAIR RELAXER SHURNEY GLENN (US) 2014-06-26 US disclosed
WO-2014100463-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2014-06-26 WO disclosed
WO-2014100818-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2014-06-26 WO disclosed
WO-2014100450-A1 BRIGHTENER-CONTAINING HAIR RELAXER SHURNEY GLENN (US) 2014-06-26 WO disclosed
US-20140179638-A1 9-AMINOMETHYL SUBSTITUTED TETRACYCLINE COMPOUNDS KBP BIOSCIENCES CO., LTD. (CN) 2014-06-26 US disclosed
US-20140179709-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2014-06-26 US disclosed
EP-1998809-B1 CAMPTOTHECIN-CELL PENETRATING PEPTIDE CONJUGATES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME DRAIS PHARMACEUTICALS INC (US) 2014-06-25 EP disclosed
CN-103889954-A Substituted 4-cyano-3-phenyl-4-(pyridin-3-yl)butanoates, processes for preparation thereof and use thereof as herbicides and plant growth regulators BAYER IP GMBH 2014-06-25 CN disclosed
US-20140171691-A1 Synthesis of Drop-in Liquid Fuels and Chemicals from Methanol, Ethanol or Syngas Using Mixed Catalysts Pioneer Energy Inc. (US) 2014-06-19 US disclosed
US-20140171432-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2014-06-19 US disclosed
US-20140171429-A1 BICYCLIC INHIBITORS OF ALK ABBVIE INC. (US) 2014-06-19 US disclosed
CN-102762625-B Polymeric materials COMMW SCIENT IND RES ORG 2014-06-18 CN disclosed
US-8754233-B2 Pyrazolylbenzothiazole derivatives and their use as therapeutic agents DERMIRA (CANADA), INC. (US) 2014-06-17 US disclosed
US-20140162361-A1 PYRIMIDINE CYCLOHEXYL GLUCOCORTICOID RECEPTOR MODULATORS CORCEPT THERAPEUTICS, INC. 2014-06-12 US disclosed
US-20140163056-A1 NOVEL SPIROINDOLINE COMPOUNDS INTERVET INC. 2014-06-12 US disclosed
WO-2014089364-A1 HISTONE DEMETHYLASE INHIBITORS QUANTICEL PHARMACEUTICALS, INC (US) 2014-06-12 WO disclosed
US-20140161801-A1 QUINAZOLINE DERIVATIVE AS TYROSINE-KINASE INHIBITOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Xuanzhu Pharma Co., Ltd. (CN) 2014-06-12 US disclosed
EP-2739678-A1 GLASS FILLED COPOLYMER PRODUCTS FOR THIN WALL AND HIGH SURFACE GLOSS ARTICLES SABIC Innovative Plastics IP B.V. (NL) 2014-06-11 EP disclosed
EP-2740720-A1 Substituted bicyclic and tricyclic pent-2-en-4-inic acid derivatives and their use for enhancing the stress tolerance in plants Bayer CropScience AG (DE) 2014-06-11 EP disclosed
EP-2740356-A1 Substituted (2Z)-5(1-Hydroxycyclohexyl)pent-2-en-4-inic acid derivatives Bayer CropScience AG (DE) 2014-06-11 EP disclosed
CN-103857664-A Method of producing 5-hydroxymethylfurfural from carbohydrates AGENCY SCIENCE TECH & RES 2014-06-11 CN disclosed
US-8748443-B2 Antiviral compounds and uses thereof ABBVIE INC. (US) 2014-06-10 US disclosed
WO-2014084944-A1 BORONIC AND BORINIC ACID COMPOUNDS AS INHIBITORS OF SULFENIC ACID-CONTAINING PROTEINS THE PENN STATE RESEARCH FOUNDATION (US) 2014-06-05 WO disclosed
US-20140155389-A1 BICYCLIC INHIBITORS OF ALK ABBVIE INC. (US) 2014-06-05 US disclosed
US-20140155382-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. (US) 2014-06-05 US disclosed
US-20140155386-A1 BRIDGED BICYCLIC ARYL AND BRIDGED BICYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2014-06-05 US disclosed
EP-2738156-A1 9-AMINOMETHYL SUBSTITUTED TETRACYCLINE COMPOUND KBP Biosciences Co., Ltd. (CN) 2014-06-04 EP disclosed
US-8741967-B2 Use of unsaturated sphingosine compounds as chemotherapeutic agents for the treatment of cancer CHILDREN'S HOSPITAL & RESEARCH CENTER AT OAKLAND (US) 2014-06-03 US disclosed
US-8741898-B2 Polycyclic heteroaryl substituted triazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2014-06-03 US disclosed
US-8741914-B2 Antiviral compounds and uses thereof ABBVIE INC. (US) 2014-06-03 US disclosed
US-20140147905-A1 Boronic and Borinic Acid Compounds as Inhibitors of Sulfenic Acid-Containing Proteins THE PENN STATE RESEARCH FOUNDATION 2014-05-29 US disclosed
US-20140148342-A1 FORMULATION COMPONENT SYNGENTA LIMITED (GB) 2014-05-29 US disclosed
EP-2734520-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Infinity Pharmaceuticals, Inc. (US) 2014-05-28 EP disclosed
EP-2734530-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Infinity Pharmaceuticals, Inc. (US) 2014-05-28 EP disclosed
US-8735418-B2 Pyrimidine-2-amine compounds and their use as inhibitors of JAK kinases RIGEL PHARMACEUTICALS, INC. (US) 2014-05-27 US disclosed
US-8735386-B2 Aminopyrazoloquinazolines BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-05-27 US disclosed
US-20140142098-A1 TRIAZOLOPYRAZINE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-05-22 US disclosed
WO-2014078575-A2 NOVEL ORALLY BIOAVAILABLE BREATHING CONTROL MODULATING COMPOUNDS, AND METHODS OF USING SAME GALLEON PHARMACEUTICALS, INC. (US) 2014-05-22 WO disclosed
US-20140142105-A1 NOVEL TRIFLUOROMETHYL-OXADIAZOLE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2014-05-22 US disclosed
US-20140142126-A1 PYRROLOPYRIMIDINE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS, INC. (US) 2014-05-22 US disclosed
WO-2014078295-A1 GEMCITABINE PRODRUGS AND USES THEREOF BoYen Therapeutics, Inc. (TW) 2014-05-22 WO disclosed
WO-2014076146-A1 TRIAZOLOPYRIDAZINE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-05-22 WO disclosed
WO-2014078578-A1 PYRROLOPYRIMIDINE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS, INC. (US) 2014-05-22 WO disclosed
WO-2014076237-A1 TRIAZOLOPYRAZINE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-05-22 WO disclosed
WO-2014076162-A1 AMINOIMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-05-22 WO disclosed
EP-2732035-A2 METHODS AND COMPOSITIONS FOR MANIPULATING TRANSLATION OF PROTEIN ISOFORMS FROM ALTERNATIVE INITIATION START SITES Sarepta Therapeutics, Inc. (US) 2014-05-21 EP disclosed
EP-2731953-A1 TRICYCLIC INHIBITORS OF KINASES USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES Abbvie Inc. (US) 2014-05-21 EP disclosed
CN-103813809-A Polymer conjugated prostaglandin analogues POLYACTIVA PTY LTD 2014-05-21 CN disclosed
CN-103814009-A Substituted 4-cyan-3-(2,6-difluorophenyl)-4-phenylbutanoates, method for the production thereof and use thereof as herbicides and plant growth regulators BAYER CROPSCIENCE AG 2014-05-21 CN disclosed
US-8729082-B2 Substituted imidazoquinoxalines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-05-20 US disclosed
US-20140135319-A1 6-SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-05-15 US disclosed
US-20140135336-A1 TRIAZOLOPYRIDAZINE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-05-15 US disclosed
US-20140134160-A1 GEMCITABINE PRODRUGS AND USES THEREOF BoYen Therapeutics, Inc. (TW) 2014-05-15 US disclosed
EP-2729454-A1 NOVEL TRIFLUOROMETHYL-OXADIAZOLE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE Novartis AG (CH) 2014-05-14 EP disclosed
EP-2729182-A1 NUCLEIC ACID COMPLEX Commonwealth Scientific and Industrial Research Organisation (AU) 2014-05-14 EP disclosed
EP-2454262-B1 PYRROLOPYRAZINE INHIBITORS OF KINASES ABBOTT LAB (US) 2014-05-14 EP disclosed
US-8722851-B2 Analgesia with minimal tolerance and dependence by a mu opioid receptor agonist that also binds filamin A PAIN THERAPEUTICS, INC. (US) 2014-05-13 US disclosed
US-8722900-B2 Process for cabazitaxel, and intermediates thereof SCINOPHARM TAIWAN, LTD. (TW) 2014-05-13 US disclosed
US-20140124709-A1 CLEAN POLYCARBONATE MATERIAL FOR USE IN HARD DISK DRIVE AND SEMICONDUCTOR APPLICATIONS SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2014-05-08 US disclosed
US-20140128331-A1 C-GLYCOSIDE DERIVATIVES Xuanzhu Pharma Co., Ltd. (CN) 2014-05-08 US disclosed
US-20140128599-A1 BENZOXAZOLE KINASE INHIBITORS AND METHODS OF USE INTELLIKINE LLC (US) 2014-05-08 US disclosed
US-20140127127-A1 HEPSIN INHIBITORS FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2014-05-08 US disclosed
US-20140128637-A1 ATROPISOMERIC 1,8-BISPHENOLNAPTHALENES AND THEIR USE IN ENANTIOSELECTIVE RECOGNITION AND ASYMMETRIC SYNTHESIS NATIONAL SCIENCE FOUNDATION 2014-05-08 US disclosed
WO-2014071105-A1 TREATMENT OF RHEUMATOID ARTHRITIS AND ASTHMA USING P13 KINASE INHIBITORS INFINITY PHARMACEUTICALS, INC. (US) 2014-05-08 WO disclosed
WO-2014071109-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS INFINITY PHARMACEUTICALS, INC. (US) 2014-05-08 WO disclosed
EP-2428515-B1 Spiro-oxindole compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC (CA) 2014-05-07 EP disclosed
EP-2121621-B1 LXR AND FXR MODULATORS EXELIXIS PATENT CO LLC (US) 2014-05-07 EP disclosed
US-8716297-B2 Chemical entities to be used for Wee1 inhibition for the treatment of cancer ABBVIE INC. (US) 2014-05-06 US disclosed
US-8716528-B2 Aryloxy amine compounds and their use as sodium channel modulators HOWARD FLOREY INSTITUTE (AU) 2014-05-06 US disclosed
US-8716529-B2 Amine derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2014-05-06 US disclosed
US-20140120060-A1 TREATMENT OF RHEUMATOID ARTHRITIS AND ASTHMA USING PI3 KINASE INHIBITORS INFINITY PHARMACEUTICALS, INC. (US) 2014-05-01 US disclosed
WO-2014066506-A2 COMPOSITIONS AND METHODS FOR JAMM PROTEIN INHIBITION CLEAVE BIOSCIENCES, INC. (US) 2014-05-01 WO disclosed
US-20140120083-A1 TREATMENT OF CANCERS USING PI3 KINASE ISOFORM MODULATORS INFINITY PHARMACEUTICALS, INC. (US) 2014-05-01 US disclosed
US-20140120087-A1 TRIAZOLOPYRIDINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-05-01 US disclosed
US-20140120058-A1 POLYMER CONJUGATED PROSTAGLANDIN ANALOGUES POLYACTIVA PTY LTD 2014-05-01 US disclosed
EP-2725031-A1 C-GLYCOSIDE DERIVATIVES Xuanzhu Pharma Co., Ltd. (CN) 2014-04-30 EP disclosed
EP-2723748-A1 HETEROCYCLYL AMINOIMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2014-04-30 EP disclosed
EP-2725015-A1 Uracil or thymine derivative for treating hepatitis c AbbVie Bahamas Ltd. (BS) 2014-04-30 EP disclosed
US-8710065-B2 Tricyclic inhibitors of kinases ABBVIE INC. (US) 2014-04-29 US disclosed
US-8710272-B2 Compounds with (1 E, 6E)-1,7-bis-(3,4-dimethoxyphenyl)-4,4-disubstituted-hepta-1,6-diene-3,5-dione structural scaffold, their biological activity, and uses thereof ANDROSCIENCE CORPORATION (US) 2014-04-29 US disclosed
US-8710055-B2 Triazolylphenyl sulfonamides as serine/threonine kinase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-04-29 US disclosed
US-8709486-B2 Administrable compositions THE UNIVERSITY OF SYDNEY (AU) 2014-04-29 US disclosed
US-20140113896-A1 ARYLAMINOALCOHOL-SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINOLINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-04-24 US disclosed
WO-2014062838-A2 PKM2 MODULATORS AND METHODS FOR THEIR USE TOLERO PHARMACEUTICALS, INC. (US) 2014-04-24 WO disclosed
US-20140113895-A1 FILAMIN A BINDING ANTI-INFLAMMATORY AND ANALGESIC PAIN THERAPEUTICS, INC. 2014-04-24 US disclosed
US-20140113901-A1 IMIDAZOPYRIDAZINES AS AKT KINASE INHIBITORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-04-24 US disclosed
US-20140113012-A1 COMPOUNDS AND METHODS FOR INDUCING CHONDROGENESIS THE SCRIPPS RESEARCH INSTITUTE (US) 2014-04-24 US disclosed
EP-2569316-B1 PYRROLOPYRIDINE AND PYRROLOPYRIMIDINE INHIBITORS OF KINASES ABBVIE INC (US) 2014-04-23 EP disclosed
US-8703822-B2 Method for removing undifferentiated and dedifferentiated stem cell NANYANG POLYTECHNIC (SG) 2014-04-22 US disclosed
US-8703805-B2 Modulators of LXR EXELIXIS PATENT COMPANY LLC (US) 2014-04-22 US disclosed
US-8703778-B2 Heterocyclic kinase inhibitors INTELLIKINE LLC (US) 2014-04-22 US disclosed
US-8703777-B2 Certain chemical entities, compositions and methods INTELLIKINE LLC (US) 2014-04-22 US disclosed
US-20140107074-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC. (US) 2014-04-17 US disclosed
US-20140107125-A1 HYDRAZONOPYRAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTICS DERMIRA (CANADA), INC. (US) 2014-04-17 US disclosed
WO-2014058794-A1 COMPOUNDS USEFUL FOR MAKING HCV PROTEASE INHIBITORS ABBVIE INC. (US) 2014-04-17 WO disclosed
EP-2719698-A1 Methods for preparing aurora kinase inhibitors MILLENNIUM PHARMACEUTICALS, INC. (US) 2014-04-16 EP disclosed
US-20140100364-A1 Compounds Useful For Making HCV Protease Inhibitors ABBVIE INC. 2014-04-10 US disclosed
WO-2014055634-A1 IDENTIFICATION OF SMALL MOLECULE INHIBITORS OF JUMONJI AT-RICH INTERACTIVE DOMAIN 1A (JARID1A) AND 1B (JARID1B) HISTONE DEMETHYLASE YALE UNIVERSITY (US) 2014-04-10 WO disclosed
WO-2014053878-A1 SUSTAINABLE ISOSORBIDE - CONTAINING POLYCARBONATE - POLYLACTIDE BLENDS SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2014-04-10 WO disclosed
US-20140100214-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2014-04-10 US disclosed
US-20140088099-A1 CHEMICAL COMPOUNDS, COMPOSITIONS AND METHODS FOR KINASE MODULATION INFINITY PHARMACEUTICALS, INC. (US) 2014-03-27 US disclosed
US-20140087949-A1 SUBSTITUTED 5-(CYCLOHEX-2-EN-1-YL)-PENTA-2,4-DIENES AND 5-(CYCLOHEX-2-EN-1-YL)-PENT-2-EN-4-INES AS ACTIVE AGENTS AGAINST ABIOTIC STRESS IN PLANTS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-03-27 US disclosed
US-20140088122-A1 METHOD OF TREATMENT OF AGE-RELATED MACULAR DEGENERATION (AMD) PRANA BIOTECHNOLOGY LIMITED (AU) 2014-03-27 US disclosed
US-20140086941-A1 SUBSTITUTED 2-BENZYLIDENE-2H-BENZO[b][1,4]THIAZIN-3(4H)-ONES, DERIVATIVES THEREOF, AND THERAPEUTIC USES THEREOF ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2014-03-27 US disclosed
US-20140087945-A1 SUBSTITUTED 4-CYAN-3-(2,6-DIFLUOROPHENYL)-4-PHENYLBUTANOATES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-03-27 US disclosed
EP-2710004-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES AS MKNK1 KINASE INHIBITORS Bayer Intellectual Property GmbH (DE) 2014-03-26 EP disclosed
EP-2710119-A1 COMPOSITIONS AND METHODS FOR JAMM PROTEIN INHIBITION Cleave Biosciences, Inc. (US) 2014-03-26 EP disclosed
CN-102424703-B Surface polymerisation process and polymer product using RAFT agent UNIV SYDNEY 2014-03-26 CN disclosed
US-20140080704-A1 SUBSTITUTED VINYL AND ALKINYL CYCLOHEXENOLS AS ACTIVE AGENTS AGAINST ABIOTIC STRESS IN PLANTS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-03-20 US disclosed
US-20140080821-A1 PYRIMIDO-PYRROLO-OXAZINE-DIONE COMPOUND INHIBITORS OF THE CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR PROTEIN AND USES THEREFOR THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-03-20 US disclosed
US-8673975-B2 Indene derivatives as pharmaceutical agents AQUINOX PHARMACEUTICALS INC. (CA) 2014-03-18 US disclosed
US-8674137-B2 Compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2014-03-18 US disclosed
US-20140073640-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC. 2014-03-13 US disclosed
EP-1807118-B1 STEROID ANALOGS AND CHARACTERIZATION AND TREATMENT METHODS HARBOR BIOSCIENCES INC (US) 2014-03-12 EP disclosed
EP-2705181-A1 COMBINATION PHARMACEUTICAL COMPOSITIONS AND USES THEREOF Intellikine, LLC (US) 2014-03-12 EP disclosed
US-20140066427-A1 S1P Receptors Modulators and Their Use Thereof AKAAL PHARMA PTY LTD. (AU) 2014-03-06 US disclosed
US-20140066462-A1 TREATMENT OF POLYCYSTIC DISEASE INTELLIKINE LLC (US) 2014-03-06 US disclosed
EP-2701505-A1 FORMULATION COMPONENT Syngenta Limited (GB) 2014-03-05 EP disclosed
US-8664266-B2 Hepsin inhibitors FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2014-03-04 US disclosed
WO-2014029983-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC. (US) 2014-02-27 WO disclosed
WO-2014029984-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC. (US) 2014-02-27 WO disclosed
EP-2308812-B1 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS ABBVIE BAHAMAS LTD (BS) 2014-02-26 EP disclosed
EP-2699575-A1 TRIAZOLOPYRIDINES Bayer Intellectual Property GmbH (DE) 2014-02-26 EP disclosed
EP-2086970-B1 2-(PYRAZIN-2-YL)-THIAZOLE AND 2-(1H PYRAZOL-3-YL)-THIAZOLE DERIVATIVES AS WELL AS RELATED COMPOUNDS AS STEAROYL-COA DESATURASE (SCD) INHIBITORS FOR THE TREATMENT OF METABOLIC, CARDIOVASCULAR AND OTHER DISORDERS NOVARTIS AG (CH) 2014-02-26 EP disclosed
US-8658606-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2014-02-25 US disclosed
US-20140051674-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-02-20 US disclosed
US-20140051689-A1 Polycyclic Agents for the Treatment of Respiratory Syncytial Virus Infections BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2014-02-20 US disclosed
US-20140051577-A1 SUBSTITUTED 5-(BICYCLO[4.1.0]HEPT-3-EN-2-YL)PENTA-2,4-DIENES AND 5-(BICYCLO[4.1.0]HEPT-3-EN-2-YL)PENT-2-ENE-4-INES AS ACTIVE AGENTS AGAINST ABIOTIC STRESSES IN PLANTS FRACKENPOHL JENS (DE) 2014-02-20 US disclosed
WO-2014028381-A1 APOPTOSIS-INDUCING AGENTS ABBVIE INC. (US) 2014-02-20 WO disclosed
CN-103596431-A Pyrimidine cyclohexyl glucocorticoid receptor modulators CORCEPT THERAPEUTICS INC 2014-02-19 CN disclosed
CN-103596923-A Substituted 5-(cyclohex-2-en-1-yl)-penta-2,4-dienes and 5-(cyclohex-2-en-1-yl)-pent-2-en-4-ines as active agents against abiotic stress in plants BAYER CROPSCIENCE AG 2014-02-19 CN disclosed
US-8653041-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2014-02-18 US disclosed
US-8653087-B2 Pyrido [5, 4-D] pyrimidines as cell proliferation inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-02-18 US disclosed
US-8653142-B2 Styrenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2014-02-18 US disclosed
US-8653068-B2 Filamin A binding anti-inflammatory and analgesic PAIN THERAPEUTICS, INC. (US) 2014-02-18 US disclosed
US-8653042-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2014-02-18 US disclosed
US-20140046018-A1 BIODEGRADABLE POLYMER - BIOACTIVE MOIETY CONJUGATES POLYACTIVA PTY LTD. (AU) 2014-02-13 US disclosed
US-20140046005-A1 HYBRID POLYMERS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2014-02-13 US disclosed
US-20140045868-A1 RAF KINASE MODULATOR COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2014-02-13 US disclosed
EP-2226632-B1 METHOD FOR SCREENING OF CELL-PROTECTING AGENT TAKEDA PHARMACEUTICAL (JP) 2014-02-12 EP disclosed
EP-2694500-A1 SUBSTITUTED IMIDAZOPYRIDINES AND INTERMEDIATES THEREOF Bayer Pharma Aktiengesellschaft (DE) 2014-02-12 EP disclosed
EP-2694055-A1 TAXANE AND ABEO-TAXANE ANALOGS Arbor Therapeutics, LLC (US) 2014-02-12 EP disclosed
EP-1799739-B1 GELS AORTECH INTERNAT PLC (GB) 2014-02-12 EP disclosed
EP-2694510-A1 IMIDAZOPYRIDAZINES AS AKT KINASE INHIBITORS Bayer Intellectual Property GmbH (DE) 2014-02-12 EP disclosed
US-20140038822-A1 USE OF SUBSTITUTED SPIROCYCLIC SULFONAMIDOCARBOXYLIC ACIDS, CARBOXYLIC ESTERS THEREOF, CARBOXAMIDES THEREOF AND CARBONITRILES THEREOF OR SALTS THEREOF FOR ENHANCEMENT OF STRESS TOLERANCE IN PLANTS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-02-06 US disclosed
WO-2014020041-A1 COMBINATIONS FOR THE TREATMENT OF CANCER BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-02-06 WO disclosed
US-20140038993-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-02-06 US disclosed
US-20140039048-A1 METHODS FOR THE TREATMENT OF DIABETIC RETINOPATHY AND OTHER OPHTHALMIC DISEASES ACUCELA INC. (US) 2014-02-06 US disclosed
US-20140038964-A1 IMIDAZOLE BASED LXR MODULATORS EXELIXIS PATENT COMPANY LLC (US) 2014-02-06 US disclosed
WO-2014020043-A1 COMBINATIONS FOR THE TREATMENT OF CANCER BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-02-06 WO disclosed
EP-2692726-A1 Anti-viral compounds Abbvie Inc. (US) 2014-02-05 EP disclosed
EP-2691375-A1 SUBSTITUTED BENZIMIDAZOLES Bayer Intellectual Property GmbH (DE) 2014-02-05 EP disclosed
EP-2692346-A1 An antiviral 1-phenyl-2,5-dibenzimidazol-5-yl-pyrrolidine derivative Abbvie Inc. (US) 2014-02-05 EP disclosed
US-20140030256-A1 BENZOXAZOLE KINASE INHIBITORS AND METHODS OF USE INTELLIKINE LLC (US) 2014-01-30 US disclosed
US-20140031395-A1 Positive Allosteric Modulators of the Alpha 7 Nicotinic Acetylcholine Receptor and uses Thereof BIONOMICS LIMITED (AU) 2014-01-30 US disclosed
EP-2078010-B1 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS INC (US) 2014-01-29 EP disclosed
CN-103547577-A Fused ring compound for use as mineralocorticoid receptor antagonist KBP BIOSCIENCES CO LTD 2014-01-29 CN disclosed
US-8637549-B2 Pyridons as PDK1 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-28 US disclosed
US-20140024583-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2014-01-23 US disclosed
WO-2014015291-A1 FUSED PYRIMIDINES AS INHIBITORS OF p97 COMPLEX ZHOU HAN-JIE (US) 2014-01-23 WO disclosed
US-20140024776-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS OLIGASIS (US) 2014-01-23 US disclosed
US-20140024661-A1 FUSED PYRIMIDINES AND SUBSTITUTED QUINAZOLINES AS INHIBITORS OF P97 CLEAVE BIOSCIENCES, INC. (US) 2014-01-23 US disclosed
US-20140023611-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. 2014-01-23 US disclosed
US-20140024821-A1 OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA SAREPTA THERAPEUTICS, INC. (US) 2014-01-23 US disclosed
US-20140024698-A1 METHODS FOR TREATING PROGEROID LAMINOPATHIES USING OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA SAREPTA THERAPEUTICS, INC. (US) 2014-01-23 US disclosed
EP-2222646-B1 URACIL OR THYMINE DERIVATIVE FOR TREATING HEPATITIS C ABBVIE BAHAMAS LTD (BS) 2014-01-22 EP disclosed
EP-2285881-B1 POLYMER MICROGEL BEADS AND PREPARATIVE METHOD THEREOF UNIV SYDNEY (AU) 2014-01-22 EP disclosed
EP-2685964-A1 FORMULATIONS OF PHENYL URACIL COMPOUNDS AbbVie Inc. (US) 2014-01-22 EP disclosed
EP-2558459-B1 PHTHALAZIN-(2H)-ONE INHIBITORS OF KINASES ABBVIE INC (US) 2014-01-22 EP disclosed
CN-101583614-B Polycyclic agents for the treatment of respiratory syncytial virus infections BIOTA SCIENT MANAGEMENT 2014-01-22 CN disclosed
US-8633265-B2 UV stabilization of isosorbide polycarbonates SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2014-01-21 US disclosed
US-8633207-B2 Quinazoline compounds and methods of use thereof AMBIT BIOSCIENCES CORPORATION (US) 2014-01-21 US disclosed
WO-2014012054-A1 ALZHEIMER'S DISEASE ASSAY IN A LIVING PATENT PAIN THERAPEUTICS, INC. (US) 2014-01-16 WO disclosed
US-20140018341-A1 METHOD OF INHIBITING TAU PHOSPHORYLATION CASSAVA SCIENCES, INC. 2014-01-16 US disclosed
US-20140017165-A1 DNA REPAIR ENZYME INHIBITOR NANOPARTICLES AND USES THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2014-01-16 US disclosed
WO-2014009219-A1 METHOD FOR PREPARING SUBSTITUTED TRIAZOLOPYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2014-01-16 WO disclosed
US-20140017761-A1 SUBSTRATE FOR IMMOBILIZING FUNCTIONAL SUBSTANCES AND METHOD FOR PREPARING THE SAME TEMASEK POLYTECHNIC (SG) 2014-01-16 US disclosed
US-20140017698-A1 ALZHEIMER'S DISEASE ASSAY IN A LIVING PATIENT WANG HOAU-YAN (US) 2014-01-16 US disclosed
US-20140017699-A1 ALZHEIMER'S DISEASE ASSAY IN A LIVING PATIENT CASSAVA SCIENCES, INC. 2014-01-16 US disclosed
WO-2014011917-A2 A METHOD OF INHIBITING TAU PHOSPHORYLATION PAIN THERAPEUTICS, INC. (US) 2014-01-16 WO disclosed
EP-2401267-B1 JAK KINASE MODULATING QUINAZOLINE DERIVATIVES AND THEIR USE IN METHODS AMBIT BIOSCIENCES CORP (US) 2014-01-15 EP disclosed
US-8624025-B2 Antiviral agents BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2014-01-07 US disclosed
WO-2014004470-A1 TREATMENT OF LUPUS, FIBROTIC CONDITIONS, AND INFLAMMATORY MYOPATHIES AND OTHER DISORDERS USING PI3 KINASE INHIBITORS INFINITY PHARMACEUTICALS, INC. (US) 2014-01-03 WO disclosed
US-20140004111-A1 POLYCYCLIC AGENTS FOR THE TREATMENT OF RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2014-01-02 US disclosed
US-20140004215-A1 COMPOSITIONS AND METHODS FOR MANAGING WEIGHT UNIGEN, INC. (KR) 2014-01-02 US disclosed
EP-2678334-A1 ANTI-VIRAL COMPOUNDS Abbvie Inc. (US) 2014-01-01 EP disclosed
EP-1723139-B1 CELL TARGETING CONJUGATES PETER MACCALLUM CANCER INST (AU) 2014-01-01 EP disclosed
EP-2678016-A2 HETEROCYCLIC COMPOUNDS AND USES THEREOF Intellikine, LLC (US) 2014-01-01 EP disclosed
CN-103492489-A High molecular weight zwitterionic polymers OLIGASIS 2014-01-01 CN disclosed
CN-101801375-B Insulin sensitisers and methods of treatment VERVA PHARMACEUTICALS LTD 2014-01-01 CN disclosed
CN-103492371-A Spiro-containing dihydropyrazole compounds KBP BIOSCIENCES CO LTD 2014-01-01 CN disclosed
US-8618331-B2 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors RIGEL PHARMACEUTICALS INC. (US) 2013-12-31 US disclosed
US-8618289-B2 RAF kinase modulator compounds and methods of use thereof AMBIT BIOSCIENCES CORPORATION (US) 2013-12-31 US disclosed
WO-2013191964-A1 SILICONE LIGANDS FOR STABILIZING QUANTUM DOT FILMS NANOSYS, INC. (US) 2013-12-27 WO disclosed
WO-2013191984-A1 FUSED THIAZIN-3-ONES AS KCA3.1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-12-27 WO disclosed
US-20130345216-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE LLC (US) 2013-12-26 US disclosed
US-20130344061-A1 TREATMENT OF LUPUS, FIBROTIC CONDITIONS, AND INFLAMMATORY MYOPATHIES AND OTHER DISORDERS USING PI3 KINASE INHIBITORS INFINITY PHARMACEUTICALS, INC. (US) 2013-12-26 US disclosed
US-20130345458-A1 SILICONE LIGANDS FOR STABILIZING QUANTUM DOT FILMS NANOSYS, INC. (US) 2013-12-26 US disclosed
US-8614324-B2 Filamin A binding anti-inflammatory and analgesic PAIN THERAPEUTICS, INC. (US) 2013-12-24 US disclosed
US-8614318-B2 Apoptosis promoters ABBVIE INC. (US) 2013-12-24 US disclosed
US-20130338133-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-12-19 US disclosed
US-20130336920-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. (US) 2013-12-19 US disclosed
US-20130336921-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. (US) 2013-12-19 US disclosed
US-20130336919-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. (US) 2013-12-19 US disclosed
US-20130336918-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. (US) 2013-12-19 US disclosed
US-20130338161-A1 AXL INHIBITORS FOR USE IN COMBINATION THERAPY FOR PREVENTING, TREATING OR MANAGING METASTATIC CANCER RIGEL PHARMACEUTICALS INC (US) 2013-12-19 US disclosed
US-20130338160-A1 Compounds with (1E, 6E)-1,7-bis-(3,4-dimethoxyphenyl)-4,4-disubstituted-hepta-1,6-diene-3,5-dione structural scaffold, their biological activity, and uses thereof Annji Pharmaceutical Co., Ltd. (TW) 2013-12-19 US disclosed
US-8610111-B2 Bistable carbazole compounds STMICROELECTRONICS S.R.L. (IT) 2013-12-17 US disclosed
US-8609661-B2 Pyrimido-pyrrolo-quinoxalinedione inhibitors of cystic fibrosis transmembrane conductance regulator protein and uses therefor THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-12-17 US disclosed
US-8609650-B2 Bridged bicyclic aryl and bridged bicyclic heteroaryl substituted triazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2013-12-17 US disclosed
US-20130330327-A1 ALKOXY-SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-12-12 US disclosed
EP-2670749-A1 NEW AZAINDOLYLPHENYL SULFONAMIDES AS SERINE/THREONINE KINASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2013-12-11 EP disclosed
US-8604032-B2 Chemical compounds, compositions and methods for kinase modulation INFINITY PHARMACEUTICALS, INC. (US) 2013-12-10 US disclosed
WO-2013181217-A2 NOVEL COMPOUNDS AND COMPOSITIONS FOR TREATMENT OF BREATHING CONTROL DISORDERS OR DISEASES GALLEON PHARMACEUTICALS, INC. (US) 2013-12-05 WO disclosed
WO-2013179024-A1 SULFONYL PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATING PROKINETICIN MEDIATED DISEASES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-12-05 WO disclosed
US-20130324576-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-12-05 US disclosed
US-20130323642-A1 Photoinduced Alkyne-Azide Click Reactions THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2013-12-05 US disclosed
WO-2013181296-A2 COMPOSITIONS AND METHODS FOR MANAGING WEIGHT UNIGEN, INC. (US) 2013-12-05 WO disclosed
US-20130326735-A1 6-(2-Aminophenyl)picolinates and their use as herbicides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-12-05 US disclosed
EP-2668178-A1 NEW 5-ALKYNYL-PYRIDINES Boehringer Ingelheim International GmbH (DE) 2013-12-04 EP disclosed
EP-2668179-A1 NEW 5-ALKYNYL-PYRIDINES Boehringer Ingelheim International GmbH (DE) 2013-12-04 EP disclosed
EP-2668189-A1 NEW PYRIMIDO[5,4-D]PYRIMIDYLAMINO PHENYL SULFONAMIDES AS SERINE/THREONINE KINASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2013-12-04 EP disclosed
US-8598194-B2 Polycyclic agents for the treatment of respiratory syncytial virus infections BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2013-12-03 US disclosed
US-8598193-B2 Polycyclic agents for the treatment of respiratory syncytial virus infections BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2013-12-03 US disclosed
US-8598157-B2 5-alkynyl-pyridines BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-12-03 US disclosed
US-20130317045-A1 THIENOPYRIDINE AND THIENOPYRIMIDINE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2013-11-28 US disclosed
US-20130317004-A1 AMINOALCOHOL SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-11-28 US disclosed
WO-2013174744-A1 THIENOPYRIMIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2013-11-28 WO disclosed
WO-2013174735-A1 SUBSTITUTED BENZOTHIENOPYRIMIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2013-11-28 WO disclosed
EP-1755373-B2 METHOD OF ALTERING THE ALKALOID COMPOSITION IN POPPY PLANTS GLAXOSMITHKLINE AUSTRALIA PTY LTD (AU) 2013-11-27 EP disclosed
EP-2665711-A1 PICOLINAMIDE INHIBITORS OF KINASES Abbvie Inc. (US) 2013-11-27 EP disclosed
EP-2491025-B1 AZAAZULENE COMPOUNDS IND TECH RES INST (TW) 2013-11-27 EP disclosed
EP-2665724-A1 BICYCLIC INHIBITORS OF ALK AbbVie Inc. (US) 2013-11-27 EP disclosed
EP-2665727-A1 BICYCLIC CARBOXAMIDE INHIBITORS OF KINASES Abbvie Inc. (US) 2013-11-27 EP disclosed
EP-2665775-A1 UV STABILIZATION OF ISOSORBIDE POLYCARBONATES SABIC Innovative Plastics IP B.V. (NL) 2013-11-27 EP disclosed
US-8592399-B2 S1P receptors modulators and their use thereof AKAAL PHARMA PTY LTD. (AU) 2013-11-26 US disclosed
US-20130310357-A1 Azolyl Urea Compounds and Methods of Use Thereof AMBIT BIOSCIENCES CORPORATION (US) 2013-11-21 US disclosed
US-8586770-B2 Unsaturated steroid compounds Harbor Therapeutics, Inc. (US) 2013-11-19 US disclosed
US-8586618-B2 Furanone compounds and lactam analogues thereof BIOSIGNAL LIMITED (AU) 2013-11-19 US disclosed
US-20130303509-A1 NAMPT INHIBITORS ABBVIE INC. (US) 2013-11-14 US disclosed
US-20130303511-A1 NAMPT INHIBITORS ABBVIE INC. (US) 2013-11-14 US disclosed
WO-2013169361-A1 IRON CHELATORS AS HIV-1 INHIBITORS HOWARD UNIVERSITY (US) 2013-11-14 WO disclosed
US-20130303508-A1 NAMPT INHIBITORS ABBVIE INC. (US) 2013-11-14 US disclosed
US-20130303532-A1 IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT HYPERPROLIFERATIVE DISORDERS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-11-14 US disclosed
US-20130303510-A1 NAMPT INHIBITORS ABBVIE INC. (US) 2013-11-14 US disclosed
US-20130303547-A1 HCV Protease Inhibitors and Uses Thereof ABBVIE INC (US) 2013-11-14 US disclosed
US-20130303533-A1 AZOLOPYRIDINE AND AZOLOPYRIMIDINE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2013-11-14 US disclosed
WO-2013170147-A1 COMPOUNDS USEFUL FOR PROMOTING PROTEIN DEGRADATION AND METHODS USING SAME YALE UNIVERSITY (US) 2013-11-14 WO disclosed
US-8580808-B2 Filamin A-binding anti-inflammatory analgesic Pain Therapeutic, Inc. (US) 2013-11-12 US disclosed
US-8580809-B2 Filamin A-binding anti-inflammatory analgesic PAIN THERAPEUTICS, INC. (US) 2013-11-12 US disclosed
US-20130296363-A1 QUINOLINE AND ISOQUINOLINE DERIVATIVES FOR USE AS JAK MODULATORS AMBIT BIOSCIENCES CORPORATION (US) 2013-11-07 US disclosed
US-20130291430-A1 Synthesis of High Caloric Fuels and Chemicals Pioneer Energy (US) 2013-11-07 US disclosed
WO-2013166449-A2 METHODS FOR THE TREATMENT OF DIABETIC RETINOPATHY AND OTHER OPHTHALMIC DISEASES ACUCELA INC. (US) 2013-11-07 WO disclosed
EP-2398797-B1 PYRIMIDO[5,4-D]PYRIMIDINE DERIVATIVES FOR THE INHIBITION OF TYROSINE KINASES BOEHRINGER INGELHEIM INT (DE) 2013-11-06 EP disclosed
EP-2507233-B1 Substituted triazolopyridines BAYER IP GMBH (DE) 2013-11-06 EP disclosed
US-8575203-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-11-05 US disclosed
US-20130288369-A1 dsRNA MOLECULES COMPRISING OLIGONUCLEOTIDE ANALOGS HAVING MODIFIED INTERSUBUNIT LINKAGES AND/OR TERMINAL GROUPS SAREPTA THERAPEUTICS, INC. (US) 2013-10-31 US disclosed
US-20130289105-A1 HEPSIN INHIBITORS FRED HUTCHINSON CANCER CENTER 2013-10-31 US disclosed
US-20130289029-A1 Fused Ring Compound For Use As Mineralocorticoid Receptor Antagonist NOVO NORDISK A/S (DK) 2013-10-31 US disclosed
US-20130289217-A1 CONDUCTING AND SEMICONDUCTING ORGANIC MATERIALS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2013-10-31 US disclosed
EP-2368890-B9 Hepatitis C virus inhibitors ABBVIE BAHAMAS LTD (BS) 2013-10-30 EP disclosed
EP-2655355-A1 NEW TRIAZOLYLPHENYL SULFONAMIDES AS SERINE/THREONINE KINASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2013-10-30 EP disclosed
EP-2655358-A1 OXINDOLOPYRIMIDINE AS IGF1R RECEPTOR INHIBITORS Boehringer Ingelheim International GmbH (DE) 2013-10-30 EP disclosed
CN-103380116-A 6-(2-aminophenyl)picolinates and their use as herbicides BAYER IP GMBH 2013-10-30 CN disclosed
US-8569352-B2 Imidazole based LXR modulators EXELIXIS PATENT COMPANY LLC (US) 2013-10-29 US disclosed
US-8569495-B2 Anthelmintic agents and their use INTERVET INTERNATIONAL B.V. (NL) 2013-10-29 US disclosed
US-8569316-B2 Pyrimido [5,4-D] pyrimidine derivatives for the inhibition of tyrosine kinases BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-10-29 US disclosed
US-8568920-B2 Electrolytic solution and lithium battery employing the same SAMSUNG SDI CO., LTD. (KR) 2013-10-29 US disclosed
US-8569323-B2 Substituted isoquinolin-1(2H)-one compounds, compositions, and methods thereof INTELLIKINE, LLC (US) 2013-10-29 US disclosed
US-8569303-B2 Diamine derivatives as inhibitors of leukotriene A4 hydrolase CELTAXSYS, INC. (US) 2013-10-29 US disclosed
US-20130281468-A1 BICYCLIC ARYL AND BICYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS MIDCAP FINANCIAL TRUST 2013-10-24 US disclosed
WO-2013158845-A1 LINEAR GLYCIDYL CARBAMATE (GC) RESINS FOR HIGHLY FLEXIBLE COATINGS NDSU RESEARCH FOUNDATION (US) 2013-10-24 WO disclosed
US-20130281460-A1 6-THIO-SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-10-24 US disclosed
EP-2651924-A1 ANTI-VIRAL COMPOUNDS Abbvie Inc. (US) 2013-10-23 EP disclosed
EP-2651920-A2 ANTI-VIRAL COMPOUNDS Abbvie Inc. (US) 2013-10-23 EP disclosed
EP-2651946-A1 2-SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS Bayer Intellectual Property GmbH (DE) 2013-10-23 EP disclosed
EP-2651945-A1 6-SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS Bayer Intellectual Property GmbH (DE) 2013-10-23 EP disclosed
EP-2651948-A1 IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT HYPERPROLIFERATIVE DISORDERS Bayer Intellectual Property GmbH (DE) 2013-10-23 EP disclosed
EP-2651950-A1 6 SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS Bayer Intellectual Property GmbH (DE) 2013-10-23 EP disclosed
EP-2651925-A2 ANTI-VIRAL COMPOUNDS Abbvie Inc. (US) 2013-10-23 EP disclosed
EP-2651944-A1 SUBSTITUTED 6-IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS Bayer Intellectual Property GmbH (DE) 2013-10-23 EP disclosed
EP-2651947-A1 6-THIO-SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS Bayer Intellectual Property GmbH (DE) 2013-10-23 EP disclosed
EP-2651885-A1 ANTI-VIRAL COMPOUNDS Abbvie Inc. (US) 2013-10-23 EP disclosed
CN-101723949-B Polycyclic agents for treatment of respiratory syncytial virus infections BIOTA SCIENT MAN 2013-10-23 CN disclosed
US-8561811-B2 Substrate for immobilizing functional substances and method for preparing the same TEMASEK POLYTECHNIC (SG) 2013-10-22 US disclosed
US-8563559-B2 Pinane-substituted pyrimidinediamine derivatives useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2013-10-22 US disclosed
WO-2013154712-A1 ASYMMETRIC SYNTHESES FOR SPIRO-OXINDOLE COMPOUNDS USEFUL AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2013-10-17 WO disclosed
US-20130274483-A1 ASYMMETRIC SYNTHESES FOR SPIRO-OXINDOLE COMPOUNDS USEFUL AS THERAPEUTIC AGENTS PACIRA PHARMACEUTICALS, INC. 2013-10-17 US disclosed
WO-2013154793-A1 F2 DERIVATIVES AS ANTIBACTERIAL AGENTS THE PENN STATE RESEARCH FOUNDATION (US) 2013-10-17 WO disclosed
WO-2013154878-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2013-10-17 WO disclosed
US-20130274285-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC 2013-10-17 US disclosed
EP-2648754-A2 METHODS OF INHIBITING METASTASIS FROM CANCER Philadelphia Health and Education Corporation D/B/A (US) 2013-10-16 EP disclosed
EP-2121639-B1 SUBSTITUTED 2,4-DIAMINO-1,3,5-TRIAZINES, METHODS FOR THE PRODUCTION THEREOF, AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2013-10-16 EP disclosed
US-8557842-B2 Cocaine analogs and methods of preparation and uses thereof Temple University—Of the Commonwealth System of Higher Education (US) 2013-10-15 US disclosed
US-8557810-B2 Imidazolothiazole compounds for the treatment of disease AMBIT BIOSCIENCES CORPORATION (US) 2013-10-15 US disclosed
US-8557737-B2 Methods of altering poppy characteristics GlaxoSmithKline Australia, Pty, Ltd (AU) 2013-10-15 US disclosed
US-8557783-B2 Phosphotetrahydropyran compounds for the treatment of wounds and fibrotic disorders Pharmaxis Pty Limited (AU) 2013-10-15 US disclosed
US-20130267527-A1 SUBSTITUTED 6-IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-10-10 US disclosed
WO-2013149909-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2013-10-10 WO disclosed
US-20130267521-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE LLC (US) 2013-10-10 US disclosed
EP-2431371-B1 THIOPHENE DERIVATIVES TIANJIN HEMAY BIO TECH CO LTD (CN) 2013-10-09 EP disclosed
EP-2646423-A1 NOVEL COMPOUNDS AS RESPIRATORY STIMULANTS FOR TREATMENT OF BREATHING CONTROL DISORDERS OR DISEASES Galleon Pharmaceuticals, Inc. (US) 2013-10-09 EP disclosed
CN-103347866-A Novel compound as respiratory stimulants for treatment of breathing control disorder or disease GALLEON PHARMACEUTICALS INC 2013-10-09 CN disclosed
CN-103342682-A Intermediate for preparing pyrimidine derivatives ASTRAZENECA AB 2013-10-09 CN disclosed
US-8551980-B2 Substituted triazolopyridines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-10-08 US disclosed
WO-2013144189-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-10-03 WO disclosed
US-20130261102-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. 2013-10-03 US disclosed
US-20130261121-A1 Compounds with (1E, 6E)-1,7-bis-(3,4-dimethoxyphenyl)-4,4-disubstituted-hepta-1,6-diene-3,5-dione structural scaffold, their biological activity, and uses thereof Annji Pharmaceutical Co., Ltd. (TW) 2013-10-03 US disclosed
EP-2642997-A1 NITRIC OXIDE DONORS IN THERAPY OF NITRIC OXIDE DEFICIENCY-INDUCED DISTURBANCES OF CEREBRAL MICROCIRCULATION Westfälische Wilhelms-Universität Münster (DE) 2013-10-02 EP disclosed
US-8546443-B2 Benzylic oxindole pyrimidines BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-10-01 US disclosed
US-8546433-B2 Axl inhibitors for use in combination therapy for preventing, treating or managing metastatic cancer RIGEL PHARMACEUTICALS, INC. (US) 2013-10-01 US disclosed
US-8546405-B2 Anti-viral compounds ABBOTT LABORATORIES (US) 2013-10-01 US disclosed
US-20130252962-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2013-09-26 US disclosed
US-20130252959-A1 NITRIC OXIDE DONORS IN THERAPY OF NITRIC OXIDE DEFICIENCY-INDUCED DISTURBANCES OF CEREBRAL MICROCIRCULATION West-Falische Wilhelms-Universitat Munster (DE) 2013-09-26 US disclosed
US-20130252922-A1 SUBSTITUTED PHENOXYPYRIDINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-09-26 US disclosed
US-20130253064-A1 STYRENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. 2013-09-26 US disclosed
EP-2640704-A1 NAMPT INHIBITORS Abbvie Inc. (US) 2013-09-25 EP disclosed
EP-2640698-A1 NAMPT AND ROCK INHIBITORS AbbVie Inc. (US) 2013-09-25 EP disclosed
EP-2640735-A1 ANTIBACTERIAL AMIINOGLYCOSIDE ANALOGS Achaogen, Inc. (US) 2013-09-25 EP disclosed
EP-1558585-B1 NEUROLOGICALLY-ACTIVE COMPOUNDS PRANA BIOTECHNOLOGY LTD (AU) 2013-09-25 EP disclosed
US-8541457-B2 Aminothiazole derivatives as human stearoyl-CoA desaturase inhibitors XENON PHARMACEUTICALS INC. (CA) 2013-09-24 US disclosed
US-8541424-B2 Anti-viral compounds ABBOTT LABORATORIES (US) 2013-09-24 US disclosed
US-8541448-B2 Compounds and methods for inhibiting NHE-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders ARDELYX, INC. (US) 2013-09-24 US disclosed
US-20130245014-A1 JAK KINASE MODULATING COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORP. (US) 2013-09-19 US disclosed
WO-2013138418-A2 PROCESS FOR MAKING CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2013-09-19 WO disclosed
WO-2013135612-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-09-19 WO disclosed
US-20130244956-A1 CAMPTOTHEAN-PEPTIDE CONJUGATES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME DRAIS PHARMACEUTICALS, INC. (US) 2013-09-19 US disclosed
US-20130245327-A1 CARBON NANOHOOPS AND METHODS OF MAKING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-09-19 US disclosed
WO-2013138413-A1 BIS-QUARTERNARY CINCHONA ALKALOID SALTS AS ASYMMETRIC PHASE TRANSFER CATALYSTS MERCK SHARP & DOHME CORP. (US) 2013-09-19 WO disclosed
EP-2639226-A1 Anti-infective pyrimidines and uses thereof ABBOTT LABORATORIES (US) 2013-09-18 EP disclosed
EP-2638044-A1 ALKOXY-SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINES Bayer Pharma Aktiengesellschaft (DE) 2013-09-18 EP disclosed
EP-2638045-A1 AMINOALCOHOL SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS Bayer Intellectual Property GmbH (DE) 2013-09-18 EP disclosed
EP-2177226-B1 Hydroxamate compositions COVIDIEN LP (US) 2013-09-18 EP disclosed
EP-2638043-A1 ARYLAMINOALCOHOL-SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINOLINES Bayer Intellectual Property GmbH (DE) 2013-09-18 EP disclosed
EP-2637669-A2 HETEROCYCLIC COMPOUNDS AND USES THEREOF Infinity Pharmaceuticals, Inc. (US) 2013-09-18 EP disclosed
US-8535655-B2 Biodegradable polymer—bioactive moiety conjugates POLYACTIVA PTY LTD. (AU) 2013-09-17 US disclosed
WO-2013133726-A1 RODENTICIDAL NORBORMIDE ANALOGUES LANDCARE RESEARCH NEW ZEALAND LIMITED (NZ) 2013-09-12 WO disclosed
US-20130237572-A1 PYRAZOLYLBENZOTHIAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS DERMIRA (CANADA), INC. (US) 2013-09-12 US disclosed
US-20130237507-A1 Novel Amide Compounds ASTRAZENECA AB INTELLECTUAL PROPERTY (GB) 2013-09-12 US disclosed
WO-2013130013-A1 NOVEL COMPOUNDS AND USES THEREOF NANYANG POLYTECHNIC (SG) 2013-09-06 WO disclosed
WO-2013127729-A1 6 - ALKYNYL PYRIDINES AS SMAC MIMETICS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-09-06 WO disclosed
EP-2632899-A1 SUBSTITUTED PHENOXYPYRIDINES Bayer Intellectual Property GmbH (DE) 2013-09-04 EP disclosed
EP-1830837-B1 HETEROCYCLIC DERIVATIVES FOR THE TREATMENT OF DISEASES MEDIATED BY STEAROYL-COA DESATURASE ENZYMES XENON PHARMACEUTICALS INC (CA) 2013-09-04 EP disclosed
US-8524689-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-09-03 US disclosed
US-8524675-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-09-03 US disclosed
US-20130225562-A1 PYRIDYLTRIAZOLES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-08-29 US disclosed
US-20130224114-A1 Translocator Protein Ligands THE UNIVERSITY OF SYDNEY (AU) 2013-08-29 US disclosed
US-20130225615-A1 2-CYCLOQUINAZOLINE DERIVATIVES AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2013-08-29 US disclosed
US-20130225579-A1 CYANOQUINOLINE DERIVATIVES TIANJIN HEMAY BIO-TECH CO., LTD. (CN) 2013-08-29 US disclosed
US-20130224083-A1 USE OF NITROANILINE DERIVATIVES FOR THE PRODUCTION OF NITRIC OXIDE STMICROELECTRONICS S.R.I. (IT) 2013-08-29 US disclosed
WO-2013126805-A2 SMALL MOLECULE COMPOUNDS TO TREAT HEARING LOSS FATE THERAPEUTICS, INC. (US) 2013-08-29 WO disclosed
US-20130225619-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS FOR DISEASE TREATMENT ACUCELA INC. (US) 2013-08-29 US disclosed
US-20130225567-A1 5-Alkynyl Pyridine BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-08-29 US disclosed
US-20130225614-A1 4-AZOLYLAMINOQUINAZOLINE DERIVATIVES AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2013-08-29 US disclosed
US-20130225578-A1 7-CYCLYLQUINAZOLINE DERIVATIVES AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2013-08-29 US disclosed
US-20130225589-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES ABBVIE INC. (US) 2013-08-29 US disclosed
CN-103270034-A NOVEL SUBSTITUTED PICOLINIC ACIDS, SALTS AND ACID DERIVATIVES THEREOF, AND USE THEREOF AS HERBICIDES BAYER IP GMBH 2013-08-28 CN disclosed
US-20130217642-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2013-08-22 US disclosed
US-20130217726-A1 INSULIN-REGULATED AMINOPEPTIDASE (IRAP) INHIBITORS AND USES THEREOF ST. VINCENT'S INSTITUTE OF MEDICAL RESEARCH (AU) 2013-08-22 US disclosed
US-20130217841-A1 CONTINUOUS FLOW POLYMERISATION PROCESS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2013-08-22 US disclosed
WO-2013123071-A1 METHODS AND COMPOSITIONS FOR JAMM PROTEASE INHIBITION CLEAVE BIOSCIENCES, INC. (US) 2013-08-22 WO disclosed
EP-2628481-A1 Trisubstituted heterocycles as replication inhibitors of hepatitis C virus HCV AbbVie Bahamas Ltd. (BS) 2013-08-21 EP disclosed
EP-2627651-A1 ANTI-VIRAL COMPOUNDS Abbvie Inc. (US) 2013-08-21 EP disclosed
EP-2454257-B1 PYRROLOPYRIDINE INHIBITORS OF KINASES ABBVIE INC (US) 2013-08-21 EP disclosed
EP-1869022-B1 NAPHTHALAMIDE DERIVATIVES HAVING ANTIPROLIFERATIVE ACTIVITY AGENCY SCIENCE TECH & RES (SG) 2013-08-21 EP disclosed
EP-1804799-B1 Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors XENON PHARMACEUTICALS INC (CA) 2013-08-21 EP disclosed
EP-1807085-B1 Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors XENON PHARMACEUTICALS INC (CA) 2013-08-21 EP disclosed
CN-101742996-B Application of ingenol in preparation of medicine for treating non-cancerous skin injury LEO LAB LTD 2013-08-21 CN disclosed
US-20130210832-A1 1H-IMIDAZO[4,5-C]QUINOLINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-08-15 US disclosed
US-20130209997-A1 COMPOSITIONS FOR STABILIZING DNA, RNA AND PROTEINS IN SALIVA AND OTHER BIOLOGICAL SAMPLES DURING SHIPPING AND STORAGE AT AMBIENT TEMPERATURES BIOMATRICA, INC. (US) 2013-08-15 US disclosed
US-20130210143-A1 NOVEL METHODS FOR PREVENTING OR TREATING DIABETES FUNDACION PUBLICA ANDALUZA PROGRESO Y SALUD (ES) 2013-08-15 US disclosed
US-20130210111-A1 SUBSTRATE FOR IMMOBILIZING FUNCTIONAL SUBSTANCES AND METHOD FOR PREPARING THE SAME TEMASEK POLYTECHNIC (SG) 2013-08-15 US disclosed
US-20130209543-A1 ENHANCED TREATMENT REGIMENS USING MTOR INHIBITORS INTELLIKINE LLC (US) 2013-08-15 US disclosed
US-20130210815-A1 SUBSTITUTED IMIDAZOPYRAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-08-15 US disclosed
US-8507539-B2 Potassium channel blockers and uses thereof BIONOMICS LIMITED (AU) 2013-08-13 US disclosed
US-8507474-B2 Anthelmintic agents and their use INTERVET INTERNATIONAL B.V. (NL) 2013-08-13 US disclosed
WO-2013116382-A1 PURINONE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS, INC. (US) 2013-08-08 WO disclosed
WO-2013116836-A1 HALOGENATED ORGANOSILICON ELECTROLYTES, METHODS OF USING THEM, AND ELECTROCHEMICAL DEVICES CONTAINING THEM SILATRONIX, INC. (US) 2013-08-08 WO disclosed
US-20130203768-A1 N-HETEROARYL COMPOUNDS WITH CYCLIC BRIDGING UNIT FOR THE TREATMENT OF PARASITIC DISEASES INTERVET INC. 2013-08-08 US disclosed
US-8501238-B2 Anti-infective agents and uses thereof ABBVIE INC. (US) 2013-08-06 US disclosed
US-8501724-B1 Purinone compounds as kinase inhibitors PHARMACYCLICS, INC. (US) 2013-08-06 US disclosed
US-8501746-B2 Organic compounds XENON PHARMACEUTICALS INC. (CA) 2013-08-06 US disclosed
US-8501889-B2 Conducting and semiconducting organic materials COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2013-08-06 US disclosed
US-20130197096-A1 ALKOXY COMPOUNDS FOR DISEASE TREATMENT ACUCELA, INC. (US) 2013-08-01 US disclosed
US-20130196993-A1 N-HETEROARYL COMPOUNDS INTERVET INC. 2013-08-01 US disclosed
US-20130196131-A1 GLASS FILLED COPOLYMER PRODUCTS FOR THIN WALL AND HIGH SURFACE GLOSS ARTICLES SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2013-08-01 US disclosed
US-20130197014-A1 PURINONE COMPOUNDS AS KINASE INHIBITORS PHARMACYCLICS, INC. (US) 2013-08-01 US disclosed
WO-2013110585-A1 5, 8 -DIHYDRO- 6H- PYRAZOLO [3, 4 -H] QUINAZOLINES AS IGF-LR/LR INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-08-01 WO disclosed
US-20130195848-A1 IMIDAZOPYRAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-08-01 US disclosed
US-8497275-B2 HCV protease inhibitors and uses thereof ABBVIE INC. (US) 2013-07-30 US disclosed
US-20130190377-A1 Novel Lactams BIOSIGNAL LIMITED (AU) 2013-07-25 US disclosed
US-20130190488-A1 APOPTOSIS PROMOTERS ABBOTT LABORATORIES (US) 2013-07-25 US disclosed
WO-2013109991-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS FOR DISEASE TREATMENT ACUCELA INC. (US) 2013-07-25 WO disclosed
WO-2013107743-A1 SPIROINDOLINE DERIVATIVES AS GONADOTROPIN- RELEASING HORMONE RECEPTOR ANTAGONISTS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-07-25 WO disclosed
US-20130190286-A1 B-RAF KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-07-25 US disclosed
US-20130190305-A1 NEW 5,8-DIHYDRO-6H-PYRAZOLO[3,4-H]QUINAZOLINES AS IGF-1R/IR INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-07-25 US disclosed
CN-103221435-A Continuous flow polymerisation process COMMW SCIENT IND RES ORG 2013-07-24 CN disclosed
US-8492379-B2 Translocator protein ligands THE UNIVERSITY OF SYDNEY (AU) 2013-07-23 US disclosed
US-8492349-B2 Analgesia with minimal tolerance and dependence by a mu opioid receptor agonist that also binds filamin A PAIN THERAPEUTICS, INC. (US) 2013-07-23 US disclosed
US-8492373-B2 Bicyclic aryl and bicyclic heteroaryl substituted triazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2013-07-23 US disclosed
US-8492354-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-07-23 US disclosed
US-8492589-B2 Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2013-07-23 US disclosed
US-8492374-B2 Azaazulene compounds INDUSTRIAL TECHNOLOGY RESEARCH INSTITUTE (TW) 2013-07-23 US disclosed
WO-2013106029-A1 TAXANE AND ABEO-TAXANE ANALOGS Arbor Therapeutics, LLC (US) 2013-07-18 WO disclosed
WO-2013106631-A1 PROCESSES FOR MAKING HCV PROTEASE INHIBITORS ABBVIE INC. (US) 2013-07-18 WO disclosed
US-20130178438-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2013-07-11 US disclosed
US-20130178630-A1 PROCESS FOR MAKING HCV PROTEASE INHIBITORS ABBVIE INC. (US) 2013-07-11 US disclosed
EP-2611502-A1 ADENOSINE A3 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2013-07-10 EP disclosed
EP-2611789-A1 QUINAZOLINE COMPOUNDS AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2013-07-10 EP disclosed
EP-2611793-A1 2-CYCLOQUINAZOLINE DERIVATIVES AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2013-07-10 EP disclosed
EP-2611812-A1 THIENOPYRIDINE AND THIENOPYRIMIDINE COMPOUNDS AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2013-07-10 EP disclosed
EP-2611809-A1 AZOLOPYRIDINE AND AZOLOPYRIMIDINE COMPOUNDS AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2013-07-10 EP disclosed
EP-2611448-A1 7-CYCLYLQUINAZOLINE DERIVATIVES AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2013-07-10 EP disclosed
US-8481502-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-07-09 US disclosed
WO-2013097773-A1 NOVEL ARYLALKENE DERIVATIVES AND USE THEREOF AS SELECTIVE ESTROGEN RECEPTOR MODULATORS CENTAURUS BIOPHARMA CO., LTD. (CN) 2013-07-04 WO disclosed
US-20130172210-A1 METHOD OF DRUG DESIGN ALCHEMIA LIMITED (AU) 2013-07-04 US disclosed
US-8476282-B2 Benzoxazole kinase inhibitors and methods of use INTELLIKINE LLC (US) 2013-07-02 US disclosed
US-8476431-B2 Benzoxazole kinase inhibitors and methods of use Itellikine LLC (US) 2013-07-02 US disclosed
US-20130165439-A1 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-27 US disclosed
EP-2607363-A1 FUSED RING COMPOUND FOR USE AS MINERALOCORTICOID RECEPTOR ANTAGONIST KBP Biosciences Co., Ltd. (CN) 2013-06-26 EP disclosed
CN-102076436-B Soil remediation process UNIV QUEENSLAND 2013-06-26 CN disclosed
US-8470782-B2 Transglutaminase inhibitors and methods of use thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2013-06-25 US disclosed
US-20130156756-A1 Substituted Triazolopyridines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-06-20 US disclosed
US-20130156761-A1 Compounds Useful for Inhibiting Metastasis from Cancer and Methods Using Same Alliance Discovery, Inc. (US) 2013-06-20 US disclosed
WO-2013087579-A1 SUBSTITUTED TRIAZOLOPYRIDINES AND THEIR USE AS TTK INHIBITORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-06-20 WO disclosed
WO-2013087581-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-06-20 WO disclosed
US-8466162-B2 5-alkynyl-pyridines BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-18 US disclosed
US-8466188-B2 Use of spiro-oxindole compounds as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2013-06-18 US disclosed
US-8466155-B2 Pyrimidines BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-18 US disclosed
US-20130150574-A1 PROCESS FOR THE MANUFACTURE OF CHIRAL CATALYSTS AND THEIR SALTS SCINOPHARM TAIWAN, LTD. (TW) 2013-06-13 US disclosed
WO-2013086441-A2 OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA SAREPTA THERAPEUTICS, INC. (US) 2013-06-13 WO disclosed
WO-2013086444-A2 METHODS FOR TREATING PROGEROID LAMINOPATHIES USING OLIGONUCLEOTIDE ANALOGUES TARGETING HUMAN LMNA SAREPTA THERAPEUTICS, INC. (US) 2013-06-13 WO disclosed
US-8461147-B2 Diaminopyridines for the treatment of diseases which are characterised by excessive or anomal cell proliferation BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-06-11 US disclosed
US-8461403-B2 Carbon nanohoops and methods of making THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-06-11 US disclosed
WO-2013081552-A1 Melamine Aldehyde Polymers AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2013-06-06 WO disclosed
EP-2598661-A2 COMPOSITIONS FOR STABILIZING DNA, RNA AND PROTEINS IN SALIVA AND OTHER BIOLOGICAL SAMPLES DURING SHIPPING AND STORAGE AT AMBIENT TEMPERATURES Biomatrica, INC. (US) 2013-06-05 EP disclosed
EP-2598660-A2 COMPOSITIONS FOR STABILIZING DNA, RNA AND PROTEINS IN BLOOD AND OTHER BIOLOGICAL SAMPLES DURING SHIPPING AND STORAGE AT AMBIENT TEMPERATURES Biomatrica, INC. (US) 2013-06-05 EP disclosed
EP-2598125-A2 NOVEL METHODS FOR PREVENTING OR TREATING DIABETES Fundación Pública Andaluza Progreso Y Salud (ES) 2013-06-05 EP disclosed
US-8455432-B2 Insulin sensitisers and methods of treatment VERVA PHARMACEUTICALS LTD. (AU) 2013-06-04 US disclosed
US-20130137804-A1 POLY(ALIPHATIC ESTER)- POLYCARBONATE COPOLYMER/POLYLACTIC ACID BLEND SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2013-05-30 US disclosed
US-20130136848-A1 POLYMERISATION PROCESS AND POLYMER PRODUCT THE UNIVERSITY OF SYDNEY (AU) 2013-05-30 US disclosed
US-20130137644-A1 CELL PENETRATING PEPTIDE CONJUGATES FOR DELIVERING OF NUCLEIC ACIDS INTO A CELL CELLECTIS (FR) 2013-05-30 US disclosed
US-20130137650-A1 METHODS OF TREATMENT USING COMBINATION THERAPY AMBIT BIOSCIENCES CORP. (US) 2013-05-30 US disclosed
WO-2013078441-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, LLC (US) 2013-05-30 WO disclosed
WO-2013076626-A1 POLY(ALIPHATIC ESTER)-POLYCARBONATE COPOLYMER/POLYLACTIC ACID BLEND SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2013-05-30 WO disclosed
WO-2013078440-A2 ENHANCED TREATMENT REGIMENS USING MTOR INHIBITORS INTELLIKINE, LLC (US) 2013-05-30 WO disclosed
EP-2595987-A1 NEW AMINOPYRAZOLOQUINAZOLINES Boehringer Ingelheim International GmbH (DE) 2013-05-29 EP disclosed
US-8450070-B2 Method for screening of cell-protecting agent TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-05-28 US disclosed
US-8450329-B2 2013-05-28 US disclosed
US-8450320-B2 Pyrrolopyrazinone inhibitors of kinases ABBVIE INC. (US) 2013-05-28 US disclosed
US-8450334-B2 Hepsin inhibitors FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2013-05-28 US disclosed
US-8450527-B2 Amine derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2013-05-28 US disclosed
US-8450480-B2 2013-05-28 US disclosed
WO-2013074834-A1 FUNCTIONALLY-MODIFIED OLIGONUCLEOTIDES AND SUBUNITS THEREOF SAREPTA THERAPEUTICS, INC. (US) 2013-05-23 WO disclosed
US-20130131286-A1 COMPOUND FOR USE IN PEPTIDE SYNTHESIS NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2013-05-23 US disclosed
US-20130131001-A1 Epirubicin Derivatives Tianjin Michele Sci-Tech Development Co., (CN) 2013-05-23 US disclosed
US-8445694-B2 Hydrazonopyrazole derivatives and their use as therapeutics DERMIRA (CANADA), INC. (US) 2013-05-21 US disclosed
US-8445476-B2 Carbacephem β-lactam antibiotics ACHAOGEN, INC. (US) 2013-05-21 US disclosed
US-8445142-B2 Organic electrolytic solution and lithium battery employing the same SAMSUNG SDI CO., LTD. (KR) 2013-05-21 US disclosed
WO-2013071264-A1 COMBINATION OF KINASE INHIBITORS AND USES THEREOF INTELLIKINE, LLC (US) 2013-05-16 WO disclosed
WO-2013067710-A1 NAMPT INHIBITORS ABBOTT LABORATORIES (US) 2013-05-16 WO disclosed
US-20130123243-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE CELTAXSYS, INC. 2013-05-16 US disclosed
US-20130121994-A1 TRIAZOLOPYRIDINE DERIVATIVES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-05-16 US disclosed
US-20130118063-A1 Synthesis of High Caloric Fuels and Chemicals Pioneer Energy (US) 2013-05-16 US disclosed
WO-2013070966-A1 SYNTHESIS OF HIGH CALORIC FUELS AND CHEMICALS Pioneer Energy (US) 2013-05-16 WO disclosed
WO-2013067579-A1 ADIPOSITY-MODULATING MOLECULES AND USES THEREFOR THE UNIVERSITY OF QUEENSLAND (AU) 2013-05-16 WO disclosed
WO-2013070976-A1 TREATMENT REGIMENS USING MULTIPLE PHARMACEUTICAL AGENTS INTELLIKINE, LLC (US) 2013-05-16 WO disclosed
WO-2013068929-A1 CLEAN POLYCARBONATE MATERIAL FOR USE IN HARD DISK DRIVE AND SEMICONDUCTOR APPLICATIONS SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2013-05-16 WO disclosed
EP-2590939-A1 COMPOUND FOR USE IN PEPTIDE SYNTHESIS Nanyang Technological University (SG) 2013-05-15 EP disclosed
EP-2590510-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT Ardelyx, Inc. (US) 2013-05-15 EP disclosed
EP-2590655-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT Ardelyx, Inc. (US) 2013-05-15 EP disclosed
EP-2590656-A2 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT Ardelyx, Inc. (US) 2013-05-15 EP disclosed
EP-2590965-A2 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT Ardelyx, Inc. (US) 2013-05-15 EP disclosed
US-8440849-B2 Use of nitroaniline derivatives for the production of nitric oxide STMICROELECTRONICS S.R.L. (IT) 2013-05-14 US disclosed
US-8440441-B2 Method of preparing a substrate for immobilization of functional substances thereon and the substrate obtained therefrom TEMASEK POLYTECHNIC (SG) 2013-05-14 US disclosed
US-20130116444-A1 PROCESS FOR CABAZITAXEL, AND INTERMEDIATES THEREOF SCINOPHARM TAIWAN, LTD. (TW) 2013-05-09 US disclosed
EP-2205592-B1 POLYCYCLIC ARYL SUBSTITUTED TRIAZOLES AND POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS INC (US) 2013-05-08 EP disclosed
US-8435980-B2 Pyrrolopyridine inhibitors of kinases ABBVIE INC. (US) 2013-05-07 US disclosed
US-8435993-B2 Methods of inhibiting metastasis from cancer PHILADELPHIA HEALTH AND EDUCATION CORPORATION (US) 2013-05-07 US disclosed
US-20130109695-A1 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2013-05-02 US disclosed
US-20130102590-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES ABBVIE INC (US) 2013-04-25 US disclosed
US-20130102633-A1 TRANSGLUTAMINASE INHIBITORS AND METHODS OF USE THEREOF THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2013-04-25 US disclosed
WO-2013059485-A1 PYRIDOPYRIMIDINONE INHIBITORS OF KINASES ABBVIE INC. (US) 2013-04-25 WO disclosed
EP-2001892-B1 IMIDAZOLOTHIAZOLE COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISEASES AMBIT BIOSCIENCES CORP (US) 2013-04-24 EP disclosed
EP-2582699-A1 SUBSTITUTED TRIAZOLOPYRIDINES Bayer Intellectual Property GmbH (DE) 2013-04-24 EP disclosed
US-8425972-B2 Antimicrobial materials and coatings COVIDIEN LP (US) 2013-04-23 US disclosed
US-8426408-B2 Pyrimidine inhibitors of kinases ABBVIE INC. (US) 2013-04-23 US disclosed
US-8426345-B2 Method of drug design ALCHEMIA LIMITED (AU) 2013-04-23 US disclosed
US-20130096335-A1 PROCESS FOR SYNTHESIS OF SILANE DIPEPTIDE ANALOGS TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2013-04-18 US disclosed
US-20130096056-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2013-04-18 US disclosed
WO-2013055897-A1 8 - CARBAMOYL - 2 - (2,3- DI SUBSTITUTED PYRID - 6 - YL) -1,2,3,4 -TETRAHYDROISOQUINOLINE DERIVATIVES AS APOPTOSIS - INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC. (US) 2013-04-18 WO disclosed
US-20130095054-A1 COPOLYMERS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2013-04-18 US disclosed
WO-2013056070-A2 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2013-04-18 WO disclosed
US-20130096121-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC. (US) 2013-04-18 US disclosed
US-20130096120-A1 APOPTOSIS-INDUCED AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC. (US) 2013-04-18 US disclosed
US-20130096113-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2013-04-18 US disclosed
EP-2421845-B1 ANTIVIRAL COMPOUNDS AND USES THEREOF ABBOTT LAB (US) 2013-04-17 EP disclosed
EP-2581372-A1 CYANOQUINOLINE DERIVATIVES Tianjin Hemay Bio-Tech Co., Ltd. (CN) 2013-04-17 EP disclosed
EP-2368890-B1 Hepatitis C virus inhibitors ABBVIE BAHAMAS LTD (BS) 2013-04-17 EP disclosed
US-8420863-B2 Styrenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA, INC. (US) 2013-04-16 US disclosed
US-20130090330-A1 N3-HETEROARYL SUBSTITUTED TRIAZOLES AND N5-HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2013-04-11 US disclosed
US-20130087736-A1 WATER SWELLABLE POLYMER MATERIALS THE UNIVERSITY OF SYDNEY (AU) 2013-04-11 US disclosed
EP-2576560-A1 SUBSTITUTED IMIDAZOPYRAZINES Bayer Intellectual Property GmbH (DE) 2013-04-10 EP disclosed
EP-2575462-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Intellikine, LLC (US) 2013-04-10 EP disclosed
US-8415351-B2 Anti-infective agents and uses thereof ABBOTT LABORATORIES (US) 2013-04-09 US disclosed
US-8415370-B2 Spiro-oxindole compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2013-04-09 US disclosed
EP-2443091-B1 ANTHELMINTIC AGENTS AND THEIR USE INTERVET INT BV (NL) 2013-04-03 EP disclosed
US-8410045-B2 Camptothecin-peptide conjugates and pharmaceutical compositions containing the same DRAIS PHARMACEUTICALS, INC. (US) 2013-04-02 US disclosed
US-8410272-B2 Pyrazolylbenzothiazole derivatives and their use as therapeutic agents DERMIRA (CANADA), INC. (US) 2013-04-02 US disclosed
US-8410126-B2 Pyrimidine inhibitors of PKTK2 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-04-02 US disclosed
WO-2013041634-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-03-28 WO disclosed
US-20130078796-A1 PROCESS FOR MAKING A PATTERNED METAL OXIDE STRUCTURE AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2013-03-28 US disclosed
US-20130079354-A1 PYRIDYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2013-03-28 US disclosed
US-20130079293-A1 NEURO-PROTECTIVE EFFECTS OF ADELOSTEMMA GRACILLIMUM AND ITS ISOLATED COMPOUNDS BIOTECHNOLOGY RESEARCH CORPORATION LIMITED (CN) 2013-03-28 US disclosed
EP-2571357-A1 CHEMICAL COMPOUNDS, COMPOSITIONS AND METHODS FOR KINASE MODULATION Intellikine, Inc. (US) 2013-03-27 EP disclosed
EP-2571877-A1 1H - IMIDAZO [4, 5 - C]QUINOLINES Boehringer Ingelheim International GmbH (DE) 2013-03-27 EP disclosed
EP-2177552-B1 Bioabsorbable surgical composition COVIDIEN LP (US) 2013-03-27 EP disclosed
US-8404674-B2 Substituted 9H-purin-2-YL compounds, compositions thereof and uses thereof BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-03-26 US disclosed
US-20130072486-A1 PYRIMIDINE CYCLOHEXYL GLUCOCORTICOID RECEPTOR MODULATORS CORCEPT THERAPEUTICS, INC. (US) 2013-03-21 US disclosed
US-20130068294-A1 DYE-SENSITISED SOLAR CELL WITH NICKEL CATHODE Commwealth Scientific and Industrial Reseach Organisation 2013-03-21 US disclosed
EP-2285882-B1 POLYMER MICROGEL BEADS UNIV SYDNEY (AU) 2013-03-20 EP disclosed
EP-2570441-A2 Bioabsorbable surgical composition Covidien LP (US) 2013-03-20 EP disclosed
EP-1799667-B1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2013-03-20 EP disclosed
US-8399419-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-03-19 US disclosed
WO-2013034570-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-03-14 WO disclosed
WO-2013036207-A1 DERIVATIVES OF XANTHONE COMPOUNDS AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2013-03-14 WO disclosed
EP-2300458-B1 SUBSTITUTED 1-(DIAZINYL) PYRAZOLE-4-YL-ACETIC ACIDS, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2013-03-13 EP disclosed
WO-2013032591-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS INC. (US) 2013-03-07 WO disclosed
EP-2564859-A1 Hydroxamate compositions Covidien LP (US) 2013-03-06 EP disclosed
US-8389557-B2 Triazole derivatives useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2013-03-05 US disclosed
US-8389771-B2 Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA, INC. (US) 2013-03-05 US disclosed
US-20130048559-A1 Method of Preparing a Substrate for Immobilization of Functional Substances Thereon and the Substrate Obtained Therefrom TEMASEK POLYTECHNIC (SG) 2013-02-28 US disclosed
US-20130052281-A1 NOVEL COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 US disclosed
US-20130053362-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLKINE, LLC (US) 2013-02-28 US disclosed
EP-2561759-A1 Fluoroalkyl-substituted 2-amidobenzimidazoles and their effect on plant growth Bayer Cropscience AG (DE) 2013-02-27 EP disclosed
EP-2560971-A1 PYRROLOPYRIDINE INHIBITORS OF KINASES Abbvie Inc. (US) 2013-02-27 EP disclosed
EP-2560967-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDES AS PDK1 INIHIBITORS Boehringer Ingelheim International GmbH (DE) 2013-02-27 EP disclosed
CN-102946877-A Neuroprotective effect of mastoid fruits (Adelostemma gracilimum) and isolated compounds thereof BIOTECHNOLOGY RES CORP LTD 2013-02-27 CN disclosed
US-8383623-B2 Phthalazin-(2H)-one inhibitors of kinases ABBOTT LABORATORIES (US) 2013-02-26 US disclosed
US-8383624-B2 Pyrrolopyrazine inhibitors of kinases ABBOTT LABORATORIES (US) 2013-02-26 US disclosed
US-8383596-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-02-26 US disclosed
US-8383873-B2 Terminal 1,1-disubstituted alkenes, method of making and using thereof THE CHINESE UNIVERSITY OF HONG KONG (CN) 2013-02-26 US disclosed
US-8383628-B2 Pyridyl derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2013-02-26 US disclosed
US-20130045522-A1 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES OLIGASIS (US) 2013-02-21 US disclosed
US-20130045955-A1 NOVEL COMPOUNDS BENNETT NICHOLAS J (GB) 2013-02-21 US disclosed
EP-2558459-A1 PHTHALAZIN-(2H)-ONE INHIBITORS OF KINASES Abbvie Inc. (US) 2013-02-20 EP disclosed
EP-2558469-A1 PYRROLOPYRAZINONE INHIBITORS OF KINASES Abbvie Inc. (US) 2013-02-20 EP disclosed
US-8377943-B2 2,4-diaminopyrimidine derivates as PTK2-inhibitors for the treatment of abnormal cell growth BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-02-19 US disclosed
US-20130040935-A1 CYCLIC KETO-ENOLS FOR THERAPY BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-02-14 US disclosed
WO-2013022793-A1 SMALL MOLECULE ACTIVATORS OF CALCIUM-ACTIVATED CHLORIDE CHANNELS AND METHODS OF USE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-02-14 WO disclosed
EP-2114954-B1 BICYCLIC ARYL AND BICYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS INC (US) 2013-02-13 EP disclosed
EP-2556058-A1 RADIOPROTECTOR COMPOUNDS AND METHODS Peter MacCallum Cancer Institute (AU) 2013-02-13 EP disclosed
EP-2114955-B1 BRIDGED BICYCLIC ARYL AND BRIDGED BICYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS INC (US) 2013-02-13 EP disclosed
CN-102933578-A Cyanoquinoline derivatives TIANJIN HEMAY BIO TECH CO LTD 2013-02-13 CN disclosed
US-8372813-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-02-12 US disclosed
US-20130035333-A1 USE OF CINNABARINIC ACID AS A MODULATOR OF IMMUNE RESPONSES IN AUTOIMMUNE DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-02-07 US disclosed
US-20130035326-A1 BIARYL COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2013-02-07 US disclosed
US-20130035324-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. 2013-02-07 US disclosed
US-20130034517-A1 TARGETED DRUG PHOSPHORYLCHOLINE POLYMER CONJUGATES OLIGASIS (US) 2013-02-07 US disclosed
WO-2013020004-A1 GLASS FILLED COPOLYMER PRODUCTS FOR THIN WALL AND HIGH SURFACE GLOSS ARTICLES SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2013-02-07 WO disclosed
EP-2552907-A1 PYRIDYLTRIAZOLES Boehringer Ingelheim International GmbH (DE) 2013-02-06 EP disclosed
EP-2552905-A1 B-RAF KINASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2013-02-06 EP disclosed
US-8367625-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2013-02-05 US disclosed
US-8367667-B2 Pyrrole derivatives as pharmaceutical agents EXELIXIS, INC. (US) 2013-02-05 US disclosed
WO-2013014579-A1 PROCESS FOR THE BORYLATION OF ORGANOHALIDES BASF SE (DE) 2013-01-31 WO disclosed
US-20130029920-A1 Metal Nanoparticles BRIMBLE MARGARET A (NZ) 2013-01-31 US disclosed
US-20130030026-A1 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. (US) 2013-01-31 US disclosed
US-20130029984-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, LLC (US) 2013-01-31 US disclosed
US-20130029993-A1 AZAINDOLYLPHENYL SULFONAMIDES AS SERINE/THREONINE KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-01-31 US disclosed
US-20130029982-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, LLC (US) 2013-01-31 US disclosed
US-20130023689-A1 PROCESS FOR THE BORYLATION OF ORGANOHALIDES BASF SE (DE) 2013-01-24 US disclosed
US-20130023523-A1 PYRIDAZINO[4,5-D]PYRIMIDIN-5(6H)-ONE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2013-01-24 US disclosed
WO-2013012681-A1 TRICYCLIC INHIBITORS OF KINASES USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES ABBOTT LABORATORIES (US) 2013-01-24 WO disclosed
WO-2013013031-A1 PYRIDAZINO [4, 5 -D] PYRIMIDIN- (6H) -ONE INHIBITORS OF WEE - 1 KINASE ABBVIE INC. (US) 2013-01-24 WO disclosed
WO-2013012918-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS INC. (US) 2013-01-24 WO disclosed
WO-2013012915-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS INC. (US) 2013-01-24 WO disclosed
WO-2013012752-A2 METHODS AND COMPOSITIONS FOR MANIPULATING TRANSLATION OF PROTEIN ISOFORMS FROM ALTERNATIVE INITIATION START SITES SAREPTA THERAPEUTICS, INC. (US) 2013-01-24 WO disclosed
US-20130023533-A1 NEW 5-ALKYNYL-PYRIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-01-24 US disclosed
US-20130023531-A1 PYRIMIDO[5,4-D]PYRIMIDYLAMINO PHENYL SULFONAMIDES AS SERINE/THREONINE KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-01-24 US disclosed
US-20130023519-A1 5-ALKYNYL-PYRIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-01-24 US disclosed
EP-2548873-A1 N-PHENYL-DIOXO-HYDROPYRIMIDINES USEFUL AS HEPATITIS C VIRUS (HCV) INHIBITORS Abbott Laboratories (US) 2013-01-23 EP disclosed
EP-1802662-B1 SURFACE POLYMERISATION PROCESS AND POLYMER PRODUCT USING RAFT AGENT UNIV SYDNEY (AU) 2013-01-23 EP disclosed
EP-2547680-A1 IMIDAZOPYRAZINES Bayer Intellectual Property GmbH (DE) 2013-01-23 EP disclosed
US-8357690-B2 Methods of treatment using combination therapy AMBIT BIOSCIENCES CORPORATION (US) 2013-01-22 US disclosed
US-20130018045-A1 New Chemical Entities To Be Used For Wee1 Inhibition For The Treatment Of Cancer ABBOTT LABORATORIES (US) 2013-01-17 US disclosed
US-20130018041-A1 PYRIMIDINE-2-AMINE COMPOUNDS AND THEIR USE AS INHIBITORS OF JAK KINASES RIGEL PHARMACEUTICAL, INC. (US) 2013-01-17 US disclosed
US-20130018077-A1 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. (US) 2013-01-17 US disclosed
WO-2013008162-A1 NOVEL TRIFLUOROMETHYL-OXADIAZOLE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2013-01-17 WO disclosed
EP-2545923-A1 Antibacterial agents Alchemia Limited (AU) 2013-01-16 EP disclosed
EP-2544542-A1 ANALGESIC COMPOUNDS, COMPOSITIONS, AND USES THEREOF Galleon Pharmaceuticals, Inc. (US) 2013-01-16 EP disclosed
EP-2546249-A1 5-Alkynyl-pyridines BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-01-16 EP disclosed
US-8354404-B2 Apoptosis promoters ABBOTT LABORATORIES (US) 2013-01-15 US disclosed
US-8354554-B2 Process for preparing organometalloids THE CHINESE UNIVERSITY OF HONGKONG (CN) 2013-01-15 US disclosed
US-20130012513-A1 HEDGEHOG INHIBITORS SELEXAGEN THERAPEUTICS, INC. 2013-01-10 US disclosed
WO-2013003887-A1 NUCLEIC ACID COMPLEX COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2013-01-10 WO disclosed
US-20130011361-A1 PYRAZOLE DERIVATIVES WHICH MODULATE STEAROYL-COA DESATURASE XENON PHARMACEUTICALS INC. (CA) 2013-01-10 US disclosed
EP-2222648-B1 PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF ASTHMA, COPD, ALLERGIC RHINITIS, ALLERGIC CONJUNCTIVITIS, ATOPIC DERMATITIS, CANCER, HEPATITIS B, HEPATITIS C, HIV, HPV, BACTERIAL INFECTIONS AND DERMATOSIS ASTRAZENECA AB (SE) 2013-01-09 EP disclosed
US-8349838-B2 Polycyclic heteroaryl substituted triazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2013-01-08 US disclosed
US-8349851-B2 JAK kinase modulating compounds and methods of use thereof AMBIT BIOSCIENCES CORP. (US) 2013-01-08 US disclosed
US-20130005736-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2013-01-03 US disclosed
EP-2540296-A1 Arminothiazole derivatives as human stearoyl-coa desaturase inhibitors Xenon Pharmaceuticals Inc. (CA) 2013-01-02 EP disclosed
EP-1904047-B1 APOPTOSIS PROMOTERS ABBOTT LAB (US) 2013-01-02 EP disclosed
WO-2012175591-A1 HETEROCYCLYL AMINOIMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-12-27 WO disclosed
US-20120329776-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, INC. 2012-12-27 US disclosed
WO-2012175514-A1 PYRIDINONE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-12-27 WO disclosed
US-20120329828-A1 Cocaine Analogs and Methods of Preparation and Uses Thereof NEW YORK UNIVERSITY (US) 2012-12-27 US disclosed
US-20120328611-A1 SUBSTITUTED TRIAZOLOPYRIDINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-12-27 US disclosed
US-20120328610-A1 TRIAZOLOPYRIDINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-12-27 US disclosed
US-20120329771-A1 BENZYLIC OXINDOLE PYRIMIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-12-27 US disclosed
EP-2536686-A1 CYCLIC KETO-ENOLS FOR THERAPY Bayer Intellectual Property GmbH (DE) 2012-12-26 EP disclosed
EP-2536485-A1 A SUBSTRATE FOR IMMOBILIZING FUNCTIONAL SUBSTANCES AND METHOD FOR PREPARING THE SAME Temasek Polytechnic (SG) 2012-12-26 EP disclosed
US-8338605-B2 Anti-viral compounds ABBOTT LABORATORIES (US) 2012-12-25 US disclosed
US-20120322803-A1 Triazolylphenyl sulfonamides as serine/threonine kinase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-12-20 US disclosed
WO-2012162742-A1 POLYMER PARTICLES THE UNIVERSITY OF SYDNEY (AU) 2012-12-06 WO disclosed
WO-2012166645-A1 PRODRUGS OF AZACITIDINE 5' -DIPHOSPHATE SYNDAX PHARMACEUTICALS, INC. (US) 2012-12-06 WO disclosed
WO-2012166658-A1 PYRIMIDO-PYRROLO-OXAZINE-DIONE COMPOUND INHIBITORS OF THE CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR PROTEIN AND USES THEREFOR THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-12-06 WO disclosed
WO-2012163942-A1 SUBSTITUTED AMINOIMIDAZOPYRIDAZINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-12-06 WO disclosed
EP-1934388-B1 METHOD OF DRUG DESIGN ALCHEMIA LTD (AU) 2012-12-05 EP disclosed
CN-102811713-A Multifunctional Zwitterionic Polymer Conjugates OLIGASIS 2012-12-05 CN disclosed
US-8324190-B2 Treatment of proliferative disorders with amino-substituted (E)-2,6- dialkoxystyryl 4-substituted benzylsulfones Temple University—Of the Commonwealth System of Higher Education (US) 2012-12-04 US disclosed
WO-2012162578-A2 ANTI-VIRAL COMPOUNDS ABBVIE INC. (US) 2012-11-29 WO disclosed
WO-2012162580-A2 ANTI-VIRAL COMPOUNDS ABBVIE INC (US) 2012-11-29 WO disclosed
WO-2012160029-A1 SUBSTITUTED TRIAZOLOPYRIDINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-11-29 WO disclosed
CN-102796147-A Compounds library ALCHEMIA LTD 2012-11-28 CN disclosed
US-8318949-B2 Organic compounds NOVARTIS AG (CH) 2012-11-27 US disclosed
US-8318685-B2 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2012-11-27 US disclosed
US-20120295856-A1 FREDERICAMYCIN DERIVATIVES ZENTOPHARM GMBH (DE) 2012-11-22 US disclosed
US-20120294930-A1 COMBINATION OF KINASE INHIBITORS AND USES THEREOF INTELLIKINE LLC (US) 2012-11-22 US disclosed
US-20120295897-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2012-11-22 US disclosed
US-20120295911-A1 Novel Compounds and Compositions for Treatment of Breathing Control Disorders or Diseases GALLEON PHARMACEUTICALS, INC. 2012-11-22 US disclosed
WO-2012156367-A1 AMINO-SUBSTITUTED IMIDAZOPYRIDAZINES AS MKNK1 KINASE INHIBITORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-11-22 WO disclosed
WO-2012158435-A1 COMPOSITIONS AND METHODS FOR JAMM PROTEIN INHIBITION ZHOU HAN-JIE (US) 2012-11-22 WO disclosed
US-8314138-B2 Pyrazole derivative as SCD1 inhibitors for the treatment of diabetes NOVARTIS AG (CH) 2012-11-20 US disclosed
US-8314103-B2 Pyridyl derivatives, their preparation and use Piramal Enterprises Limited (IN) 2012-11-20 US disclosed
WO-2012154610-A1 REACTIVE PI3K KINASE INHIBITORS AND USES THEREOF INTELLIKINE, LLC (US) 2012-11-15 WO disclosed
WO-2012154608-A1 REACTIVE MTOR AND PI3 KINASE INHIBITORS AND USES THEREOF INTELLIKINE, LLC (US) 2012-11-15 WO disclosed
US-20120289457-A1 PEPTIDE OLIGONUCLEOTIDE CONJUGATES AVI BIOPHARMA, INC. (US) 2012-11-15 US disclosed
EP-2121608-B1 DIHYDROPYRIDINE DERIVATIVES USEFUL AS PROTEIN KINASE INHIBITORS BAYER IP GMBH (DE) 2012-11-14 EP disclosed
EP-2521451-A1 HEDGEHOG INHIBITORS Selexagen Therapeutics, Inc. (US) 2012-11-14 EP disclosed
US-8309557-B2 Pyrimidin-4-ylpropanedinitrile derivatives, processes for their preparation and their use as herbicides and plant growth regulators BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-11-13 US disclosed
US-8309566-B2 Pyrimidine-2-amine compounds and their use as inhibitors of JAK kinases RIGEL PHARMACEUTICALS, INC. (US) 2012-11-13 US disclosed
US-8309545-B2 Benzofuran potassium channel blockers and uses thereof BIONOMICS LIMITED (AU) 2012-11-13 US disclosed
US-20120283209-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-11-08 US disclosed
US-20120283207-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-11-08 US disclosed
US-20120283208-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-11-08 US disclosed
WO-2012151562-A1 COMBINATION PHARMACEUTICAL COMPOSITIONS AND USES THEREOF INTELLIKINE, LLC (US) 2012-11-08 WO disclosed
EP-1789079-B1 Insulin-regulated aminopeptidase (IRAP) inhibitors and uses thereof FLOREY HOWARD INST (AU) 2012-11-07 EP disclosed
WO-2012146888-A1 FORMULATION COMPONENT SYNGENTA LIMITED (GB) 2012-11-01 WO disclosed
CN-101945851-B peptidyl nitriles and their use as dipeptidyl peptidase I inhibitors ASTRAZENECA AB 2012-10-31 CN disclosed
CN-102762625-A Polymeric materials COMMW SCIENT IND RES ORG 2012-10-31 CN disclosed
US-8299307-B2 Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC. (US) 2012-10-30 US disclosed
US-8298994-B2 Substituted 1-(diazinyl)pyrazol-4-ylacetic acids, processes for their preparation and their use as herbicides and plant growth regulators BAYER CROPSCIENCE AG (DE) 2012-10-30 US disclosed
WO-2012142670-A1 NUCLEAR MAGNETIC RESONANCE AGENT THE UNIVERSITY OF QUEENSLAND (AU) 2012-10-26 WO disclosed
WO-2012143329-A1 TRIAZOLOPYRIDINES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-10-26 WO disclosed
US-20120269804-A1 SUBSTITUTED BENZOSULPHONAMIDES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-10-25 US disclosed
US-20120269831-A1 SUBSTITUTED PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONES AND THERAPEUTIC USES THEREOF TEMPLE UNIVERSITY- OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2012-10-25 US disclosed
US-20120269803-A1 SUBSTITUTED BENZOSULPHONAMIDES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-10-25 US disclosed
US-20120270901-A1 INDENE DERIVATIVES AS PHARMACEUTICAL AGENTS AQUINOX PHARMACEUTICALS INC. (CA) 2012-10-25 US disclosed
US-20120270859-A1 INDOLINE DERIVATIVES AND THEIR USE IN TREATING DISEASE-STATES SUCH AS CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-10-25 US disclosed
EP-2514423-A2 Method of treatment of age-related macular degeneration (AMD) Prana Biotechnology Ltd (AU) 2012-10-24 EP disclosed
EP-1651606-B1 PYRIDYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2012-10-24 EP disclosed
CN-102746239-A Uracil or thymine derivatives for the treatment of hepatitis C ABBOTT LAB 2012-10-24 CN disclosed
CN-102746240-A Anti-infective pyrimidines and uses thereof ABBOTT LAB 2012-10-24 CN disclosed
US-8293812-B2 Containing thermoplastic resin having solid particles dispersed throughout; controlling particle size; modulus; high tensile strength The University of Queensland St. Lucia (AU) 2012-10-23 US disclosed
US-8293738-B2 Indazole inhibitors of kinase ABBOTT LABORATORIES (US) 2012-10-23 US disclosed
US-8293768-B2 Organic compounds NOVARTIS AG (CH) 2012-10-23 US disclosed
US-20120264740-A1 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2012-10-18 US disclosed
US-20120263670-A1 COMPOUNDS AND METHODS FOR INHIBITING NHE-MEDIATED ANTIPORT IN THE TREATMENT OF DISORDERS ASSOCIATED WITH FLUID RETENTION OR SALT OVERLOAD AND GASTROINTESTINAL TRACT DISORDERS ARDELYX, INC. (US) 2012-10-18 US disclosed
US-20120263708-A1 SUBSTITUTED AMINOQUINOXALINES AS TYROSINE THREONINE KINASE INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-10-18 US disclosed
US-20120263714-A1 SUBSTITUTED HALOPHENOXYBENZAMIDE DERIVATIVES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-10-18 US disclosed
EP-2511255-A1 Substituted prop-2-in-1-ol and prop-2-en-1-ol derivatives Bayer CropScience AG (DE) 2012-10-17 EP disclosed
EP-2510786-A1 Substituted Prop-2-in-1-ol and Prop-2-en-1-ol derivatives Bayer CropScience AG (DE) 2012-10-17 EP disclosed
CN-102741363-A Water swellable polymer materials UNIV SYDNEY 2012-10-17 CN disclosed
US-8288382-B2 Diaminothiazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2012-10-16 US disclosed
WO-2012136776-A1 IMIDAZOPYRIDAZINES AS AKT KINASE INHIBITORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-10-11 WO disclosed
WO-2012136531-A1 SUBSTITUTED IMIDAZOPYRIDINES AND INTERMEDIATES THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-10-11 WO disclosed
US-20120258925-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-10-11 US disclosed
EP-2507235-A1 TRIAZOLOPYRIDINES Bayer Intellectual Property GmbH (DE) 2012-10-10 EP disclosed
EP-2507233-A1 SUBSTITUTED TRIAZOLOPYRIDINES Bayer Intellectual Property GmbH (DE) 2012-10-10 EP disclosed
EP-2507236-A1 TRIAZOLOPYRIDINE DERIVATIVES Bayer Intellectual Property GmbH (DE) 2012-10-10 EP disclosed
EP-2507280-A1 POLYMERIC MATERIALS Commonwealth Scientific and Industrial Research Organisation (AU) 2012-10-10 EP disclosed
EP-1971611-B1 ANTI-VIRAL COMPOUNDS ABBOTT LAB (US) 2012-10-10 EP disclosed
EP-2507322-A1 WATER SWELLABLE POLYMER MATERIALS The University Of Sydney (AU) 2012-10-10 EP disclosed
WO-2012130905-A1 SUBSTITUTED BENZIMIDAZOLES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-10-04 WO disclosed
EP-2504374-A1 WATER CURABLE RESIN FORMULATIONS Petroliam Nasional Berhad (PETRONAS) (MY) 2012-10-03 EP disclosed
US-20120245169-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE LLC 2012-09-27 US disclosed
US-20120245284-A1 WATER CURABLE RESIN FORMULATIONS PETROLIAM NASIONAL BERHAD (PETRONAS) (MY) 2012-09-27 US disclosed
US-20120244119-A1 ANTI-INFECTIVE AGENTS AND USES THEREOF ABBOTT LABORATORIES (US) 2012-09-27 US disclosed
WO-2012129099-A1 FORMULATIONS OF PHENYL URACIL COMPOUNDS ABBOTT LABORATORIES (US) 2012-09-27 WO disclosed
US-8273403-B2 Generation of surface coating diversity BIO-LAYER PTY LTD. (AU) 2012-09-25 US disclosed
US-20120237951-A1 ANALGESIA WITH MINIMAL TOLERANCE AND DEPENDENCE BY A MU OPIOID RECEPTOR AGONIST THAT ALSO BINDS FILAMIN A PAIN THERAPEUTICS 2012-09-20 US disclosed
US-20120238706-A1 POLYMERIC MATERIALS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2012-09-20 US disclosed
US-20120238542-A1 AMINOPYRAZOLOQUINAZOLINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-09-20 US disclosed
EP-2498600-A1 FILAMIN A-BINDING ANTI-INFLAMMATORY ANALGESIC Pain Therapeutics, Inc. (US) 2012-09-19 EP disclosed
EP-2498599-A1 ANALGESIC THAT BINDS FILAMIN A Pain Therapeutics, Inc. (US) 2012-09-19 EP disclosed
CN-102675290-A Bicyclic dihydropyrazole compounds SHANDONG HENGLI MEDICAL TECHNOLOGY CO LTD 2012-09-19 CN disclosed
CN-101278079-B Drug design method ALCHEMIA LTD 2012-09-19 CN disclosed
US-8268990-B2 Compounds ASTRAZENECA AB (SE) 2012-09-18 US disclosed
US-8263606-B2 Spiro-oxindole compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2012-09-11 US disclosed
US-8263775-B2 Insulin-regulated aminopeptidase (IRAP) inhibitors and uses thereof HOWARD FLOREY INSTITUTE (AU) 2012-09-11 US disclosed
US-8258160-B2 SCD1 inhibitors triazole and tetrazole compounds NOVARTIS AG (CH) 2012-09-04 US disclosed
US-20120220572-A1 TRICYCLIC INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2012-08-30 US disclosed
US-20120220562-A1 Anti-Viral Compounds Abbott Labaoratories (US) 2012-08-30 US disclosed
WO-2012116237-A2 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, LLC (US) 2012-08-30 WO disclosed
WO-2012116257-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. (US) 2012-08-30 WO disclosed
EP-2491016-A1 SUBSTITUTED BENZOSULPHONAMIDES Bayer Pharma Aktiengesellschaft (DE) 2012-08-29 EP disclosed
EP-2491014-A1 SUBSTITUTED HALOPHENOXYBENZAMIDE DERIVATIVES Bayer Pharma Aktiengesellschaft (DE) 2012-08-29 EP disclosed
EP-2491015-A1 SUBSTITUTED BENZOSULPHONAMIDES Bayer Pharma Aktiengesellschaft (DE) 2012-08-29 EP disclosed
EP-2491025-A1 AZAAZULENE COMPOUNDS Industrial Technology Research Institute (TW) 2012-08-29 EP disclosed
US-8252723-B2 Substituted 1-(3-pyridinyl)pyrazol-4-ylacetic acids, processes for their preparation and their use as herbicides and plant growth regulators BAYER CROPSCIENCE AG (DE) 2012-08-28 US disclosed
US-20120214759-A1 TREATMENT OF KLEBSIELLA PNEUMONIAE INFECTIONS WITH ANTIBACTERIAL AMINOGLYCOSIDE COMPOUNDS ACHAOGEN, INC. (US) 2012-08-23 US disclosed
US-20120214852-A1 Alkoxy Compounds for Disease Treatment ACUCELA INC. (US) 2012-08-23 US disclosed
US-20120214760-A1 TREATMENT OF URINARY TRACT INFECTIONS WITH ANTIBACTERIAL AMINOGLYCOSIDE COMPOUNDS ACHAOGEN, INC. (US) 2012-08-23 US disclosed
US-20120213733-A1 ANTI-INFECTIVE AGENTS AND USES THEREOF ABBOTT LABORATORIES (US) 2012-08-23 US disclosed
EP-2488177-A1 FILAMIN A BINDING ANTI-INFLAMMATORY AND ANALGESIC Pain Therapeutics, Inc. (US) 2012-08-22 EP disclosed
US-8247424-B2 Water soluble groups on ring A; antitumor antibiotics; 1-Desoxy-5-C-[(8R)-4',9,9'-trihydroxy-6'-methoxy-1,1',3',5',8'-pentaoxo-1,1',2,3',5',6,7,8'-octahydrospiro[cyclopenta[g]isoquinoline-8,2'-cyclopenta[b]-naphthalene]-3-yl]pentitol; topoisomerase inhibitors; cyclodextrin inclusions; stereoisomers ZENTOPHARM GMBH (DE) 2012-08-21 US disclosed
US-20120208781-A1 AMINOGLYCOSIDE DOSING REGIMENS ACHAOGEN, INC. (US) 2012-08-16 US disclosed
US-20120208822-A1 PYRIMIDO-PYRROLO-QUINOXALINEDIONE INHIBITORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR PROTEIN AND USES THEREFOR THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-08-16 US disclosed
EP-2486044-A2 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS Achaogen, Inc. (US) 2012-08-15 EP disclosed
US-20120202877-A1 ANTI-INFLUENZA AGENTS GRIFFITH UNIVERSITY (AU) 2012-08-09 US disclosed
WO-2012104388-A1 NEW AZAINDOLYLPHENYL SULFONAMIDES AS SERINE/THREONINE KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-08-09 WO disclosed
US-20120202860-A2 Analgesic Compounds, Compositions and Uses Thereof GALLEON PHARMACEUTICALS, INC. (US) 2012-08-09 US disclosed
EP-2483264-A1 PYRAZOLE DERIVATIVES WHICH MODULATE STEAROYL-COA DESATURASE Novartis AG (CH) 2012-08-08 EP disclosed
EP-2483249-A1 PYRIMIDINE DERIVATIVES AS PROTEIN TYROSINE KINASE 2 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2012-08-08 EP disclosed
EP-2484679-A2 N3-heteroaryl substituted triazoles and n5-heteroaryl substitued triazoles useful as axl inhibitors Rigel Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
US-8236852-B2 Drugs/cosmetics having at least one (substituted phenyl)-propenal moiety; bioavailability' water solubility; antiandrogens; antiinflammatory and wound healing agents; antiarthritic agents; acne; alopecia, hirsutism; anticarcinogenic agents; cancer of the bladder, liver, breast; Kennedy's disease ANDROSCIENCE CORPORATION (US) 2012-08-07 US disclosed
US-8236950-B2 Anti-viral compounds ABBOTT LABORATORIES (US) 2012-08-07 US disclosed
US-8236835-B2 Heterocyclic inhibitors of stearoyl-CoA desaturase NOVARTIS AG (CH) 2012-08-07 US disclosed
US-20120196791-A1 COMBINATION THERAPIES USING ANTIBACTERIAL AMINOGLYCOSIDE COMPOUNDS ACHAOGEN, INC. (US) 2012-08-02 US disclosed
WO-2012101184-A1 NEW 5-ALKYNYL-PYRIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-08-02 WO disclosed
WO-2012101238-A1 NEW PYRIMIDO[5,4-D]PYRIMIDYLAMINO PHENYL SULFONAMIDES AS SERINE/THREONINE KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-08-02 WO disclosed
WO-2012101186-A1 NEW 5-ALKYNYL-PYRIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-08-02 WO disclosed
EP-1888543-B1 APOPTOSIS PROMOTERS ABBOTT LAB (US) 2012-08-01 EP disclosed
US-8232246-B2 Anti-viral compounds ABBOTT LABORATORIES (US) 2012-07-31 US disclosed
US-20120189546-A1 Radiolabelling Method Using Cycloalkyl Groups BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-07-26 US disclosed
US-20120189580-A1 ANTI-INFECTIVE AGENTS AND USES THEREOF ABBOTT LABORATORIES (US) 2012-07-26 US disclosed
US-20120189548-A1 2-ARYLPYRAZOLO[L,5-ALPHA]PYRIMIDIN-3-YL ACETAMIDE DERIVATIVES AS LIGANDS FOR TRANSLOCATOR PROTEIN (18 KDA) THE UNIVERSITY OF SYDNEY (AU) 2012-07-26 US disclosed
US-20120190681-A1 PICOLINAMIDE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2012-07-26 US disclosed
WO-2012097684-A1 BICYCLIC CARBOXAMIDE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2012-07-26 WO disclosed
WO-2012100135-A1 PICOLINAMIDE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2012-07-26 WO disclosed
WO-2012098513-A1 UV STABILIZATION OF ISOSORBIDE POLYCARBONATES SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2012-07-26 WO disclosed
WO-2012097682-A1 BICYCLIC INHIBITORS OF ALK ABBOTT LABORATORIES (US) 2012-07-26 WO disclosed
CN-102612514-A Anti -influenza agents UNIV GRIFFITH 2012-07-25 CN disclosed
US-20120184501-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-07-19 US disclosed
US-20120184651-A1 UV Stabilization of Isosorbide Polycarbonates SHPP GLOBAL TECHNOLOGIES B.V. (NL) 2012-07-19 US disclosed
US-20120184568-A1 PROCESSES FOR PREPARING ISOQUINOLINONES AND SOLID FORMS OF ISOQUINOLINONES HCR COLLATERAL MANAGEMENT, LLC 2012-07-19 US disclosed
WO-2012097049-A2 DNA REPAIR ENZYME INHIBITOR NANOPARTICLES AND USES THEREOF THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2012-07-19 WO disclosed
EP-2476679-A2 Substituted triazoles useful as AXL inhibitors Rigel Pharmaceuticals, Inc. (US) 2012-07-18 EP disclosed
EP-1905773-B1 Compounds and methods for inhibiting mitotic progression by inhibition of aurora kinase MILLENNIUM PHARM INC (US) 2012-07-18 EP disclosed
CN-101460525-B Polymer products and interfacial polymerization process using RAFT agents UNIV SYDNEY 2012-07-18 CN disclosed
US-20120178726-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2012-07-12 US disclosed
EP-2473478-A2 NOVEL USES Nanyang Polytechnic (SG) 2012-07-11 EP disclosed
EP-2473498-A1 SUBSTITUTED AMINOQUINOXALINES AS TYROSINE THREONINE KINASE INHIBITORS Bayer Pharma Aktiengesellschaft (DE) 2012-07-11 EP disclosed
US-8217171-B2 Antiviral agents BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2012-07-10 US disclosed
US-8217189-B2 Chromenone potassium channel blockers and uses thereof BIONOMICS LIMITED (AU) 2012-07-10 US disclosed
US-20120172290-A1 Anti-Viral Compounds ABBOTT LABORATORIES (US) 2012-07-05 US disclosed
US-20120172332-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-07-05 US disclosed
EP-2471363-A1 Use of aryl-, heteroaryl- and benzylsulfonamide carboxylic acids, -carboxylic acid esters, -carboxylic acid amides and -carbonitriles and/or its salts for increasing stress tolerance in plants Bayer CropScience AG (DE) 2012-07-04 EP disclosed
EP-2471536-A1 STEROID ANALOGS AND CHARACTERIZATION AND TREATMENT METHODS Harbor BioSciences, Inc. (US) 2012-07-04 EP disclosed
EP-2471776-A1 Pyridin-2-ylpropandinitriles and their use as herbicides Bayer CropScience AG (DE) 2012-07-04 EP disclosed
EP-2471787-A1 New compounds Boehringer Ingelheim International GmbH (DE) 2012-07-04 EP disclosed
US-20120165282-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-06-28 US disclosed
WO-2012085126-A1 OXINDOLOPYRIMIDINE AS IGF1R RECEPTOR INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-28 WO disclosed
WO-2012083866-A1 QUINOLINE DERIVATIVES AS ANTI-CANCER AGENTS THE HONG KONG POLYTECHNIC UNIVERSITY (CN) 2012-06-28 WO disclosed
WO-2012085127-A1 NEW TRIAZOLYLPHENYL SULFONAMIDES AS SERINE/THREONINE KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-28 WO disclosed
US-20120165370-A1 QUINOLINE DERIVATIVES AS ANTI-CANCER AGENTS THE HONG KONG POLYTECHNIC UNIVERSITY (CN) 2012-06-28 US disclosed
EP-2468269-A1 Nitric oxide donors in therapy of nitric oxide deficiency-induced disturbances of cerebral microcirculation Universitätsklinikum Münster (DE) 2012-06-27 EP disclosed
EP-2467141-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Intellikine, Inc. (US) 2012-06-27 EP disclosed
EP-2467137-A1 BIARYL COMPOUNDS AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2012-06-27 EP disclosed
US-8207245-B2 Gels AORTECH INTERNATIONAL PLC (GB) 2012-06-26 US disclosed
US-8207179-B2 Substituted indolines as tyrosine kinase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-26 US disclosed
WO-2012083058-A2 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2012-06-21 WO disclosed
WO-2012080232-A1 2-SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-06-21 WO disclosed
WO-2012083164-A1 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2012-06-21 WO disclosed
WO-2012080229-A1 IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT HYPERPROLIFERATIVE DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-06-21 WO disclosed
WO-2012083048-A2 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2012-06-21 WO disclosed
WO-2012083170-A1 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2012-06-21 WO disclosed
WO-2012080236-A1 6-SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-06-21 WO disclosed
US-20120157314-A1 NOVEL SUBSTITUTED PICOLINIC ACIDS, SALTS AND ACID DERIVATIVES THEREOF, AND USE THEREOF AS HERBICIDES BAYER CROPSCIENCE AG (DE) 2012-06-21 US disclosed
WO-2012080234-A1 SUBSTITUTED 6-IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-06-21 WO disclosed
US-20120157306-A1 Substituted Fused Pyrimidinones and Dihydropyrimidinones BAYER CROPSCIENCE AG (DE) 2012-06-21 US disclosed
WO-2012080230-A1 6 SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-06-21 WO disclosed
WO-2012080228-A1 6-THIO-SUBSTITUTED IMIDAZOPYRAZINES FOR USE AS MPS-1 AND TKK INHIBITORS IN THE TREATMENT OF HYPERPROLIFERATIVE DISORDERS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-06-21 WO disclosed
EP-2464354-A1 PYRIMIDO-PYRROLO-QUINOXALINEDIONE INHIBITORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR PROTEIN AND USES THEREFOR The Regents of the University of California (US) 2012-06-20 EP disclosed
US-8202997-B2 Compositions and methods for treating or preventing hypoxic or ischemic injury IKARIA, INC. (US) 2012-06-19 US disclosed
US-8202905-B2 Compounds with (substituted phenyl)-propenal moiety, their derivatives, biological activity, and use thereof ANDROSCIENCE CORPORATION (US) 2012-06-19 US disclosed
US-8203001-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-19 US disclosed
US-8202513-B2 Aryl potassium channel blockers and uses thereof BIONOMICS LIMITED (AU) 2012-06-19 US disclosed
WO-2012078633-A2 METHODS OF INHIBITING METASTASIS FROM CANCER PHILADELPHIA HEALTH AND EDUCATION CORPORATION, D/B/A DREXEL UNIVERSITY COLLEGE OF MEDICENE (US) 2012-06-14 WO disclosed
US-20120149701-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE, INC. 2012-06-14 US disclosed
US-8198456-B2 e.g. 1,4-dihydro-4-(1H-indazol-5-yl)-2,6-dimethyl-3,5-pyridinedicarbonitrile; c-Met tyrosine kinase inhibitor; antitumor agent; lung, liver, gastric and breast solid tumors; pancreatic cancer, glioma, and hepatocellular carcinoma BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-06-12 US disclosed
US-8198308-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-12 US disclosed
WO-2012074999-A1 NOVEL COMPOUNDS AS RESPIRATORY STIMULANTS FOR TREATMENT OF BREATHING CONTROL DISORDERS OR DISEASES GALLEON PHARMACEUTICALS, INC. (US) 2012-06-07 WO disclosed
WO-2012074931-A2 PHOTOLINDUCED ALKYNE-AZIDE CLICK REACTIONS THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2012-06-07 WO disclosed
US-20120142647-A1 Novel Compounds as Respiratory Stimulants for Treatment of Breathing Control Disorders or Diseases GALLEON PHARMACEUTICALS, INC. 2012-06-07 US disclosed
US-20120141471-A1 Methods of Inhibiting Metastasis from Cancer Alliance Discovery, Inc. 2012-06-07 US disclosed
US-8193182-B2 Substituted isoquinolin-1(2H)-ones, and methods of use thereof INTELLIKINE, INC. (US) 2012-06-05 US disclosed
US-20120135948-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-05-31 US disclosed
US-20120135945-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-05-31 US disclosed
US-20120135946-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-05-31 US disclosed
WO-2012069620-A1 NITRIC OXIDE DONORS IN THERAPY OF NITRIC OXIDE DEFICIENCY-INDUCED DISTURBANCES OF CEREBRAL MICROCIRCULATION Westfälische Wilhelms-Universität Münster (DE) 2012-05-31 WO disclosed
EP-2456444-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS Intellikine, Inc. (US) 2012-05-30 EP disclosed
EP-2456842-A1 IONIC LIQUID FLAME RETARDANTS H & C Scientific Resources International, LLC (US) 2012-05-30 EP disclosed
US-8188104-B2 Anti-infective agents and uses thereof ABBOTT LABORATORIES (US) 2012-05-29 US disclosed
US-8188112-B2 Naphthalamide derivatives having antiproliferative activity AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2012-05-29 US disclosed
US-20120128662-A1 SUBSTITUTED IMIDAZOQUINOXALINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-05-24 US disclosed
US-20120129833-A1 CYCLIC KETOENOLS FOR THERAPY BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-05-24 US disclosed
US-20120129894-A1 Alkoxy Compounds for Disease Treatment ACUCELA INC. (US) 2012-05-24 US disclosed
US-20120129860-A1 STYRENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2012-05-24 US disclosed
US-20120129850-A1 IMIDAZOLOTHIAZOLE COMPOUNDS FOR THE TREATMENT OF DISEASE AMBIT BIOSCIENCES CORPORATION 2012-05-24 US disclosed
WO-2012067978-A1 ANTIBACTERIAL AMIINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-05-24 WO disclosed
US-20120128743-A1 POLYMER PARTICLES THE UNIVERSITY OF SYDNEY (AU) 2012-05-24 US disclosed
WO-2012067963-A1 NAMPT INHIBITORS ABBOTT LABORATORIES (US) 2012-05-24 WO disclosed
WO-2012067965-A1 NAMPT AND ROCK INHIBITORS ABBOTT LABORATORIES (US) 2012-05-24 WO disclosed
EP-2455376-A1 Heterocyclic compounds as inhibitors of hepatitis C virus (HCV) Abbott Laboratories (US) 2012-05-23 EP disclosed
EP-2454230-A1 RADIOLABELLING METHOD USING CYCLOALKYL GROUPS Bayer Pharma Aktiengesellschaft (DE) 2012-05-23 EP disclosed
EP-2454248-A1 ANTI -INFLUENZA AGENTS Griffith University (AU) 2012-05-23 EP disclosed
WO-2012062745-A1 ALKOXY-SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-05-18 WO disclosed
WO-2012062748-A1 AMINOALCOHOL SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINAZOLINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-05-18 WO disclosed
WO-2012064973-A2 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed
WO-2012062743-A1 ARYLAMINOALCOHOL-SUBSTITUTED 2,3-DIHYDROIMIDAZO[1,2-C]QUINOLINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-05-18 WO disclosed
US-20120122924-A1 NAMPT INHIBITORS ABBOTT LABORATORIES (US) 2012-05-17 US disclosed
US-20120122842-A1 NAMPT AND ROCK INHIBITORS ABBOTT LABORATORIES (US) 2012-05-17 US disclosed
US-20120122938-A1 Alkoxy Compounds for Disease Treatment ACUCELA INC. (US) 2012-05-17 US disclosed
US-20120122809-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-05-17 US disclosed
US-20120122838-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. 2012-05-17 US disclosed
US-20120122909-A9 SPIRO-OXINDOLE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2012-05-17 US disclosed
CN-102459186-A Anthelmintic agents and uses thereof ANTHELMINTIC AGENTS AND THEIR USE 2012-05-16 CN disclosed
CN-102459306-A Novel amide derivatives of steroidal [3,2-C ] pyrazole compounds having glucocorticoid activity ASTRAZENECA AB 2012-05-16 CN disclosed
US-8178548-B2 Anti-infective agents and uses thereof ABBOTT LABORATORIES (US) 2012-05-15 US disclosed
US-20120115918-A1 Anti-Viral Compounds ABBOTT LABORATORIES (US) 2012-05-10 US disclosed
EP-2448569-A2 PHARMACOLOGY OF VISUAL CYCLE MODULATORS Acucela, Inc. (US) 2012-05-09 EP disclosed
CN-102448920-A Antiviral compounds and uses thereof ABBOTT LAB 2012-05-09 CN disclosed
CN-102448952-A Antiviral compounds and uses thereof ABBOTT LAB 2012-05-09 CN disclosed
US-8173811-B2 Apoptosis promoters ABBOTT LABORATORIES (US) 2012-05-08 US disclosed
WO-2012055953-A1 SUBSTITUTED PHENOXYPYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-05-03 WO disclosed
US-20120107269-A1 THIOPHENE DERIVATIVES Tianjin Hemay Biotech Co., Ltd (CN) 2012-05-03 US disclosed
EP-1651616-B1 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2012-05-02 EP disclosed
EP-1651605-B1 PYRIDYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2012-05-02 EP disclosed
CN-102439049-A Polymer particles UNIV SYDNEY 2012-05-02 CN disclosed
US-8168636-B2 Polycyclic heteroaryl substituted triazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2012-05-01 US disclosed
WO-2012054110-A2 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. (US) 2012-04-26 WO disclosed
US-20120100104-A1 Antiviral Compounds And Uses Thereof ABBOTT LABORATORIES (US) 2012-04-26 US disclosed
CN-102424703-A Surface polymerisation process and polymer product using RAFT agent UNIV SYDNEY 2012-04-25 CN disclosed
US-8163724-B2 Glucocorticosteroids, processes for their preparation, pharmaceutical compositions containing them and their use in therapy ASTRAZENECA AB (SE) 2012-04-24 US disclosed
WO-2012051361-A1 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2012-04-19 WO disclosed
US-20120094981-A1 ANTHELMINTIC AGENTS AND THEIR USE INTERVET INTERNATIONAL B.V. (NL) 2012-04-19 US disclosed
US-20120094976-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-04-19 US disclosed
US-20120094975-A1 PYRIDO [5, 4-D] PYRIMIDINES AS CELL PROLIFERATION INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-04-19 US disclosed
US-20120094963-A1 TARGETING PRODRUGS AND COMPOSITIONS FOR THE TREATMENT OF GASTROINTESTINAL DISEASES of Queen Elizabeth near Dublin 2012-04-19 US disclosed
EP-2440548-A1 2- ( LH-PYRAZOL-4 -YLAMINO ) -PYRIMIDINE AS KINASE INHIBITORS Abbott Laboratories (US) 2012-04-18 EP disclosed
US-20120088768-A1 PINANE-SUBSTITUTED PYRIMIDINEDIAMINE DERIVATIVES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2012-04-12 US disclosed
WO-2012045196-A1 PHOSPHOGLYCERATE KINASE INHIBITORS ABBOTT LABORATORIES (US) 2012-04-12 WO disclosed
EP-1851205-B1 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2012-04-11 EP disclosed
US-8153741-B2 Furanone copolymers TYCO HEALTHCARE GROUP LP (US) 2012-04-10 US disclosed
US-8153636-B2 Pyridyl derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2012-04-10 US disclosed
US-8153593-B2 Transglutaminase inhibitors and methods of use thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2012-04-10 US disclosed
US-8153788-B2 Substituted 2,4-diamino-1,3,5-triazines, processes for their use as herbicides and crop growth regulators BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2012-04-10 US disclosed
US-20120083532-A1 NOVEL USES NANYANG POLYTECHNIC (SG) 2012-04-05 US disclosed
US-20120082646-A1 Antiviral Compounds And Uses Thereof ABBOTT LABORATORIES (US) 2012-04-05 US disclosed
EP-2435411-A1 2, 4 -DIAMINOPYRIMIDINES FOR THE TREATMENT OF DISEASES CHARACTERISED BY EXCESSIVE OR ABNORMAL CELL PROLIFERATION Boehringer Ingelheim International GmbH (DE) 2012-04-04 EP disclosed
US-8148378-B2 Pyridazine derivatives and their use as inhibitors of stearoyl-CoA desaturase-1 activity in a mammal XENON PHARMACEUTICALS INC. (CA) 2012-04-03 US disclosed
US-8143284-B2 2-cyclohexyl-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide; allergic encephalitis, arthritis, cardiac and kidney toxicities from doxorubicin-based and platinum-based antineoplastic agents, carcinoma of the breast, central nervous system inflammation, cervical carcinoma, ABBOTT LABORATORIES (US) 2012-03-27 US disclosed
WO-2012037217-A1 TRANSFER HYDROGENATION OF CYCLOPAMINE ANALOGS INFINITY PHARMACEUTICALS, INC. (US) 2012-03-22 WO disclosed
US-20120071681-A1 PROCESS FOR PREPARING ORGANOMETALLOIDS THE CHINESE UNIVERSITY OF HONGKONG (CN) 2012-03-22 US disclosed
EP-2431371-A1 THIOPHENE DERIVATIVES Tianjin Hemay Bio-Tech Co., Ltd. (CN) 2012-03-21 EP disclosed
US-8138337-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2012-03-20 US disclosed
US-20120065169-A1 OLIGONUCLEOTIDE ANALOGUES HAVING MODIFIED INTERSUBUNIT LINKAGES AND/OR TERMINAL GROUPS JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2012-03-15 US disclosed
US-20120065399-A1 Transfer Hydrogenation of Cyclopamine Analogs INFINITY PHARMACEUTICALS, INC. (US) 2012-03-15 US disclosed
US-20120065400-A1 Transfer Hydrogenation of Cyclopamine Analogs INFINITY PHARMACEUTICALS, INC. (US) 2012-03-15 US disclosed
EP-2428515-A1 Spiro-oxindole compounds and their uses as therapeutic agents Xenon Pharmaceuticals Inc. (CA) 2012-03-14 EP disclosed
EP-2427195-A2 HETEROCYCLIC COMPOUNDS AND USES THEREOF Intellikine, Inc. (US) 2012-03-14 EP disclosed
CN-102372710-A Fused cyclic compound being taken as mineral corticoid recept antagonist KBP BIOSCIENCES CO LTD 2012-03-14 CN disclosed
US-20120059000-A1 CHEMICAL COMPOUNDS, COMPOSITIONS AND METHODS FOR KINASE MODULATION INFINITY PHARMACEUTICALS, INC. 2012-03-08 US disclosed
US-20120058989-A1 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS ACHAOGEN, INC. (US) 2012-03-08 US disclosed
WO-2012031243-A2 dsRNA MOLECULES COMPRISING OLIGONUCLEOTIDE ANALOGS HAVING MODIFIED INTERSUBUNIT LINKAGES AND/OR TERMINAL GROUPS AVI BIOPHARMA, INC. (US) 2012-03-08 WO disclosed
WO-2012030948-A1 QUINAZOLINE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2012-03-08 WO disclosed
WO-2012030918-A1 ADENOSINE A3 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2012-03-08 WO disclosed
WO-2012030910-A1 2-CYCLOQUINAZOLINE DERIVATIVES AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2012-03-08 WO disclosed
WO-2012030924-A1 AZOLOPYRIDINE AND AZOLOPYRIMIDINE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2012-03-08 WO disclosed
WO-2012030912-A1 7-CYCLYLQUINAZOLINE DERIVATIVES AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2012-03-08 WO disclosed
WO-2012030894-A1 THIENOPYRIDINE AND THIENOPYRIMIDINE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2012-03-08 WO disclosed
EP-2424537-A1 SUBSTITUTED IMIDAZOQUINOXALINES Bayer Pharma Aktiengesellschaft (DE) 2012-03-07 EP disclosed
US-8129190-B2 Via violanthrone compounds APPLIED NANOTECH HOLDINGS, INC. (US) 2012-03-06 US disclosed
US-8129374-B2 Method of using imidazolothiazole compounds for the treatment of disease AMBIT BIOSCIENCE CORPORATION (US) 2012-03-06 US disclosed
US-20120053174-A1 QUINAZOLINE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION 2012-03-01 US disclosed
US-20120052572-A1 COMPOSITIONS FOR STABILIZING DNA, RNA AND PROTEINS IN BLOOD AND OTHER BIOLOGICAL SAMPLES DURING SHIPPING AND STORAGE AT AMBIENT TEMPERATURES EXACT SCIENCES CORPORATION 2012-03-01 US disclosed
US-20120053176-A1 ADENOSINE A3 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORP. (US) 2012-03-01 US disclosed
EP-1542997-B1 PYRAZOLYLBENZOTHIAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS DERMIRA CANADA INC (CA) 2012-02-29 EP disclosed
WO-2011044502-A9 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-02-23 WO disclosed
US-20120046270-A1 PYRIMIDO [5,4-D] PYRIMIDINE DERIVATIVES FOR THE INHIBITION OF TYROSINE KINASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-02-23 US disclosed
US-20120045455-A1 PHOSPHOTETRAHYDROPYRAN COMPOUNDS FOR THE TREATMENT OF WOUNDS AND FIBROTIC DISORDERS Pharmaxis Pty Limited (AU) 2012-02-23 US disclosed
WO-2012024583-A2 OXYSTEROL COMPOUNDS FATE THERAPEUTICS, INC. (US) 2012-02-23 WO disclosed
WO-2012022776-A1 SUBSTITUTED THIOPENES OR FURANS AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2012-02-23 WO disclosed
EP-2419404-A1 ANTI-VIRAL COMPOUNDS Abbott Laboratories (US) 2012-02-22 EP disclosed
CN-102361889-A Raft polymerisation COMMW SCIENT IND RES ORG 2012-02-22 CN disclosed
WO-2012021146-A1 IONIC LIQUID FLAME RETARDANTS H & C Scientific Resources International, LLC (US) 2012-02-16 WO disclosed
US-20120041039-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. (US) 2012-02-16 US disclosed
US-20120041038-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. (US) 2012-02-16 US disclosed
US-20120041064-A1 SKIN TREATMENT PEPLIN RESEARCH PTY LTD (AU) 2012-02-16 US disclosed
EP-2073806-B1 USE OF SPIRO-OXINDOLE COMPOUNDS AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2012-02-15 EP disclosed
US-20120035161-A1 Novel Compositions and Methods of Treating Diseases Using the Same CORRIDOR PHARMACEUTICALS, INC. 2012-02-09 US disclosed
WO-2012018638-A2 COMPOSITIONS FOR STABILIZING DNA, RNA AND PROTEINS IN BLOOD AND OTHER BIOLOGICAL SAMPLES DURING SHIPPING AND STORAGE AT AMBIENT TEMPERATURES BIOMATRICA, INC. (US) 2012-02-09 WO disclosed
WO-2011044503-A9 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-02-09 WO disclosed
WO-2012018639-A2 COMPOSITIONS FOR STABILIZING DNA, RNA AND PROTEINS IN SALIVA AND OTHER BIOLOGICAL SAMPLES DURING SHIPPING AND STORAGE AT AMBIENT TEMPERATURES BIOMATRICA, INC. (US) 2012-02-09 WO disclosed
WO-2011044498-A9 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-02-09 WO disclosed
US-20120034270-A1 S1P Receptors Modulators AKAAL PHARMA PTY LTD (AU) 2012-02-09 US disclosed
US-20120035199-A9 SPIROHETEROCYCLIC COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2012-02-09 US disclosed
EP-2410987-A1 METHODS OF TREATMENT USING COMBINATION THERAPY Ambit Biosciences Corporation (US) 2012-02-01 EP disclosed
EP-1888595-B1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2012-02-01 EP disclosed
US-8106087-B2 Spiro-oxindole compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2012-01-31 US disclosed
WO-2012010704-A1 NEW AMINOPYRAZOLOQUINAZOLINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-26 WO disclosed
EP-2408752-A1 SUBSTITUTED PYRIMIDINES FOR THE TREATMENT OF CANCER Boehringer Ingelheim International GmbH (DE) 2012-01-25 EP disclosed
US-8101647-B2 Spiro-oxindole compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2012-01-24 US disclosed
US-20120014906-A1 ORGANIC COMPOUNDS XENON PHARMACEUTICALS INC. (CA) 2012-01-19 US disclosed
WO-2012009263-A1 COCAINE ANALOGS AND METHODS OF PREPARATION AND USES THEREOF TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2012-01-19 WO disclosed
EP-1979348-B1 ANTI-VIRAL COMPOUNDS ABBOTT LAB (US) 2012-01-18 EP disclosed
US-8097630-B2 Pinane-substituted pyrimidinediamine derivatives derivatives and pharmaceutical compositions containing the dthe activity of the receptor protein tyrosine kinase Axl. Methods of using erivatives are disclosed as being useful in inhibiting activity of enzyme RIGEL PHARMACEUTICALS, INC. (US) 2012-01-17 US disclosed
WO-2012006477-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. (US) 2012-01-12 WO disclosed
WO-2012006474-A2 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. (US) 2012-01-12 WO disclosed
WO-2012005691-A1 COMPOUND FOR USE IN PEPTIDE SYNTHESIS NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2012-01-12 WO disclosed
US-20120010124-A9 Cell Penetrating Peptide Conjugates for Delivering of Nucleic Acids into a Cell DIATOS (FR) 2012-01-12 US disclosed
US-20120010135-A1 SPIRO DERIVATIVES FOR THE MODULATION OF STEAROYL-COA DESATURASE XENON PHARMACEUTICALS INC. (CA) 2012-01-12 US disclosed
WO-2012006473-A1 COMPOUNDS AND METHODS FOR INHIBITING PHOSPHATE TRANSPORT ARDELYX, INC. (US) 2012-01-12 WO disclosed
CN-102316866-A Skin treatment PEPLIN RESEARCH PTY LTD 2012-01-11 CN disclosed
US-8093227-B2 Monosaccharide compounds and methods therefor ALCHEMIA PTY LTD (AU) 2012-01-10 US disclosed
US-8093396-B2 Benzthiazole inhibitors of poly(ADP-ribose)polymerase ABBOTT LABORATORIES (US) 2012-01-10 US disclosed
US-20120004164-A1 ORGANIC COMPOUNDS XENON PHARMACEUTICALS INC. (CA) 2012-01-05 US disclosed
US-20120004381-A1 RAFT POLYMERISATION COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2012-01-05 US disclosed
US-20120004269-A1 Alkynyl Phenyl Derivative Compounds for Treating Ophthalmic Diseases and Disorders ACUCELA INC. (US) 2012-01-05 US disclosed
US-20120004196-A1 Anti-Viral Compounds Abbott Labaoratories (US) 2012-01-05 US disclosed
EP-2401304-A1 POLYMER PARTICLES The University Of Sydney (AU) 2012-01-04 EP disclosed
EP-2401267-A1 JAK KINASE MODULATING QUINAZOLINE DERIVATIVES AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2012-01-04 EP disclosed
EP-2402334-A1 Inhibitors of E1 Activating Enzymes Millennium Pharmaceuticals, Inc. (US) 2012-01-04 EP disclosed
CN-102304300-A Polymer product and interfacial polymerisation process using raft agent UNIV SYDNEY 2012-01-04 CN disclosed
US-20110319366-A1 Plasma Carboxypeptidase B Inhibitors BUCKMAN BRAD (US) 2011-12-29 US disclosed
US-20110318388-A1 S1P Receptors Modulators and Their Use Thereof AKAAL PHARMA PTY LTD (AU) 2011-12-29 US disclosed
US-20110319393-A1 ANTHELMINTIC AGENTS AND THEIR USE INTERVET INTERNATIONAL B.V. (NL) 2011-12-29 US disclosed
EP-2398797-A1 PYRIMIDO [5,4-D]PYRIMIDINE DERIVATIVES FOR THE INHIBITION OF TYROSINE KINASES Boehringer Ingelheim International GmbH (DE) 2011-12-28 EP disclosed
US-8084607-B2 Apoptosis promoters ABBOTT LABORATORIES (US) 2011-12-27 US disclosed
US-8084503-B2 Indene derivatives as pharmaceutical agents AQUINOX PHARMACEUTICALS INC. (CA) 2011-12-27 US disclosed
US-20110312939-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-12-22 US disclosed
US-20110313156-A1 HETEROCYCLYL CARBONIC ACID AMIDES AS ANTIPROLIFERATIVE AGENTS, PDKL INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-12-22 US disclosed
WO-2011157688-A1 SUBSTITUTED TRIAZOLOPYRIDINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-12-22 WO disclosed
EP-1763350-B1 NICOTINAMIDE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2011-12-21 EP disclosed
EP-2395996-A1 COMPOUNDS AND METHODS FOR INHIBITING MMP2 AND MMP9 Indiana University Research and Technology Corporation (US) 2011-12-21 EP disclosed
US-8080657-B2 Compounds of reverse turn mimetics and the use thereof CHOONGWAE PHARMA CORPORATION (KR) 2011-12-20 US disclosed
CN-102281875-A Combination therapy using AXL inhibitors for the prevention, treatment or management of metastatic cancer 2011-12-14 CN disclosed
US-8076516-B2 Amine derivative compounds for treating ophthalmic diseases and disorders ACUCELA, INC. (US) 2011-12-13 US disclosed
WO-2011151259-A1 SUBSTITUTED IMIDAZOPYRAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-12-08 WO disclosed
US-20110301128-A1 Pyrrole Derivatives As Pharmaceutical Agents EXELIXIS, INC. (US) 2011-12-08 US disclosed
US-8071603-B2 Contacting a source of hSCD with N-(2-Cyclopropyl-ethyl)-4-[4-(5-fluoro-2-trifluoromethyl-benzoyl)-piperazin-1-yl]-benzamide; elevated lipid levels, cardiovascular disease, diabetes, obesity, metabolic syndrome XENON PHARMACEUTICALS INC. (CA) 2011-12-06 US disclosed
US-8071764-B2 Compounds of reverse turn mimetics and the use thereof (2) CHOONGWAE PHARMA CORPORATION (KR) 2011-12-06 US disclosed
US-20110293744-A1 BENZOXAZOLE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE ABBOTT LABORATORIES (US) 2011-12-01 US disclosed
US-20110293643-A1 COMPOUNDS AND METHODS FOR INHIBITING MMP2 AND MMP9 INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION 2011-12-01 US disclosed
US-20110294842-A9 SPIRO (FURO [3, 2-C] PYRIDINE-3-3' -INDOL) -2' (1'H)-ONE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF SODIUM-CHANNEL MEDIATED DISEASES, SUCH AS PAIN XENON PHARMACEUTICALS INC. (CA) 2011-12-01 US disclosed
US-20110294766-A1 16 Alpha, 17 Alpha-Acetal Glucocorticosteroidal Derivatives and their Use ASTRAZENECA AB (SE) 2011-12-01 US disclosed
US-20110294664-A1 USE OF DERIVATIVES OF (1-CYANOCYCLOPROPYL)PHENYLPHOSPHINIC ACID, ESTERS THEREOF AND/OR SALTS THEREOF FOR ENHANCING TOLERANCE IN PLANTS TO ABIOTIC STRESS BAYER CROPSCIENCE AG (DE) 2011-12-01 US disclosed
WO-2011150198-A1 AZOLYL UREA COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2011-12-01 WO disclosed
WO-2011150201-A2 AZOLYL AMIDE COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2011-12-01 WO disclosed
WO-2011149937-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, INC. (US) 2011-12-01 WO disclosed
CN-102264737-A Anti-viral compounds 2011-11-30 CN disclosed
US-8067611-B2 Substituted 1-(thiazolyl)-and 1-(isothiazolyl)pyrazol-4-ylacetic acids, processes for their preparation and their use as herbicides and plant growth regulators BAYER CROPSCIENCE AG (DE) 2011-11-29 US disclosed
US-8067409-B2 Protein kinase inhibitors ABBOTT LABORATORIES (US) 2011-11-29 US disclosed
WO-2011144725-A2 NOVEL METHODS FOR PREVENTING OR TREATING DIABETES FUNDACIÓN PÚBLICA ANDALUZA PROGRESO Y SALUD (ES) 2011-11-24 WO disclosed
US-20110288109-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-24 US disclosed
US-20110288041-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2011-11-24 US disclosed
US-20110286995-A1 Drug Therapy for Celiac Sprue THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2011-11-24 US disclosed
US-20110288071-A1 SUBSTITUTED PYRIMIDINES FOR THE TREATMENT OF DISEASES SUCH AS CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-24 US disclosed
WO-2011144622-A1 1H - IMIDAZO [4, 5 - C] QUINOLINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-24 WO disclosed
WO-2011146842-A1 PROCESS FOR SYNTHESIS OF SILANE DIPEPTIDE ANALOGS TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2011-11-24 WO disclosed
WO-2011146882-A1 CHEMICAL COMPOUNDS, COMPOSITIONS AND METHODS FOR KINASE MODULATION INTELLIKINE, INC. (US) 2011-11-24 WO disclosed
EP-2387395-A1 AXL INHIBITORS FOR USE IN COMBINATION THERAPY FOR PREVENTING, TREATING OR MANAGING METASTATIC CANCER Rigel Pharmaceuticals, Inc. (US) 2011-11-23 EP disclosed
US-8063093-B2 Derivatives of 5-(halo)alkanoyl-6-hydroxy- benozofuran, benzothiophene, or indole; autoimmune diseases; systemic lupus erythematosis, rheumatoid arthritis, multiple sclerosis and psoriasis, transplant rejection; antiproliferative, anticarcinogenic, antidiabetic, antiinflammatory and antiulcer agents HARVEY ANDREW J (AU) 2011-11-22 US disclosed
US-8063051-B2 9-substituted-8-oxo-adenine compounds as toll-like receptor (TLR7) modulators ASTRAZENECA AB (SE) 2011-11-22 US disclosed
US-8063053-B2 1-(arylsulfonyl)-4-(piperazin-1-yl)-1H-benzimidazoles as 5-hydroxytryptamine-6 ligands WYETH LLC (US) 2011-11-22 US disclosed
US-8063084-B2 Heterocyclic compounds suitable for the treatment of diseases related to elevated lipid levels NOVARTIS AG (CH) 2011-11-22 US disclosed
US-20110281866-A1 HETEROCYCLIC KINASE INHIBITORS INTELLIKINE, INC. (US) 2011-11-17 US disclosed
US-20110280824-A1 Furanone Copolymers TYCO HEALTHCARE GROUP LP (US) 2011-11-17 US disclosed
US-20110281846-A1 BRIDGED BICYCLIC ARYL AND BRIDGED BICYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2011-11-17 US disclosed
US-20110281868-A1 INDAZOLE INHIBITORS OF KINASE ABBOTT LABORATORIES (US) 2011-11-17 US disclosed
US-20110281842-A1 PYRROLOPYRIDINE AND PYRROLOPYRIMIDINE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2011-11-17 US disclosed
CN-102245604-A Antiviral compounds ABBOTT LAB 2011-11-16 CN disclosed
US-20110275633-A1 2,4-DIAMINOPYRIMIDINE DERIVATES AS PTK2- INHIBITORS FOR THE TREATMENT OF ABNORMAL CELL GROWTH BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-10 US disclosed
US-20110274713-A1 ANTIGEN-PRESENTING SCAFFOLDS THE UNIVERSITY OF QUEENSLAND (AU) 2011-11-10 US disclosed
US-20110275586-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2011-11-10 US disclosed
EP-1651620-B1 PIPERAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2011-11-09 EP disclosed
EP-2069353-B1 POLYCYCLIC AGENTS FOR THE TREATMENT OF RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENT MANAGEMENT (AU) 2011-11-09 EP disclosed
CN-102239166-A Substituted 1- (thiazolyl) -and 1- (isothiazolyl) pyrazol-4-ylacetic acids, method for the production thereof and use thereof as herbicides and plant growth regulators BAYER CROPSCIENCE AG 2011-11-09 CN disclosed
US-20110269779-A1 METHODS AND COMPOSITIONS FOR TREATMENT OF OPHTHALMIC CONDITIONS INTELLIKINE, INC. (US) 2011-11-03 US disclosed
US-20110269740-A1 JAK KINASE MODULATING COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION 2011-11-03 US disclosed
US-20110269958-A1 PYRIDONS AS PDK1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-03 US disclosed
WO-2010132760-A9 ANTIBACTERIAL DERIVATIVES OF TOBRAMYCIN ACHAOGEN, INC. (US) 2011-11-03 WO disclosed
US-8049016-B2 Thiazole derivatives which inhibit stearoyl-CoA desaturase enzymes NOVARTIS AG (CH) 2011-11-01 US disclosed
US-8049008-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2011-11-01 US disclosed
US-20110263565-A1 COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-10-27 US disclosed
WO-2011133388-A1 PYRROLOPYRIDINE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2011-10-27 WO disclosed
WO-2011131741-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDES AS PDK1 INIHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-10-27 WO disclosed
EP-2181985-B1 Antiviral Agent SHIONOGI & CO (JP) 2011-10-26 EP disclosed
EP-2139894-B1 9-SUBSTITUTED-8-OXO-ADENINE COMPOUNDS AS TOLL-LIKE RECEPTOR (TLR7) MODULATORS ASTRAZENECA AB (SE) 2011-10-26 EP disclosed
US-8044067-B2 Isoquinolines as IGF-1R inhibitors ANALYTECON S.A. (CH) 2011-10-25 US disclosed
US-8044061-B2 Parkinson's disease, catalepsy, dystonia, dyskinetic syndrome, restless legs syndrome, migraine, pain, dementia, neurodegenerative disorders, alcohol withdrawal and/or ischemic conditions such as e.g. stroke or cardiac ischemia. UCB PHARMA GMBH (DE) 2011-10-25 US disclosed
US-20110257152-A1 PYRROLOPYRIDINE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2011-10-20 US disclosed
US-20110257187-A1 PHTHALAZIN-(2H)-ONE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2011-10-20 US disclosed
US-20110257189-A1 PYRROLOPYRAZINONE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2011-10-20 US disclosed
US-20110257014-A1 1-(Heteroaryl)pyrazol-4-ylacetic acids, processes for their preparation and their use as herbicides and plant growth regulators BAYER CROPSCIENCE AG (DE) 2011-10-20 US disclosed
US-20110256129-A1 APOPTOSIS PROMOTERS ABBOTT LABORATORIES 2011-10-20 US disclosed
WO-2011130478-A1 PHTHALAZIN-(2H)-ONE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2011-10-20 WO disclosed
WO-2011130481-A1 PYRROLOPYRAZINONE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2011-10-20 WO disclosed
EP-2377854-A1 N-phenyl-dioxo-hydropyrimidines useful as hepatitis C virus (HCV) inhibitors Abbott Laboratories (US) 2011-10-19 EP disclosed
EP-2377869-A1 Synthesis of Bortezomib MILLENNIUM PHARMACEUTICALS, INC. (US) 2011-10-19 EP disclosed
US-8040491-B2 Exposure method, substrate stage, exposure apparatus, and device manufacturing method NIKON CORPORATION (JP) 2011-10-18 US disclosed
US-20110251224-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2011-10-13 US disclosed
WO-2011123890-A1 RADIOPROTECTOR COMPOUNDS AND METHODS PETER MACCALLUM CANCER INSTITUTE (AU) 2011-10-13 WO disclosed
WO-2010132765-A9 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2011-10-13 WO disclosed
EP-1534755-B1 GENERATION OF SURFACE COATING DIVERSITY BIO LAYER PTY LTD (AU) 2011-10-12 EP disclosed
US-20110243884-A1 BIODEGRADABLE POLYMER - BIOACTIVE MOIETY CONJUGATES THE BIONICS INSTITUTE OF AUSTRALIA (AU) 2011-10-06 US disclosed
EP-2370416-A1 2,4-DIAMINOPYRIMIDINE DERIVATES AS PTK2- INHIBITORS FOR THE TREATMENT OF ABNORMAL CELL GROWTH Boehringer Ingelheim International GmbH (DE) 2011-10-05 EP disclosed
EP-1648874-B1 PIPERAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2011-10-05 EP disclosed
US-8030488-B2 Piperazine derivatives as stearoyl-coa desaturase inhibitors and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2011-10-04 US disclosed
US-20110237598-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-09-29 US disclosed
US-20110237783-A1 HYDRAZONOPYRAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTICS Valocor Therapeutics, Inc. (CA) 2011-09-29 US disclosed
WO-2011117382-A1 PYRIDYLTRIAZOLES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-09-29 WO disclosed
WO-2011117381-A1 B-RAF KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-09-29 WO disclosed
US-20110237567-A9 TRICYCLIC SPIRO-OXINDOLE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2011-09-29 US disclosed
EP-2367799-A1 NEW COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2011-09-28 EP disclosed
EP-2367800-A2 NEW COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2011-09-28 EP disclosed
EP-2368890-A1 Hepatitis C virus inhibitors Abbott Laboratories (US) 2011-09-28 EP disclosed
EP-2368882-A1 ANTI-INFECTIVE PYRIMIDINES AND USES THEREOF ABBOTT LABORATORIES (US) 2011-09-28 EP disclosed
CN-102203058-A Sulfur-linked compounds for the treatment of ophthalmic diseases and disorders ACUCELA INC 2011-09-28 CN disclosed
US-8026237-B2 For modulating activity of one or more steroid nuclear receptors and for treatment, prevention, or amelioration of symptoms of disease or disorder related to the activity of receptors; 5-benzo[b]thiophen-2-yl-1,4-dimethyl-1H-pyrrole-3-carboxylic acid (4-methanesulfonyl-phenyl)-amide EXELIXIS, INC. (US) 2011-09-27 US disclosed
US-8026360-B2 Substituted pyridazines as stearoyl-CoA desaturase inhibitors XENON PHARMACEUTICALS INC. (CA) 2011-09-27 US disclosed
WO-2011114220-A1 NEURO-PROTECTIVE EFFECTS OF ADELOSTEMMA GRACILLIMUM AND ITS ISOLATED COMPOUNDS BIOTECHNOLOGY RESEARCH CORPORATION LIMITED (CN) 2011-09-22 WO disclosed
US-20110230350-A1 ARYL-AND HETARYLSULFONAMIDES AS ACTIVE INGREDIENTS AGAINST ABIOTIC PLANT STRESS BAYER CROPSCIENCE AG (DE) 2011-09-22 US disclosed
WO-2011113862-A1 IMIDAZOPYRAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-09-22 WO disclosed
EP-1846035-B1 COMBINATION THERAPY XENON PHARMACEUTICALS INC (CA) 2011-09-21 EP disclosed
EP-1487428-B1 AMINO-SUBSTITUTED (E)-2,6-DIALKOXYSTYRYL 4-SUBSTITUTED BENZYLSULFONES FOR TREATING PROLIFERATIVE DISORDERS UNIV TEMPLE (US) 2011-09-21 EP disclosed
WO-2010147836-A9 COMBINATION THERAPIES USING ANTIBACTERIAL AMINOGLYCOSIDE COMPOUNDS ACHAOGEN, INC. (US) 2011-09-15 WO disclosed
WO-2010132839-A9 AMINOGLYCOSIDE DOSING REGIMENS ACHAOGEN, INC. (US) 2011-09-15 WO disclosed
US-20110224186-A1 CARBACEPHEM BETA-LACTAM ANTIBIOTICS ACHAOGEN, INC. (US) 2011-09-15 US disclosed
WO-2010132768-A9 ANTIBACTERIAL DERIVATIVES OF SISOMICIN ACHAOGEN, INC. (US) 2011-09-15 WO disclosed
WO-2011112602-A1 ANALGESIC COMPOUNDS, COMPOSITIONS, AND USES THEREOF GALLEON PHARMACEUTICALS, INC. (US) 2011-09-15 WO disclosed
US-20110224269-A1 Analgesic Compounds, Compositions, and Uses Thereof GALLEON PHARMACEUTICALS, INC. 2011-09-15 US disclosed
US-8017599-B2 Sequence selective pyrrole and imidazole polyamide metallocomplexes UNIVERSITY OF WESTERN SYDNEY (AU) 2011-09-13 US disclosed
WO-2010132759-A9 ANTIBACTERIAL DERIVATIVES OF DIBEKACIN ACHAOGEN, INC. (US) 2011-09-09 WO disclosed
US-20110218103-A1 Fluoroalkyl-substituted 2-amidobenzimidazoles BAYER CROPSCIENCE AG (DE) 2011-09-08 US disclosed
EP-2363419-A1 Polymer product formed using raft agent The University of Sydney (AU) 2011-09-07 EP disclosed
US-8012965-B2 e.g. 1-(2-chloro-7-methylthieno[3,2-d]pyrimidin-4-yl)-N3-(5,7-ethano-5,7,8-trihydro-6-methyl-1,6-naphthyridin-3-yl)-1H-1,2,4-triazole-3,5-diamine; angiogenesis inhibitor, antiproliferative agent RIGEL PHARMACEUTICALS, INC. (US) 2011-09-06 US disclosed
US-8013001-B2 Modulators of LXR EXELIXIS, INC. (US) 2011-09-06 US disclosed
US-20110212966-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2011-09-01 US disclosed
CN-101193921-B Carbon-bridged cyclopentadienyl-fluorenyl ligands TOTAL PETROCHEMICALS RES FELUY 2011-08-31 CN disclosed
US-8008325-B2 Plasma carboxypeptidase B inhibitors BAYER SCHERING PHARMA AG (DE) 2011-08-30 US disclosed
WO-2011102807-A1 A SUBSTRATE FOR IMMOBILIZING FUNCTIONAL SUBSTANCES AND METHOD FOR PREPARING THE SAME TEMASEK POLYTECHNIC (SG) 2011-08-25 WO disclosed
WO-2010132757-A9 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2011-08-25 WO disclosed
US-20110207699-A1 Anti-Viral Compounds Abbott Labaoratories (US) 2011-08-25 US disclosed
WO-2011098433-A1 CYCLIC KETO-ENOLS FOR THERAPY BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-08-18 WO disclosed
US-20110201581-A1 Novel Compounds 010 ASTRAZENECA AB (SE) 2011-08-18 US disclosed
US-20110201840-A1 TERMINAL 1,1-DISUBSTITUTED ALKENES, METHOD OF MAKING AND USING THEREOF THE CHINESE UNIVERSITY OF HONG KONG (CN) 2011-08-18 US disclosed
EP-2355814-A2 PYRONES FOR THE TREATMENT OF METABOLIC DISORDERS Limerick BioPharma, Inc. (US) 2011-08-17 EP disclosed
US-7999010-B2 Indene derivatives as pharmaceutical agents AQUINOX PHARMACEUTICALS INC. (CA) 2011-08-16 US disclosed
US-7999051-B2 Furanone copolymers TYCO HEALTHCARE GROUP LP (US) 2011-08-16 US disclosed
US-7998995-B2 LXR and FXR modulators EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed
US-20110196088-A1 POLYMER PRODUCT AND INTERFACIAL POLYMERISATION PROCESS USING RAFT AGENT THE UNIVERSITY OF SYDNEY (AU) 2011-08-11 US disclosed
US-20110195305-A1 Organic electrolyte and lithium battery including the same SAMSUNG SDI CO., LTD. (KR) 2011-08-11 US disclosed
EP-2203431-B1 ANTI-INFECTIVE PYRIMIDINES AND USES THEREOF ABBOTT LAB (US) 2011-08-10 EP disclosed
US-7994346-B2 such as methyl 2-({(4S,5R)-5-[(1E,3E,7E)-(S)-10-(4-fluorophenoxy)-9-hydroxydeca-1,3,7-trien-5-yn-1-yl]-2,2-dimethyl-1,3-dioxolan-4-yl}methoxy)acetate, useful in treating inflammatory and autoimmune disorders in humans BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-08-09 US disclosed
US-20110190566-A1 POLYMER MICROGEL BEADS UNIVERSITY OF SYDNEY (AU) 2011-08-04 US disclosed
US-20110190514-A1 PYRONE ANALOG COMPOSITIONS AND METHODS LIMERICK BIOPHARMA, INC. (US) 2011-08-04 US disclosed
EP-2349236-A2 COMPOSITIONS AND METHODS FOR TREATING OR PREVENTING HYPOXIC OR ISCHEMIC INJURY Ikaria, Inc. (US) 2011-08-03 EP disclosed
EP-2350083-A1 PYRIDO [5, 4-D]PYRIMIDINES AS CELL PROLIFERATION INHIBITORS Boehringer Ingelheim International GmbH (DE) 2011-08-03 EP disclosed
EP-2350090-A2 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2011-08-03 EP disclosed
EP-2350052-A2 ANTIPROLIFERATIVE COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2011-08-03 EP disclosed
EP-2350091-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2011-08-03 EP disclosed
US-7989422-B2 Antibacterial agents ALCHEMIA LIMITED (AU) 2011-08-02 US disclosed
US-7989656-B2 Biaryl carboxylic acid apoptosis promoters ABBOTT LABORATORIES (US) 2011-08-02 US disclosed
US-20110183952-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-28 US disclosed
US-20110183986-A1 POLYCYCLIC ARYL SUBSTITUTED TRIAZOLES AND POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2011-07-28 US disclosed
US-20110182670-A1 SOIL REMEDIATION PROCESS THE UNIVERSITY OF QUEENSLAND (AU) 2011-07-28 US disclosed
WO-2011091131-A2 ESLICARBAZEPINE ACETATE AND ITS POLYMORPHS DR. REDDY'S LABORATORIES LTD. (IN) 2011-07-28 WO disclosed
EP-2346508-A1 HETEROCYCLIC KINASE INHIBITORS Intellikine, Inc. (US) 2011-07-27 EP disclosed
EP-1534284-B1 AMINO-SUBSTITUTED SULFONANILIDES AND DERIVATIVES THEREOF FOR TREATING PROLIFERATIVE DISORDERS UNIV TEMPLE (US) 2011-07-27 EP disclosed
US-20110178126-A1 PYRAZOLYLBENZOTHIAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS Valocor Therapeutics, Inc. (CA) 2011-07-21 US disclosed
US-20110177002-A1 CYLIC POLYAMINES FOR BINDING PHOSPHATIDYLSERINE BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-07-21 US disclosed
EP-2345652-A1 Antiviral compounds Abbott Laboratories (US) 2011-07-20 EP disclosed
EP-2344451-A2 SULFUR-LINKED COMPOUNDS FOR TREATING OPTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2011-07-20 EP disclosed
US-7981885-B2 N-[3-substituted piperazino] alkylphenothiazines; antiproliferative agents, apoptotic agents; 5-HT receptor antagonists IMMUNE CONTROL INC. (US) 2011-07-19 US disclosed
US-7982071-B2 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2011-07-19 US disclosed
WO-2011085261-A1 HEDGEHOG INHIBITORS SELEXAGEN THERAPEUTICS, INC. (US) 2011-07-14 WO disclosed
WO-2011085128-A1 HEDGEHOG INHIBITORS SELEXAGEN THERAPEUTICS, INC. (US) 2011-07-14 WO disclosed
US-20110172126-A1 LIBRARIES OF PEPTIDE CONJUGATES AND METHODS FOR MAKING THEM XENOME LTD (AU) 2011-07-14 US disclosed
US-20110172282-A9 USE OF SPIRO-OXINDOLE COMPOUNDS AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2011-07-14 US disclosed
US-20110172258-A9 INDENE DERIVATIVES AS PHARMACEUTICAL AGENTS AQUINOX PHARMACEUTICALS INC. (CA) 2011-07-14 US disclosed
US-20110172228-A1 KINASE INHIBITORS AND METHODS OF USE INTELLIKINE LLC 2011-07-14 US disclosed
EP-2343294-A1 Substituted triazolopyridines Bayer Schering Pharma AG (DE) 2011-07-13 EP disclosed
EP-2343297-A1 Triazolopyridines Bayer Schering Pharma AG (DE) 2011-07-13 EP disclosed
EP-2343295-A1 Triazolopyridine derivates Bayer Schering Pharma AG (DE) 2011-07-13 EP disclosed
US-7977489-B2 Benzylthiazolone inhibitors of estrogen-related receptors (ERR) EXELIXIS, INC. (US) 2011-07-12 US disclosed
US-20110166298-A1 CONDUCTING AND SEMICONDUCTING ORGANIC MATERIALS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL ORGANISATION (AU) 2011-07-07 US disclosed
US-20110166390-A1 CARBON NANOHOOPS AND METHODS OF MAKING LAWRENCE BERKELEY NATIONAL LABORATORY (US) 2011-07-07 US disclosed
US-20110166130-A1 NOVEL POTASSIUM CHANNEL BLOCKERS AND USES THEREOF BIONOMICS LIMITED (AU) 2011-07-07 US disclosed
EP-2340242-A2 COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2011-07-06 EP disclosed
EP-2340271-A1 POLYMER-BIOACTIVE AGENT CONJUGATES The Bionic Ear Institute (AU) 2011-07-06 EP disclosed
US-7973161-B2 Apoptosis promoters ABBOTT LABORATORIES (US) 2011-07-05 US disclosed
US-7973171-B2 Process for synthesis of dialkoxyorganoboranes BURKHARDT ELIZABETH 2011-07-05 US disclosed
US-20110155996-A1 BISTABLE CARBAZOLE COMPOUNDS STMICROELECTRONICS S.R.L. (IT) 2011-06-30 US disclosed
US-20110160233-A1 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2011-06-30 US disclosed
WO-2011076687-A1 PYRIDINONE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-06-30 WO disclosed
EP-2337781-A2 ANTI-VIRAL COMPOUNDS TO TREAT HCV INFECTION Abbott Laboratories (US) 2011-06-29 EP disclosed
CN-102112453-A Novel potassium channel blockers and uses thereof BIONOMICS LTD 2011-06-29 CN disclosed
WO-2011075185-A1 TARGETED DRUG PHOSPHORYLCHOLINE POLYMER CONJUGATES OLIGASIS (US) 2011-06-23 WO disclosed
US-7964591-B2 Pyridazine derivatives and their use as therapeutic agents NOVARTIS PHARMA AG (CH) 2011-06-21 US disclosed
US-20110142757-A1 NOVEL COMPOUNDS AND THEIR USES IN DIAGNOSIS THE UNIVERSITY OF SYDNEY 2011-06-16 US disclosed
US-20110144112-A9 APOPTOSIS PROMOTERS ABBVIE INC. 2011-06-16 US disclosed
US-20110144128-A1 Heterocyclic Carboxamide Compounds as Steroid Nuclear Receptors Ligands EXELIXIS, INC. (US) 2011-06-16 US disclosed
US-20110144139-A1 HEPSIN INHIBITORS FRED HUTCHINSON CANCER RESEARCH CENTER 2011-06-16 US disclosed
EP-2331556-A1 BISTABLE CARBAZOLE COMPOUNDS STMicroelectronics S.r.l. (IT) 2011-06-15 EP disclosed
EP-2331514-A2 CYCLIC POLYAMINES FOR BINDING PHOSPHATIDYLSERINE Bayer Schering Pharma Aktiengesellschaft (DE) 2011-06-15 EP disclosed
EP-2203430-B1 N-PHENYL-DIOXO-HYDROPYRIMIDINES USEFUL AS HEPATITIS C VIRUS (HCV) INHIBITORS ABBOTT LAB (US) 2011-06-15 EP disclosed
US-20110137633-A1 ANTI-VIRAL COMPOUNDS AND METHODS OF IDENTIFYING THE SAME ABBOTT LABORATORIES (US) 2011-06-09 US disclosed
WO-2011066616-A1 POLYMERIC MATERIALS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2011-06-09 WO disclosed
WO-2011066608-A1 WATER SWELLABLE POLYMER MATERIALS THE UNIVERSITY OF SYDNEY (AU) 2011-06-09 WO disclosed
US-20110136988-A1 CONDENSATION POLYMERS WITH MODIFIED PROPERTIES Commonwealth Scientific an dIndustrial Research Organisation (AU) 2011-06-09 US disclosed
US-20110137057-A1 Unsaturated Steroid Compounds BIOVIE INC. 2011-06-09 US disclosed
US-7956185-B2 Cyclobut-3-ene-1,2,-dione inhibitors of polo-like kinases ABBOTT LABORATORIES (US) 2011-06-07 US disclosed
WO-2011065813-A1 WATER CURABLE RESIN FORMULATIONS PETROLIAM NASIONAL BERHAD (PETRONAS) (MY) 2011-06-03 WO disclosed
WO-2011064328-A1 TRIAZOLOPYRIDINE DERIVATIVES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-06-03 WO disclosed
WO-2011063907-A1 SUBSTITUTED TRIAZOLOPYRIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-06-03 WO disclosed
WO-2011063908-A1 TRIAZOLOPYRIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-06-03 WO disclosed
US-20110130401-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-06-02 US disclosed
US-20110129417-A1 ADMINISTRABLE COMPOSITIONS UNIVERSITY OF SYDNEY (AU) 2011-06-02 US disclosed
EP-2326641-A2 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS Rigel Pharmaceuticals, Inc. (US) 2011-06-01 EP disclosed
US-7951805-B2 Heterocyclic derivatives and their use as mediators of stearoyl-CoA desaturase XENON PHARMACEUTICALS INC. (CA) 2011-05-31 US disclosed
EP-2324012-A1 NEW COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2011-05-25 EP disclosed
EP-2323986-A2 HETOEROCYCLYL CARBONIC ACID AMIDES AS ANTIPROLIFERATIVE AGENTS, PDKL INHIBITORS Boehringer Ingelheim International GmbH (DE) 2011-05-25 EP disclosed
CN-102076436-A Soil remediation process UNIV QUEENSLAND 2011-05-25 CN disclosed
US-7947854-B2 Phospholipase inhibitor; prevention or therapy of microbial infection; bactericides; fungicides; viricides; parasiticides; using quaternary or phosphonium group containing compounds THE UNIVERSITY OF SYDNEY (AU) 2011-05-24 US disclosed
US-7947733-B2 Phosphorylated pyrone analogs and methods LIMERICK BIOPHARMA (US) 2011-05-24 US disclosed
US-20110118533-A1 POLYMER MICROGEL BEADS AND PREPARATIVE METHOD THEREOF UNIVERSITY OF SYDNEY (AU) 2011-05-19 US disclosed
US-20110118245-A1 RAF KINASE MODULATOR COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORP. 2011-05-19 US disclosed
EP-2321299-A2 PYRIDONS AS PDK1 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2011-05-18 EP disclosed
US-20110112162-A9 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2011-05-12 US disclosed
US-20110105487-A1 FILAMIN A BINDING ANTI-INFLAMMATORY AND ANALGESIC PAIN THERAPEUTICS 2011-05-05 US disclosed
US-20110105484-A1 FILAMIN A-BINDING ANTI-INFLAMMATORY ANALGESIC PAIN THERAPEUTICS 2011-05-05 US disclosed
US-20110105547-A1 FILAMIN A-BINDING ANTI-INFLAMMATORY ANALGESIC PAIN THERAPEUTICS 2011-05-05 US disclosed
US-20110105481-A1 FILAMIN A BINDING ANTI-INFLAMMATORY AND ANALGESIC PAIN THERAPEUTICS 2011-05-05 US disclosed
US-20110105511-A1 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2011-05-05 US disclosed
US-20110105530-A1 ORGANIC COMPOUNDS XENON PHARMACEUTICALS INC. (CA) 2011-05-05 US disclosed
US-20110105496-A1 Methods For The Treatment Of Myosin Heavy Chain-Mediated Conditions Using 4,7-Dihydrothieno[2,3-B]Pyridine Compounds GILEAD COLORADO, INC. 2011-05-05 US disclosed
EP-2316458-A1 Pyridazine derivatives for inhibiting human stearoyl-coa-desaturase Xenon Pharmaceuticals Inc. (CA) 2011-05-04 EP disclosed
EP-2316457-A1 Pyridine derivatives for inhibiting human stearoyl-coa-desaturase Xenon Pharmaceuticals Inc. (CA) 2011-05-04 EP disclosed
EP-2316827-A1 Piperazine derivatives and their use as therapeutic agents Xenon Pharmaceuticals Inc. (CA) 2011-05-04 EP disclosed
EP-2316825-A1 Pyridyl derivatives and their use as therapeutic agents Xenon Pharmaceuticals Inc. (CA) 2011-05-04 EP disclosed
EP-2316828-A1 Piperazine derivatives and their use as therapeutic agents Xenon Pharmaceuticals Inc. (CA) 2011-05-04 EP disclosed
EP-2316826-A1 Pyridazine derivatives and their use as therapeutics agents Xenon Pharmaceuticals Inc. (CA) 2011-05-04 EP disclosed
US-7935693-B2 Polycyclic aryl substituted triazoles and polycyclic heteroaryl substituted triazoles useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2011-05-03 US disclosed
US-7935721-B2 Spiro-oxindole compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2011-05-03 US disclosed
US-20110098274-A1 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2011-04-28 US disclosed
WO-2011047788-A1 SUBSTITUTED BENZOSULPHONAMIDES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-04-28 WO disclosed
WO-2011047795-A1 SUBSTITUTED BENZOSULPHONAMIDES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-04-28 WO disclosed
WO-2011047796-A1 SUBSTITUTED HALOPHENOXYBENZAMIDE DERIVATIVES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-04-28 WO disclosed
US-20110098305-A1 ARYLSULFONAMIDE COMPOUNDS, COMPOSITIONS AND METHODS OF USE BAELL JONATHAN BAYLDON 2011-04-28 US disclosed
US-20110098317-A1 USE OF UNSATURATED SPHINGOSINE COMPOUNDS AS CHEMOTHERAPEUTIC AGENTS FOR THE TREATMENT OF CANCER CHILDREN'S HOSPITAL & RESEARCH CENTER AT OAKLAND (US) 2011-04-28 US disclosed
EP-2314582-A1 Heterocyclic compounds as antiviral agents Biota Scientific Management Pty Ltd (AU) 2011-04-27 EP disclosed
EP-2313414-A2 KINASE INHIBITORS AND METHODS OF USE Intellikine, Inc. (US) 2011-04-27 EP disclosed
US-20110092502-A1 DIAMINOTHIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2011-04-21 US disclosed
US-20110092415-A1 Anti-Viral Compounds Abbott Labaoratories (US) 2011-04-21 US disclosed
US-7928255-B2 Intermediates for the preparation of lipoxin A4 analogs BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-04-19 US disclosed
WO-2011044501-A2 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2011-04-14 WO disclosed
WO-2011044498-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2011-04-14 WO disclosed
WO-2011044502-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2011-04-14 WO disclosed
WO-2011044503-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2011-04-14 WO disclosed
EP-2308812-A2 N-acylsulfonamide apoptosis promoters Abbott Laboratories (US) 2011-04-13 EP disclosed
EP-2307379-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2011-04-13 EP disclosed
EP-2307013-A1 PAIN-RELIEVING COMPOSITIONS OF FUROXAN NO DONORS AND USES THEREOF The University Of Queensland (AU) 2011-04-13 EP disclosed
CN-102015750-A 16 alpha, 17 beta-acetal glucocorticoid derivative and application thereof ASTRAZENECA AB 2011-04-13 CN disclosed
US-7923439-B2 Hydroxamate compositions TYCO HEALTHCARE GROUP LP (US) 2011-04-12 US disclosed
US-7923445-B2 10-{3-[4-(2-Amino)ethylpiperazinyl]propyl}2-trifluoromethylphenothiazine and analogues and derivatives; antiproliferative agents; serotonin receptor antagonists; apoptosis in activated lymphocytes, including T, B, and and mylenoma cells; asthma; antiarthritic agents; rheumatic diseeases IMMUNE CONTROL, INC. (US) 2011-04-12 US disclosed
WO-2011039344-A1 PYRIMIDINE DERIVATIVES AS PROTEIN TYROSINE KINASE 2 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-04-07 WO disclosed
WO-2011039358-A1 PYRAZOLE DERIVATIVES WHICH MODULATE STEAROYL-COA DESATURASE NOVARTIS AG (CH) 2011-04-07 WO disclosed
US-20110082131-A1 TRIAZOLE DERIVATIVES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2011-04-07 US disclosed
EP-1888592-B1 SPIROHETEROCYCLIC COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2011-04-06 EP disclosed
CN-101198615-B Method for synthesizing dialkoxyorganoborane BASF AG 2011-04-06 CN disclosed
CN-102007124-A Pyrimidine-2-amine compounds and their use as inhibitors of jak kinases RIGEL PHARMACEUTICALS INC 2011-04-06 CN disclosed
US-7919484-B2 Combination therapy XENON PHARMACEUTICALS INC. (CA) 2011-04-05 US disclosed
US-7919496-B2 5-[4-(2-Trifluoromethylbenzoyl)piperazin-1-yl]-[1,3,4]thiadiazole-2-carboxylic acid ethyl ester; metabolic disorders type II diabetes, impaired glucose tolerance, insulin resistance, obesity, fatty liver, non-alcoholic steatohepatitis, dyslipidemia and metabolic syndrome; cardiovascular disorders XENON PHARMACEUTICALS INC. (CA) 2011-04-05 US disclosed
US-20110073331-A1 Ionic Liquid Flame Retardants H & C Scientific Resources International, LLC 2011-03-31 US disclosed
US-20110077252-A1 PYRIDYL DERIVATIVES, THEIR PREPARATION AND USE Piramal Enterprises Limited (IN) 2011-03-31 US disclosed
CN-101993451-A Process for synthesis of dialkoxyorganoboranes BASF SE 2011-03-30 CN disclosed
US-7915411-B2 Anti-viral compounds ABBOTT LABORATORIES (US) 2011-03-29 US disclosed
US-20110070193-A1 Anti-Infective Agents and Uses Thereof ABBOTT LABORATORIES (US) 2011-03-24 US disclosed
US-20110071167-A1 METHOD OF TREATMENT OF AGE-RELATED MACULAR DEGENERATION (AMD) PRANA BIOTECHNOLOGY LIMITED (AU) 2011-03-24 US disclosed
US-20110071158-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-03-24 US disclosed
US-20110071133-A1 BICYCLIC ARYL AND BICYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2011-03-24 US disclosed
US-7910742-B2 Survivin inhibitors ABBOTT LABORATORIES (US) 2011-03-22 US disclosed
US-7910755-B2 Stem cell expansion and uses HARBOR BIOSCIENCES, INC. (US) 2011-03-22 US disclosed
US-7910595-B2 Anti-viral compounds ABBOTT LABORATORIES (US) 2011-03-22 US disclosed
WO-2011031745-A1 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS ACHAOGEN, INC. (US) 2011-03-17 WO disclosed
WO-2011031743-A1 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS ACHAOGEN, INC. (US) 2011-03-17 WO disclosed
US-20110064673-A1 New L-Glutamic acid and L-Glutamine derivative (III), use thereof and method for obtaining them PIRAMAL IMAGING SA (CH) 2011-03-17 US disclosed
WO-2011031740-A1 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS ACHAOGEN, INC. (US) 2011-03-17 WO disclosed
WO-2011031744-A1 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS ACHAOGEN, INC. (US) 2011-03-17 WO disclosed
US-20110059938-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-03-10 US disclosed
WO-2011026579-A1 SUBSTITUTED AMINOQUINOXALINES AS TYROSINE THREONINE KINASE INHIBITORS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-03-10 WO disclosed
US-20110060163-A1 Process for Synthesis of Dialkoxyorganoboranes BASF SE (DE) 2011-03-10 US disclosed
EP-2291175-A1 ADMINISTRABLE COMPOSITIONS THE UNIVERSITY OF SYDNEY (AU) 2011-03-09 EP disclosed
US-7902181-B2 Compounds 010 ASTRAZENECA AB (SE) 2011-03-08 US disclosed
EP-2289510-A1 Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-coa desaturase enzymes Xenon Pharmaceuticals Inc. (CA) 2011-03-02 EP disclosed
WO-2011022473-A1 BIARYL COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2011-02-24 WO disclosed
US-20110044898-A1 TRANSLOCATOR PROTEIN LIGANDS UNIVERSITY OF SYDNEY (AU) 2011-02-24 US disclosed
US-20110046165-A1 CERTAIN CHEMICAL ENTITLES, COMPOSITIONS AND METHODS INTELLIKINE LLC 2011-02-24 US disclosed
WO-2011022439-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, INC. (US) 2011-02-24 WO disclosed
EP-2285882-A1 POLYMER MICROGEL BEADS THE UNIVERSITY OF SYDNEY (AU) 2011-02-23 EP disclosed
EP-2287167-A1 Polycyclic agents for the treatment of respiratory syncytial virus infections BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2011-02-23 EP disclosed
EP-2285784-A1 1-(ARYLSULFONYL)-4-(PIPERAZIN-1-YL)-1H-BENZIMIDAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS Wyeth LLC (US) 2011-02-23 EP disclosed
EP-2285881-A1 POLYMER MICROGEL BEADS AND PREPARATIVE METHOD THEREOF THE UNIVERSITY OF SYDNEY (AU) 2011-02-23 EP disclosed
WO-2011019737-A1 PYRIMIDO-PYRROLO-QUINOXALINEDIONE INHIBITORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR PROTEIN AND USES THEREFOR THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2011-02-17 WO disclosed
US-20110039467-A1 Ionic liquid flame retardants H&C Chemical (US) 2011-02-17 US disclosed
EP-1615866-B1 INDENE DERIVATIVES AS PHARMACEUTICAL AGENTS AQUINOX PHARMACEUTICALS INC (CA) 2011-02-16 EP disclosed
EP-2282981-A1 {F-19} -LABELED L-GLUTAMIC ACID AND L-GLUTAMINE DERIVATIVE (III), USE THEREOF AND METHOD FOR OBTAINING THEM Bayer Schering Pharma Aktiengesellschaft (DE) 2011-02-16 EP disclosed
US-20110034500-A1 SPIROHETEROCYCLIC COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2011-02-10 US disclosed
EP-1379508-B9 N-(ARYL)-2-ARYLETHENESULFONAMIDES AND THERAPEUTIC USES THEREOF UNIV TEMPLE (US) 2011-02-09 EP disclosed
US-7884119-B2 protein tyrosine kinase receptor inhibitors such as 3-amino -1-(1H-indol-5-yl)carbonyl-5-[4-2-(pyrrolidin-1-yl)ethoxy]phenylamino]-1H-1,2,4-triazole, used for treating diseases and conditions associated with neovascularization and/or cell proliferation RIGEL PHARMACEUTICALS, INC. (US) 2011-02-08 US disclosed
US-20110028437-A1 PHOSPHORYLATED PYRONE ANALOGS AND METHODS LIMERICK BIOPHARMA, INC. (US) 2011-02-03 US disclosed
WO-2011014888-A1 NOVEL HEDGEHOG INHIBITORS SELEXAGEN THERAPEUTICS (US) 2011-02-03 WO disclosed
EP-2279174-A2 ARYLSULFONAMIDE COMPOUNDS, COMPOSITIONS AND METHODS OF USE Genentech, Inc. (US) 2011-02-02 EP disclosed
US-7879856-B2 5-(quinoxalin-2-yl)-N2-(3,4,5-trimethoxyphenyl)thiazole-2,4-diamine; useful in inhibiting the activity of the receptor protein tyrosine kinase Axl; rheumatoid arthritis, vascular disease, vascular injury, psoriasis, visual impairment due to macular degeneration, diabetic retinopathy, retinopathy RIGEL PHARMACEUTICALS, INC. (US) 2011-02-01 US disclosed
US-20110021577-A1 ARYLOXY AMINE COMPOUNDS AND THEIR USE AS SODIUM CHANNEL MODULATORS HOWARD FLOREY INSTITUTE (AU) 2011-01-27 US disclosed
US-20110020731-A1 POLYMER ELECTROLYTE COMPOSITION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2011-01-27 US disclosed
US-20110021563-A1 INSULIN-REGULATED AMINOPEPTIDASE (IRAP) INHIBITORS AND USES THEREOF HOWARD FLOREY INSTITUTE (AU) 2011-01-27 US disclosed
US-20110021506-A1 ANTHELMINTIC AGENTS AND THEIR USE INTERVET INTERNATIONAL B.V. (NL) 2011-01-27 US disclosed
US-20110021530-A1 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS IN THE TREATMENT OF SKIN DISORDERS XENON PHARMACEUTICALS INC. (CA) 2011-01-27 US disclosed
EP-2277848-A1 Indene derivatives as pharmaceutical agents Aquinox Pharmaceuticals Inc. (CA) 2011-01-26 EP disclosed
EP-1697377-B1 POLYCYCLIC AGENTS FOR THE TREATMENT OF RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENT MANAGEMENT (AU) 2011-01-26 EP disclosed
EP-2094663-B1 PYRIDINE DERIVATIVES FOR THE TREATMENT OF METABOLIC DISORDERS RELATED TO INSULIN RESISTANCE OR HYPERGLYCEMIA PIRAMAL LIFE SCIENCES LTD (IN) 2011-01-26 EP disclosed
EP-1572660-B1 ISOQUINOLINONE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS X CEPTOR THERAPEUTICS INC (US) 2011-01-26 EP disclosed
US-7875728-B2 tert-butyl-[5-methyl-4-(phenylhydrazono)-4H-pyrazol-3-yl]amine; 4-(3-fluorophenylhydrazono)-5-methyl-2H-pyrazol-3-ylamine; demonstrate anti-proliferative activity, and may promote apoptosis in cells lacking normal regulation of cell cycle and death Valocor Therapeutics, Inc. (CA) 2011-01-25 US disclosed
US-7875631-B2 e.g.1-(3,5-dichlorophenyl)-2-formyl-6-methoxy-1,2,3,4-tetrahydroisoquinoline; to prevent and/or treat cancer and other abnormal cell growth, and metabolic as well as blood vessel proliferate disorders, in which uncontrolled expression of insulin-like growth factor-1 receptor is observed ANALYTECON S.A. (CH) 2011-01-25 US disclosed
WO-2011008302-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE, INC. (US) 2011-01-20 WO disclosed
WO-2011006208-A1 ANTI -INFLUENZA AGENTS GRIFFITH UNIVERSITY (AU) 2011-01-20 WO disclosed
US-20110015173-A1 PYRROLOPYRIDINE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2011-01-20 US disclosed
WO-2011006621-A1 RADIOLABELLING METHOD USING CYCLOALKYL GROUPS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-01-20 WO disclosed
US-20110015172-A1 PYRROLOPYRAZINE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2011-01-20 US disclosed
EP-1608623-B1 METAL ION CHELATORS AND THERAPEUTIC USE THEREOF RICHARDSON DESI RAYMOND (AU) 2011-01-19 EP disclosed
US-7872000-B2 angiogenesis and/or cell proliferation, carcinoma, myeloid leukemia, endometriosis; inhibitors of the receptor protein tyrosine kinase; N3-(3-cyclopentyl-1,2,3,4,5,6-hexahydrobenzo[d]azocin-8-yl)-1-(6-fluoroquinazolin-4-yl)-1H-1,2,4-triazole-3,5-diamine RIGEL PHARMACEUTICALS, INC. (US) 2011-01-18 US disclosed
US-20110009439-A1 INDENE DERIVATIVES AS PHARMACEUTICAL AGENTS AQUINOX PHARMACEUTICALS INC. (CA) 2011-01-13 US disclosed
US-20110009414-A9 HETEROCYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2011-01-13 US disclosed
EP-1827438-B1 PYRIDINE DERIVATIVES FOR INHIBITING HUMAN STEAROYL-COA-DESATURASE XENON PHARMACEUTICALS INC (CA) 2011-01-12 EP disclosed
CN-101945851-A Peptidyl nitriles and their use as dipeptidyl peptidase I inhibitors ASTRAZENECA AB 2011-01-12 CN disclosed
US-20110003895-A1 Pharmacology of Visual Cycle Modulators ACUCELA, INC. (US) 2011-01-06 US disclosed
US-20110003740-A1 INSULIN SENSITISERS AND METHODS OF TREATMENT VERVA PHARMACEUTICALS LTD. (AU) 2011-01-06 US disclosed
WO-2011003103-A2 PHARMACOLOGY OF VISUAL CYCLE MODULATORS ACUCELA, INC. (US) 2011-01-06 WO disclosed
EP-2269610-A2 Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors Xenon Pharmaceuticals Inc. (CA) 2011-01-05 EP disclosed
EP-2270104-A1 POLYMER ELECTROLYTE COMPOSITION Sumitomo Chemical Company, Limited (JP) 2011-01-05 EP disclosed
EP-2268623-A1 QUINAZOLINE DERIVATIVES AS RAF KINASE MODULATORS AND METHODS OF USE THEREOF Ambit Biosciences Corporation (US) 2011-01-05 EP disclosed
US-7863298-B2 Bridged ring structures as pharmaceutical agents EXELIXIS, INC. (US) 2011-01-04 US disclosed
US-20100331295-A1 MODULATORS OF LXR EXELIXIS, INC. (US) 2010-12-30 US disclosed
US-20100330155-A1 METHODS AND COMPOSITIONS FOR IMPROVED THERAPEUTIC EFFECTS WITH siRNA FLAGSHIP VENTURES (US) 2010-12-30 US disclosed
EP-2266566-A2 Nicotinamide derivatives and their use as therapeutic agents Xenon Pharmaceuticals Inc. (CA) 2010-12-29 EP disclosed
EP-2265607-A1 PYRIMIDINE-2-AMINE COMPOUNDS AND THEIR USE AS INHIBITORS OF JAK KINASES Rigel Pharmaceuticals, Inc. (US) 2010-12-29 EP disclosed
EP-2266569-A2 Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors Xenon Pharmaceuticals Inc. (CA) 2010-12-29 EP disclosed
EP-2265654-A1 POLYURETHANES Commonwealth Scientific and Industrial Research Organisation (AU) 2010-12-29 EP disclosed
EP-2265661-A1 CONDENSATION POLYMERS WITH MODIFIED PROPERTIES Commonwealth Scientific and Industrial Research Organisation (AU) 2010-12-29 EP disclosed
US-7858827-B2 Process for synthesis of dialkoxyorganoboranes BASF SE (DE) 2010-12-28 US disclosed
WO-2010147836-A1 COMBINATION THERAPIES USING ANTIBACTERIAL AMINOGLYCOSIDE COMPOUNDS ACHAOGEN, INC. (US) 2010-12-23 WO disclosed
US-20100323981-A1 TREATMENT OF STATIN SIDE EFFECTS MAGRAL LIMITED (AU) 2010-12-23 US disclosed
EP-2078723-B1 Process for synthesis of organo-oxazaborolidines BASF SE (DE) 2010-12-22 EP disclosed
EP-2262797-A1 INSULIN-REGULATED AMINOPEPTIDASE (IRAP) INHIBITORS AND USES THEREOF Howard Florey Institute (AU) 2010-12-22 EP disclosed
CN-101925584-A Pyrimidine Derivatives for the Treatment of Asthma, COPD, Allergic Rhinitis, Allergic Conjunctivitis, Atopic Dermatitis, Cancer, Hepatitis B, Hepatitis C, HIV, HPV, Bacterial Infections and Skin Diseases ASTRAZENECA AB 2010-12-22 CN disclosed
WO-2010144059-A2 NOVEL USES NANYANG POLYTECHNIC (SG) 2010-12-16 WO disclosed
WO-2010144055-A1 NOVEL COMPOUNDS AND USES THEREOF NANYANG POLYTECHNIC (SG) 2010-12-16 WO disclosed
US-20100317680-A1 PYRIMIDINE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2010-12-16 US disclosed
US-20100317568-A1 Anti-Viral Compounds Abbott Labaoratories (US) 2010-12-16 US disclosed
WO-2010144646-A2 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2010-12-16 WO disclosed
WO-2010144468-A1 2- ( LH-PYRAZOL-4 -YLAMINO ) -PYRIMIDINE AS KINASE INHIBITORS ABBOTT LABORATORIES (US) 2010-12-16 WO disclosed
US-20100317659-A1 JAK KINASE MODULATING COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORP. 2010-12-16 US disclosed
CN-101917980-A Amine derivative compounds for the treatment of ophthalmic diseases and disorders ACUCELA INC 2010-12-15 CN disclosed
CN-101918369-A Uracil or thymine derivatives for the treatment of hepatitis C ABBOTT LAB 2010-12-15 CN disclosed
US-20100311763-A1 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS NOVARTIS PHARMA AG (US) 2010-12-09 US disclosed
US-20100311721-A1 COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-12-09 US disclosed
EP-2257291-A2 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS IN THE TREATMENT OF SKIN DISORDERS Xenon Pharmaceuticals Inc. (CA) 2010-12-08 EP disclosed
US-7847101-B2 such as (4-Benzothiazol-2-yl-1H-pyrazol-3-yl)-[2-(1H-imidazol-4-yl)-ethyl]-amine, used in the treatment of disorders associated with hyperproliferation and tissue remodelling or repair, inflammation, cell migration and invasion, and renal diseases, or as protein kinase inhibitors Valocor Therapeutics, Inc. (CA) 2010-12-07 US disclosed
US-20100305099-A1 DIAMINOPYRIDINES FOR THE TREATMENT OF DISEASES WHICH ARE CHARACTERISED BY EXCESSIVE OR ANOMAL CELL PROLIFERATION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-12-02 US disclosed
US-20100305138-A1 PYRIDYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2010-12-02 US disclosed
WO-2010136559-A1 2, 4 -DIAMINOPYRIMIDINES FOR THE TREATMENT OF DISEASES CHARACTERISED BY EXCESSIVE OR ABNORMAL CELL PROLIFERATION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-12-02 WO disclosed
US-7842661-B2 Glycopegylated erythropoietin formulations NOVO NORDISK A/S (DK) 2010-11-30 US disclosed
US-7842743-B2 Stabiliser composition for halide-containing polymers SUN ACE KAKOH (PTE.) LTD. (SG) 2010-11-30 US disclosed
US-7842681-B2 Treatment of myeoproliferative diseases ABBOTT LABORATORIES (US) 2010-11-30 US disclosed
US-20100297077-A1 NOVEL ARYL POTASSIUM CHANNEL BLOCKERS AND USES THEREOF BIONOMICS LIMITED (AU) 2010-11-25 US disclosed
US-20100297020-A1 PHOSPHORYLATED AND PHOSPHONATED PYRONE ANALOGS FOR THERAPEUTIC TREATMENT LIMERICK BIOPHARMA, INC. (US) 2010-11-25 US disclosed
US-20100298313-A1 METHOD OF USING IMIDAZOLOTHIAZOLE COMPOUNDS FOR THE TREATMENT OF DISEASE AMBIT BIOSCIENCES CORPORATION 2010-11-25 US disclosed
US-20100297508-A1 Organic electrolytic solution and lithium battery employing the same SAMSUNG SDI CO., LTD. (KR) 2010-11-25 US disclosed
US-20100297046-A1 Compositions and Methods Related to Fructosamine-3-Kinase Inhibitors DYNAMIS THERAPEUTICS, INC. (US) 2010-11-25 US disclosed
WO-2010132765-A2 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010132770-A1 TREATMENT OF KLEBSIELLA PNEUMONIAE INFECTIONS WITH ANTIBACTERIAL AMINOGLYCOSIDE COMPOUNDS ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010132777-A2 TREATMENT OF URINARY TRACT INFECTIONS WITH ANTIBACTERIAL AMINOGLYCOSIDE COMPOUNDS ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010132839-A2 AMINOGLYCOSIDE DOSING REGIMENS ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010132760-A1 ANTIBACTERIAL DERIVATIVES OF TOBRAMYCIN ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010132759-A1 ANTIBACTERIAL DERIVATIVES OF DIBEKACIN ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
WO-2010132757-A2 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
US-20100292177-A1 Methods of treatment using combination therapy AMBIT BIOSCIENCES CORP. 2010-11-18 US disclosed
US-20100292342-A1 Compounds with (substituted phenyl)-propenal moiety, their derivatives, biological activity, and use thereof Annji Pharmaceutical Co., Ltd. (TW) 2010-11-18 US disclosed
WO-2010132352-A2 SPIRO COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2010-11-18 WO disclosed
WO-2010132768-A1 ANTIBACTERIAL DERIVATIVES OF SISOMICIN ACHAOGEN, INC. (US) 2010-11-18 WO disclosed
EP-2250171-A2 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS Achaogen, Inc. (US) 2010-11-17 EP disclosed
CN-101888989-A Novel aryl potassium channel blockers and uses thereof BIONOMICS LTD 2010-11-17 CN disclosed
CN-101889017-A Alkoxy compounds for the treatment of diseases ACUCELA INC 2010-11-17 CN disclosed
US-20100286094-A1 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF CHOONGWAE PHARMA CORPORATION (KR) 2010-11-11 US disclosed
WO-2007143597-A9 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2010-11-11 WO disclosed
US-20100285374-A1 Electrolytic solution and lithium battery employing the same SAMSUNG SDI CO., LTD. (KR) 2010-11-11 US disclosed
WO-2010129816-A2 HETEROCYCLIC COMPOUNDS AND USES THEREOF INTELLIKINE, INC. (US) 2010-11-11 WO disclosed
EP-1996217-B1 NOVEL ANTIBIOTIC COMPOSITIONS CAMBRIDGE ENTPR LTD (GB) 2010-11-10 EP disclosed
CN-101883778-A Steroidal [3, 2-C] pyrazole compounds, with glucocorticoid activity ASTRAZENECA AB 2010-11-10 CN disclosed
US-7829712-B2 Pyridazine derivatives for inhibiting human stearoyl-CoA-desaturase XENON PHARMACEUTICALS INC. (CA) 2010-11-09 US disclosed
US-20100279311-A1 METHOD FOR SCREENING OF CELL-PROTECTING AGENT TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-11-04 US disclosed
US-20100280012-A1 AZAAZULENE COMPOUNDS INDUSTRIAL TECHNOLOGY RESEARCH INSTITUTE (TW) 2010-11-04 US disclosed
US-20100280061-A1 NOVEL ANALGESIC THAT BINDS FILAMIN A BARBIER LINDSAY BURNS 2010-11-04 US disclosed
US-20100279996-A1 NOVEL ANALGESIC THAT BINDS FILAMIN A BARBIER LINDSAY BURNS 2010-11-04 US disclosed
US-20100280057-A1 NOVEL ANALGESIC THAT BINDS FILAMIN A BURNS BARBIER LINDSAY 2010-11-04 US disclosed
US-20100279997-A1 ANALGESIC THAT BINDS FILAMIN A PAIN THERAPEUTICS 2010-11-04 US disclosed
WO-2010124648-A1 AZAAZULENE COMPOUNDS INDUSTRIAL TECHNOLOGY RESEARCH INSTITUTE (CN) 2010-11-04 WO disclosed
WO-2010124826-A1 SUBSTITUTED IMIDAZOQUINOXALINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-11-04 WO disclosed
EP-1916889-B1 METHODS OF ALTERING POPPY CHARACTERISTICS GLAXOSMITHKLINE AUSTRALIA PTY (AU) 2010-11-03 EP disclosed
EP-2029572-B1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2010-11-03 EP disclosed
WO-2010123997-A1 CARBACEPHEM BETA-LACTAM ANTIBIOTICS ACHAOGEN, INC. (US) 2010-10-28 WO disclosed
US-7820657-B2 receptor kinase inhibitors such as 3-(2-{4-[3-(5-tert-Butyl-isoxazol-3-yl)-ureido]-phenyl}-benzo[d]imidazo[2,1-b]thiazol-7-yl)-N-(2-morpholin-4-yl-ethyl)-propionamide; flk inhibitors AMBIT BIOSCIENCES CORPORATION (US) 2010-10-26 US disclosed
US-20100267634-A1 Anti-Viral Compounds Abbott Labaoratories (US) 2010-10-21 US disclosed
US-20100267686-A1 CARBACEPHEM BETA-LACTAM ANTIBIOTICS ACHAOGEN, INC. (US) 2010-10-21 US disclosed
WO-2010118471-A1 REACTOR AND METHOD FOR PERFORMING A CHEMICAL REACTION THE UNIVERSITY OF QUEENSLAND (AU) 2010-10-21 WO disclosed
WO-2010118575-A1 RACEMIC ENANTIOMERS RESOLUTING CHENGDU ORGANIC CHEMICALS CO., LTD, CHINESE ACADEMY OF SCIENCE (CN) 2010-10-21 WO disclosed
WO-2010120935-A1 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2010-10-21 WO disclosed
EP-2240451-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS Intellikine, Inc. (US) 2010-10-20 EP disclosed
EP-2240452-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS Intellikine, Inc. (US) 2010-10-20 EP disclosed
US-20100256139-A1 Anti-Viral Compounds ABBOTT LABORATORIES (US) 2010-10-07 US disclosed
US-20100256105-A1 NOVEL COMPOUNDS ASTRAZENECA R&D 2010-10-07 US disclosed
US-20100256104-A1 NOVEL AMIDE COMPOUNDS ASTRAZENECA R&D (SE) 2010-10-07 US disclosed
WO-2010111172-A1 METHODS OF TREATMENT USING COMBINATION THERAPY AMBIT BIOSCIENCES CORPORATION (US) 2010-09-30 WO disclosed
EP-2231620-A1 DIAMINOPYRIDINES FOR THE TREATMENT OF DISEASES WHICH ARE CHARACTERISED BY EXCESSIVE OR ANOMAL CELL PROLIFERATION Boehringer Ingelheim International GmbH (DE) 2010-09-29 EP disclosed
US-20100240662-A1 REVERSE-TURN MIMETICS AND METHOD RELATING THERETO CHOONGWAE PHARMA CORPORATION (KR) 2010-09-23 US disclosed
WO-2010106097-A1 SUBSTITUTED PYRIMIDINES FOR THE TREATMENT OF CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-23 WO disclosed
US-20100240715-A1 Apoptosis promoters ABBOTT LABORATORIES 2010-09-23 US disclosed
US-20100240536-A1 PYRIMIDIN-4-YLPROPANEDINITRILE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2010-09-23 US disclosed
US-20100240657-A1 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-23 US disclosed
US-20100239520-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2010-09-23 US disclosed
US-20100240713-A1 AROMATIC AND HETEROAROMATIC COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2010-09-23 US disclosed
EP-2229813-A1 Pyrimidine-4-ylpropandinitrile derivatives, method for their manufacture and their use as herbicides and plant growth regulators Bayer CropScience AG (DE) 2010-09-22 EP disclosed
CN-101842360-A Anti-infective pyrimidines and uses thereof ABBOTT LAB 2010-09-22 CN disclosed
US-7799798-B2 Spiroheterocyclic compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2010-09-21 US disclosed
US-20100233116-A1 ORGANIC COMPOUNDS XENON PHARMACEUTICALS INC. (CA) 2010-09-16 US disclosed
US-20100234456-A1 APOPTOSIS PROMOTERS ABBOTT LABORATORIES (US) 2010-09-16 US disclosed
US-20100228027-A1 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF (2) CHOONGWAE PHARMA CORPORATION (KR) 2010-09-09 US disclosed
EP-2226632-A1 METHOD FOR SCREENING OF CELL-PROTECTING AGENT Takeda Pharmaceutical Company Limited (JP) 2010-09-08 EP disclosed
WO-2010096867-A1 POLYMER PARTICLES THE UNIVERSITY OF SYDNEY (AU) 2010-09-02 WO disclosed
US-20100222303-A1 REVERSE-TURN MIMETICS AND METHOD RELATING THERETO CHOONGWAE PHARMA CORPORATION (KR) 2010-09-02 US disclosed
WO-2010099379-A1 JAK KINASE MODULATING QUINAZOLINE DERIVATIVES AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2010-09-02 WO disclosed
US-20100222331-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 US disclosed
EP-2222682-A1 IMIDAZO-THIAZOLE DERIVATIVES AS PROTEIN KINASE INHIBITORS Abbott Laboratories (US) 2010-09-01 EP disclosed
EP-1379508-B1 N-(ARYL)-2-ARYLETHENESULFONAMIDES AND THERAPEUTIC USES THEREOF UNIV TEMPLE (US) 2010-09-01 EP disclosed
WO-2010094695-A1 PYRIMIDO [5,4-D] PYRIMIDINE DERIVATIVES FOR THE INHIBITION OF TYROSINE KINASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-08-26 WO disclosed
WO-2010096619-A1 PROCESS, PURIFICATION AND CRYSTALLIZATION OF 1-(4-{[4-(DIMETHYLAMINO)PIPERIDIN-1-YL]CARBONYL}PHENYL)-3-[4-(4,6-DIMORPHOLIN-4-YL-1,3,5-TRIAZIN-2-YL)PHENYL]UREA WYETH LLC (US) 2010-08-26 WO disclosed
US-20100210644-A1 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-08-19 US disclosed
US-20100209345-A1 Fluorinated Ligands for Targeting Peripheral Benzodiazepine Receptors AUSTRALIAN NUCLEAR SCIENCE & TECHNOLOGY ORGANISATION 2010-08-19 US disclosed
WO-2010093607-A1 COMPOUNDS AND METHODS FOR INHIBITING MMP2 AND MMP9 INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2010-08-19 WO disclosed
WO-2010091472-A1 SKIN TREATMENT PEPLIN RESEARCH PTY LTD (AU) 2010-08-19 WO disclosed
US-20100210630-A1 Diamine Derivatives as Inhibitors of Leukotriene A4 Hydrolase ESTRELLITA PHARMACEUTICALS, LLC 2010-08-19 US disclosed
EP-2217265-A2 MODIFIED INSULIN POLYPEPTIDES AND THEIR USES Ambrx, Inc. (US) 2010-08-18 EP disclosed
EP-2217610-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS Achaogen, Inc. (US) 2010-08-18 EP disclosed
US-7777036-B2 Heterocyclic derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2010-08-17 US disclosed
US-7777076-B2 Macrocyclic inhibitors of BCL proteins ABBOTT LABORATORIES (US) 2010-08-17 US disclosed
US-20100204318-A1 TREATMENT OF VIRALLY INDUCED LESIONS PEPLIN RESEARCH PTY LTD (AU) 2010-08-12 US disclosed
US-20100204089-A1 PHOSPHORYLATED PYRONE ANALOGS AND METHODS LIMERICK BIOPHARMA, INC. 2010-08-12 US disclosed
CN-101801935-A Uracil or thymine derivatives for the treatment of hepatitis C ABBOTT LAB 2010-08-11 CN disclosed
CN-101801375-A Insulin sensitisers and methods of treatment VERVA PHARMACEUTICALS LTD 2010-08-11 CN disclosed
US-7772231-B2 Substituted pyrazolo[3,4-d]pyrimidines as protein kinase inhibitors ABBOTT LABORATORIES (US) 2010-08-10 US disclosed
US-20100196511-A1 AXL INHIBITORS FOR USE IN COMBINATION THERAPY FOR PREVENTING, TREATING OR MANAGING METASTATIC CANCER RIGEL PHARMACEUTICALS, INC. (US) 2010-08-05 US disclosed
US-20100197501-A1 SUBSTITUTED 1-(THIAZOLYL)-AND 1-(ISOTHIAZOLYL)PYRAZOL-4-YLACETIC ACIDS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2010-08-05 US disclosed
EP-2212330-A2 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF (3) Choongwae Pharma Corporation (KR) 2010-08-04 EP disclosed
EP-2212329-A2 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF (1) Choongwae Pharma Corporation (KR) 2010-08-04 EP disclosed
EP-2212328-A2 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF (2) Choongwae Pharma Corporation (KR) 2010-08-04 EP disclosed
US-7767684-B2 Apoptosis promoters ABBOTT LABORATORIES (US) 2010-08-03 US disclosed
US-7767677-B2 Heterocyclic derivatives and their use as stearoyl-CoA desaturase inhibitors XENON PHARMACEUTICALS INC. (CA) 2010-08-03 US disclosed
US-20100189653-A1 Pyrone analogs for therapeutic treatment LIMERICK BIOPHARMA, INC. 2010-07-29 US disclosed
US-20100190749-A1 Benzoxazole kinase inhibitors and methods of use FAETH THERAPEUTICS, INC. 2010-07-29 US disclosed
EP-2210892-A2 Neurologically-active compounds Prana Biotechnology Limited (AU) 2010-07-28 EP disclosed
EP-1979349-B1 ANTI-VIRAL COMPOUNDS ABBOTT LAB (US) 2010-07-28 EP disclosed
US-7763731-B2 Anti-viral compounds ABBOTT LABORATORIES (US) 2010-07-27 US disclosed
US-7763618-B2 1-Pentyl-3-{6-[4-(2-trifluoromethylbenzoyl)piperazin-1-yl]-pyridin-3-yl}urea; inhibitors of stearoyl-CoA desaturase; cardiovascular disease, diabetes, obesity, metabolic syndrome XENON PHARMACEUTICALS INC. (CA) 2010-07-27 US disclosed
US-20100184747-A1 INDOLINE DERIVATIVES AND THEIR USE IN TREATING DISEASE-STATES SUCH AS CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-07-22 US disclosed
US-20100183743-A1 BENZTHIAZOLE INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE ABBOTT LABORATORIES (US) 2010-07-22 US disclosed
WO-2010083465-A1 AXL INHIBITORS FOR USE IN COMBINATION THERAPY FOR PREVENTING, TREATING OR MANAGING METASTATIC CANCER RIGEL PHARMACEUTICALS, INC. (US) 2010-07-22 WO disclosed
US-20100184607-A1 MONOSACCHARIDE COMPOUNDS AND METHODS THEREFOR ALCHEMIA PTY LTD. (AU) 2010-07-22 US disclosed
US-20100184760-A1 Benzoxazole kinase inhibitors and methods of use FAETH THERAPEUTICS, INC. 2010-07-22 US disclosed
CN-101784188-A Alkynyl phenyl derivative compounds for the treatment of ophthalmic diseases and disorders ACUCELA INC 2010-07-21 CN disclosed
US-7759348-B2 Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2010-07-20 US disclosed
EP-2205600-A1 CARBACEPHEM ß -LACTAM ANTIBIOTICS Achaogen, Inc. (US) 2010-07-14 EP disclosed
EP-2205592-A1 POLYCYCLIC ARYL SUBSTITUTED TRIAZOLES AND POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS Rigel Pharmaceuticals, Inc. (US) 2010-07-14 EP disclosed
US-7754711-B2 Antidiabetic agents; disease of glucose tolerance; insulin resistance; obesity; dyslipidemia; metabolic disorders; liver disorders XENON PHARMACEUTICALS INC. (CA) 2010-07-13 US disclosed
US-20100173967-A1 USE OF SPIRO-OXINDOLE COMPOUNDS AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2010-07-08 US disclosed
EP-2204373-A1 Phosphonic acid as Plasma Carboxypeptidase B Inhibitors Bayer Schering Pharma Aktiengesellschaft (DE) 2010-07-07 EP disclosed
EP-2203431-A1 ANTI-INFECTIVE PYRIMIDINES AND USES THEREOF Abbott Laboratories (US) 2010-07-07 EP disclosed
US-7750004-B2 Apoptosis promoters ABBOTT LABORATORIES (US) 2010-07-06 US disclosed
WO-2010072734-A2 TARGETING PRODRUGS AND COMPOSITIONS FOR THE TREATMENT OF GASTROINTESTINAL DISEASES THE PROVOST FELLOWS AND SCHOLARS OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2010-07-01 WO disclosed
US-20100168416-A1 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2010-07-01 US disclosed
US-20100168170-A1 Piperidinones Useful in the Treatment of Inflammation BIOLIPOX AB (SE) 2010-07-01 US disclosed
US-20100168384-A1 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2010-07-01 US disclosed
US-20100168138-A1 Anti-Viral Compounds ABBOTT LABORATORIES (US) 2010-07-01 US disclosed
US-20100168167-A1 Piperidinones Useful in the Treatment of Inflammation BIOLIPOX AB (SE) 2010-07-01 US disclosed
US-7744889-B2 Alpha, beta-unsaturated sulfoxides for treating proliferative disorders TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2010-06-29 US disclosed
US-7745553-B2 Aqueous dispersions of polymer particles UNIVERSITY OF SYDNEY (AU) 2010-06-29 US disclosed
US-20100160362-A1 SPIRO (FURO [3, 2-C] PYRIDINE-3-3' -INDOL) -2' (1'H)-ONE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF SODIUM-CHANNEL MEDIATED DISEASES, SUCH AS PAIN XENON PHARMACEUTICALS INC. (CA) 2010-06-24 US disclosed
WO-2010040345-A9 ECDYSONE DERIVATIVES AND THE USE THEREOF VERDEVITAL BERATUNGS-, IMPORT- UND VERTRIEBSGESELLSCHAFT MBH (DE) 2010-06-24 WO disclosed
US-20100160355-A1 Anti-Viral Compounds ABBOTT LABORATORIES (US) 2010-06-24 US disclosed
US-20100160164-A1 SUBSTITUTED 1-(DIAZINYL)PYRAZOL-4-YLACETIC ACIDS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2010-06-24 US disclosed
US-20100160291-A1 TRICYCLIC SPIRO-OXINDOLE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2010-06-24 US disclosed
US-20100160346-A1 NEUROLOGICALLY ACTIVE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED (AU) 2010-06-24 US disclosed
US-20100152220-A1 INDENE DERIVATIVES AS PHARMACEUTICAL AGENTS AQUINOX PHARMACEUTICALS INC. (CA) 2010-06-17 US disclosed
US-20100152187-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2010-06-17 US disclosed
CN-101742996-A Treatment of viral-induced lesions PEPLIN RESEARCH PTY LTD 2010-06-16 CN disclosed
US-7737159-B2 Antibacterial compounds ABBOTT LABORATORIES (US) 2010-06-15 US disclosed
US-7737145-B2 Diamine derivatives as inhibitors of leukotriene A4 hydrolase ESTRELLITA PHARMACEUTICALS, LLC (US) 2010-06-15 US disclosed
US-20100144612-A1 PHOSPHORYLATED PYRONE ANALOGS AND METHODS LIMERICK BIOPHARMA, INC. 2010-06-10 US disclosed
US-20100144693-A1 METHOD OF TREATMENT OF AGE-RELATED MACULAR DEGENERATION (AMD) PRANA BIOTECHNOLOGY LIMITED (AU) 2010-06-10 US disclosed
US-20100144665-A1 TREATMENT OF STATIN SIDE EFFECTS MAGRAL LIMITED (AU) 2010-06-10 US disclosed
EP-2194052-A1 Substituted 1.(1-thiazolyl)- and 1-(isothiazolyl)pyrazol-4-yl acetic acids, method for their production and their use as herbicides and plant growth regulators Bayer CropScience AG (DE) 2010-06-09 EP disclosed
CN-101723949-A Polycyclic agents for the treatment of respiratory syncytial virus infections BIOTA SCIENT MAN 2010-06-09 CN disclosed
US-20100137299-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2010-06-03 US disclosed
WO-2010058030-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-05-27 WO disclosed
WO-2010058032-A2 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-05-27 WO disclosed
WO-2010059593-A1 METHODS AND COMPOSITIONS FOR TREATMENT OF OPHTHALMIC CONDITIONS INTELLIKINE, INC. (US) 2010-05-27 WO disclosed
US-20100130457-A1 Phenothiazine Derivatives for Treatment of Asthma IMMUNE CONTROL, INC. 2010-05-27 US disclosed
US-20100130487-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2010-05-27 US disclosed
US-20100130713-A1 FURANONE COPOLYMERS COVIDIEN LP 2010-05-27 US disclosed
US-20100130555-A1 COMPOSITIONS AND METHODS FOR TREATING OR PREVENTING HYPOXIC OR ISCHEMIC INJURY IKARIA, INC. (US) 2010-05-27 US disclosed
WO-2010056644-A1 1- (ARYLSULFONYL) -4- (PI PERAZIN-I -YL) -IH-BENZ IMIDAZOLES AS δ-HYDROXYTRYPTAMINE- 6 LIGANDS WYETH LLC (US) 2010-05-20 WO disclosed
WO-2010055117-A1 2,4-DIAMINOPYRIMIDINE DERIVATES AS PTK2- INHIBITORS FOR THE TREATMENT OF ABNORMAL CELL GROWTH BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-05-20 WO disclosed
US-20100125072-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2010-05-20 US disclosed
WO-2010056979-A1 PHENOTHIAZINE DERIVATIVES FOR TREATMENT OF ASTHMA IMMUNE CONTROL, INC. (US) 2010-05-20 WO disclosed
WO-2010053998-A1 SPIRO-CONDENSED INDOLE DERIVATIVES AS SODIUM CHANNEL INHIBITORS XENON PHARMACEUTICALS, INC. (CA) 2010-05-14 WO disclosed
US-20100120779-A1 1-(ARYLSULFONYL)-4-(PIPERAZIN-1-YL)-1H-BENZIMIDAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS WYETH (US) 2010-05-13 US disclosed
US-20100119695-A1 ANTIMICROBIAL MATERIALS AND COATINGS COVIDIEN LP 2010-05-13 US disclosed
EP-2182957-A2 PHOSPHORYLATED PYRONE ANALOGS AND METHODS Limerick BioPharma, Inc. (US) 2010-05-12 EP disclosed
EP-2182801-A1 PYRONE ANALOG COMPOSITIONS AND METHODS Limerick BioPharma, Inc. (US) 2010-05-12 EP disclosed
WO-2010051497-A1 FILAMIN A BINDING ANTI-INFLAMMATORY AND ANALGESIC PAIN THERAPEUTICS, INC. (US) 2010-05-06 WO disclosed
WO-2010051374-A1 ANALGESIC THAT BINDS FILAMIN A PAIN THERAPEUTICS, INC. (US) 2010-05-06 WO disclosed
US-20100113539-A1 COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2010-05-06 US disclosed
WO-2010051476-A1 FILAMIN A-BINDING ANTI-INFLAMMATORY ANALGESIC PAIN THERAPEUTICS, INC. (US) 2010-05-06 WO disclosed
EP-2181108-A2 3-HETROCYCLYLIDENE-INDOLINONE DERIVATIVES AS INHIBITORS OF SPECIFIC CELL CYCLE KINASES Boehringer Ingelheim International GmbH (DE) 2010-05-05 EP disclosed
US-7709482-B2 angiogenesis and/or cell proliferation, carcinoma, myeloid leukemia, endometriosis; inhibitors of the receptor protein tyrosine kinase; N3-(3-cyclopentyl-1,2,3,4,5,6-hexahydrobenzo[d]azocin-8-yl)-1-(6-fluoroquinazolin-4-yl)-1H-1,2,4-triazole-3,5-diamine RIGEL PHARMACEUTICALS, INC. (US) 2010-05-04 US disclosed
US-20100105685-A1 S-Nitrosothiol Compounds and Related Derivatives GALLEON PHARMACEUTICALS, INC. 2010-04-29 US disclosed
WO-2010048332-A2 COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2010-04-29 WO disclosed
WO-2010045251-A2 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS, INC. (CA) 2010-04-22 WO disclosed
US-20100099728-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2010-04-22 US disclosed
US-20100099661-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2010-04-22 US disclosed
WO-2010045197-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS, INC. (CA) 2010-04-22 WO disclosed
WO-2010045582-A2 COMPOSITIONS AND METHODS FOR TREATING OR PREVENTING HYPOXIC OR ISCHEMIC INJURY IKARIA, INC. (US) 2010-04-22 WO disclosed
EP-2177226-A1 Hydroxamate compositions Tyco Healthcare Group LP (US) 2010-04-21 EP disclosed
EP-2177554-A2 Hydroxamate-initiated polymers Tyco Healthcare Group LP (US) 2010-04-21 EP disclosed
EP-2176249-A2 NEW CHEMICAL COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-04-21 EP disclosed
EP-2177552-A1 Bioabsorbable surgical composition Tyco Healthcare Group LP (US) 2010-04-21 EP disclosed
EP-2177235-A2 Coating compositions Tyco Healthcare Group LP (US) 2010-04-21 EP disclosed
US-7700641-B2 Spiro-oxindole compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2010-04-20 US disclosed
US-20100093865-A1 SULPHUR-LINKED COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2010-04-15 US disclosed
WO-2010040187-A1 POLYMER-BIOACTIVE AGENT CONJUGATES THE BIONIC EAR INSTITUTE (AU) 2010-04-15 WO disclosed
US-20100093846-A1 HYDROXAMATE COMPOSITIONS TYCO HEALTHCARE GROUP LP 2010-04-15 US disclosed
WO-2010040345-A2 ECDYSONE DERIVATIVES AND THE USE THEREOF VERDEVITAL BERATUNGS-, IMPORT- UND VERTRIEBSGESELLSCHAFT MBH (DE) 2010-04-15 WO disclosed
US-20100094338-A1 HYDROXAMATE-INITIATED POLYMERS TYCO HEALTHCARE GROUP LP 2010-04-15 US disclosed
US-20100092533-A1 Bioabsorbable Surgical Composition COVIDIEN LP 2010-04-15 US disclosed
US-20100094340-A1 COATING COMPOSITIONS TYCO HEALTHCARE GROUP LP 2010-04-15 US disclosed
WO-2010042851-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2010-04-15 WO disclosed
WO-2010042886-A2 PYRONE ANALOGS FOR THERAPEUTIC TREATMENT LIMERICK BIOPHARMA, INC. (US) 2010-04-15 WO disclosed
WO-2010042850-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2010-04-15 WO disclosed
EP-2173734-A2 CHEMICAL COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-04-14 EP disclosed
US-20100087443-A1 9-SUBSTITUTED-8-OXO-ADENINE COMPOUNDS AS TOLL-LIKE RECEPTOR (TLR7) MODULATORS ASTRAZENECA AB (SE) 2010-04-08 US disclosed
US-20100087430-A1 NOVEL BENZOFURAN POTASSIUM CHANNEL BLOCKERS AND USES THEREOF BIONOMICS LIMITED (AU) 2010-04-08 US disclosed
WO-2010037169-A1 PROCESS FOR EXTRACTION OF MINED MATERIAL THE UNIVERSITY OF QUEENSLAND (AU) 2010-04-08 WO disclosed
EP-2172457-A2 Fredericamycin derivatives Biofrontera Discovery Gmbh (DE) 2010-04-07 EP disclosed
EP-2170884-A2 CHEMICAL COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-04-07 EP disclosed
EP-2172491-A1 Polymer obtained by the use of RAFT-agents and process of encapsulating of particulate material by said polymer. The University of Sydney (AU) 2010-04-07 EP disclosed
US-7692011-B2 8-hydroxy and 8-mercapto quinazolinones PRANA BIOTECHNOLOGY LIMITED (AU) 2010-04-06 US disclosed
WO-2010036380-A1 HETEROCYCLIC KINASE INHIBITORS INTELLIKINE, INC. (US) 2010-04-01 WO disclosed
WO-2010034838-A2 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO disclosed
EP-2167465-A1 INDOLINONE DERIVATIVES AND THEIR USE IN TREATING DISEASE-STATES SUCH AS CANCER Boehringer Ingelheim International GmbH (DE) 2010-03-31 EP disclosed
CN-101686665-A styrenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC 2010-03-31 CN disclosed
WO-2009141090-A9 {F-19} -LABELED L-GLUTAMIC ACID AND L-GLUTAMINE DERIVATIVE (III), USE THEREOF AND METHOD FOR OBTAINING THEM BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-03-25 WO disclosed
US-20100075964-A1 IMIDAZOLE BASED LXR MODULATORS EXELIXIS, INC. (US) 2010-03-25 US disclosed
EP-1755373-B1 METHOD OF ALTERING THE ALKALOID COMPOSITION IN POPPY PLANTS GLAXOSMITHKLINE AUSTRALIA PTY (AU) 2010-03-24 EP disclosed
WO-2010030811-A2 CARBACEPHEM β-LACTAM ANTIBIOTICS ACHAOGEN, INC. (US) 2010-03-18 WO disclosed
US-20100069367-A1 LXR and FXR Modulators EXELIXIS, INC. (US) 2010-03-18 US disclosed
US-20100068204-A1 4-ARYLOXYQUINOLIN-2(1H)-ONES AS MTOR KINASE AND PI3 KINASE INHIBITORS, FOR USE AS ANTI-CANCER AGENTS WYETH (US) 2010-03-18 US disclosed
WO-2010028836-A1 BISTABLE CARBAZOLE COMPOUNDS STMICROELECTRONICS S.R.L. (IT) 2010-03-18 WO disclosed
WO-2010030810-A1 CARBACEPHEM BETA-LACTAM ANTIBIOTICS ACHAOGEN, INC. (US) 2010-03-18 WO disclosed
WO-2010030727-A1 3-SUBSTITUTED-1H-INDOLE, 3-SUBSTITUTED-1H-PYRROLO[2,3-B]PYRIDINE AND 3-SUBSTITUTED-1H-PYRROLO[3,2-B]PYRIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH LLC (US) 2010-03-18 WO disclosed
WO-2010030704-A2 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2010-03-18 WO disclosed
WO-2010030967-A1 4-ARYLOXYQUINOLIN-2(1H)-ONES AS MTOR KINASE AND PI3 KINASE INHIBITORS, FOR USE AS ANTI-CANCER AGENTS WYETH LLC (US) 2010-03-18 WO disclosed
WO-2010028088-A2 SULFUR-LINKED COMPOUNDS FOR TREATING OPTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2010-03-11 WO disclosed
US-20100059363-A1 SURFACE TREATMENT OF ALUMINA FILMS NATIONAL UNIVERSITY OF SINGAPORE (SG) 2010-03-11 US disclosed
US-20100061982-A1 3-SUBSTITUTED-1H-INDOLE, 3-SUBSTITUTED-1H-PYRROLO[2,3-B]PYRIDINE AND 3-SUBSTITUTED-1H-PYRROLO[3,2-B]PYRIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2010-03-11 US disclosed
WO-2010026262-A1 PYRIDO [5, 4-D] PYRIMIDINES AS CELL PROLIFERATION INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-03-11 WO disclosed
EP-2160192-A1 ANTIMICROBIAL MATERIALS AND COATINGS Tyco Healthcare Group LP (US) 2010-03-10 EP disclosed
EP-2160193-A1 FURANONE COPOLYMERS Tyco Healthcare Group LP (US) 2010-03-10 EP disclosed
US-7674569-B2 Optical recording material and optical recording medium ADEKA CORPORATION (JP) 2010-03-09 US disclosed
US-20100056582-A1 Modulators of LXR X-CEPTOR THERAPEUTICS, INC. (US) 2010-03-04 US disclosed
US-7671054-B1 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2010-03-02 US disclosed
WO-2010020008-A1 POLYMER COATINGS POLYMERS CRC LIMITED (AU) 2010-02-25 WO disclosed
US-20100048750-A1 VESICULATED POLYMER PARTICLES THE UNIVERSITY OF SYDNEY (AU) 2010-02-25 US disclosed
US-20100048584-A1 PYRIDYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2010-02-25 US disclosed
US-20100041613-A1 NOVEL ANTIBIOTIC COMPOSITIONS CAMBRIDGE ENTERPRISE LTD. (GB) 2010-02-18 US disclosed
EP-2152261-A1 TREATMENT OF VIRALLY INDUCED LESIONS Peplin Research Pty Ltd. (AU) 2010-02-17 EP disclosed
US-20100036123-A1 PROCESS FOR THE PREPARATION OF 2,4-DICHLORO-7H-PYRROLO[2,3H]QUINAZOLINE WYETH (US) 2010-02-11 US disclosed
US-20100035948-A1 Furanone compounds and lactam analogues thereof UNILEVER PLC (GB) 2010-02-11 US disclosed
US-20100035858-A1 Novel Compositions and Methods for Binding and Inhibiting 5-HT4 Receptor IMMUNE CONTROL, INC. 2010-02-11 US disclosed
WO-2010015037-A1 THERAPEUTIC METHODS AND COMPOSITIONS HOWARD FLOREY INSTITUTE (AU) 2010-02-11 WO disclosed
US-20100028368-A1 SULFIDE, SULFOXIDE AND SULFONE CHALCONE ANALOGUES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF TEMPLE UNIVERSITY- OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2010-02-04 US disclosed
US-20100029686-A1 HCV PROTEASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2010-02-04 US disclosed
US-20100029718-A1 ORGANIC COMPOUNDS NOVARTIS AG 2010-02-04 US disclosed
US-20100029722-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2010-02-04 US disclosed
WO-2010012747-A1 NEW COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-02-04 WO disclosed
US-20100021458-A1 POLYCYCLIC AGENTS FOR THE TREATMENT OF RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2010-01-28 US disclosed
US-20100022773-A1 APOPTOSIS PROMOTERS ABBVIE INC. 2010-01-28 US disclosed
US-20100022557-A1 RADIOPROTECTOR COMPOUNDS AND RELATED METHODS PETER MACCALLUM CANCER INSTITUTE (AU) 2010-01-28 US disclosed
WO-2010011620-A1 4-PHENOXY-6-ARYL-1H-PYRAZOLO[3,4-D]PYRIMIDINE AND N-ARYL-6-ARYL-1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2010-01-28 WO disclosed
EP-2147919-A1 Heterocyclic substituted amides, method for their manufacture and their use as herbicides Bayer CropScience Aktiengesellschaft (DE) 2010-01-27 EP disclosed
WO-2010007116-A2 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-21 WO disclosed
US-20100015136-A1 CAMPTOTHECIN-PEPTIDE CONJUGATES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME DIATOS, S.A. (FR) 2010-01-21 US disclosed
US-20100015141-A1 4-PHENOXY-6-ARYL-1H-PYRAZOLO[3,4-D]PYRIMIDINE AND N-ARYL-6-ARYL-1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2010-01-21 US disclosed
WO-2010007114-A2 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-21 WO disclosed
WO-2010006755-A2 A COMPOUND FOR IMAGING CELL DEATH BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-01-21 WO disclosed
EP-1675812-B1 BRIDGED RING STRUCTURES AS PHARMACEUTICAL AGENTS X CEPTOR THERAPEUTICS INC (US) 2010-01-20 EP disclosed
CN-101631788-A 8-alkynyl xanthine and derivative SANOL ARZNEI SCHWARZ GMBH 2010-01-20 CN disclosed
CN-100582109-C Polycyclic agents for the treatment of respiratory syncytial virus infection BIOTA SCIENT MAN 2010-01-20 CN disclosed
US-7648966-B2 Mannose-6-phosphonate compounds for the treatment of inflammatory diseases Pharmaxis Pty Limited (AU) 2010-01-19 US disclosed
WO-2010005876-A2 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2010-01-14 WO disclosed
WO-2010005851-A1 COMBINATION THERAPY FOR TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2010-01-14 WO disclosed
WO-2010006086-A2 KINASE INHIBITORS AND METHODS OF USE INTELLIKINE, INC. (US) 2010-01-14 WO disclosed
US-7645760-B2 1-(4-Benzyl-piperazin-1-yl)-3-phenyl-propenone derivatives NOVARTIS AG. (CH) 2010-01-12 US disclosed
WO-2010000019-A1 PAIN-RELIEVING COMPOSITIONS OF FUROXAN NO DONORS AND USES THEREOF THE UNIVERSITY OF QUEENSLAND (AU) 2010-01-07 WO disclosed
WO-2010000008-A1 THIOSEMICARBAZONE COMPOUNDS AND USE THEREOF RICHARDSON DESI RAYMOND (AU) 2010-01-07 WO disclosed
US-20100004333-A1 COMPOSITIONS AND METHODS FOR TREATING CARDIOVASCULAR DISORDERS STOCKER ROLAND O 2010-01-07 US disclosed
WO-2010002472-A1 JAK KINASE MODULATING COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2010-01-07 WO disclosed
EP-2139894-A1 9-SUBSTITUTED-8-OXO-ADENINE COMPOUNDS AS TOLL-LIKE RECEPTOR (TLR7) MODULATORS AstraZeneca AB (SE) 2010-01-06 EP disclosed
EP-2141163-A1 Substituted thiazolidinones, their production and utilisation as medicine Bayer Schering Pharma AG (DE) 2010-01-06 EP disclosed
US-7642260-B2 N-acylsulfonamide derivatives; BCL-X1 protein inhibitors; anticarcinogenic agents; bladder cancer; for example, N-(4-(4-((4'-chloro(1,1'-biphenyl)-2-yl)methyl)piperazin-1-yl)benzoyl)-4-(((1R)-3-(dimethylamino)-1-((phenylsulfanyl)methyl)-propyl)amino)-3-nitrobenzenesulfonamide ABBOTT LABORATORIES, INC. (US) 2010-01-05 US disclosed
US-20090326074-A1 Alkoxy compounds for disease treatment ACUCELA INC. (US) 2009-12-31 US disclosed
US-20090326017-A1 PAIN-RELIEVING COMPOSITIONS AND USES THEREFOR THE UNIVERSITY OF QUEENSLAND (AU) 2009-12-31 US disclosed
US-20090325906-A1 Methods and compositions for therapeutic treatment LIMERICK BIOPHARMA, INC. 2009-12-31 US disclosed
WO-2009156484-A2 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-12-30 WO disclosed
EP-2137150-A1 PIPERIDINONES USEFUL IN THE TREATMENT OF INFLAMMATION Biolipox AB (SE) 2009-12-30 EP disclosed
EP-2135865-A1 Substituted 1-(diazinyl)pyrazol-4-yl acetic acids, method for their production and their use as herbicides and plant growth regulators Bayer CropScience AG (DE) 2009-12-23 EP disclosed
EP-2134723-A1 9H- PURINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF PROLIFERATIVE DISEASES Boehringer Ingelheim International GmbH (DE) 2009-12-23 EP disclosed
EP-2134686-A1 PIPERIDINONES USEFUL IN THE TREATMENT OF INFLAMMATION Biolipox AB (SE) 2009-12-23 EP disclosed
US-20090312260-A1 DRUG THERAPY FOR CELIAC SPRUE THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2009-12-17 US disclosed
US-20090312319-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE 2009-12-17 US disclosed
WO-2009151920-A2 HEPSIN INHIBITORS FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2009-12-17 WO disclosed
US-20090312272-A1 Transglutaminase inhibitors and methods of use thereof THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY; AND THE WASHINGTON UNIVERSITY 2009-12-17 US disclosed
US-20090311176-A1 2-Arylpyrazolo[L,5-Alpha] Pyrimidin-3-YL Acetamide Derivatives as Ligands for Translocator Protein (18 Kda) THE UNIVERSITY OF SYDNEY (AU) 2009-12-17 US disclosed
US-7632946-B2 Naphthyridine-based antibacterial compositions ABBOTT LABORATORIES (US) 2009-12-15 US disclosed
US-20090306042-A1 Novel Compounds 010 ASTRAZENECA AB (SE) 2009-12-10 US disclosed
US-20090306373-A1 4,7-DIHYDROTHIENO[2,3-B]PYRIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS GILEAD COLORADO, INC. 2009-12-10 US disclosed
US-20090306090-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2009-12-10 US disclosed
CN-100567271-C 4,4 ' (5 ')-di-t-butyl hexamethylene also-the improvement purification process of hexaoxacyclooctadecane-6-6 PG RES FOUNDATION (US) 2009-12-09 CN disclosed
US-20090298931-A1 NOVEL CHROMENONE POTASSIUM CHANNEL BLOCKERS AND USES THEREOF BIONOMICS LIMITED (AU) 2009-12-03 US disclosed
US-7625579-B2 Antimicrobial coatings UNISEARCH LIMITED (AU) 2009-12-01 US disclosed
WO-2009141090-A1 {F-19} -LABELED L-GLUTAMIC ACID AND L-GLUTAMINE DERIVATIVE (III), USE THEREOF AND METHOD FOR OBTAINING THEM BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-11-26 WO disclosed
WO-2009143246-A2 ARYLSULFONAMIDE COMPOUNDS, COMPOSITIONS AND METHODS OF USE GENENTECH, INC. (US) 2009-11-26 WO disclosed
US-20090291957-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2009-11-26 US disclosed
EP-2121671-A1 2-SUBSTITUTED 5-MEMBERED HETEROCYCLES AS SCD INHIBITORS Novartis AG (CH) 2009-11-25 EP disclosed
EP-2121621-A1 LXR AND FXR MODULATORS Exelixis, Inc. (US) 2009-11-25 EP disclosed
EP-2121608-A1 DIHYDROPYRIDINE DERIVATIVES USEFUL AS PROTEIN KINASE INHIBITORS Bayer Schering Pharma AG (DE) 2009-11-25 EP disclosed
EP-2123620-A1 {F-19}-labeled L-Glutamic acid and L-Glutamine derivative (III), use thereof and method for obtaining them Bayer Schering Pharma Aktiengesellschaft (DE) 2009-11-25 EP disclosed
WO-2009137888-A1 POLYMER MICROGEL BEADS AND PREPARATIVE METHOD THEREOF THE UNIVERSITY OF SYDNEY (AU) 2009-11-19 WO disclosed
WO-2009137890-A1 ADMINISTRABLE COMPOSITIONS THE UNIVERSITY OF SYDNEY (AU) 2009-11-19 WO disclosed
WO-2009137889-A1 POLYMER MICROGEL BEADS THE UNIVERSITY OF SYDNEY (AU) 2009-11-19 WO disclosed
US-20090286835-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2009-11-19 US disclosed
CN-101583614-A Polycyclic agents for the treatment of respiratory syncytial virus infections BIOTA SCIENT MAN (AU) 2009-11-18 CN disclosed
US-7619091-B2 Treating nervous system disorders such as mild cognitive impairment, Alzheimer's disease or dementia associated with Down syndrome; e.g. use of 5,7-dichloro-8-hydroxy-2-(2-pyridyl)-quinoline (PBT 1052) PRANA BIOTECHNOLOGY LIMITED (AU) 2009-11-17 US disclosed
WO-2009137130-A2 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS ACHAOGEN, INC. (US) 2009-11-12 WO disclosed
US-20090281149-A1 Amine Derivative Compounds for Treating Ophthalmic Diseases and Disorders ACUCELA, INC. (US) 2009-11-12 US disclosed
US-20090281066-A1 Treatment of proliferative disorders with amino-substituted (E)-2,6- dialkoxystyryl 4-substituted benzylsulfones TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2009-11-12 US disclosed
EP-2114896-A1 RADIOPROTECTOR COMPOUNDS AND RELATED METHODS Peter MacCallum Cancer Institute (AU) 2009-11-11 EP disclosed
EP-2114954-A1 BICYCLIC ARYL AND BICYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS Rigel Pharmaceuticals, Inc. (US) 2009-11-11 EP disclosed
WO-2009133045-A1 NEW BORANE-AMINE COMPLEXES AND THEIR APPLICATION IN SUZUKI-TYPE CROSS -COUPLING REACTIONS BASF SE (DE) 2009-11-05 WO disclosed
US-20090275557-A1 Novel Composition for Treatment of Diseases Related to Activated Lymphocytes IMMUNE CONTROL, INC. (US) 2009-11-05 US disclosed
EP-2111223-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2009-10-28 EP disclosed
WO-2009127011-A1 MODIFIED CONDENSATION POLYMERS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2009-10-22 WO disclosed
WO-2009127009-A1 CONDENSATION POLYMERS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2009-10-22 WO disclosed
WO-2009127012-A1 POLYURETHANES COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2009-10-22 WO disclosed
WO-2009127010-A1 CONDENSATION POLYMERS WITH MODIFIED PROPERTIES COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2009-10-22 WO disclosed
US-20090264444-A1 Organic compounds XENON PHARMACEUTICALS INC. (CA) 2009-10-22 US disclosed
US-7605161-B2 1-Pentyl-3-{6-[4-(2-trifluoromethylbenzoyl)piperazin-1-yl]-pyridin-3-yl}urea; inhibitors of stearoyl-CoA desaturase; cardiovascular disease, diabetes, obesity, metabolic syndrome XENON PHARMACEUTICALS INC. (CA) 2009-10-20 US disclosed
US-7605150-B2 Drug therapy for Celiac Sprue THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2009-10-20 US disclosed
US-20090258864-A1 PYRIMIDINE-2-AMINE COMPOUNDS AND THEIR USE AS INHIBITORS OF JAK KINASES RIGEL PHARMACEUTICALS, INC. (US) 2009-10-15 US disclosed
US-20090258939-A1 PYRONE ANALOG COMPOSITIONS AND METHODS LIMERICK BIOPHARMA, INC. 2009-10-15 US disclosed
US-20090258979-A1 POLYMER PRODUCT AND INTERFACIAL POLYMERISATION PROCESS USING RAFT AGENT THE UNIVERSITY OF SYDNEY (AU) 2009-10-15 US disclosed
US-20090256111-A1 DIALKYLBORANE AMINE COMPLEXES BASF SE PATENTS, TRADEMARKS AND LICENSES (DE) 2009-10-15 US disclosed
US-20090258857-A1 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-10-15 US disclosed
CN-101558065-A Oxazole derivatives as positive allosteric modulators of metabotropic glutamate receptors ADDEX PHARMACEUTICALS SA (CH) 2009-10-14 CN disclosed
US-7601874-B2 Antiinflammatory agents; antiarthritic agents; brain disorders; multiple sclerosis; gout; inflammatory bowel disorders; gastrointestinal disorders; psoriasis; antiallergens; autoimmune disease AQUINOX PHARMACEUTICALS INC. (CA) 2009-10-13 US disclosed
US-20090253723-A1 PROTEIN KINASE INHIBITORS ABBOTT LABORATORIES (US) 2009-10-08 US disclosed
EP-2106260-A1 INSULIN SENSITISERS AND METHODS OF TREATMENT Verva Pharmaceuticals Ltd (AU) 2009-10-07 EP disclosed
US-7598401-B2 Multifunctional cationic photoinitiators, their preparation and use SUN CHEMICAL CORPORATION (US) 2009-10-06 US disclosed
US-7598232-B2 Amino-substituted (E)-2,6-dialkoxystyryl 4-substituted-benzylsulfones for treating proliferative disorders TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2009-10-06 US disclosed
EP-2104659-A1 COMPOUNDS WITH (SUBSTITUTED PHENYL)-PROPENAL MOIETY, THEIR DERIVATIVES, BIOLOGICAL ACTIVITY, AND USES THEREOF AndroScience Corporation (US) 2009-09-30 EP disclosed
CN-101547703-A S-nitrosothiol compounds and related derivatives GALLEON PHARMACEUTICALS INC (US) 2009-09-30 CN disclosed
WO-2009117080-A1 QUINAZOLINE DERIVATIVES AS RAF KINASE MODULATORS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATON (US) 2009-09-24 WO disclosed
WO-2009114981-A1 PROCESS FOR PREPARING SULFOXIDE COMPOUNDS CHENGDU LIKAI CHIRAL TECH CO., LTD (CN) 2009-09-24 WO disclosed
EP-2101765-A1 USE OF EPOTHILONES IN THE TREATMENT OF OSTEOPOROSIS AND RELATED DISEASES Bayer Schering Pharma AG (DE) 2009-09-23 EP disclosed
US-7592343-B2 Pyridazine-piperazine compounds and their use as stearoyl-CoA desaturase inhibitors XENON PHARMACEUTICALS INC. (CA) 2009-09-22 US disclosed
WO-2009111830-A1 CONJUGATED UNSATURATED COMPOUNDS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2009-09-17 WO disclosed
CN-101535317-A Dialkylborane amine complexes BASF SE (DE) 2009-09-16 CN disclosed
EP-1519724-B1 FREDERICAMYCIN DERIVATIVES AS MEDICAMENTS FOR TREATING TUMOURS ZENTOPHARM GMBH (DE) 2009-09-09 EP disclosed
CN-101528226-A Fluorinated ligands targeting peripheral benzodiazepine receptors AUSTRALIAN NUCLEAR SCIENCE TEC (AU) 2009-09-09 CN disclosed
US-20090221624-A1 4-AMINOQUINOLINE COMPOUNDS FOR TREATING VIRUS-RELATED CONDITIONS OLIVO PAUL D 2009-09-03 US disclosed
WO-2009106991-A2 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2009-09-03 WO disclosed
US-20090220554-A1 Transglutaminase Inhibitors and Methods of Use Thereof PHARMIX CORPORATION 2009-09-03 US disclosed
EP-1838714-A4 METHODS OF TREATING PAIN UNIV QUEENSLAND (AU) 2009-09-02 EP disclosed
EP-1893622-B1 PROCESS FOR SYNTHESIS OF DIALKOXYORGANOBORANES BASF SE (DE) 2009-09-02 EP disclosed
WO-2009103360-A1 POLYISOPRENOID EPOXIDES USEFUL FOR DECREASING CHOLESTEROL AND/OR INCREASING COENZYME Q BIOSYNTHESIS NEWBIOTECHNIC, S.A. (ES) 2009-08-27 WO disclosed
US-20090215884-A1 METHOD FOR WOUND HEALING PEPLIN RESEARCH PTY LTD. (AU) 2009-08-27 US disclosed
US-20090215817-A1 Novel Triazolopyridine Compounds for the Treatment of Inflammation PFIZER INC 2009-08-27 US disclosed
EP-2091955-A1 ALKOXY COMPOUNDS FOR DISEASE TREATMENT Acucela, Inc. (US) 2009-08-26 EP disclosed
EP-1802662-A4 SURFACE POLYMERISATION PROCESS AND POLYMER PRODUCT USING RAFT AGENT UNIV SYDNEY (AU) 2009-08-26 EP disclosed
EP-2093222-A1 Polyisoprenoid epoxides useful for decreasing cholesterol and/or increasing coenzyme Q biosynthesis NEWBIOTECHNIC, S.A. (ES) 2009-08-26 EP disclosed
EP-1539700-B1 8-HYDROXY QUINOLINE DERIVATIVES PRANA BIOTECHNOLOGY LTD (AU) 2009-08-26 EP disclosed
US-7579313-B2 Administering to a patient an effective dose of [(S)-1-[(3-Bromo-4,5-dihydro-isoxazol-5-ylmethyl)-methyl-carbamoyl]-2-(4-hydroxy-phenyl)-ethyl]-carbamic acid benzyl ester; treatment of glioblastoma, meningioma, melanoma and colon cancer THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2009-08-25 US disclosed
US-7579465-B2 For treatment of picornavirus infections in mammals BIOTA SCIENTIFIC MANAGMENT PTY. LTD. (AU) 2009-08-25 US disclosed
WO-2009103032-A1 PYRIMIDINE-2-AMINE COMPOUNDS AND THEIR USE AS INHIBITORS OF JAK KINASES RIGEL PHARMACEUTICALS, INC. (US) 2009-08-20 WO disclosed
US-20090209577-A1 Novel Triazolopyridine Compounds PFIZER INC. (US) 2009-08-20 US disclosed
US-20090209524-A1 Novel Compounds ASTRAZENECA AB (SE) 2009-08-20 US disclosed
EP-1628987-B1 MANNOSE-6-PHOSPHONATE COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISEASES PHARMAXIS PTY LTD (AU) 2009-08-19 EP disclosed
CN-101511853-A Preparation of diphenyl-bridged substituted cyclopentadienyl-fluorenyl ligands TOTAL PETROCHEMICALS RES FELUY (BE) 2009-08-19 CN disclosed
US-20090203728-A1 Naphthalamide derivatives having antiproliferative activity AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2009-08-13 US disclosed
EP-2086970-A2 2-(PYRAZIN-2-YL)-THIAZOLE AND 2-(1H PYRAZOL-3-YL)-THIAZOLE DERIVATIVES AS WELL AS RELATED COMPOUNDS AS STEAROYL-COA DESATURASE (SCD) INHIBITORS FOR THE TREATMENT OF METABOLIC, CARDIOVASCULAR AND OTHER DISORDERS Novartis AG (CH) 2009-08-12 EP disclosed
EP-1996217-A4 NOVEL ANTIBIOTIC COMPOSITIONS INFLAZYME PHARM LTD (CA) 2009-08-12 EP disclosed
US-7572938-B2 Precursors for ketones and aldehydes GIVAUDAN SA (CH) 2009-08-11 US disclosed
US-20090197890-A1 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2009-08-06 US disclosed
US-20090197894-A1 NICOTINAMIDE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2009-08-06 US disclosed
US-20090197870-A1 Pharmaceutical Compositions EXELIXIS, INC. (US) 2009-08-06 US disclosed
US-20090191284-A1 USE OF NITROANILINE DERIVATIVES FOR THE PRODUCTION OF NITRIC OXIDE STMICROELECTRONICS S.R.I. (IT) 2009-07-30 US disclosed
US-20090191579-A1 ANALGESIA WITH MINIMAL TOLERANCE AND DEPENDENCE BY A MU OPIOID RECEPTOR AGONIST THAT ALSO BINDS FILAMIN A PAIN THERAPEUTICS, INC. 2009-07-30 US disclosed
US-20090191193-A1 Aryl Vinyl Sulfides, Sulfones, Sulfoxides and Sulfonamides, Derivatives Thereof and Therapeutic Uses Thereof TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2009-07-30 US disclosed
US-20090186912-A1 ANTI-INFECTIVE AGENTS AND USES THEREOF ABBOTT LABORATORIES (US) 2009-07-23 US disclosed
US-20090186901-A1 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-07-23 US disclosed
US-20090186802-A1 Cell Penetrating Peptide Conjugates for Delivering of Nucleic Acids into a Cell DIATOS (FR) 2009-07-23 US disclosed
EP-2079736-A1 SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS Rigel Pharmaceuticals, Inc. (US) 2009-07-22 EP disclosed
EP-2079737-A1 PYRIDOPYRIMIDINONE COMPOUNDS USEFUL IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2009-07-22 EP disclosed
EP-1503988-B1 FREDERICAMYCIN DERIVATIVES BIOFRONTERA DISCOVERY GMBH (DE) 2009-07-22 EP disclosed
WO-2009088990-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE, INC. (US) 2009-07-16 WO disclosed
WO-2009088986-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS INTELLIKINE, INC. (US) 2009-07-16 WO disclosed
US-20090182337-A1 Antimicrobial Coatings TYCO HEALTHCARE GROUP LP 2009-07-16 US disclosed
US-20090182133-A1 BENZOPYRANONE DERIVATIVES AND THEIR USE AS ANTI-VIRAL AGENTS SINGAPORE POLYTECHNIC 2009-07-16 US disclosed
EP-1794172-B1 ANTIVIRAL 4'-AZIDO-NUCLEOSIDES HOFFMANN LA ROCHE (CH) 2009-07-15 EP disclosed
EP-2078010-A2 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS Rigel Pharmaceuticals, Inc. (US) 2009-07-15 EP disclosed
EP-2078723-A1 Process for synthesis of organo-oxazaborolidines BASF SE (DE) 2009-07-15 EP disclosed
EP-1740587-A4 SELECTIVE ANTAGONISTS OF A-2A- ADENOSINE RECEPTORS ADENOSINE THERAPEUTICS LLC (US) 2009-07-15 EP disclosed
US-20090176784-A1 ANTI-INFECTIVE AGENTS AND USES THEREOF ABBOTT LABORATORIES (US) 2009-07-09 US disclosed
EP-2076124-A2 STYRENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2009-07-08 EP disclosed
EP-2076514-A1 SPIRO (FURO Ý3, 2-C¨PYRIDINE-3-3 ' -INDOL) -2' (1'H)-ONE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF SODIUM-CHANNEL MEDIATED DISEASES, SUCH AS PAIN XENON PHARMACEUTICALS INC. (CA) 2009-07-08 EP disclosed
EP-2076122-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2009-07-08 EP disclosed
EP-2076518-A1 TRICYCLIC SPIRO-OXINDOLE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2009-07-08 EP disclosed
US-7557118-B2 Preparation of fused polycyclic alkaloids by ring closure of azomethine ylides, novel compounds thereof and their use as chemotherapeutic agents THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2009-07-07 US disclosed
US-20090170841-A1 Styrenyl Derivative Compounds for Treating Ophthalmic Diseases and Disorders ACUCELA INC. (US) 2009-07-02 US disclosed
EP-1507549-A4 DRUG THERAPY FOR CELIAC SPRUE UNIV LELAND STANFORD JUNIOR (US) 2009-07-01 EP disclosed
EP-2074115-A1 N3-HETEROARYL SUBSTITUTED TRIAZOLES AND N5-HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS Rigel Pharmaceuticals, Inc. (US) 2009-07-01 EP disclosed
EP-2073806-A2 USE OF SPIRO-OXINDOLE COMPOUNDS AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2009-07-01 EP disclosed
US-20090163373-A1 Method of Drug Design ALCHEMIA LIMITED (AU) 2009-06-25 US disclosed
WO-2009076598-A1 USE OF UNSATURATED SPHINGOSINE COMPOUNDS AS CHEMOTHERAPEUTIC AGENTS FOR THE TREATMENT OF CANCER CHILDREN'S HOSPITAL & RESEARCH CENTER AT OAKLAND (US) 2009-06-18 WO disclosed
US-20090156615-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-06-18 US disclosed
EP-2069353-A1 POLYCYCLIC AGENTS FOR THE TREATMENT OF RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2009-06-17 EP disclosed
EP-2068855-A2 AROMATIC AND HETEROAROMATIC COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2009-06-17 EP disclosed
US-7547698-B2 Bicyclic heterocyclic derivatives and their use as inhibitors of stearoyl-coadesaturase (SCD) XENON PHARMACEUTICALS INC. (CA) 2009-06-16 US disclosed
WO-2009071535-A1 DIAMINOPYRIDINES FOR THE TREATMENT OF DISEASES WHICH ARE CHARACTERISED BY EXCESSIVE OR ANOMAL CELL PROLIFERATION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-06-11 WO disclosed
EP-2066664-A1 HETEROCYCLIC ORGANIC COMPOUNDS Novartis AG (CH) 2009-06-10 EP disclosed
EP-1869022-A4 NAPHTHALAMIDE DERIVATIVES HAVING ANTIPROLIFERATIVE ACTIVITY AGENCY SCIENCE TECH & RES (SG) 2009-06-10 EP disclosed
US-20090143417-A1 METHODS OF TREATING PAIN THE UNIVERSITY OF QUEENSLAND (AU) 2009-06-04 US disclosed
WO-2009070516-A1 IMIDAZO-THIAZOLE DERIVATIVES AS PROTEIN KINASE INHIBITORS ABBOTT LABORATORIES (US) 2009-06-04 WO disclosed
US-20090138041-A1 Halogenated Cyclic Lactones and Polymers Made Therefrom TYCO HEALTHCARE GROUP LP 2009-05-28 US disclosed
US-20090137653-A1 SUBSTITUTED BENZYLAMINES AS CYP2A INHIBITORS AND USES THEREOF TO TREAT NICOTINE DEPENDENCE INFLAYZME PHARMACEUTICALS LTD. (CA) 2009-05-28 US disclosed
WO-2009067636-A2 MODIFIED INSULIN POLYPEPTIDES AND THEIR USES AMBRX, INC. (US) 2009-05-28 WO disclosed
WO-2009065169-A1 INSULIN-REGULATED AMINOPEPTIDASE (IRAP) INHIBITORS AND USES THEREOF HOWARD FLOREY INSTITUTE (AU) 2009-05-28 WO disclosed
WO-2009067692-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2009-05-28 WO disclosed
EP-2061560-A2 BCL INHIBITORS FOR TREATING PLATELET EXCESS Abbott Laboratories (US) 2009-05-27 EP disclosed
EP-2061754-A1 BIARYL AND BIHETEROARYL COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2009-05-27 EP disclosed
EP-2061755-A1 TRICYCLIC COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2009-05-27 EP disclosed
CN-101443334-A Anti-viral compounds ABBOTT LAB (US) 2009-05-27 CN disclosed
US-20090131447-A1 COMBINATION THERAPY XENON PHARMACEUTICALS INC. (CA) 2009-05-21 US disclosed
EP-2059496-A1 ACETYLENIC COMPOUNDS Commonwealth Scientific and Industrial Research Organisation (AU) 2009-05-20 EP disclosed
EP-2056816-A2 LIPOXIN A4 ANALOGS FOR THE TREATMENT AND PREVENTION OF INTESTINAL FIBROSIS Bayer Schering Pharma Aktiengesellschaft (DE) 2009-05-13 EP disclosed
WO-2009059225-A2 ANALGESIA WITH MINIMAL TOLERANCE AND DEPENDENCE BY A MU OPIOID RECEPTOR AGONIST THAT ALSO BINDS FILAMIN A PAIN THERAPEUTICS, INC. (US) 2009-05-07 WO disclosed
US-20090118455-A1 SILOXANE-CONTAINING POLYURETHANE-UREA COMPOSITIONS AORTECH BIOMATERIAL PTY LTD. 2009-05-07 US disclosed
WO-2009055869-A1 ARYLOXY AMINE COMPOUNDS AND THEIR USE AS SODIUM CHANNEL MODULATORS HOWARD FLOREY INSTITUTE (AU) 2009-05-07 WO disclosed
WO-2009058216-A1 AMINE DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2009-05-07 WO disclosed
US-7528173-B2 Plasma carboxypeptidase B inhibitors SCHERING AKTIENGESELLSHAFT (DE) 2009-05-05 US disclosed
WO-2009054864-A1 POLYCYCLIC ARYL SUBSTITUTED TRIAZOLES AND POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2009-04-30 WO disclosed
US-20090111816-A1 POLYCYCLIC ARYL SUBSTITUTED TRIAZOLES AND POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2009-04-30 US disclosed
WO-2009055696-A1 CARBACEPHEM β-LACTAM ANTIBIOTICS ACHAOGEN, INC. (US) 2009-04-30 WO disclosed
US-20090110842-A1 Boron-based wood preservatives and treatment of wood with boron-based preservatives THE UNIVERSITY OF MELBOUME (AU) 2009-04-30 US disclosed
WO-2009051399-A2 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF (1) CHOONGWAE PHARMA CORPORATION (KR) 2009-04-23 WO disclosed
WO-2009051397-A2 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF (3) CHOONGWAE PHARMA CORPORATION (KR) 2009-04-23 WO disclosed
WO-2009051398-A2 NOVEL COMPOUNDS OF REVERSE TURN MIMETICS AND THE USE THEREOF (2) CHOONGWAE PHARMA CORPORATION (KR) 2009-04-23 WO disclosed
US-20090099133-A1 Isoquinolines Derivatives as Igf-1R Inhibitors ANALYTECON S.A. (CH) 2009-04-16 US disclosed
US-20090099229-A1 Isoquinolines as IGF-1R Inhibitors ANALYTECON S.A (CH) 2009-04-16 US disclosed
WO-2009045479-A1 ALKOXY COMPOUNDS FOR DISEASE TREATMENT ACUCELA INC. (US) 2009-04-09 WO disclosed
US-20090093520-A1 PLASMA CARBOXYPEPTIDASE B INHIBITORS BUCKMAN BRAD 2009-04-09 US disclosed
EP-2044938-A2 Radioprotectors Peter MacCallum Cancer Institute (AU) 2009-04-08 EP disclosed
US-7514436-B2 Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2009-04-07 US disclosed
EP-2041116-A1 PHENYL SUBSTITUTED HETEROARYL-DERIVATIVES AND USE THEREOF AS ANTI-TUMOR AGENTS Boehringer Ingelheim International GmbH (DE) 2009-04-01 EP disclosed
US-20090082400-A1 SOLUBLE PYRONE ANALOGS METHODS AND COMPOSITIONS LIMERICK BIOPHARMA, INC. 2009-03-26 US disclosed
WO-2009039134-A1 ANTI-INFECTIVE PYRIMIDINES AND USES THEREOF ABBOTT LABORATORIES (US) 2009-03-26 WO disclosed
US-20090075822-A1 Method of Altering the Alkaloid Composition in Poppy Plants GLAXOSMITHKLINE AUSTRALIA PTY LTD (AU) 2009-03-19 US disclosed
EP-2035421-A1 2-ARYLPYRAZOLO[L,5-alpha]PYRIMIDIN-3-YL ACETAMIDE DERIVATIVES AS LIGANDS FOR TRANSLOCATOR PROTEIN (18 KDA) THE UNIVERSITY OF SYDNEY (AU) 2009-03-18 EP disclosed
US-20090069273-A1 PHOSPHORYLATED PYRONE ANALOGS AND METHODS LIMERICK BIOPHARMA, INC. 2009-03-12 US disclosed
US-20090069408-A1 TRICYCLIC COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2009-03-12 US disclosed
EP-2032583-A1 NEW CHEMICAL COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2009-03-11 EP disclosed
EP-1916889-A4 METHODS OF ALTERING POPPY CHARACTERISTICS GLAXOSMITHKLINE AUSTRALIA PTY (AU) 2009-03-11 EP disclosed
CN-101384592-A Antiviral compounds ABBOTT LAB (US) 2009-03-11 CN disclosed
CN-101384591-A Antiviral compounds ABBOTT LAB (US) 2009-03-11 CN disclosed
US-20090062353-A1 Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA, INC. 2009-03-05 US disclosed
EP-1472209-B1 LIPOXIN A4 ANALOGS BAYER SCHERING PHARMA AG (DE) 2009-03-04 EP disclosed
EP-2029572-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2009-03-04 EP disclosed
EP-2029138-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2009-03-04 EP disclosed
US-20090054482-A1 Method of making and administering quinoline derivatives as anti-cancer agents THE HONG KONG POLYTECHNIC UNIVERSITY (HK) 2009-02-26 US disclosed
EP-2026825-A2 FURANONE-INITIATED POLYMERS Tyco Healthcare Group, LP (US) 2009-02-25 EP disclosed
US-20090048461-A1 Regulators of Bacterial Signalling Pathways BIOSIGNAL LIMITED (AU) 2009-02-19 US disclosed
EP-2024370-A1 SPIRO- (THO) BENZOPYRAN-2, 4' -PIPERIDINE-AND CYCLOHEXANE DERIVATIVES AS INHIBITORS OF SPECIFIC CELL CYCLE ENZYMES Boehringer Ingelheim International GmbH (DE) 2009-02-18 EP disclosed
EP-2024113-A1 ANTIMICROBIAL COATINGS Tyco Healthcare Group LP (US) 2009-02-18 EP disclosed
US-20090042848-A1 COPPER COMPLEXES LAY PETER 2009-02-12 US disclosed
US-20090042806-A1 TRANSGLUTAMINASE INHIBITORS AND METHODS OF USE THEREOF THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2009-02-12 US disclosed
WO-2009018320-A1 PYRONE ANALOG COMPOSITIONS AND METHODS LIMERICK BIOPHARMA, INC. (US) 2009-02-05 WO disclosed
WO-2009018326-A2 SOLUBLE PYRONE ANALOGS METHODS AND COMPOSITIONS LIMERICK BIOPHARMA, INC. (US) 2009-02-05 WO disclosed
WO-2009018350-A1 PYRONE ANALOG COMPOSITIONS AND METHODS LIMERICK BIOPHARMA, INC. (US) 2009-02-05 WO disclosed
US-20090036310-A1 Substituted 1-(3-pyridinyl)pyrazol-4-ylacetic Acids, Processes for Their Preparation and Their Use as Herbicides and Plant Growth Regulators BAYER CORPSCIENCE GMBH (DE) 2009-02-05 US disclosed
WO-2009018338-A2 PHOSPHORYLATED PYRONE ANALOGS AND METHODS LIMERICK BIOPHARMA, INC. (US) 2009-02-05 WO disclosed
CN-101360506-A Methods for wound healing PEPLIN RESEARCH PTY LTD (AU) 2009-02-04 CN disclosed
US-7485667-B2 Acetylenic aryl sulfonate hydroxamic acid tace and matrix metalloproteinase inhibitors WYETH HOLDINGS CORPORATION (US) 2009-02-03 US disclosed
US-20090030008-A1 PIPERAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2009-01-29 US disclosed
US-20090030000-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2009-01-29 US disclosed
US-20090030123-A1 STABILISER COMPOSITION FOR HALIDE-CONTAINING POLYMERS SUN ACE KAKOH (PTE.) LTD. (SG) 2009-01-29 US disclosed
EP-2018373-A1 FURANONE ENDCAPPED POLYMERS Tyco Healthcare Group, LP (US) 2009-01-28 EP disclosed
EP-2018361-A1 HALOGENATED CYCLIC LACTONES AND POLYMERS MADE THEREFROM Tyco Healthcare Group, LP (US) 2009-01-28 EP disclosed
US-7482366-B2 Modulators of LXR X-CEPTOR THERAPEUTICS, INC. (US) 2009-01-27 US disclosed
US-7482488-B2 Aryl and heteroaryl propene amides, derivatives thereof and therapeutic uses thereof TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2009-01-27 US disclosed
US-20090022824-A1 Pesticidal formulations AKHIL TECHNOLOGIES PTY LTD (AU) 2009-01-22 US disclosed
US-20090023669-A1 Antibacterial Agents ALCHEMIA LIMITED (AU) 2009-01-22 US disclosed
EP-2017264-A1 Substituted phenyl propargyl compounds, method for their manufacture and their use as herbicides and plant growth regulators BAYER CROPSCIENCE AG (DE) 2009-01-21 EP disclosed
US-7479471-B2 2-Amino-4-bicyclylamino-6H-1,3,5-triazines, processes for their preparation and their use as herbicides and plant growth regulators BAYER CROPSCIENCE GMBH (DE) 2009-01-20 US disclosed
EP-2012789-A1 METHOD OF TREATMENT OF AGE-RELATED MACULAR DEGENERATION(AMD) Prana Biotechnology Limited (AU) 2009-01-14 EP disclosed
WO-2009003998-A2 ANTIPROLIFERATIVE COMPOUNDS BASED ON 5-MEMBERED HETEROCYCLES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-01-08 WO disclosed
WO-2009003999-A2 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-01-08 WO disclosed
WO-2009005794-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2009-01-08 WO disclosed
US-20090005250-A1 Substituted 2,4-diamino-1,3,5-triazines, processes for their use as herbicides and crop growth regulators BAYER CROPSCIENCE AG (DE) 2009-01-01 US disclosed
EP-2007790-A1 COMPOUNDS AND METHODS FOR THE TREATMENT OF PAIN THE UNIVERSITY OF QUEENSLAND (AU) 2008-12-31 EP disclosed
EP-1149075-B1 SYNTHESIS OF DITHIOESTER CHAIN TRANSFER AGENTS COMMW SCIENT IND RES ORG (AU) 2008-12-31 EP disclosed
WO-2009000832-A2 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-12-31 WO disclosed
US-20080318942-A1 Fredericamycin Derivatives BIOAGENCY AG (DE) 2008-12-25 US disclosed
US-20080318417-A1 METHOD OF FORMING RUTHENIUM FILM FOR METAL WIRING STRUCTURE ASM JAPAN K.K. (JP) 2008-12-25 US disclosed
US-20080311040-A1 METHODS AND COMPOSITIONS FOR IMPROVED THERAPEUTIC EFFECTS WITH siRNA FLAGSHIP VENTURES (US) 2008-12-18 US disclosed
WO-2008152013-A1 INDOLINONE DERIVATIVES AND THEIR USE IN TREATING DISEASE-STATES SUCH AS CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-12-18 WO disclosed
WO-2008152014-A2 3-HETROCYCLYLIDENE-INDOLINONE DERIVATIVES AS INHIBITORS OF SPECIFIC CELL CYCLE KINASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-12-18 WO disclosed
EP-2001911-A1 POLYMER PRODUCT AND INTERFACIAL POLYMERISATION PROCESS USING RAFT AGENT The University of Sydney (AU) 2008-12-17 EP disclosed
EP-2001892-A2 IMIDAZOLOTHIAZOLE COMPOUNDS FOR THE TREATMENT OF DISEASE Ambit Biosciences Corporation (US) 2008-12-17 EP disclosed
EP-1968569-A4 BENZOPYRANONE DERIVATIVES AND THEIR USE AS ANTI-CORONAVIRAL AGENTS SINGAPORE POLYTECHNIC (SG) 2008-12-17 EP disclosed
WO-2008151288-A2 AROMATIC AND HETEROAROMATIC COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2008-12-11 WO disclosed
EP-1998809-A2 CAMPTOTHECIN-CELL PENETRATING PEPTIDE CONJUGATES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Diatos S.A. (FR) 2008-12-10 EP disclosed
WO-2008147864-A2 METHODS OF USING PIPERAZINE COMPOUNDS IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-12-04 WO disclosed
US-20080299170-A1 Medical Devices and Coatings Therefor ASTON UNIVERSITY (GB) 2008-12-04 US disclosed
EP-1996217-A2 NOVEL ANTIBIOTIC COMPOSITIONS Inflazyme Pharmaceuticals, Ltd. (CA) 2008-12-03 EP disclosed
US-7459462-B2 Fredericamycin derivatives BIOFRONTERA DISCOVERY GMBH (DE) 2008-12-02 US disclosed
WO-2008144248-A1 FURANONE COPOLYMERS TYCO HEALTHCARE GROUP LP (US) 2008-11-27 WO disclosed
US-20080293844-A1 Gels AORTECH BIOMATERIALS PTY LTD (AU) 2008-11-27 US disclosed
WO-2008144247-A1 ANTIMICROBIAL MATERIALS AND COATINGS TYCO HEALTHCARE GROUP LP (US) 2008-11-27 WO disclosed
US-7456180-B2 Piperazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2008-11-25 US disclosed
US-20080280916-A1 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-11-13 US disclosed
US-20080281016-A1 Polymer Composite MILLER WASTE MILLS INC. DBA RTP COMPANY 2008-11-13 US disclosed
US-20080280985-A1 Methods and Compositions Using Certain Phenolic Derivatives for the Treatment of Diabetes STOCKER, ROLAND (AU) 2008-11-13 US disclosed
WO-2008134547-A1 METHODS OF USING HYDROXYCYCLOHEXANE AND HYDROXYPIPERIDINE COMPOUNDS IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-11-06 WO disclosed
WO-2008131491-A1 TREATMENT OF VIRALLY INDUCED LESIONS PEPLIN RESEARCH PTY LTD (AU) 2008-11-06 WO disclosed
WO-2008134553-A1 METHODS OF USING BICYCLIC COMPOUNDS IN TREATING SODIUM CHANNEL-MEDIATED DISEASES XENON PHARMACEUTICALS INC. (CA) 2008-11-06 WO disclosed
US-20080275003-A1 Bis-Cationic Compounds and Use Thereof THE UNIVERSITY OF SYDNEY (AU) 2008-11-06 US disclosed
WO-2008131368-A2 STYRENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA INC. (US) 2008-10-30 WO disclosed
US-20080269058-A1 Methods of Altering Poppy Characteristics SUN PHARMACEUTICAL INDUSTRIES (AUSTRALIA) PTY LTD (AU) 2008-10-30 US disclosed
US-20080269247-A1 Chemokine Inhibiting Piperazine Derivatives and Their Use to Treat Myocarditis BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-10-30 US disclosed
US-20080268250-A1 Polymerisation Process and Polymer Product THE UNIVERSITY OF SYDNEY (AU) 2008-10-30 US disclosed
WO-2008127381-A2 ARTEMISININ DERIVATIVES JOHNS HOPKINS UNIVERSITY (US) 2008-10-23 WO disclosed
EP-1981844-A1 NOVEL LACTAMS Biosignal Limited (AU) 2008-10-22 EP disclosed
EP-1979349-A2 ANTI-VIRAL COMPOUNDS Abbott Laboratories (US) 2008-10-15 EP disclosed
US-7435484-B2 a ruthenium(Ru) thin film on a substrate in a reaction chamber, includes: (i) supplying a gas of a ruthenium precursor into the reaction chamber so that the gas of the ruthenium precursor is adsorbed onto the substrate, wherein the ruthenium precursor a ruthenium complex contains a non-cyclic diene ASM JAPAN K.K. (JP) 2008-10-14 US disclosed
WO-2008121861-A2 PYRAZOLE AND PYRROLE COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2008-10-09 WO disclosed
WO-2008121859-A1 METHODS OF USING TRICYCLIC COMPOUNDS IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-10-09 WO disclosed
EP-1976828-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE Schering Aktiengesellschaft (DE) 2008-10-08 EP disclosed
EP-1363880-A4 SYNTHESIS FOR THE PREPARATION OF COMPOUNDS FOR SCREENING AS POTENTIAL TUBULIN BINDING AGENTS UNIV AUSTRALIAN (AU) 2008-10-08 EP disclosed
EP-1478628-B1 2-AMINO-4-BICYCLYL AMINO-6H-1.3.5-TRIAZINES, METHOD FOR THE PRODUCTION AND USE THEREOF AS HERBICIDES AND PLANT GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2008-10-08 EP disclosed
CN-101282935-A Isoquinoline derivatives as insulin-like growth factor-1 receptor inhibitors ANALYTECON SA (CH) 2008-10-08 CN disclosed
WO-2008118946-A1 METHODS AND COMPOSITIONS USING CERTAIN PHENOLIC DERIVATIVES FOR THE TREATMENT OF DIABETES ATHEROGENICS, INC. (US) 2008-10-02 WO disclosed
WO-2008118790-A1 DIHYDROINDAZOLE COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2008-10-02 WO disclosed
EP-1973917-A2 PROTEIN KINASE INHIBITORS Abbott Laboratories (US) 2008-10-01 EP disclosed
WO-2008114006-A1 9-SUBSTITUTED-8-OXO-ADENINE COMPOUNDS AS TOLL-LIKE RECEPTOR (TLR7) MODULATORS ASTRAZENECA AB (SE) 2008-09-25 WO disclosed
US-20080234270-A1 Pyrrole Derivatives As Pharmaceutical Agents EXELIXIS, INC. (US) 2008-09-25 US disclosed
US-20080234327-A1 DIHYDROINDAZOLE COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2008-09-25 US disclosed
US-20080233102-A1 Drug Therapy for Celiac Sprue THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2008-09-25 US disclosed
WO-2008115999-A1 BIARYL AND BIHETEROARYL COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2008-09-25 WO disclosed
US-20080234384-A1 BIARYL AND BIHETEROARYL COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2008-09-25 US disclosed
EP-1971611-A1 ANTI-VIRAL COMPOUNDS Abbott Laboratories (US) 2008-09-24 EP disclosed
WO-2008113006-A1 METHODS OF USING QUINOLINONE COMPOUNDS IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-09-18 WO disclosed
US-20080227789-A1 DIAMINOTHIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2008-09-18 US disclosed
WO-2008110794-A1 PIPERIDINONES USEFUL IN THE TREATMENT OF INFLAMMATION BIOLIPOX AB (SE) 2008-09-18 WO disclosed
WO-2008110793-A1 PIPERIDINONES USEFUL IN THE TREATMENT OF INFLAMMATION BIOLIPOX AB (SE) 2008-09-18 WO disclosed
EP-1968643-A2 CELL PENETRATING PEPTIDE CONJUGATES FOR DELIVERING OF NUCLEIC ACIDS INTO A CELL Diatos (FR) 2008-09-17 EP disclosed
EP-1968979-A2 9-MEMBERED HETEROBICYCLIC COMPOUNDS AS INHIBITORS OF PROTEIN KINASES ABBOTT LABORATORIES (US) 2008-09-17 EP disclosed
EP-1495003-B1 FREDERICAMYCIN DERIVATIVES BIOFRONTERA DISCOVERY GMBH (DE) 2008-09-17 EP disclosed
EP-1968569-A1 BENZOPYRANONE DERIVATIVES AND THEIR USE AS ANTI-CORONAVIRAL AGENTS Singapore Polytechnic (SG) 2008-09-17 EP disclosed
WO-2008109105-A2 METHODS AND COMPOSITIONS FOR IMPROVED THERAPEUTIC EFFECTS WITH SIRNA FLAGSHIP VENTURES (US) 2008-09-12 WO disclosed
WO-2008107444-A1 9H- PURINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF PROLIFERATIVE DISEASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-09-12 WO disclosed
WO-2008109840-A1 TRICYCLIC COMPOUNDS USEFUL IN TREATING IRON DISORDERS XENON PHARMACEUTICALS INC. (CA) 2008-09-12 WO disclosed
WO-2008109856-A2 METHODS OF USING DIAZEPINONE COMPOUNDS IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-09-12 WO disclosed
US-20080221134-A1 8-ALKYNYLXANTHINES AND DERIVATIVES RHEINISCHE FRIEDRICH-WILHELMS-UNIVERSITAET BONN (DE) 2008-09-11 US disclosed
US-20080221194-A1 Novel Potassium channel Blockers and Uses Thereof HARVEY ANDREW J 2008-09-11 US disclosed
EP-1294705-B1 SYNTHESIS OF CYCLIC COMPOUNDS BIOSIGNAL LTD (AU) 2008-09-10 EP disclosed
EP-1965796-A2 4,7-DIHYDROTHIENO[2,3-B]PYRIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS Gilead Colorado, Inc. (US) 2008-09-10 EP disclosed
EP-1965818-A1 METHODS FOR WOUND HEALING Peplin Research Pty Ltd. (AU) 2008-09-10 EP disclosed
WO-2008106633-A1 METHODS OF USING BENZODIOXINE COMPOUNDS IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-09-04 WO disclosed
EP-1962840-A1 USE OF 4, 7-DIHYDROTHIENO [2, 3-B]PYRIDINE COMPOUNDS IN THE TREATMENT OF CARDIOVASCULAR DISEASES Gilead Colorado, Inc. (US) 2008-09-03 EP disclosed
EP-1962864-A1 ANTIBACTERIAL AGENTS Alchemia Limited (AU) 2008-09-03 EP disclosed
CN-101258130-A Isoquinolines as insulin-like growth factor-1 receptor inhibitors ANALYTECON SA (CH) 2008-09-03 CN disclosed
US-20080207587-A1 Pyridazine Derivatives for Inhibiting Human Stearoyl-Coa-Desaturase XENON PHARMACEUTICALS INC. (CA) 2008-08-28 US disclosed
US-7417129-B2 Combinatorial libraries of monosaccharides ALCHEMIA PTY LTD (AU) 2008-08-26 US disclosed
WO-2008101029-A2 USE OF THIAZOLE, OXAZOLE AND IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-08-21 WO disclosed
US-20080200728-A1 Process for Synthesis of Dialkoxyorganoboranes BASF AKTIENGESELLSCHAFT (DE) 2008-08-21 US disclosed
US-20080194636-A1 Enzyme Inhibitors and Uses Thereof HOWARD FLOREY INSTITUTE OF EXPERIMENTAL PHYSIOLOGY AND MEDICINE (AU) 2008-08-14 US disclosed
WO-2008097991-A1 PYRIDOPYRIMIDINONE COMPOUNDS USEFUL IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-08-14 WO disclosed
US-20080194616-A1 PYRIDOPYRIMIDINONE COMPOUNDS USEFUL IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-08-14 US disclosed
US-20080194691-A1 Apoptosis Promoters ABBOTT LABORATORIES (US) 2008-08-14 US disclosed
EP-1954285-A2 TRANSGLUTAMINASE INHIBITORS AND METHODS OF USE THEREOF Alvine Pharmaceuticals, Inc. (US) 2008-08-13 EP disclosed
US-20080188455-A1 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2008-08-07 US disclosed
WO-2008094909-A2 QUINAZOLINONE AND FUSED PYRIMIDINONE COMPOUNDS AND THEIR USE IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-08-07 WO disclosed
US-20080188488-A1 Heterocyclic Derivatives and Their Use as Stearoyl-Coa Desaturase Inhibitors XENON PHARMACEUTICALS INC. (CA) 2008-08-07 US disclosed
US-20080188454-A1 angiogenesis and/or cell proliferation, carcinoma, myeloid leukemia, endometriosis; inhibitors of the receptor protein tyrosine kinase; N3-(3-cyclopentyl-1,2,3,4,5,6-hexahydrobenzo[d]azocin-8-yl)-1-(6-fluoroquinazolin-4-yl)-1H-1,2,4-triazole-3,5-diamine RIGEL PHARMACEUTICALS, INC. (US) 2008-08-07 US disclosed
US-20080188557-A1 Compounds with (substituted phenyl)-propenal moiety, their derivatives, biological activity, and use thereof Annji Pharmaceutical Co., Ltd. (TW) 2008-08-07 US disclosed
US-20080188474-A1 e.g. 1-phenyl-N3-(4-(2-(piperidin-1-yl)ethoxy)phenyl)-1H-1,2,4-triazole-3,5-diamine; receptor protein tyrosine kinase (AXL) antagonist; antiinflammatory, anticarcinogenic , antidiabetic agent; rheumatoid arthritis, vascular disease; breast, renal, endometrial, ovarian carcinoma, or myeloid leukemia RIGEL PHARMACEUTICALS, INC. (US) 2008-08-07 US disclosed
EP-1773768-A4 PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS EXELIXIS INC (US) 2008-08-06 EP disclosed
EP-1476149-B1 SUBSTITUTED HYDRAZONES AS INHIBITORS OF CYCLOOXYGENASE-2 UNIV TEMPLE (US) 2008-08-06 EP disclosed
US-20080182837-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-31 US disclosed
US-20080182834-A1 Multi-Nuclear Metal Complexes Partially Encapsulated by Cucurbit[7-12]Urils NEWSOUTH INNOVATIONS PTY LIMITED (AU) 2008-07-31 US disclosed
WO-2008089521-A1 INSULIN SENSITISERS AND METHODS OF TREATMENT VERVA PHARMACEUTICALS LTD (AU) 2008-07-31 WO disclosed
US-20080182862-A1 N3-HETEROARYL SUBSTITUTED TRIAZOLES AND N5-HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2008-07-31 US disclosed
EP-1725558-A4 METHOD FOR PREPARING COMPOUNDS COMPRISING CUCURBITURIL GROUPS NEWSOUTH INNOVATIONS PTY LTD (AU) 2008-07-30 EP disclosed
WO-2008089439-A2 METHODS AND COMPOSITIONS FOR ENHANCING LIFESPAN INVOLVING SIRTUIN-MODULATING COMPOUNDS AND CHALCOGENIDES FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2008-07-24 WO disclosed
US-20080176858-A1 SELECTIVE ANTAGONISTS OF A2A ADENOSINE RECEPTORS ADENOSINE THERAPEUTICS, LLC (US) 2008-07-24 US disclosed
US-20080176833-A1 DIHYDROPYRIDINE DERIVATIVES AS USEFUL AS PROTEIN KINASE INHIBITORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2008-07-24 US disclosed
US-20080176847-A1 BRIDGED BICYCLIC ARYL AND BRIDGED BICYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2008-07-24 US disclosed
EP-1296673-B1 ANTIMICROBIAL COATINGS BIOSIGNAL AUSTRALIA PTY LTD (AU) 2008-07-23 EP disclosed
WO-2008085984-A1 COMPOUNDS WITH (SUBSTITUTED PHENYL)-PROPENAL MOIETY, THEIR DERIVATIVES, BIOLOGICAL ACTIVITY, AND USES THEREOF ANDROSCIENCE CORPORATION (US) 2008-07-17 WO disclosed
EP-1054004-B1 NOVEL PYRIMIDINE-5-CARBOXAMIDE DERIVATIVES ASTELLAS PHARMA INC (JP) 2008-07-16 EP disclosed
US-20080167321-A1 Pyridine Derivatives For Inhibiting Human Stearoyl-Coa-Desaturase XENON PHARMACEUTICALS INC. (CA) 2008-07-10 US disclosed
WO-2008083356-A1 SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2008-07-10 WO disclosed
WO-2008083353-A1 BICYCLIC ARYL AND BICYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2008-07-10 WO disclosed
WO-2008083354-A1 N3-HETEROARYL SUBSTITUTED TRIAZOLES AND N5-HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2008-07-10 WO disclosed
WO-2008083367-A2 POLYCYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2008-07-10 WO disclosed
EP-1940796-A1 ISOQUINOLINES DERIVATIVES AS IGF-1R INHIBITORS Analytecon S.A. (CH) 2008-07-09 EP disclosed
CN-100400531-C 2-oxabicyclo 3.3.0 octane compounds, process for producing the same, optical resolver, method of separating diastereomer mixture, and method of optically resolving alcohol ZEON CORP (JP) 2008-07-09 CN disclosed
WO-2008080134-A2 4-AMIN0-2- (HETERO) ARYLAMINO-5- (HETERO) ARYLTHIAZOLES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed
US-20080161353-A1 8-Hydroxy quinoline derivatives PRANA BIOTECHNOLOGY LIMITED (AU) 2008-07-03 US disclosed
EP-1939197-A1 8-ethinylxanthine derivatives as selective A2A receptor antagonists SCHWARZ PHARMA AG (DE) 2008-07-02 EP disclosed
EP-1937719-A2 GLYCOPEGYLATED FACTOR VII AND FACTOR VIIA Neose Technologies, Inc. (US) 2008-07-02 EP disclosed
EP-1938686-A1 Substituted 1-(3-pyridinyl)pyrazol-4-yl-acetic acids, process for their preparation and their use as herbicide and plant growth regulator. Bayer CropScience AG (DE) 2008-07-02 EP disclosed
EP-1558585-A4 NEUROLOGICALLY-ACTIVE COMPOUNDS PRANA BIOTECHNOLOGY LTD (AU) 2008-07-02 EP disclosed
US-7393869-B2 Methods of using thiazolidine derivatives to treat cancer or inflammation QLT INC. (CA) 2008-07-01 US disclosed
WO-2008074078-A1 SELECTIVELY DELIVERABLE ISATIN-BASED CYTOTOXIC AGENTS UNIVERSITY OF WOLLONGONG (AU) 2008-06-26 WO disclosed
WO-2008074835-A1 2-SUBSTITUTED 5-MEMBERED HETEROCYCLES AS SCD INHIBITORS NOVARTIS AG (CH) 2008-06-26 WO disclosed
WO-2008074091-A1 RADIOPROTECTOR COMPOUNDS AND RELATED METHODS PETER MACCALLUM CANCER INSTITUTE (AU) 2008-06-26 WO disclosed
US-20080153815-A1 PINANE-SUBSTITUTED PYRIMIDINEDIAMINE DERIVATIVES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2008-06-26 US disclosed
EP-1934388-A1 METHOD OF DRUG DESIGN Alchemia Ltd (AU) 2008-06-25 EP disclosed
WO-2008071451-A1 DIHYDROPYRIDINE DERIVATIVES USEFUL AS PROTEIN KINASE INHIBITORS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-06-19 WO disclosed
WO-2008073825-A1 LXR AND FXR MODULATORS EXELIXIS, INC. (US) 2008-06-19 WO disclosed
US-20080146626-A1 USE OF EPOTHILONES IN THE TREATMENT OF OSTEOPOROSIS AND RELATED DISEASES BAYER SCHERING PHARMA AG (DE) 2008-06-19 US disclosed
EP-1678133-A4 SEQUENCE SELECTIVE PYRROLE AND IMIDAZOLE POLYAMIDE METALLOCOMPLEXES UNIV WESTERN SYDNEY (AU) 2008-06-18 EP disclosed
EP-1931205-A2 TRANSGLUTAMINASE INHIBITORS AND METHODS OF USE THEREOF THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2008-06-18 EP disclosed
CN-101203230-A Modulation of angiogenesis with NOD factors such as glucosamine oligosaccharides RICHARD PARISH CHRISTOPHER (AU) 2008-06-18 CN disclosed
WO-2008070741-A1 COMPOSITIONS AND METHODS FOR ENHANCING SURVIVAL AND REDUCING INJURY UNDER ISCHEMIC OR HYPOXIC CONDITIONS IKARIA, INC. (US) 2008-06-12 WO disclosed
WO-2008068043-A1 USE OF EPOTHILONES IN THE TREATMENT OF OSTEOPOROSIS AND RELATED DISEASES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-06-12 WO disclosed
EP-1930004-A1 Use of epothilones in the treatment of osteoporosis and related diseases Bayer Schering Pharma Aktiengesellschaft (DE) 2008-06-11 EP disclosed
CN-101198615-A Method for synthesizing dialkoxyorganoborane BASF AG (DE) 2008-06-11 CN disclosed
WO-2008064432-A1 POLYCYCLIC MOLECULAR COMPOUNDS THE UNIVERSITY OF SYDNEY (AU) 2008-06-05 WO disclosed
US-20080132521-A1 Isoquinolinone Derivatives and Their Use As Therapeutic Agents EXELIXIS, INC. (US) 2008-06-05 US disclosed
US-20080132697-A1 Novel compositions for treatment of diseases related to activated lymphocytes IMMUNE CONTROL, INC. (US) 2008-06-05 US disclosed
CN-101193921-A Carbon-bridged cyclopentadienyl-fluorenyl ligands TOTAL PETROCHEMICALS RES FELUY (BE) 2008-06-04 CN disclosed
US-20080125434-A1 Heterocyclic Derivatives and Their Use as Strearoyl-Coa Desaturase Inhibitors XENON PHARMACEUTICALS INC. (CA) 2008-05-29 US disclosed
US-20080124484-A1 METHOD OF FORMING RU FILM AND METAL WIRING STRUCTURE ASM JAPAN K.K. (JP) 2008-05-29 US disclosed
US-20080125415-A1 Novel methods for treatment of diseases related to activated lymphocytes IMMUNE CONTROL, INC. (US) 2008-05-29 US disclosed
EP-1274420-A4 MICROBIAL INHIBITORY COMPOSITIONS BIOSIGNAL AUSTRALIA PTY LTD (AU) 2008-05-28 EP disclosed
WO-2008060789-A2 USE OF SPIRO-OXINDOLE COMPOUNDS AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-05-22 WO disclosed
US-20080118982-A1 Tagged Petroleum Products and Methods of Detecting Same AUTHENTIX, INC. (US) 2008-05-22 US disclosed
US-20080119471-A1 Piperazine urea derivatives for the treatment of endometriosis BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-05-22 US disclosed
US-20080119488-A1 Modulators Of Nuclear Receptors EXELIXIS, INC. (US) 2008-05-22 US disclosed
US-20080119439-A1 Treatment and prevention of intestinal fibrosis BAYER SCHERING PHARMA AKTIENGESELLSCHAFT 2008-05-22 US disclosed
EP-1922310-A2 TRIAZOLE DERIVATIVES USEFUL AS AXL INHIBITORS Rigel Pharmaceuticals, Inc. (US) 2008-05-21 EP disclosed
EP-1765755-A4 REGULATORS OF BACTERIAL SIGNALLING PATHWAYS BIOSIGNAL LTD (AU) 2008-05-21 EP disclosed
US-7371755-B1 Antiviral agents BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2008-05-13 US disclosed
US-20080108659-A1 POLY(ADP-RIBOSE)POLYMERASE INHIBITORS ABBVIE INC. 2008-05-08 US disclosed
US-20080108629-A1 Heterocyclic Derivatives for the Treatment of Diseases Mediated by Stearoyl-Coa Desaturase Enzymes XENON PHARMACEUTICALS INC. (CA) 2008-05-08 US disclosed
EP-1916889-A1 METHODS OF ALTERING POPPY CHARACTERISTICS Glaxosmithkline Australia PTY Ltd. (AU) 2008-05-07 EP disclosed
EP-1755373-A4 METHOD OF ALTERING THE ALKALOID COMPOSITION IN POPPY PLANTS GLAXOSMITHKLINE AUSTRALIA PTY (AU) 2008-05-07 EP disclosed
US-20080103191-A1 ENTACAPONE-DERIVATIVES SCHWARZ PHARMA AG (DE) 2008-05-01 US disclosed
US-20080103151-A9 Heterocyclic compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2008-05-01 US disclosed
WO-2008046156-A1 VESICULATED POLYMER PARTICLES THE UNIVERSITY OF SYDNEY (AU) 2008-04-24 WO disclosed
WO-2008046155-A1 METHODS FOR REGULATING GLUCOSE HOMEOSTASIS AND AGENTS THEREFOR DIA-B TECH LIMITED (AU) 2008-04-24 WO disclosed
US-20080096895-A1 Heterocyclic Derivatives and Their Use as Stearoyl-Coa Desaturase Inhibitors XENON PHARMACEUTICALS INC. (CA) 2008-04-24 US disclosed
WO-2008046049-A1 SPIRO (FURO [3, 2-C] PYRIDINE-3-3 ' -INDOL) -2' (1'H)-ONE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF SODIUM-CHANNEL MEDIATED DISEASES, SUCH AS PAIN XENON PHARMACEUTICALS INC. (CA) 2008-04-17 WO disclosed
WO-2008046087-A2 SPIRO COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-04-17 WO disclosed
WO-2008046046-A1 TRICYCLIC SPIRO-OXINDOLE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-04-17 WO disclosed
WO-2008046084-A2 SPIROHETEROCYCLIC COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-04-17 WO disclosed
WO-2008046082-A2 USE OF HETEROCYCLIC COMPOUNDS AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-04-17 WO disclosed
WO-2008046083-A2 USE OF OXINDOLE COMPOUNDS AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-04-17 WO disclosed
WO-2008045978-A1 PINANE-SUBSTITUTED PYRIMIDINEDIAMINE DERIVATIVES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2008-04-17 WO disclosed
WO-2008046065-A1 SPIROHETEROCYCLIC COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-04-17 WO disclosed
EP-1910307-A1 PYRAZOLE BASED LXR MODULATORS Exelixis, Inc. (US) 2008-04-16 EP disclosed
EP-1910308-A1 IMIDAZOLE BASED LXR MODULATORS Exelixis, Inc. (US) 2008-04-16 EP disclosed
EP-1907027-A2 MEDICAL DEVICES AND COATINGS THEREFOR Aston University (GB) 2008-04-09 EP disclosed
US-20080081917-A1 MULTIFUNCTIONAL CATIONIC PHOTOINITIATORS, THEIR PREPARATION AND USE SUN CHEMICAL CORPORATION (US) 2008-04-03 US disclosed
WO-2008037011-A1 POLYCYCLIC AGENTS FOR THE TREATMENT OF RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2008-04-03 WO disclosed
EP-1904047-A2 APOPTOSIS PROMOTERS ABBOTT LABORATORIES (US) 2008-04-02 EP disclosed
US-20080076779-A1 Reducing platelets in mammals blood and preventing/treating pro-thrombotic conditions and diseases via inhibitors of anti-apoptotic Bcl-2 family protein members ABBVIE INC. 2008-03-27 US disclosed
WO-2008034895-A2 ANSAMYCIN DERIVATIVES DISCOVERY PARTNERS INTERNATIONAL GMBH (DE) 2008-03-27 WO disclosed
WO-2008036715-A1 HETEROCYCLIC ORGANIC COMPOUNDS NOVARTIS AG (CH) 2008-03-27 WO disclosed
EP-1366015-A4 BENZENE-1 2-DIOL MANNICH BASES LIGANDS POLYMERS AND METHOD OF SELECTIVE METAL IONS REMOVAL TECH RESOURCES PTY LTD (AU) 2008-03-26 EP disclosed
WO-2008031157-A1 ACETYLENIC COMPOUNDS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2008-03-20 WO disclosed
EP-1697377-A4 POLYCYCLIC AGENTS FOR THE TREATMENT OF RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENT MANAGEMENT (AU) 2008-03-19 EP disclosed
WO-2008030836-A2 BCL INHIBITORS TREATING PLATELET EXCESS ABBOTT LABORATORIES (US) 2008-03-13 WO disclosed
US-20080054472-A1 a ruthenium(Ru) thin film on a substrate in a reaction chamber, includes: (i) supplying a gas of a ruthenium precursor into the reaction chamber so that the gas of the ruthenium precursor is adsorbed onto the substrate, wherein the ruthenium precursor a ruthenium complex contains a non-cyclic diene ASM JAPAN K.K. (JP) 2008-03-06 US disclosed
EP-1893622-A2 PROCESS FOR SYNTHESIS OF DIALKOXYORGANOBORANES BASF SE (DE) 2008-03-05 EP disclosed
WO-2008022807-A2 LIPOXIN A4 ANALOGS FOR THE TREATMENT AND PREVENTION OF INTESTINAL FIBROSIS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-02-28 WO disclosed
WO-2008024390-A2 2- (PYRAZIN-2-YL) -THIAZOLE AND 2- (1H-PYRAZ0L-3-YL) -THIAZOLE DERIVATIVES AS WELL AS RELATED COMPOUNDS AS STEAROYL-COA DESATURASE (SCD) INHIBITORS FOR THE TREATMENT OF METABOLIC, CARDIOVASCULAR AND OTHER DISORDERS NOVARTIS AG (CH) 2008-02-28 WO disclosed
US-7335658-B2 Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2008-02-26 US disclosed
US-20080044401-A1 DRUG THERAPY FOR CELIAC SPRUE THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2008-02-21 US disclosed
EP-1888098-A2 GLYCOPEGYLATED ERYTHROPOIETIN FORMULATIONS Neose Technologies, Inc. (US) 2008-02-20 EP disclosed
EP-1888543-A1 APOPTOSIS PROMOTERS ABBOTT LABORATORIES (US) 2008-02-20 EP disclosed
EP-1888595-A2 SPIRO-OXINDOLE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-02-20 EP disclosed
EP-1888592-A1 SPIROHETEROCYCLIC COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-02-20 EP disclosed
US-20080039522-A1 Composition Containing a Complex Comprising a Metal Ion and a Carboxylate Ligand Having Anti-Inflammatory Activity MEDICAL THERAPIES LIMITED (AU) 2008-02-14 US disclosed
US-20080033179-A1 Optical Recording Material and Optical Recording Medium ADEKA CORPORATION (JP) 2008-02-07 US disclosed
EP-1879892-A2 2-PYRROLIDONE DERIVATIVES AND THEIR USES FOR THE TREATMENT OF INFLAMMATORY CONDITIONS AND PAIN XENON PHARMACEUTICALS INC. (CA) 2008-01-23 EP disclosed
EP-1732898-B1 TETRAHYDROISOQUINOLINE- AND TETRAHYDROBENZAZEPINE DERIVATIVES AS IGF-1R INHIBITORS ANALYTECON SA (CH) 2008-01-23 EP disclosed
US-20080015230-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-01-17 US disclosed
US-20080015192-A1 INHIBITORS OF POLO-LIKE KINASES ABBVIE INC. 2008-01-17 US disclosed
EP-1877481-A2 STABILISER COMPOSITION FOR HALIDE-CONTAINING POLYMERS Sun Ace Kakoh (Pte.) Ltd. (SG) 2008-01-16 EP disclosed
EP-1877378-A2 OXINDOLE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2008-01-16 EP disclosed
WO-2008003770-A1 PHENYL SUBSTITUTED HETEROARYL-DERIVATIVES AND USE THEREOF AS ANTI-TUMOR AGENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-01-10 WO disclosed
WO-2008004986-A1 CATALYST SYSTEM FOR OLIGOMERIZATION OF OLEFINS NATIONAL UNIVERSITY OF SINGAPORE (SG) 2008-01-10 WO disclosed
US-20080009418-A1 Selective Inhibitors ALCHEMIA LTD. (AU) 2008-01-10 US disclosed
EP-1874322-A1 USE OF TAFI INHIBITORS FOR ENHANCED MYOCARDIAL REPERFUSION AND FACILITATED PCI Bayer Schering Pharma Aktiengesellschaft (DE) 2008-01-09 EP disclosed
EP-1871357-A2 SUBSTITUTED BENZYLAMINES AS CYP2A INHIBITORS AND USES THEREOF TO TREAT NICOTINE DEPENDENCE Inflazyme Pharmaceuticals, Ltd. (CA) 2008-01-02 EP disclosed
EP-1871392-A1 MODULATING ANGIOGENESIS WITH NOD FACTORS SUCH AS GLUCOSAMINE OLIGOSACCHARIDES Parish, Christopher Richard (AU) 2008-01-02 EP disclosed
US-20070297980-A1 Geldanamycin and Derivatives Inhibit Cancer Invasion and Identify Novel Targets MICHIGAN STATE UNIVERSITY 2007-12-27 US disclosed
US-20070299081-A1 Heterocyclic Derivatives and Their Use as Mediators of Stearoyl-Coa Desaturase XENON PHARMACEUTICALS INC. (CA) 2007-12-27 US disclosed
EP-1869022-A1 NAPHTHALAMIDE DERIVATIVES HAVING ANTIPROLIFERATIVE ACTIVITY Agency for Science, Technology and Research (SG) 2007-12-26 EP disclosed
EP-1868995-A1 COPPER COMPLEXES MEDICAL THERAPIES LIMITED (AU) 2007-12-26 EP disclosed
US-7312194-B2 Delivery systems ALCHEMIA PTY. LTD. (AU) 2007-12-25 US disclosed
WO-2007144370-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-12-21 WO disclosed
US-20070292477-A1 Association of Antimicrobial Compounds with Surfaces and Polymers BIOSIGNAL LIMITED (AT) 2007-12-20 US disclosed
US-20070293399-A1 SUBSTITUTED DIAMINO-1,3,5-TRIAZINES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND CROP GROWTH REGULATORS BAYER CROPSCIENCE AG (DE) 2007-12-20 US disclosed
US-20070287836-A1 Method for Preparing Compounds Comprising Cucurbituril Groups NEWSOUTH INNOVATIONS PTY LIMITED (AU) 2007-12-13 US disclosed
US-20070287700-A1 Polycyclic agents for the treatment of respiratory syncytial virus infections BIOTA SCIENTFIC MANAGEMENMT PTY LTD. (AU) 2007-12-13 US disclosed
US-20070287855-A1 Process for Preparing Fluorinated Molecules BAYER CROPSCIENCE AG (DE) 2007-12-13 US disclosed
WO-2007143597-A2 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2007-12-13 WO disclosed
WO-2007136746-A2 MACROCYCLIC COMPOUNDS AND THEIR USES AS STEAROYL-COA DESATURASE XENON PHARMACEUTICALS INC. (CA) 2007-11-29 WO disclosed
WO-2007134362-A1 2-ARYLPYRAZOLO[L,5-α]PYRIMIDIN-3-YL ACETAMIDE DERIVATIVES AS LIGANDS FOR TRANSLOCATOR PROTEIN (18 KDA) THE UNIVERSITY OF SYDNEY (AU) 2007-11-29 WO disclosed
WO-2007133777-A1 FURANONE ENDCAPPED POLYMERS TYCO HEALTHCARE GROUP LP (US) 2007-11-22 WO disclosed
WO-2007133783-A1 HALOGENATED CYCLIC LACTONES AND POLYMERS MADE THEREFROM TYCO HEALTHCARE GROUP LP (US) 2007-11-22 WO disclosed
WO-2007133782-A1 ANTIMICROBIAL COATINGS TYCO HEALTHCARE GROUP LP (US) 2007-11-22 WO disclosed
WO-2007133781-A2 FURANONE-INITIATED POLYMERS TYCO HEALTHCARE GROUP LP (US) 2007-11-22 WO disclosed
US-20070265240-A1 Sequence Selective Pyrrole and Imidazole Polyamide Metallocomplexes UNIVERSITY OF WESTERN SYDNEY (AU) 2007-11-15 US disclosed
WO-2007128782-A1 SPIRO- (THO) BENZOPYRAN-2, 4' -PIPERIDINE-AND CYCLOHEXANE DERIVATIVES AS INHIBITORS OF SPECIFIC CELL CYCLE ENZYMES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-11-15 WO disclosed
WO-2007130075-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2007-11-15 WO disclosed
EP-1689706-A4 ALPHA, BETA-UNSATURATED SULFOXIDES FOR TREATING PROLIFERATIVE DISORDERS UNIV TEMPLE (US) 2007-11-14 EP disclosed
EP-1851205-A2 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-11-07 EP disclosed
WO-2007118276-A1 METHOD OF TREATMENT OF AGE-RELATED MACULAR DEGENERATION(AMD) PRANA BIOTECHNOLOGY LTD (AU) 2007-10-25 WO disclosed
EP-1846035-A2 COMBINATION THERAPY XENON PHARMACEUTICALS INC. (CA) 2007-10-24 EP disclosed
US-20070244134-A1 Selective antagonists of A2A adenosine receptors ADENOSINE THERAPEUTICS, LLC 2007-10-18 US disclosed
WO-2007117394-A2 COMPOSITIONS AND METHODS RELATED TO FRUCTOSAMINE-3-KINASE INHIBITORS DYNAMIS THERAPEUTICS, INC. (US) 2007-10-18 WO disclosed
EP-1844009-A1 COMPOSITIONS AND METHODS FOR TREATING CARDIOVASCULAR DISORDERS Stocker, Roland O. (AU) 2007-10-17 EP disclosed
EP-1844020-A1 HETEROCYCLIC CARBOXAMIDE COMPOUNDS AS STEROID NUCLEAR RECEPTOR LIGANDS Exelixis, Inc. (US) 2007-10-17 EP disclosed
WO-2007112492-A1 COMPOUNDS AND METHODS FOR THE TREATMENT OF PAIN THE UNIVERSITY OF QUEENSLAND (AU) 2007-10-11 WO disclosed
WO-2007113687-A2 CAMPTOTHECIN-CELL PENETRATING PEPTIDE CONJUGATES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME DIATOS S.A. (FR) 2007-10-11 WO disclosed
WO-2007112503-A1 POLYMER PRODUCT AND INTERFACIAL POLYMERISATION PROCESS USING RAFT AGENT THE UNIVERSITY OF SYDNEY (AU) 2007-10-11 WO disclosed
WO-2007110745-A1 COMBINATION THERAPY FOR TREATMENT OF CANCER MEDICAL THERAPIES LIMITED (AU) 2007-10-04 WO disclosed
US-20070232627-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. 2007-10-04 US disclosed
US-20070232604-A1 receptor kinase inhibitors such as 3-(2-{4-[3-(5-tert-Butyl-isoxazol-3-yl)-ureido]-phenyl}-benzo[d]imidazo[2,1-b]thiazol-7-yl)-N-(2-morpholin-4-yl-ethyl)-propionamide; flk inhibitors AMBIT BIOSCIENCES CORPORATION 2007-10-04 US disclosed
WO-2007109845-A1 PROPHYLAXIS OR TREATMENT OF DIABETES MEDICAL THERAPIES LIMITED (AU) 2007-10-04 WO disclosed
WO-2007109843-A1 METAL COMPLEXES HAVING ANTI-INFLAMMATORY ACTIVITY MEDICAL THERAPIES LIMITED (AU) 2007-10-04 WO disclosed
WO-2007109844-A1 ANTI-INFLAMMATORY METAL COMPLEXES MEDICAL THERAPIES LIMITED (AU) 2007-10-04 WO disclosed
US-20070232645-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. 2007-10-04 US disclosed
EP-1838772-A2 METHOD FOR TRANSFORMATION OF CONVENTIONAL AND COMMERCIALLY IMPORTANT POLYMERS INTO DURABLE AND RECHARGEABLE ANTIMICROBIAL POLYMERIC MATERIALS Board of Regents, The University of Texas System (US) 2007-10-03 EP disclosed
EP-1838714-A1 METHODS OF TREATING PAIN THE UNIVERSITY OF QUEENSLAND (AU) 2007-10-03 EP disclosed
EP-1734945-A4 A COMPOSITION CONTAINING A COMPLEX COMPRISING A METAL ION AND A CARBOXYLATE LIGAND HAVING ANTI-INFLAMMATORY ACTIVITY MEDICAL THERAPIES LTD (AU) 2007-10-03 EP disclosed
US-20070225377-A1 Bridged Ring Structures as Pharmaceutical Agents X-CEPTOR THERAPEUTICS, INC. (US) 2007-09-27 US disclosed
WO-2007109120-A2 IMIDAZOLOTHIAZOLE COMPOUNDS FOR THE TREATMENT OF DISEASE AMBIT BIOSCIENCES CORPORATION (US) 2007-09-27 WO disclosed
WO-2007109324-A2 POTENT AND SELECTIVE NAV 1.7 SODIUM CHANNEL BLOCKERS XENON PHARMACEUTICALS, INC. (CA) 2007-09-27 WO disclosed
US-20070219211-A1 Bicyclic Heterocyclic Derivatives and Their Use as Inhibitors of Stearoyl-Coadesaturase (Scd) XENON PHARMACEUTICALS INC. (CA) 2007-09-20 US disclosed
WO-2007103548-A2 NOVEL ANTIBIOTIC COMPOSITIONS INFLAZYME PHARMACEUTICALS LTD. (CA) 2007-09-13 WO disclosed
US-20070213375-A1 Triazole derivatives useful as Axl inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2007-09-13 US disclosed
US-7268140-B2 Piperazine derivatives and their use as anti-inflammatory agents SCHERING AG (DE) 2007-09-11 US disclosed
EP-1827438-A2 PYRIDINE DERIVATIVES FOR INHIBITING HUMAN STEAROYL-COA-DESATURASE XENON PHARMACEUTICALS INC. (CA) 2007-09-05 EP disclosed
EP-1689698-A4 BIS-CATIONIC COMPOUNDS AND USE THEREOF UNIV SYDNEY (AU) 2007-09-05 EP disclosed
US-7265093-B2 Drug therapy for Celiac Sprue THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2007-09-04 US disclosed
US-7265131-B2 Isoquinolinone derivatives and their use as therapeutic agents EXELIXIS, INC. (US) 2007-09-04 US disclosed
US-20070203143-A1 PROTEIN KINASE INHIBITORS ABBVIE INC. 2007-08-30 US disclosed
WO-2007095696-A1 POLYKETIDE XANTHONES AND USES THEREOF THE UNIVERSITY OF QUEENSLAND (AU) 2007-08-30 WO disclosed
US-20070197558-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. 2007-08-23 US disclosed
US-20070196270-A1 Compounds As Ccri Antagonists HENG RICHARD 2007-08-23 US disclosed
EP-1343488-B1 TREATMENT OF STATIN SIDE EFFECTS MAGRAL LTD (AU) 2007-08-15 EP disclosed
EP-1817041-A2 TAFI INHIBITORS AND THEIR USE TO TREAT PULMONARY FIBROSIS Bayer Schering Pharma Aktiengesellschaft (DE) 2007-08-15 EP disclosed
EP-1814551-A2 PYRIDAZINE DERIVATIVES FOR INHIBITING HUMAN STEAROYL-COA-DESATURASE XENON PHARMACEUTICALS INC. (CA) 2007-08-08 EP disclosed
EP-0980867-B1 KETONE DERIVATIVES AND MEDICINAL USE THEREOF TORAY INDUSTRIES (JP) 2007-08-08 EP disclosed
WO-2007085042-A1 NOVEL LACTAMS BIOSIGNAL LIMITED (AU) 2007-08-02 WO disclosed
EP-1809281-A2 USE OF EPOTHILONES IN THE TREATMENT OF BONE METASTASES AND BONE TUMORS OR CANCERS Bayer Schering Pharma Aktiengesellschaft (DE) 2007-07-25 EP disclosed
WO-2007081517-A2 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2007-07-19 WO disclosed
EP-1807085-A2 HETEROCYCLIC DERIVATIVES AND THEIR USE AS STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2007-07-18 EP disclosed
EP-1608623-A4 METAL ION CHELATORS AND THERAPEUTIC USE THEREOF NEWSOUTH INNOVATIONS PTY LTD (AU) 2007-07-18 EP disclosed
US-7244741-B2 Fredericamycin derivatives as medicaments for treating tumours BIOFRONTERA DISCOVERY GMBH (DE) 2007-07-17 US disclosed
WO-2007079164-A2 PROTEIN KINASE INHIBITORS ABBOTT LABORATORIES (US) 2007-07-12 WO disclosed
WO-2007079003-A2 AMIDE INHIBITORS OF LEUKOTRIENE A4 HYDROLASE BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-07-12 WO disclosed
WO-2007079078-A1 DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-07-12 WO disclosed
EP-1804792-A1 BICYCLIC HETEROCYCLIC DERIVATIVES AND THEIR USE AS INHIBITORS OF STEAROYL-COA-DESATURASE (SCD) XENON PHARMACEUTICALS INC. (CA) 2007-07-11 EP disclosed
EP-1539675-A4 ARYL AND HETEROARYL PROPENE AMIDES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF UNIV TEMPLE (US) 2007-07-11 EP disclosed
EP-1805154-A2 PHARMACEUTICAL COMPOSITIONS Exelixis, Inc. (US) 2007-07-11 EP disclosed
EP-1558617-A4 AMIDINE COMPOUNDS UNIV MONASH (AU) 2007-07-11 EP disclosed
EP-1804799-A2 HETEROCYCLIC DERIVATIVES AND THEIR USE AS STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2007-07-11 EP disclosed
CN-1325476-C Preparation of fused polycyclic alkaloids by ring closure of azomethine ylides, noval compounds thereof and their use as chemotherapeutic agents UNIV AUSTRALIAN (AU) 2007-07-11 CN disclosed
US-20070155726-A1 Diamine derivatives as inhibitors of leukotriene A4 hydrolase SCHERING AKTIENGESELLSCHAFT (DE) 2007-07-05 US disclosed
WO-2007075145-A1 BENZOPYRANONE DERIVATIVES AND THEIR USE AS ANTI-CORONAVIRAL AGENTS SINGAPORE POLYTECHNIC (SG) 2007-07-05 WO disclosed
WO-2007076035-A2 ANTI-VIRAL COMPOUNDS ABBOTT LABORATORIES (US) 2007-07-05 WO disclosed
US-20070155727-A1 Amide inhibitors of leukotriene A4 hydrolase SCHERING AKTIENGESSELLSCHAFT (DE) 2007-07-05 US disclosed
US-20070155834-A1 Acetylenic aryl sulfonate hydroxamic acid tace and matrix metalloproteinase inhibitors WYETH HOLDINGS CORPORATION (US) 2007-07-05 US disclosed
WO-2007076379-A2 4,7-DIHYDROTHIENO[2,3-B]PYRIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS GILEAD COLORADO, INC. (US) 2007-07-05 WO disclosed
EP-1802662-A1 SURFACE POLYMERISATION PROCESS AND POLYMER PRODUCT USING RAFT AGENT The University of Sydney (AU) 2007-07-04 EP disclosed
EP-1802590-A1 SUBSTITUTED N-ALKYLPYRIMIDINONES Pharmacia & Upjohn Company LLC (US) 2007-07-04 EP disclosed
WO-2007070947-A1 ANTIBACTERIAL AGENTS ALCHEMIA LTD (AU) 2007-06-28 WO disclosed
US-20070149530-A1 For treatment of picornavirus infections in mammals BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2007-06-28 US disclosed
WO-2007073555-A1 USE OF 4, 7-DIHYDROTHIENO [2, 3-B] PYRIDINE COMPOUNDS IN THE TREATMENT OF CARDIOVASCULAR DISEASES GILEAD COLORADO, INC. (US) 2007-06-28 WO disclosed
US-20070148124-A1 Cellulose and acrylic based polymers and the use thereof for the treatment of infectious diseases NOVAFLUX INC. 2007-06-28 US disclosed
EP-1799739-A1 GELS AorTech Biomaterials Pty Ltd (AU) 2007-06-27 EP disclosed
EP-1799664-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2007-06-27 EP disclosed
EP-1799668-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS MEDIATORS OF STEAROYL-COA DESATURASE XENON PHARMACEUTICALS INC. (CA) 2007-06-27 EP disclosed
EP-1799667-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-06-27 EP disclosed
US-20070142353-A1 ANTIBACTERIAL COMPOUNDS ABBVIE INC. 2007-06-21 US disclosed
WO-2007069068-A2 CELL PENETRATING PEPTIDE CONJUGATES FOR DELIVERING NUCLEIC ACIDS INTO CELLS DIATOS (FR) 2007-06-21 WO disclosed
US-20070140970-A1 Cell targeting conjugates PETER MACCALLUM CANCER INSTITUTE 2007-06-21 US disclosed
EP-1797428-A1 SELECTIVE INHIBITORS Alchemia Pty Ltd (AU) 2007-06-20 EP disclosed
EP-1797901-A1 Cell penetrating peptide conjugates for delivering nucleic acids into cells Diatos (FR) 2007-06-20 EP disclosed
CN-1321644-C Process for preparing substituted pyrazoles PHARMACIA CORP (US) 2007-06-20 CN disclosed
WO-2007067781-A2 9-MEMBERED HETEROBICYCLIC COMPOUNDS AS INHIBITORS OF PROTEIN KINASES ABBOTT LABORATORIES (US) 2007-06-14 WO disclosed
US-20070135387-A1 Inhibitors of protein kinases ABBOTT LABORATORIES 2007-06-14 US disclosed
US-20070135392-A1 Apoptosis promoters ABBVIE INC. 2007-06-14 US disclosed
EP-1794164-A2 BRIDGED PIPERAZINE AND PIPERIDINE DERIVATIVES AS CCR1 ANTAGONISTS Novartis AG (CH) 2007-06-13 EP disclosed
US-20070129399-A1 Tetrahydroisoquinoline-and tetrahydrobenzazepine derivatives as igf-1r inhibitors ANALYTECON S.A. (CH) 2007-06-07 US disclosed
WO-2007059584-A1 METHODS FOR WOUND HEALING PEPLIN RESEARCH PTY LTD (AU) 2007-05-31 WO disclosed
EP-1789079-A1 ENZYME INHIBITORS AND USES THEREOF HOWARD FLOREY INSTITUTE OF EXPERIMENTAL PHYSIOLOGY AND MEDICINE (AU) 2007-05-30 EP disclosed
US-7223798-B2 Lipoxin A4 analogs SCHERING AKTIENGESELLSCHAFT (DE) 2007-05-29 US disclosed
US-7220881-B2 Process for production of acid anhydride TOKUYAMA CORPORATION (JP) 2007-05-22 US disclosed
US-7217702-B2 Selective antagonists of A2A adenosine receptors ADENOSINE THERAPEUTICS, LLC (US) 2007-05-15 US disclosed
WO-2007051255-A1 PROCESS FOR THE PREPARATION OF COMPOUNDS CONTAINING AN AZACYCLIC RING SYSTEM THE UNIVERSITY OF SYDNEY (AU) 2007-05-10 WO disclosed
US-20070105862-A1 Heat-shock protein binders ABBOTT LABORATORIES 2007-05-10 US disclosed
US-20070105820-A1 Oxindole compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2007-05-10 US disclosed
US-20070105949-A1 Intermediates for the preparation of lipoxin A4 analogs SCHERING AKTIENGESELLSCHAFT (DE) 2007-05-10 US disclosed
EP-1334092-B1 PROCESS FOR PREPARATION OF BICYCLIC AND POLYCYCLIC MOLECULES UNIV MONASH (AU) 2007-05-09 EP disclosed
WO-2007050124-A1 FUSED PIPERIDINE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-05-03 WO disclosed
WO-2007050795-A2 TRANSGLUTAMINASE INHIBITORS AND METHODS OF USE THEREOF ALVINE PHARMACEUTICALS, INC. (US) 2007-05-03 WO disclosed
WO-2007046868-A2 THIAZOLIDINE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-04-26 WO disclosed
WO-2007046867-A2 PIPERIDINE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-04-26 WO disclosed
WO-2007044085-A2 HETEROARYL COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-04-19 WO disclosed
US-20070087363-A1 Therapeutic methods, compounds and compositions MYRIAD GENETICS, INCORPORATED (US) 2007-04-19 US disclosed
US-20070088040-A1 Antibacterial compounds ABBVIE INC. 2007-04-19 US disclosed
EP-1773768-A2 PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS Exelixis, Inc. (US) 2007-04-18 EP disclosed
EP-1773337-A2 MODULATORS OF NUCLEAR RECEPTORS Exelixis, Inc. (US) 2007-04-18 EP disclosed
US-20070082850-A1 Mannose-6-phosphonate compounds for the treatment of inflammatory diseases PHARMAXIX PTY LTD (AU) 2007-04-12 US disclosed
WO-2007038829-A1 METHOD OF DRUG DESIGN ALCHEMIA LTD (AU) 2007-04-12 WO disclosed
US-20070077201-A1 Stem cell expansion and uses BIOVIE INC. 2007-04-05 US disclosed
US-7199155-B2 Acetylenic aryl sulfonate hydroxamic acid TACE and matrix metalloproteinase inhibitors WYETH HOLDINGS CORPORATION (US) 2007-04-03 US disclosed
US-7199129-B2 Derivatives of morphine-like opioid compounds MONASH UNIVERSITY (AU) 2007-04-03 US disclosed
US-20070072860-A1 N-acylsulfonamide derivatives; BCL-X1 protein inhibitors; anticarcinogenic agents; bladder cancer; for example, N-(4-(4-((4'-chloro(1,1'-biphenyl)-2-yl)methyl)piperazin-1-yl)benzoyl)-4-(((1R)-3-(dimethylamino)-1-((phenylsulfanyl)methyl)-propyl)amino)-3-nitrobenzenesulfonamide ABBOTT LABORATORIES 2007-03-29 US disclosed
US-20070072833-A1 Survivin inhibitors ABBVIE INC. 2007-03-29 US disclosed
EP-1765755-A1 REGULATORS OF BACTERIAL SIGNALLING PATHWAYS Biosignal Limited (AU) 2007-03-28 EP disclosed
US-7196200-B2 Antibacterial compounds ABBOTT LABORATORIES (US) 2007-03-27 US disclosed
EP-1483253-A4 AN ANTIMICROBIAL AGENT UNIV GRIFFITH (AU) 2007-03-21 EP disclosed
EP-1763350-A1 NICOTINAMIDE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-03-21 EP disclosed
WO-2007030680-A2 TRIAZOLE DERIVATIVES USEFUL AS AXL INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2007-03-15 WO disclosed
WO-2007029107-A1 ISOQUINOLINES DERIVATIVES AS IGF-1R INHIBITORS ANALYTECON SA (CH) 2007-03-15 WO disclosed
US-20070060551-A1 Methods of using isothiazole derivatives to treat cancer or inflammation QLT, INC. (CA) 2007-03-15 US disclosed
WO-2007026240-A1 SUNSCREEN AND COSMETIC COMPOSITIONS FOR PROPHYLAXIS OR TREATMENT OF SKIN CANCERS MEDICAL THERAPIES LIMITED (AU) 2007-03-08 WO disclosed
WO-2007024744-A2 HETEROCYCLIC CARBOXAMIDE COMPOUNDS AS STEROID NUCLEAR RECEPTOR LIGANDS EXELIXIS, INC. (US) 2007-03-01 WO disclosed
WO-2007025247-A2 TRANSGLUTAMINASE INHIBITORS AND METHODS OF USE THEREOF THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2007-03-01 WO disclosed
WO-2007022561-A1 METHODS OF ALTERING POPPY CHARACTERISTICS GLAXOSMITHKLINE AUSTRALIA PTY LTD (AU) 2007-03-01 WO disclosed
EP-1755373-A1 METHOD OF ALTERING THE ALKALOID COMPOSITION IN POPPY PLANTS Glaxosmithkline Australia PTY Ltd. (AU) 2007-02-28 EP disclosed
WO-2007022512-A2 GLYCOPEGYLATED FACTOR VII AND FACTOR VIIA NEOSE TECHNOLOGIES, INC. (US) 2007-02-22 WO disclosed
EP-1754703-A2 N-Heterocyclic derivatives as nos inhibitors Berlex, Inc. (US) 2007-02-21 EP disclosed
US-20070037864-A1 Intermediates for the preparation of lipoxin A4 analogs SCHERING AKTIENGESELLSCHAFT (DE) 2007-02-15 US disclosed
US-7176207-B2 Anticoagulants; antithrombotic agents in the treatment and prevention of thrombosis SCHERING AKTIENGESELLSCHAFT (DE) 2007-02-13 US disclosed
EP-1749041-A2 CELLULOSE AND ACRYLIC BASED POLYMERS AND THE USE THEREOF FOR THE TREATMENT OF INFECTIOUS DISEASES Nova Flux Biosciences, Inc. (US) 2007-02-07 EP disclosed
US-20070027285-A1 Polyurethanes COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2007-02-01 US disclosed
CN-1297537-C Sulfonium salt compound WAKO PURE CHEM IND LTD (JP) 2007-01-31 CN disclosed
WO-2007010201-A2 MEDICAL DEVICES AND COATINGS THEREFOR ASTON UNIVERSITY (GB) 2007-01-25 WO disclosed
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
US-7166604-B2 N-Heterocyclic derivatives; picornavirus infections in mammals; human rhinovirus BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2007-01-23 US disclosed
US-20070015787-A1 Apoptosis promoters ABBVIE INC. 2007-01-18 US disclosed
WO-2007008627-A2 APOPTOSIS PROMOTERS ABBOTT LABORATORIES (US) 2007-01-18 WO disclosed
US-20070014719-A1 Steroid analogs and characterization and treatment methods BIOVIE INC. 2007-01-18 US disclosed
CN-1898247-A Polycyclic agents for the treatment of respiratory syncytial virus infection BIOTA SCIENT MAN (AU) 2007-01-17 CN disclosed
EP-1740587-A2 SELECTIVE ANTAGONISTS OF A-2A- ADENOSINE RECEPTORS Adenosine Therapeutics, LLC (US) 2007-01-10 EP disclosed
US-7161031-B2 Amino-substituted sulfonanilides and derivatives thereof for treating proliferative disorders TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2007-01-09 US disclosed
WO-2007002559-A1 PYRAZOLE BASED LXR MODULATORS EXELIXIS, INC. (US) 2007-01-04 WO disclosed
WO-2007001240-A1 SURFACE TREATMENT OF ALUMINA FILMS NATIONAL UNIVERSITY OF SINGAPORE (SG) 2007-01-04 WO disclosed
WO-2007002563-A1 IMIDAZOLE BASED LXR MODULATORS EXELIXIS, INC. (US) 2007-01-04 WO disclosed
EP-1737825-A1 GELDANAMYCIN AND DERIVATIVES INHIBIT CANCER INVASION AND IDENTIFY NOVEL TARGETS Van Andel Research Institute (US) 2007-01-03 EP disclosed
US-20060293308-A1 Pyridyl derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2006-12-28 US disclosed
EP-1734945-A1 A COMPOSITION CONTAINING A COMPLEX COMPRISING A METAL ION AND A CARBOXYLATE LIGAND HAVING ANTI-INFLAMMATORY ACTIVITY THE UNIVERSITY OF SYDNEY (AU) 2006-12-27 EP disclosed
WO-2006134074-A2 PROCESS FOR SYNTHESIS OF DIALKOXYORGANOBORANES BASF AKTIENGESELLSCHAFT (DE) 2006-12-21 WO disclosed
US-20060287224-A1 Conjugates between erythropoietin and polyoxyethylene glycol groups, linked via an intact glycosyl linking group interposed between and covalently attached to the peptide and the modifying group; enhancing red blood cell production; treating a tissue injury NEOSE TECHNOLOGIES, INC. (US) 2006-12-21 US disclosed
US-20060287307-A1 Antibacterial compounds HINMAN MIRA M 2006-12-21 US disclosed
US-20060280746-A1 (1E)-1-{[(3-amino-4-methoxyphenyl)methyl]sulfinyl}-2-(2,4,6-trimethoxyphenyl)ethene; antiproliferative agents; offers protection from the cytotoxic effects of ionizing radiation and of cytotoxic chemotherapeutic agents ONCONOVA THERAPEUTICS INC. 2006-12-14 US disclosed
US-20060281798-A1 Methods of using thiazolidinedithione derivatives QLT INC. (CA) 2006-12-14 US disclosed
EP-1727526-A2 PIPERAZINE UREA DERIVATIVES FOR THE TREATMENT OF ENDOMETRIOSIS Schering Aktiengesellschaft (DE) 2006-12-06 EP disclosed
WO-2006127910-A2 GLYCOPEGYLATED ERYTHROPOIETIN FORMULATIONS NEOSE TECHNOLOGIES, INC. (US) 2006-11-30 WO disclosed
WO-2006127364-A1 APOPTOSIS PROMOTERS ABBOTT LABORATORIES (US) 2006-11-30 WO disclosed
EP-1725558-A1 METHOD FOR PREPARING COMPOUNDS COMPRISING CUCURBITURIL GROUPS Newsouth Innovations Pty Limited (AU) 2006-11-29 EP disclosed
CN-1871247-A Novel sulfenamides UNIV GRIFFITH (AU) 2006-11-29 CN disclosed
CN-1871248-A Novel sulfenamide oxides UNIV GRIFFITH (AU) 2006-11-29 CN disclosed
WO-2006125180-A1 PIPERAZINE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-11-23 WO disclosed
WO-2006125194-A2 PIPERAZINE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-11-23 WO disclosed
WO-2006125181-A2 PIPERIDINE DERIVATIVES AND THEIR USE AS STEAROYL-COA DESATURASE MODULATORS XENON PHARMACEUTICALS INC. (CA) 2006-11-23 WO disclosed
WO-2006122344-A1 POLYMERISATION AGENT NEWSOUTH INNOVATIONS PTY LTD (AU) 2006-11-23 WO disclosed
WO-2006125178-A2 TRICYCLIC PYRIDAZINE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-11-23 WO disclosed
WO-2006125179-A1 TRICYCLIC COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-11-23 WO disclosed
US-7138418-B2 For therapy of atherosclerosis and hypercholesterolemia; 5-Pentafluorophenylsulfonamidoindazole for example; increasing LDL receptor gene expression in a cell AMGEN, INC. (US) 2006-11-21 US disclosed
US-20060258657-A1 Apoptosis promoters ABBVIE INC. 2006-11-16 US disclosed
US-20060258659-A1 Heterocyclic compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2006-11-16 US disclosed
EP-0968206-B1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LAB (US) 2006-11-15 EP disclosed
US-7135468-B2 Antibacterial compounds ABBOTT LABORATORIES (US) 2006-11-14 US disclosed
US-20060252812-A1 Spiro-oxindole compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2006-11-09 US disclosed
US-20060252798-A1 Metal ion chelators and therapeutic use thereof RICHARDSON, DESI (AU) 2006-11-09 US disclosed
WO-2006116817-A1 PESTICIDAL FORMULATIONS AKHIL TECHNOLOGIES PTY LTD (AU) 2006-11-09 WO disclosed
US-20060252767-A1 Piperazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2006-11-09 US disclosed
US-20060252758-A1 Spiroheterocyclic compounds and their uses as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2006-11-09 US disclosed
US-20060247210-A1 such as (4-Benzothiazol-2-yl-1H-pyrazol-3-yl)-[2-(1H-imidazol-4-yl)-ethyl]-amine, used in the treatment of disorders associated with hyperproliferation and tissue remodelling or repair, inflammation, cell migration and invasion, and renal diseases, or as protein kinase inhibitors QLT INC. (CA) 2006-11-02 US disclosed
US-20060247213-A1 Plasma carboxypeptidase b inhibitors SCHERING AKTIENGESELLSCHAFT (DE) 2006-11-02 US disclosed
WO-2006113875-A2 2 - PYRROLIDONE DERIVATIVES AND THEIR USES FOR THE TREATMENT OF INFLAMMATORY CONDITIONS AND PAIN XENON PHARMACEUTICALS INC. (CA) 2006-10-26 WO disclosed
WO-2006113247-A1 USE OF TAFI INHIBITORS FOR ENHANCED MYOCARDIAL REPERFUSION AND FACILITATED PCI BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2006-10-26 WO disclosed
WO-2006113864-A2 OXINDOLE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-10-26 WO disclosed
EP-1713483-A1 CHEMOKINE INHIBITING PIPERAZINE DERIVATIVES AND THEIR USE TO TREAT MULTIPLE MYELOMA Schering Aktiengesellschaft (DE) 2006-10-25 EP disclosed
US-20060234986-A1 Use of TAFI inhibitors for enhanced myocardial reperfusion and facilitated PCI SCHERING AKTIENGESELLSCHAFT (DE) 2006-10-19 US disclosed
WO-2006110917-A2 SPIRO-OXINDOLE COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-10-19 WO disclosed
WO-2006110918-A1 PYRROLE COMPOUNDS AND USES THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2006-10-19 WO disclosed
WO-2006110112-A2 STABILISER COMPOSITION FOR HALIDE-CONTAINING POLYMERS SUN ACE KAKOH (PTE.) LTD. (SG) 2006-10-19 WO disclosed
WO-2006110654-A1 SPIROHETEROCYCLIC COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-10-19 WO disclosed
US-20060235061-A1 Methods of using benzothiophenone derivatives to treat cancer or inflammation QLT,INC. (CA) 2006-10-19 US disclosed
EP-1078010-B1 NON-ELASTOMERIC POLYURETHANE COMPOSITIONS AORTECH BIOMATERIALS PTY LTD (AU) 2006-10-18 EP disclosed
US-7122570-B2 Tetrahydrocarbazol derivatives as ligands for G-protein-coupled receptors (GPCR) ZENTARIS AG (DE) 2006-10-17 US disclosed
US-7122571-B2 Substituted hydrazones as inhibitors of cyclooxygenase-2 TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2006-10-17 US disclosed
US-7122694-B2 Hydroboronation process BORON MOLECULAR PTY LIMITED (AU) 2006-10-17 US disclosed
US-7122699-B2 Process for preparing organic boronic acid derivatives using diboronic acid BORON MOLECULAR LIMITED (AU) 2006-10-17 US disclosed
WO-2006108149-A2 SUBSTITUTED BENZYLAMINES AS CYP2A INHIBITORS AND USES THEREOF TO TREAT NICOTINE DEPENDENCE INFLAZYME PHARMACEUTICALS LTD. (CA) 2006-10-12 WO disclosed
US-20060229310-A1 Antibacterial compounds ABBOTT LABORATORIES 2006-10-12 US disclosed
US-7119203-B2 Piperidinyl- and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors PHARMACIA CORPORATION (US) 2006-10-10 US disclosed
WO-2006104461-A1 NAPHTHALAMIDE DERIVATIVES HAVING ANTIPROLIFERATIVE ACTIVITY AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2006-10-05 WO disclosed
WO-2006102717-A1 MODULATING ANGIOGENESIS WITH NOD FACTORS SUCH AS GLUCOSAMINE OLIGOSACCHARIDES PARISH CHRISTOPHER RICHARD (AU) 2006-10-05 WO disclosed
US-20060223936-A1 Polymerization of a dispersion having a continuous aqueous phase and a dispersed organic phase of an unsaturated monomer(s), and an amphiphilic RAFT agent, which is an addition polymer residue capped with a compound containing a dithio ester or a trithiocarbonate group; paint, filler, adhesive, seals UNIVERSITY OF SYDNEY (AU) 2006-10-05 US disclosed
EP-1423392-B1 DERIVATIVES OF MORPHINE-LIKE OPIOID COMPOUNDS NEURO THERAPEUTICS LTD (AU) 2006-10-04 EP disclosed
EP-1706129-A1 DRUG THERAPY FOR CELIAC SPRUE The Board of Trustees of The Leland Stanford Junior University (US) 2006-10-04 EP disclosed
CN-1277855-C Novel fluoroalkyl polymers containing cationic segment 3M INNOVATIVE PROPERTIES CO (US) 2006-10-04 CN disclosed
US-7115632-B1 Sulfonyl aryl or heteroaryl hydroxamic acid compounds G. D. SEARLE & CO. (US) 2006-10-03 US disclosed
WO-2006101521-A2 HETEROCYCLIC DERIVATIVES AND THEIR USE AS STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2006-09-28 WO disclosed
WO-2006099685-A1 METHOD FOR THE PROPHYLAXIS OR TREATMENT OF CARCINOMAS MEDICAL THERAPIES LIMITED (AU) 2006-09-28 WO disclosed
WO-2006099677-A1 METAL COMPLEXES MEDICAL THERAPIES LIMITED (AU) 2006-09-28 WO disclosed
WO-2006099684-A1 COPPER COMPLEXES MEDICAL THERAPIES LIMITED (AU) 2006-09-28 WO disclosed
EP-1701988-A1 POLYURETHANES COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2006-09-20 EP disclosed
US-20060205713-A1 Antidiabetic agents; disease of glucose tolerance; insulin resistance; obesity; dyslipidemia; metabolic disorders; liver disorders; [4-(6-Phenethyloxy-pyridazin-3-yl)piperazin-1-yl]-(2-trifluoromethyl-phenyl)-methanone; stearoyl-CoA desaturase modulators XENON PHARMACEUTICALS INC. (CA) 2006-09-14 US disclosed
US-7105563-B2 Indolinone derivatives and their use in treating disease-states such as cancer SCHERING AKTIENGESELLSCHAFT (DE) 2006-09-12 US disclosed
WO-2006093518-A2 THIENYL COMPOUNDS FOR TREATING VIRUS-RELATED CONDITIONS APATH, LLC (US) 2006-09-08 WO disclosed
US-20060199802-A1 Pyridyl derivatives and their use as therapeutic agents DISCOVERY PARTNERS INTERNATIONAL, INC. 2006-09-07 US disclosed
EP-1697377-A1 POLYCYCLIC AGENTS FOR THE TREATMENT OF RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2006-09-06 EP disclosed
EP-1515943-B1 USE OF ALKYLAMIDOMANDELATES AS FLAVOURINGS SYMRISE GMBH & CO KG (DE) 2006-08-30 EP disclosed
WO-2006086447-A2 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-08-17 WO disclosed
WO-2006086445-A2 COMBINATION THERAPY XENON PHARMACEUTICALS INC. (CA) 2006-08-17 WO disclosed
US-20060183782-A1 Methods of using thiazolidine derivatives to treat cancer or inflammation QLT INC. (CA) 2006-08-17 US disclosed
EP-1689698-A1 BIS-CATIONIC COMPOUNDS AND USE THEREOF THE UNIVERSITY OF SYDNEY (AU) 2006-08-16 EP disclosed
EP-1534284-A4 AMINO-SUBSTITUTED SULFONANILIDES AND DERIVATIVES THEREOF FOR TREATING PROLIFERATIVE DISORDERS UNIV TEMPLE (US) 2006-08-16 EP disclosed
EP-1689388-A1 ASSOCIATION OF ANTIMICROBIAL COMPOUNDS WITH SURFACES AND POLYMERS Biosignal Limited (AU) 2006-08-16 EP disclosed
EP-1689706-A2 ALPHA, BETA-UNSATURATED SULFOXIDES FOR TREATING PROLIFERATIVE DISORDERS Temple University of the Commonwealth System of Higher Education (US) 2006-08-16 EP disclosed
EP-1689743-A2 PIPERIDINYL-AND PIPERAZINYL-SULFONYLMETHYL HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS Pharmacia Corporation (US) 2006-08-16 EP disclosed
US-7091338-B2 Purification of 4,4′(5′)- di-t-butylcyclohexano-18-crown-6 PG RESEARCH FOUNDATION (US) 2006-08-15 US disclosed
US-20060173004-A1 1-(4-Benzyl-piperazin-1-yl)-3-phenyl-propenone derivatives NOVARTIS AG (CH) 2006-08-03 US disclosed
EP-1685119-A1 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS Abbott Laboratories (US) 2006-08-02 EP disclosed
US-20060167271-A1 Purified compounds that inhibit intracellular alphax4/paxillin binding GINSBERG MARK 2006-07-27 US disclosed
US-20060167317-A1 Aryl and heteroaryl propene amides, derivatives thereof and therapeutic uses thereof TEMPLE UNIVERSITY- OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2006-07-27 US disclosed
US-20060167000-A1 Neurologically-active compounds PRANA BIOTECHNOLOGY LIMITED (AU) 2006-07-27 US disclosed
WO-2006076202-A1 HETEROCYCLIC CARBOXAMIDE COMPOUNDS AS STEROID NUCLEAR RECEPTORS LIGANDS EXELIXIS, INC. (US) 2006-07-20 WO disclosed
EP-1680401-A2 INDOLINONE DERIVATIVES AND THEIR USE IN TREATING DISEASE-STATES SUCH AS CANCER Schering Aktiengesellschaft (DE) 2006-07-19 EP disclosed
US-7078403-B1 Antiviral agents BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2006-07-18 US disclosed
WO-2006074455-A2 METHOD FOR TRANSFORMATION OF CONVENTIONAL AND COMMERCIALLY IMPORTANT POLYMERS INTO DURABLE AND RECHARGEABLE ANTIMICROBIAL POLYMERIC MATERIALS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2006-07-13 WO disclosed
EP-1678133-A1 SEQUENCE SELECTIVE PYRROLE AND IMIDAZOLE POLYAMIDE METALLOCOMPLEXES University of Western Sydney (AU) 2006-07-12 EP disclosed
US-20060148848-A1 Compounds and methods for treating cancer and inflammation QLT, INC. 2006-07-06 US disclosed
EP-1675812-A2 BRIDGED RING STRUCTURES AS PHARMACEUTICAL AGENTS X-Ceptor Therapeutics, Inc. (US) 2006-07-05 EP disclosed
WO-2006066362-A1 METHODS OF TREATING PAIN THE UNIVERSITY OF QUEENSLAND (AU) 2006-06-29 WO disclosed
EP-1539700-A4 8-HYDROXY QUINOLINE DERIVATIVES PRANA BIOTECHNOLOGY LTD (AU) 2006-06-28 EP disclosed
CN-1795185-A Process for preparing substituted pyrazoles PHARMACIA CORP (US) 2006-06-28 CN disclosed
US-7067670-B2 Sulfamato hydroxamic acid metalloprotease inhibitor WARNER LAMBERT COMPANY (US) 2006-06-27 US disclosed
US-20060135532-A1 Platelet adenosine diphosphate receptor antagonists SCHERING AKTIENGESELLSCHAFT (DE) 2006-06-22 US disclosed
US-20060135487-A1 Piperazine derivatives and their use as anti-inflammatory agents BAUMAN JOHN G 2006-06-22 US disclosed
WO-2006063408-A1 COMPOSITIONS AND METHODS FOR TREATING CARDIOVASCULAR DISORDERS STOCKER RONALD O (AU) 2006-06-22 WO disclosed
US-20060128706-A1 Apoptosis promoters ABBVIE INC. 2006-06-15 US disclosed
US-20060128608-A1 Novel chemical compounds and their use BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2006-06-15 US disclosed
EP-1664071-A1 NOVEL SULFENAMIDE OXIDES GRIFFITH UNIVERSITY (AU) 2006-06-07 EP disclosed
EP-1664072-A1 NOVEL SULFENAMIDES GRIFFITH UNIVERSITY (AU) 2006-06-07 EP disclosed
EP-1296673-A4 ANTIMICROBIAL COATINGS UNISEARCH LTD (AU) 2006-06-07 EP disclosed
US-7057049-B2 Process for making substituted pyrazoles PHARMACIA CORPORATION (US) 2006-06-06 US disclosed
EP-1660089-A1 CHEMOKINE INHIBITING PIPERAZINE DERIVATIVES AND THEIR USE TO TREAT MYOCARDITIS SCHERING AKTIENGESELLSCHAFT (DE) 2006-05-31 EP disclosed
US-20060111309-A1 Chalcomycin derivatives BIOFRONTERA DISCOVERY GMBH (DE) 2006-05-25 US disclosed
US-20060111381-A1 Amidine compounds MONASH UNIVERSITY (AU) 2006-05-25 US disclosed
US-20060105995-A1 TAFI inhibitors and their use to treat pulmonary fibrosis SCHERING AKTIENGESELLSCHAFT (DE) 2006-05-18 US disclosed
EP-1463765-A4 AQUEOUS DISPERSIONS OF POLYMER PARTICLES UNIV SYDNEY (AU) 2006-05-10 EP disclosed
WO-2006047269-A2 PHARMACEUTICAL COMPOSITIONS EXELIXIS, INC. (US) 2006-05-04 WO disclosed
EP-1651605-A2 PYRIDYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-05-03 EP disclosed
EP-1651606-A2 PYRIDYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-05-03 EP disclosed
EP-1651616-A2 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-05-03 EP disclosed
EP-1651620-A2 PIPERAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-05-03 EP disclosed
US-20060089380-A1 8-Hydroxy quinoline derivatives PRANA BIOTECHNOLOGY LTD. (AU) 2006-04-27 US disclosed
EP-1648874-A2 PIPERAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-04-26 EP disclosed
US-20060083678-A1 Radio-labeled compounds, compositions, and methods of making the same NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2006-04-20 US disclosed
WO-2006025979-A9 MODULATORS OF NUCLEAR RECEPTORS EXELIXIS INC (US) 2006-04-20 WO disclosed
US-20060083858-A1 Generation of surface coating diversity ANTEO TECHNOLOGIES PTY LTD (AU) 2006-04-20 US disclosed
WO-2006040666-A1 SUBSTITUTED N-ALKYLPYRIMIDINONES PHARMACIA & UPJOHN COMPANY LLC (US) 2006-04-20 WO disclosed
US-20060084688-A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor BARTA THOMAS E 2006-04-20 US disclosed
WO-2006041808-A2 TAFI INHIBITORS AND THEIR USE TO TREAT PULMONARY FIBROSIS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2006-04-20 WO disclosed
EP-1487428-A4 AMINO-SUBSTITUTED (E)-2,6-DIALKOXYSTYRYL 4-SUBSTITUTED BENZYLSULFONES FOR TREATING PROLIFERATIVE DISORDERS UNIV TEMPLE (US) 2006-04-19 EP disclosed
WO-2006037159-A1 SELECTIVE INHIBITORS ALCHEMIA LIMITED (AU) 2006-04-13 WO disclosed
WO-2006037161-A1 SURFACE POLYMERISATION PROCESS AND POLYMER PRODUCT USING RAFT AGENT THE UNIVERSITY OF SYDNEY (AU) 2006-04-13 WO disclosed
WO-2006037185-A1 NOVEL SULFENAMIDES AND SULFENAMIDE OXIDES GRIFFITH UNIVERSITY (AU) 2006-04-13 WO disclosed
US-7026323-B2 Platelet adenosine diphosphate receptor antagonists SCHERING AKTIENGESELLSCHAFT (DE) 2006-04-11 US disclosed
US-7026423-B2 Silicon-based polycarbonates AORTECH BIOMATERIALS PTY LTD. (AU) 2006-04-11 US disclosed
US-20060074243-A1 Hydroxamic acid and amide compounds and their use as protease inhibitors PHARMACIA CORPORATION 2006-04-06 US disclosed
WO-2006034547-A1 GELS AORTECH BIOMATERIALS PTY LTD (AU) 2006-04-06 WO disclosed
WO-2006032537-A2 USE OF EPOTHILONES IN THE TREATMENT OF BONE METASTASES AND BONE TUMORS OR CANCERS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2006-03-30 WO disclosed
WO-2006034441-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2006-03-30 WO disclosed
WO-2006034312-A1 BICYCLIC HETEROCYCLIC DERIVATIVES AND THEIR USE AS INHIBITORS OF STEAROYL-COA-DESATURASE (SCD) XENON PHARMACEUTICALS INC. (CA) 2006-03-30 WO disclosed
WO-2006034446-A2 PYRIDINE DERIVATIVES FOR INHIBITING HUMAN STEAROYL-COA-DESATURASE XENON PHARMACEUTICALS INC. (CA) 2006-03-30 WO disclosed
WO-2006034279-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-03-30 WO disclosed
US-20060069136-A1 Use of Epothilones in the treatment of bone metastasis BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2006-03-30 US disclosed
WO-2006034338-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS MEDIATORS OF STEAROYL-COA DESATURASE XENON PHARMACEUTICALS INC. (CA) 2006-03-30 WO disclosed
WO-2006034440-A2 HETEROCYCLIC DERIVATIVES AND THEIR USE AS STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2006-03-30 WO disclosed
WO-2006034341-A2 PYRIDAZINE DERIVATIVES FOR INHIBITING HUMAN STEAROYL-COA-DESATURASE XENON PHARMACEUTICALS INC. (CA) 2006-03-30 WO disclosed
EP-1640004-A1 Use of epothilones in the treatment of bone metastases and bone tumors or cancers Schering Aktiengesellschaft (DE) 2006-03-29 EP disclosed
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed
US-7019000-B1 Method of treating a disease condition caused or exacerbated by an HPV INSTITUTE OF MOLECULAR & CELL BIOLOGY (SG) 2006-03-28 US disclosed
WO-2006026832-A1 ENZYME INHIBITORS AND USES THEREOF HOWARD FLOREY INSTITUTE OF EXPERIMENTAL PHYSIOLOGY AND MEDICINE (AU) 2006-03-16 WO disclosed
US-7012142-B2 Process for preparation of bicyclic and polycyclic molecules MONASH UNIVERSITY (AU) 2006-03-14 US disclosed
US-20060052308-A1 Administering to a patient an effective dose of [(S)-1-[(3-Bromo-4,5-dihydro-isoxazol-5-ylmethyl)-methyl-carbamoyl]-2-(4-hydroxy-phenyl)-ethyl]-carbamic acid benzyl ester; treatment of glioblastoma, meningioma, melanoma and colon cancer THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2006-03-09 US disclosed
WO-2006025979-A2 MODULATORS OF NUCLEAR RECEPTORS EXELIXIS, INC. (US) 2006-03-09 WO disclosed
WO-2006024068-A1 POLYMER COMPOSITE THE UNIVERSITY OF QUEENSLAND (AU) 2006-03-09 WO disclosed
EP-1628987-A2 MANNOSE-6-PHOSPHONATE COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISEASES Pharmaxis Pty Ltd. (AU) 2006-03-01 EP disclosed
US-20060035838-A1 Drug therapy for celiac sprue THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2006-02-16 US disclosed
WO-2006014168-A1 NICOTINAMIDE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-02-09 WO disclosed
US-6995156-B2 Platelet adenosine diphosphate receptor antagonists SCHERING AKTIENGESELLSCHAFT (DE) 2006-02-07 US disclosed
WO-2006012642-A2 PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS EXELIXIS, INC. (US) 2006-02-02 WO disclosed
EP-1621533-A1 Preparation of fused polycyclic alkaloids by ring closure of azomethine ylides, novel compounds thereof and their use as chemotherapeutic agents THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2006-02-01 EP disclosed
EP-1615866-A1 INDENE DERIVATIVES AS PHARMACEUTICAL AGENTS Inflazyme Pharmaceuticals, Ltd. (CA) 2006-01-18 EP disclosed
US-20060009459-A1 Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2006-01-12 US disclosed
EP-1613616-A2 PROCESS FOR MAKING SUBSTITUTED PYRAZOLES Pharmacia Corporation (US) 2006-01-11 EP disclosed
WO-2005123645-A1 REGULATORS OF BACTERIAL SIGNALLING PATHWAYS BIOSIGNAL LIMITED (AU) 2005-12-29 WO disclosed
EP-1478760-A4 ESTERASES WITH LIPASE ACTIVITY COMMW SCIENT IND RES ORG (AU) 2005-12-28 EP disclosed
EP-1379508-A4 N-(ARYL)-2-ARYLETHENESULFONAMIDES AND THERAPEUTIC USES THEREOF UNIV TEMPLE (US) 2005-12-28 EP disclosed
EP-1332138-B1 RADIOPHARMACEUTICALS FOR DIAGNOSING ALZHEIMER'S DISEASE SCHERING AG (DE) 2005-12-28 EP disclosed
EP-1608623-A1 METAL ION CHELATORS AND THERAPEUTIC USE THEREOF UNISEARCH LIMITED (AU) 2005-12-28 EP disclosed
US-20050282831-A1 Selective antagonists of A2A adenosine receptors ADENOSINE THERAPEUTICS, LLC 2005-12-22 US disclosed
US-6977258-B2 Piperazine derivatives and their use as anti-inflammatory agents SCHERING AKTIENGESELLSCHAFT (DE) 2005-12-20 US disclosed
US-20050272709-A1 Immugenic compositions and diagnostic and therapeutic uses thereof DERMIRA (CANADA), INC. 2005-12-08 US disclosed
US-6972290-B2 Piperazine derivatives and their use as anti-inflammatory agents SCHERING AKTIENGESELLSCHAFT (DE) 2005-12-06 US disclosed
WO-2005111112-A2 CELLULOSE AND ACRYLIC BASED POLYMERS AND THE USE THEREOF FOR THE TREATMENT OF INFECTIOUS DISEASES NOVA FLUX BIOSCIENCES, INC. (US) 2005-11-24 WO disclosed
WO-2005107436-A1 METHOD OF ALTERING THE ALKALOID COMPOSITION IN POPPY PLANTS GLAXOSMITHKLINE AUSTRALIA PTY LTD (AU) 2005-11-17 WO disclosed
US-20050256066-A1 Water soluble groups on ring A; antitumor antibiotics; 1-Desoxy-5-C-[(8R)-4',9,9'-trihydroxy-6'-methoxy-1,1',3',5',8'-pentaoxo-1,1',2,3',5',6,7,8'-octahydrospiro[cyclopenta[g]isoquinoline-8,2'-cyclopenta[b]-naphthalene]-3-yl]pentitol; topoisomerase inhibitors; cyclodextrin inclusions; stereoisomers BIOFRONTERA DISCOVERY GMBH (DE) 2005-11-17 US disclosed
US-20050256150-A1 Enantioselective acyl transfer catalysts and their use in kinetic resolution of alcohols and desymmetrization of meso-diols WASHINGTON UNIVERSITY 2005-11-17 US disclosed
EP-0981517-B1 PREPARATION OF FUSED POLYCYCLIC ALKALOIDS BY RING CLOSURE OF AZOMETHINE YLIDES UNIV AUSTRALIAN (AU) 2005-11-16 EP disclosed
CN-1227229-C Ethylene derivatives and pesticides containing the same NISSAN CHEMICAL IND LTD (JP) 2005-11-16 CN disclosed
US-20050250674-A1 Nutritional and food supplement preparation comprising creatine and orotic acid complexes, derivatives and analogs AMATO DANIEL 2005-11-10 US disclosed
US-6962929-B2 Pentafluorobenzenesulfonamides and analogs TULARIK INC. (US) 2005-11-08 US disclosed
WO-2005103054-A2 BRIDGED PIPERAZINE AND PIPERIDINE DERIVATIVES AS CCRI ANTAGONISTS NOVARTIS AG (CH) 2005-11-03 WO disclosed
US-6958145-B2 Synthesis of cyclic compounds UNISEARCH LIMITED (AU) 2005-10-25 US disclosed
US-20050234053-A1 9-oxo-3,4,6,9-tetrahydro-2H-[1,4]-(oxazino, thiazino, or pyrazino)[3,2-b][1,8]naphthyridine-8-carboxylic acids; fish or mammals; bacterial protein biosynthesis inhibitors ABBVIE INC. 2005-10-20 US disclosed
WO-2005097140-A2 SELECTIVE ANTAGONISTS OF A2A ADENOSINE RECEPTORS ADENOSINE THERAPEUTICS, LLC (US) 2005-10-20 WO disclosed
WO-2005094809-A1 A COMPOSITION CONTAINING A COMPLEX COMPRISING A METAL ION AND A CARBOXYLATE LIGAND HAVING ANTI-INFLAMMATORY ACTIVITY MEDICAL THERAPIES LIMITED (AU) 2005-10-13 WO disclosed
WO-2005095347-A1 GELDANAMYCIN AND DERIVATIVES INHIBIT CANCER INVASION AND IDENTIFY NOVEL TARGETS VAN ANDEL RESEARCH INSTITUTE (US) 2005-10-13 WO disclosed
CN-1678602-A 2-oxabicyclo [3.3.0] octane compounds, process for producing the same, optical resolution agent, process for separating diastereomer mixture, and process for optically resolving alcohol ZEON CORP (JP) 2005-10-05 CN disclosed
US-20050215772-A1 Furanone derivatives and methods of making same BIOSIGNAL LIMITED (AT) 2005-09-29 US disclosed
US-20050215579-A1 Fredericamycin derivatives as medicaments for treating tumours BIOFRONTERA DISCOVERY GMBH (DE) 2005-09-29 US disclosed
WO-2005090351-A1 METHOD FOR PREPARING COMPOUNDS COMPRISING CUCURBITURIL GROUPS NEWSOUTH INNOVATIONS PTY LIMITED (AU) 2005-09-29 WO disclosed
CN-1220676-C Method for producing acid anhydride TOKUYAMA CORP (JP) 2005-09-28 CN disclosed
US-20050208084-A1 Use of alkylamidomandelates as flavourings SYMRISE GMBH & CO. KG (DE) 2005-09-22 US disclosed
US-20050209278-A1 Piperidinyl- and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors PHARMACIA CORPORATION 2005-09-22 US disclosed
EP-1572660-A1 ISOQUINOLINONE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS X-Ceptor Therapeutics, Inc. (US) 2005-09-14 EP disclosed
EP-1476149-A4 SUBSTITUTED HYDRAZONES AS INHIBITORS OF CYCLOOXYGENASE-2 UNIV TEMPLE (US) 2005-09-14 EP disclosed
EP-1112250-A4 THERAPEUTIC COMPOUNDS AND METHODS INST OF MOLECUL & CELL BIOLOGY (SG) 2005-09-14 EP disclosed
WO-2005082873-A2 1,4-BENZOTHIAZEPANS AND DERIVATIVES THEREOF BIOAGENCY AG (DE) 2005-09-09 WO disclosed
WO-2005079769-A2 PIPERAZINE DERIVATIVES FOR THE TREATMENT OF ENDOMETRIOSIS SCHERING AKTIENGESELLSCHAFT (DE) 2005-09-01 WO disclosed
US-20050192282-A1 Chemokine inhibiting piperazine derivatives and their use to treat multiple myeloma SCHERING AKTIENGESELLSCHAFT (DE) 2005-09-01 US disclosed
US-20050191385-A1 Natural product derivatives as food supplements and pharmaceuticals AMATO DANIEL K (US) 2005-09-01 US disclosed
WO-2005080549-A2 TRIOXACARCINS AND THEIR USE AGAINST INFECTIONS BIOFRONTERA DISCOVERY GMBH (DE) 2005-09-01 WO disclosed
WO-2005077372-A1 CHEMOKINE INHIBITING PIPERAZINE DERIVATIVES AND THEIR USE TO TREAT MULTIPLE MYELOMA SCHERING AKTIENGESELLSCHAFT (DE) 2005-08-25 WO disclosed
EP-1565459-A2 HETEROARYLSULFONYLMETHYL HYDROXAMIC ACIDS AND AMIDES AND THEIR USE AS PROTEASE INHIBITORS Pharmacia Corporation (US) 2005-08-24 EP disclosed
CN-1215835-C Ketone derivatives and medical use thereof TORAY INDUSTRIES (JP) 2005-08-24 CN disclosed
CN-1216056-C Sulfamidohydroxamic acid metalloprotease inhibitor SEARLE & CO (US) 2005-08-24 CN disclosed
WO-2005075527-A1 HYPERBRANCHED POLYMERS THE GENERAL HOSPITAL CORPORATION (US) 2005-08-18 WO disclosed
WO-2005075477-A1 ANTIBACTERIAL COMPOUNDS ABBOTT LABORATORIES (US) 2005-08-18 WO disclosed
EP-1534755-A4 GENERATION OF SURFACE COATING DIVERSITY BIO LAYER PTY LTD (AU) 2005-08-17 EP disclosed
EP-1562928-A1 AROMATIC SULFONE HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS Pharmacia Corporation (US) 2005-08-17 EP disclosed
US-20050176118-A1 Esterases with lipase activity COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2005-08-11 US disclosed
WO-2005072731-A1 3-PHENYL-N- ((1, 3, 4) THIADIAZOL-2-YL) -ACRYLAMIDE DERIVATIVES AND RELATED COMPOUNDS AS MODULATORS OF ESTROGEN-RELATED RECEPTORS FOR THE TREATMENT OF E.G. CANCER, RHEUMATOID ARTHRITIS OR NEUROLOGICAL DISORDERS X-CEPTOR THERAPEUTICS, INC. (US) 2005-08-11 WO disclosed
EP-1558585-A1 NEUROLOGICALLY-ACTIVE COMPOUNDS Prana Biotechnology Ltd (AU) 2005-08-03 EP disclosed
EP-1558594-A2 1-(4-BENZYL-PIPERAZIN-1-YL)-3-PHENYL-PROPENONE DERIVATIVES Novartis AG (CH) 2005-08-03 EP disclosed
EP-1558617-A1 AMIDINE COMPOUNDS Monash University (AU) 2005-08-03 EP disclosed
US-20050164999-A1 Benzamides and compositions benzamides for use as fungicizide E. I. DU PONT DE NEMOURS AND COMPANY 2005-07-28 US disclosed
US-20050159423-A1 Antibacterial compounds ABBOTT LABORATORIES 2005-07-21 US disclosed
US-20050159427-A1 N-acylsulfonamide apoptosis promoters ABBOTT LABORATORIES 2005-07-21 US disclosed
US-20050154004-A1 Preparation of fused polycyclic alkaloids by ring closure of azomethine ylides, novel compounds thereof and their use as chemotherapeutic agents AUSTRALIAN NATIONAL UNIVERSITY, THE (AU) 2005-07-14 US disclosed
US-20050153997-A1 Fredericamycin derivatives BIOFRONTERA DISCOVERY GMBH (DE) 2005-07-14 US disclosed
US-6916805-B2 Quinoxalinones as serine protease inhibitors WARNER-LAMBERT COMPANY LLC (US) 2005-07-12 US disclosed
WO-2005061485-A1 PROCESS FOR MAKING SUBSTITUTED PYRAZOLES PHARMACIA CORPORATION (US) 2005-07-07 WO disclosed
WO-2005061513-A1 POLYCYCLIC AGENTS FOR THE TREATMENT OF RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2005-07-07 WO disclosed
US-20050148669-A1 Amino acid esters as nutrient supplements and methods of use AMATO DANIEL (US) 2005-07-07 US disclosed
EP-1542997-A2 PYRAZOLYLBENZOTHIAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS QLT, Inc. (CA) 2005-06-22 EP disclosed
US-20050130942-A1 Amino-substituted (e)-2,6-dialkoxystyryl 4-substituted-benzylsulfones for treating proliferative disorders TEMPLE UNIVERSITY OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2005-06-16 US disclosed
US-20050130221-A1 Synthesis for the preparation of compounds for screening as potential tubulin binding agents THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2005-06-16 US disclosed
WO-2005053684-A1 ASSOCIATION OF ANTIMICROBIAL COMPOUNDS WITH SURFACES AND POLYMERS BIOSIGNAL LIMITED (AU) 2005-06-16 WO disclosed
EP-1539700-A1 8-HYDROXY QUINOLINE DERIVATIVES Prana Biotechnology Ltd (AU) 2005-06-15 EP disclosed
EP-1539675-A2 ARYL AND HETEROARYL PROPENE AMIDES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF Temple University of the Commonwealth System of Higher Education (US) 2005-06-15 EP disclosed
WO-2005052019-A1 POLYURETHANES COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2005-06-09 WO disclosed
US-20050124559-A1 Antimicrobial agent UNIVERSITY, MONASH (AU) 2005-06-09 US disclosed
WO-2005051960-A2 HYDROCARBYL AMINOHYDROCARBONOATES AND AMINOHYDROCARBONOL HYDROCARBONOATES AS ANTIMICROBIAL AND ANTIVIRAL AGENTS MIDWEST RESEARCH LABORATORIES, LLC (US) 2005-06-09 WO disclosed
EP-1121365-B1 ORGANOBORON DERIVATIVES AND PROCESS FOR COUPLING ORGANIC COMPOUNDS COMMW SCIENT IND RES ORG (AU) 2005-06-08 EP disclosed
EP-1019414-B1 PROCESS FOR PREPARING ORGANIC BORONIC ACID DERIVATIVES USING DIBORONIC ACID COMMW SCIENT IND RES ORG (AU) 2005-06-08 EP disclosed
CN-1205198-C Cyclic ketone derivative and pharmaceutical use thereof TORAY INDUSTRIES (JP) 2005-06-08 CN disclosed
US-20050119461-A1 Novel receptor, and compounds which bind thereto THE UNIVERSITY OF MELBOURNE 2005-06-02 US disclosed
WO-2005049064-A1 DRUG THERAPY FOR CELIAC SPRUE THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2005-06-02 WO disclosed
WO-2005049593-A2 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS ABBOTT LABORATORIES (US) 2005-06-02 WO disclosed
US-20050119251-A1 Nicotinamide derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2005-06-02 US disclosed
WO-2005049594-A1 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS ABBOTT LABORATORIES (US) 2005-06-02 WO disclosed
EP-1534284-A2 AMINO-SUBSTITUTED SULFONANILIDES AND DERIVATIVES THEREOF FOR TREATING PROLIFERATIVE DISORDERS Temple University of the Commonwealth System of Higher Education (US) 2005-06-01 EP disclosed
EP-1534755-A1 GENERATION OF SURFACE COATING DIVERSITY Bio-Layer Pty Limited (AU) 2005-06-01 EP disclosed
WO-2005046599-A2 ALPHA, BETA-UNSATURATED SULFOXIDES FOR TREATING PROLIFERATIVE DISORDERS TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2005-05-26 WO disclosed
US-20050113274-A1 Hydrocarbyl aminohydrocarbonoates and aminohydrocarbonol hydrocarbonoates as antimicrobial and antiviral agents MIDWEST RESEARCH LABORATORIES, LLC 2005-05-26 US disclosed
WO-2005047230-A1 BIS-CATIONIC COMPOUNDS AND USE THEREOF THE UNIVERSITY OF SYDNEY (AU) 2005-05-26 WO disclosed
EP-1254899-B1 Piperazine derivatives and their use as anti-inflammatory agents SCHERING AG (DE) 2005-05-25 EP disclosed
US-6897318-B2 Process for making substituted pyrazoles PHARMACIA CORPORATION (US) 2005-05-24 US disclosed
WO-2005042521-A2 PIPERIDINYL-AND PIPERAZINYL-SULFONYLMETHYL HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2005-05-12 WO disclosed
US-20050101641-A1 Aromatic sulfone hydroxamic acids and their use as protease inhibitors PHARMACIA CORPORATION 2005-05-12 US disclosed
CN-1615303-A Improved purification process for 4,4 '(5') -di-tert-butylcyclohexa-18-crown-6 PG RES FOUNDATION (US) 2005-05-11 CN disclosed
US-6890937-B2 Aromatic sulfone hydroxamic acid metalloprotease inhibitor PHARMACIA CORPORATION (US) 2005-05-10 US disclosed
US-6890928-B2 Aromatic sulfone hydroxamic acids and their use as protease inhibitors PHARMACIA CORPORATION (US) 2005-05-10 US disclosed
WO-2005040116-A2 INDOLINONE DERIVATIVES AND THEIR USE IN TREATING DISEASE-STATES SUCH AS CANCER SCHERING AKTIENGESELLSCHAFT (DE) 2005-05-06 WO disclosed
US-20050096484-A1 Amino-substituted sulfonanilides and derivatives thereof for treating proliferative disorders ONCONOVA THERAPEUTICS, INC. 2005-05-05 US disclosed
US-6887865-B2 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2005-05-03 US disclosed
WO-2005037755-A2 BRIDGED RING STRUCTURES AS PHARMACEUTICAL AGENTS X-CEPTOR THERAPEUTICS, INC. (US) 2005-04-28 WO disclosed
US-20050090541-A1 Indolinone derivatives and their use in treating disease-states such as cancer SCHERING AKTIENGESELLSCHAFT (DE) 2005-04-28 US disclosed
US-20050080111-A1 Modulators of LXR X-CEPTOR THERAPEUTICS, INC. (US) 2005-04-14 US disclosed
WO-2005033077-A1 SEQUENCE SELECTIVE PYRROLE AND IMIDAZOLE POLYAMIDE METALLOCOMPLEXES UNIVERSITY OF WESTERN SYDNEY (AU) 2005-04-14 WO disclosed
EP-1521577-A1 METHODS OF USING ISOTHIAZOLE DERIVATIVES TO TREAT CANCER OR INFLAMMATION QLT, Inc. (CA) 2005-04-13 EP disclosed
US-6878690-B2 Compounds and methods PHARMAXIS PTY LTD. (AU) 2005-04-12 US disclosed
US-20050075374-A1 Sulfonyl aryl or heteroaryl hydroxamic acid compounds PHARMACIA CORPORATION 2005-04-07 US disclosed
EP-1519724-A1 FREDERICAMYCIN DERIVATIVES AS MEDICAMENTS FOR TREATING TUMOURS Biofrontera Pharmaceuticals Holding AG (DE) 2005-04-06 EP disclosed
US-6872381-B1 Radiopharmaceuticals for diagnosing Alzheimer's disease SCHERING AG (DE) 2005-03-29 US disclosed
US-20050065143-A1 Pyridazine derivatives and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2005-03-24 US disclosed
US-20050065163-A1 Platelet adenosine diphosphate receptor antagonists SCHERING AKTIENGESELLSCHAFT (DE) 2005-03-24 US disclosed
EP-1515951-A1 ARYLSULFONYLHYDROXAMIC ACID AND AMIDE DERIVATIVES AND THEIR USE AS PROTEASE INHIBITORS Pharmacia Corporation (US) 2005-03-23 EP disclosed
EP-1187859-A4 POLYMER GELS, METHODS FOR THEIR PREPARATION AND THEIR USE IN ELECTROPHORETIC APPLICATIONS UNIV MELBOURNE (AU) 2005-03-23 EP disclosed
EP-1515943-A1 USE OF ALKYLAMIDOMANDELATES AS FLAVOURINGS Symrise GmbH & Co. KG (DE) 2005-03-23 EP disclosed
US-20050054722-A1 Inhibition of two-component signal transduction systems UNISEARCH LIMITED, (AU) 2005-03-10 US disclosed
WO-2005021547-A2 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD. (AU) 2005-03-10 WO disclosed
EP-1511743-A1 PYRAZOLE-DERIVATIVES AS P38 KINASE INHIBITORS Pharmacia Corporation (US) 2005-03-09 EP disclosed
US-6864263-B2 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2005-03-08 US disclosed
US-6864368-B2 N-heterocyclic derivatives as NOS inhibitors BERLAX LABORATORIES, INC. (US) 2005-03-08 US disclosed
WO-2005018642-A1 CHEMOKINE INHIBITING PIPERAZINE DERIVATIVES AND THEIR USE TO TREAT MYOCARDITIS SCHERING AKTIENGESELLSCHAFT (DE) 2005-03-03 WO disclosed
WO-2005019237-A1 NOVEL SULFENAMIDES GRIFFITH UNIVERSITY (AU) 2005-03-03 WO disclosed
WO-2005019236-A1 NOVEL SULFENAMIDE OXIDES GRIFFITH UNIVERSITY (AU) 2005-03-03 WO disclosed
US-20050049280-A1 Sulfamato hydroxamic acid metalloprotease inhibitor PHARMACIA CORPORATION 2005-03-03 US disclosed
US-6861424-B2 Platelet adenosine diphosphate receptor antagonists SCHERING AKTIENGESELLSCHAFT (DE) 2005-03-01 US disclosed
US-20050043318-A1 Chemokine inhibiting piperazine derivatives and their use to treat myocarditis SCHERING AKTIEGESELLSCHAFT (DE) 2005-02-24 US disclosed
US-20050043533-A1 Process for making alpha-substituted hydroxamic acids PHARMACIA CORPORATION 2005-02-24 US disclosed
EP-1507772-A1 METHODS OF USING THIAZOLIDINEDITHIONE DERIVATIVES QLT, Inc. (CA) 2005-02-23 EP disclosed
EP-1507549-A2 DRUG THERAPY FOR CELIAC SPRUE The Board of Trustees of The Leland Stanford Junior University (US) 2005-02-23 EP disclosed
US-6858680-B2 Shape memory polyurethane or polyurethane-urea polymers AORTECH BIOMATERIALS PTY LTD (AU) 2005-02-22 US disclosed
US-20050038037-A1 Platelet adenosine diphosphate receptor antagonists SCHERING AKTIENGESELLSCHAFT (DE) 2005-02-17 US disclosed
EP-1506213-A1 AN ANTIMICROBIAL AGENT GRIFFITH UNIVERSITY (AU) 2005-02-16 EP disclosed
EP-1505970-A1 METHODS OF USING THIAZOLIDINE DERIVATIVES TO TREAT CANCER OR INFLAMMATION QLT Inc. (CA) 2005-02-16 EP disclosed
US-6855726-B1 Quinolones as serine protease inhibitors WARNER-LAMBERT COMPANY LLC (US) 2005-02-15 US disclosed
WO-2005011656-A2 PYRIDYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2005-02-10 WO disclosed
WO-2005011657-A2 PIPERAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2005-02-10 WO disclosed
WO-2005011654-A2 PYRIDYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2005-02-10 WO disclosed
WO-2005011655-A2 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2005-02-10 WO disclosed
WO-2005011653-A2 PYRIDAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2005-02-10 WO disclosed
EP-1453813-A4 IMPROVED PURIFICATION OF 4, 4'(5')-DI- i t /i -BUTYLCYCLOHEXANO-18-CROWN-6 PG RES FOUNDATION (US) 2005-02-09 EP disclosed
EP-0934310-B1 THIO ACID DERIVED MONOCYCLIC N-HETEROCYCLICS AS ANTICOAGULANTS SCHERING AG (DE) 2005-02-09 EP disclosed
EP-1294705-A4 SYNTHESIS OF CYCLIC COMPOUNDS UNISEARCH LTD (AU) 2005-02-09 EP disclosed
US-6852795-B2 Prepolymeric (meth)acrylates with polycyclic or aromatic segments 3M ESPE AG (DE) 2005-02-08 US disclosed
EP-1501827-A2 PIPERIDINYL-AND PIPERAZINYL-SULFONYLMETHYL HYDROXAMIC ACID AND THEIR USE AS PROTEASE INHIBITORS Pharmacia Corporation (US) 2005-02-02 EP disclosed
CN-1575176-A Process for preparing substituted pyrazoles PHARMACIA CORP (US) 2005-02-02 CN disclosed
US-6849739-B2 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2005-02-01 US disclosed
EP-0983267-B1 AMIDOAROMATIC RING SULFONAMIDE HYDROXAMIC ACID COMPOUNDS PHARMACIA CORP (US) 2005-01-26 EP disclosed
US-6846829-B2 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2005-01-25 US disclosed
US-20050014840-A1 Thiol sulfonamide metalloprotease inhibitors PHARMACIA CORPORATION 2005-01-20 US disclosed
US-20050013939-A1 Boron-based wood preservatives and treatment of wood with boron-based preservatives THE UNIVERSITY OF MELBOURNE (AU) 2005-01-20 US disclosed
EP-1497300-A2 PLASMA CARBOXYPEPTIDASE B INHIBITORS Schering Aktiengesellschaft (DE) 2005-01-19 EP disclosed
EP-0857067-A4 RADIOPROTECTORS PETER MACCALLUM CANCER INST (AU) 2005-01-19 EP disclosed
US-20050009838-A1 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors PHARMACIA CORPORATION 2005-01-13 US disclosed
EP-1495003-A1 FREDERICAMYCIN DERIVATIVES Biofrontera Discovery Gmbh (DE) 2005-01-12 EP disclosed
US-6841674-B2 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2005-01-11 US disclosed
US-6841673-B2 N-heterocyclic derivatives as nos inhibitors BERLEX LABORATORIES, INC. (US) 2005-01-11 US disclosed
US-20050000889-A1 Substrate with interstitial gaps having a polymeric membrane that is thinner than cross-sectional thickness of substrate SOLOMON DAVID HENRY (AU) 2005-01-06 US disclosed
US-20050004086-A1 Antiinflammatory agents; antiarthritic agents; brain disorders; multiple sclerosis; gout; inflammatory bowel disorders; gastrointestinal disorders; psoriasis; antiallergens; autoimmune disease INFLAZYME PHARMACEUTICALS LTD. (CA) 2005-01-06 US disclosed
EP-1353911-A4 ANTIVIRAL AGENTS BIOTA SCIENT MANAGEMENT (AU) 2005-01-05 EP disclosed
EP-1000108-B1 AQUEOUS POLYIMIDE PROCESS COMMW SCIENT IND RES ORG (AU) 2005-01-05 EP disclosed
EP-1284979-B1 PREPOLYMERIC (METH)ACRYLATES WITH POLYCYCLIC OR AROMATIC SEGMENTS 3M ESPE AG (DE) 2004-12-29 EP disclosed
EP-1487428-A2 AMINO-SUBSTITUTED (E)-2,6-DIALKOXYSTYRYL 4-SUBSTITUTED BENZYLSULFONES FOR TREATING PROLIFERATIVE DISORDERS Temple University of the Commonwealth System of Higher Education (US) 2004-12-22 EP disclosed
US-6831186-B2 Antiinflammatory agents; autoimmune disease SCHERING AKTIENGESELLSCHFT (DE) 2004-12-14 US disclosed
EP-1483253-A1 AN ANTIMICROBIAL AGENT GRIFFITH UNIVERSITY (AU) 2004-12-08 EP disclosed
US-20040242929-A1 Process for production of acid anhydride TOKUYAMA CORPORATION (JP) 2004-12-02 US disclosed
WO-2004104015-A2 MANNOSE-6-PHOSPHONATE COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISEASES PHARMAXIS PTY LTD. (AU) 2004-12-02 WO disclosed
US-20040242616-A1 Derivatives of morphine-like opioid compounds NEURO THERAPEUTICS LIMITED (AU) 2004-12-02 US disclosed
EP-0977745-B1 THIOARYL SULFONAMIDE HYDROXAMIC ACID COMPOUNDS PHARMACIA CORP (US) 2004-12-01 EP disclosed
US-20040235818-A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor PHARMACIA CORPORATION 2004-11-25 US disclosed
EP-1478760-A1 ESTERASES WITH LIPASE ACTIVITY COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2004-11-24 EP disclosed
EP-1476149-A2 SUBSTITUTED HYDRAZONES AS INHIBITORS OF CYCLOOXYGENASE-2 Temple University of the Commonwealth System of Higher Education (US) 2004-11-17 EP disclosed
EP-1423392-A4 DERIVATIVES OF MORPHINE-LIKE OPIOID COMPOUNDS POLYCHIP PHARMACEUTICALS PTY (AU) 2004-11-17 EP disclosed
US-6818718-B2 IMPROVED SEPARATION OF PROTEINS, ENZYMES, PEPTIDES, OLIGONUCLEOTIDES, POLYNUCLEOTIDES, AND CARBOHYDRATES THE UNIVERSITY OF MELBOURNE (AU) 2004-11-16 US disclosed
WO-2004096766-A1 A METHOD OF INDOLE SYNTHESIS THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2004-11-11 WO disclosed
EP-1472209-A2 LIPOXIN A4 ANALOGS SCHERING AKTIENGESELLSCHAFT (DE) 2004-11-03 EP disclosed
EP-1472244-A1 AROMATIC SULFONE HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS Pharmacia Corporation (US) 2004-11-03 EP disclosed
WO-2004091549-A2 PROCESS FOR MAKING ALPHA-SUBSTITUTED HYDROXAMIC ACIDS PHARMACIA CORPORATION (US) 2004-10-28 WO disclosed
WO-2004092100-A1 INDENE DERIVATIVES AS PHARMACEUTICAL AGENTS INFLAZYME PHARMACEUTICALS LTD. (CA) 2004-10-28 WO disclosed
EP-1005453-B1 SUBSTITUTED BENZENE COMPOUNDS AS ANTIPROLIFERATIVE LOWERING AGENTS TULARIK INC (US) 2004-10-27 EP disclosed
US-20040209914-A1 Aromatic sulfone hydroxamic acids and their use as protease inhibitors PHARMACIA CORPORATION 2004-10-21 US disclosed
US-20040204447-A1 Isoquinolinone derivatives and their use as therapeutic agents X-CEPTOR THERAPEUTICS INC. 2004-10-14 US disclosed
WO-2004087074-A2 PROCESS FOR MAKING SUBSTITUTED PYRAZOLES PHARMACIA CORPORATION (US) 2004-10-14 WO disclosed
CN-1537097-A Method for producing acid anhydride ��ʽ�����ɽ 2004-10-13 CN disclosed
WO-2004085551-A1 CORROSION INHIBITING COATING MONASH UNIVERSITY (AU) 2004-10-07 WO disclosed
EP-1463765-A1 AQUEOUS DISPERSIONS OF POLYMER PARTICLES University of Sydney (AU) 2004-10-06 EP disclosed
US-6800646-B1 Sulfamato hydroxamic acid metalloprotease inhibitor PHARMACIA CORPORATION 2004-10-05 US disclosed
US-6794511-B2 AN ENZYME INHIBITORS OF METALLOPROTEASE; TREATING CONNECTIVE TISSUE DEGRADATION CAUSED BY INFLAMMATION OR TUMOR G. D. SEARLE 2004-09-21 US disclosed
US-20040176281-A1 Delivery systems ALCHEMIA LIMITED (AU) 2004-09-09 US disclosed
EP-1453803-A2 TETRAHYDROCARBOZOLE DERIVATIVES AS LIGANDS FOR G-PROTEIN COUPLED RECEPTORS (GPCR) Zentaris GmbH (DE) 2004-09-08 EP disclosed
EP-1453813-A2 IMPROVED PURIFICATION OF 4, 4'(5')-DI- i t /i -BUTYLCYCLOHEXANO-18-CROWN-6 PG Research Foundation (US) 2004-09-08 EP disclosed
US-20040171516-A1 Precursors for ketones and aldehydes GIVAUDAN SA (CH) 2004-09-02 US disclosed
EP-1450791-A1 HYDRAZONOPYRAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTICS Kinetek Pharmaceuticals, Inc. (CA) 2004-09-01 EP disclosed
US-6783809-B2 LOW VISCOSITY PHOTOCURABLE COMPOSITIONS WHICH, WHEN FULLY CURED, GIVE MOULDED ARTICLES OF EXCELLENT FLEXIBILITY HUNTSMAN ADVANCED MATERIALS AMERICAS INC. 2004-08-31 US disclosed
US-20040167182-A1 Hydroxamic acid and amide compounds and their use as protease inhibitors PHARMACIA CORPORATION 2004-08-26 US disclosed
US-20040167069-A1 Drug therapy for Celiac Sprue NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2004-08-26 US disclosed
CN-1524095-A Novel fluoroalkyl polymers containing cationic segment 3M 2004-08-25 CN disclosed
WO-2004069801-A1 METAL ION CHELATORS AND THERAPEUTIC USE THEREOF UNISEARCH LIMITED (AU) 2004-08-19 WO disclosed
US-20040162433-A1 Lipoxin A4 analogs SCHERING AKTIENGESELLSCHAFT (DE) 2004-08-19 US disclosed
EP-1334092-A4 PROCESS FOR PREPARATION OF BICYCLIC AND POLYCYCLIC MOLECULES UNIV MONASH (AU) 2004-08-11 EP disclosed
WO-2004065334-A1 METHOD OF REMOVING ORGANOTIN RESIDUE CHIROGEN PTY LIMITED (AU) 2004-08-05 WO disclosed
WO-2004065335-A1 ENANTIOSELECTIVE REDUCTION METHOD CHIROGEN PTY LIMITED (AU) 2004-08-05 WO disclosed
US-20040147595-A1 Biofilm degrading or sloughing compositions and methods UNISEARCH LIMITED (AU) 2004-07-29 US disclosed
US-20040142979-A1 Heteroarylsulfonylmethyl hydroxamic acids and amides and their use as protease inhibitors PHARMACIA CORPORATION 2004-07-22 US disclosed
US-20040142877-A1 Ligands of the $g(a)v$g(b)6 integrin MERCK PATENT GMBH (DE) 2004-07-22 US disclosed
US-20040138488-A1 Benzene-1 2-diol mannich bases ligands polymers and method of selective metal ions removal TECHNOLOGICAL RESOURCES PTY LTD. (AU) 2004-07-15 US disclosed
WO-2004058717-A1 ISOQUINOLINONE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS X-CEPTOR THERAPEUTICS, INC. (US) 2004-07-15 WO disclosed
US-20040133028-A1 Hydroboronation process COMMONWEALTH SCIENTIFIC 2004-07-08 US disclosed
US-20040127524-A1 Acetylenic aryl sulfonate hydroxamic acid TACE and matrix metalloproteinase inhibitors WYETH HOLDINGS CORPORATION 2004-07-01 US disclosed
US-20040127539-A1 Antiangiogenic combination therapy for the treatment of cancer PHARMACIA CORPORATION 2004-07-01 US disclosed
WO-2004054988-A1 ARYLTHIOETHERPYRIMIDINE AND ARYLOXYETHERPYRIMIDINE DERIVATIVES AND THEIR THERAPEUTIC USES ACTIVE PASS PHARMACEUTICALS, INC. (CA) 2004-07-01 WO disclosed
EP-1429773-A1 PROCESS FOR MAKING SUBSTITUTED PYRAZOLES Pharmacia Corporation (US) 2004-06-23 EP disclosed
WO-2004050677-A1 NOVEL CHEMICAL COMPUNDS AND THEIR USE BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2004-06-17 WO disclosed
US-6750233-B2 SELECTIVITY PHARMACIA CORPORATION 2004-06-15 US disclosed
US-20040110727-A1 Aldehyde-releasing compounds LA TROBE UNIVERSITY (AU) 2004-06-10 US disclosed
WO-2004048368-A2 HETEROARYLSULFONYLMETHYL HYDROXAMIC ACIDS AND AMIDES AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2004-06-10 WO disclosed
US-20040110805-A1 Aromatic sulfone hydroxamic acids and their use as protease inhibitors PHARMACIA CORPORATION 2004-06-10 US disclosed
US-20040110966-A1 Synthesis of cyclic compounds UNISEARCH LIMITED (AU) 2004-06-10 US disclosed
US-6747031-B2 MUSCLE RELAXANTS, CONTROLLING IMMUNOLOGY, STROKES, ANTIDIABETIC AGENTS BERLEX LABORATORIES, INC. 2004-06-08 US disclosed
US-6747027-B1 SELECTIVELY INHIBITS IN VITRO ACTIVITY OF HUMAN MATRIX METALLOPROTEASE-13 OVER IN VITRO ACTIVITY OF HUMAN MATRIX METALLOPROTEASE-1 PHARMACIA CORPORATION 2004-06-08 US disclosed
EP-1423392-A1 DERIVATIVES OF MORPHINE-LIKE OPIOID COMPOUNDS Polychip Pharmaceuticals Pty. Ltd. (AU) 2004-06-02 EP disclosed
CN-1501827-A Ligands of the alpha-v-beta 6 integrin Ĭ��ר�����޹�˾ 2004-06-02 CN disclosed
WO-2004043350-A2 PURIFIED COMPOUNDS THAT INHIBIT INTRACELLULAR α4/PAXILLIN BINDING THE SCRIPPS RESEARCH INSTITUTE (US) 2004-05-27 WO disclosed
WO-2004043943-A1 AROMATIC SULFONE HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2004-05-27 WO disclosed
US-20040097487-A1 Aromatic sulfonyl alpha-cycloamino hydroxamic acid compounds G.D. SEARLE & CO. 2004-05-20 US disclosed
US-6737111-B2 POLYMERIC MEMBRANE COMPONENTS RESIDE WITHIN THE INTERSTITIAL GAPS OF THE SUBSTRATE; ULTRA-THIN; POLYMERIZATION AND CROSSLINKING OF POLYACRYLAMIDE GEL GRADIPORE LIMITED (AU) 2004-05-18 US disclosed
WO-2004037796-A2 1-(4-BENZYL-PIPERAZIN-1-YL)-3-PHENYL-PROPENONE DERIVATIVES NOVARTIS AG (CH) 2004-05-06 WO disclosed
WO-2004037751-A2 ARYL AND HETEROARYL PROPENE AMIDES, DERIVATIVES THEREOF AND THERAPEUTIC USES THEREOF TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2004-05-06 WO disclosed
EP-1414526-A2 ANTIANGIOGENIC COMBINATION THERAPY FOR THE TREATMENT OF CANCER Pharmacia Corporation (US) 2004-05-06 EP disclosed
US-20040082551-A1 Novel pyrazoles and their use as p38 kinase inhibitors PHARMACIA CORPORATION 2004-04-29 US disclosed
WO-2004035598-A2 CHALCOMYCIN DERIVATIVES BIOFRONTERA DISCOVERY GMBH (DE) 2004-04-29 WO disclosed
EP-1413572-A1 PROCESS FOR PRODUCING ACID ANHYDRIDE Tokuyama Corporation (JP) 2004-04-28 EP disclosed
EP-0888271-B1 BENZAMIDINE DERIVATIVES SUBSTITUTED BY AMINO ACID AND HYDROXY ACID DERIVATIVES AND THEIR USE AS ANTI-COAGULANTS BERLEX LAB (US) 2004-04-28 EP disclosed
CN-1147294-C Pentafluorobenzenesulfonamides and analogs �㽭�пؼ����ɷ����޹�˾ 2004-04-28 CN disclosed
WO-2004033458-A1 AMIDINE COMPOUNDS MONASH UNIVERSITY (AU) 2004-04-22 WO disclosed
US-20040077633-A1 N-Heterocyclic derivatives; picornavirus infections in mammals; human rhinovirus BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2004-04-22 US disclosed
WO-2004031198-A1 ENANTIOSELECTIVE REDUCTIVE METHODS USING CHIRAL ORGANOSTANNANES CHIROGEN PTY LIMITED (AU) 2004-04-15 WO disclosed
WO-2004031161-A1 NEUROLOGICALLY-ACTIVE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED (AU) 2004-04-15 WO disclosed
EP-1301522-A4 NOVEL COMPOUNDS AND METHODS PHARMAXIS PTY LTD (AU) 2004-04-14 EP disclosed
EP-1406602-A2 USE OF SULFONYL ARYL OR HETEROARYL HYDROXAMIC ACIDS AND DERIVATIVES THEREOF AS AGGRECANASE INHIBITORS Pharmacia Corporation (US) 2004-04-14 EP disclosed
EP-1406626-A2 SULPHONYL ARYL HYDROXAMATES AND THEIR USE AS MMP INHIBITORS Pharmacia Corporation (US) 2004-04-14 EP disclosed
EP-1127060-B1 HYDROBORONATION PROCESS COMMW SCIENT IND RES ORG (AU) 2004-04-07 EP disclosed
CN-1144793-C Polar-substituted hydrocarbons ˮ�ɺ� 2004-04-07 CN disclosed
US-6716844-B2 ENZYME INHIBITORS; ANTIINFLAMMATORY AGENTS, ANTIARTHRITIC AGENTS PHARMACIA CORPORATION 2004-04-06 US disclosed
US-20040063661-A1 Treatment of statin side effects MAGRAL LIMITED (AU) 2004-04-01 US disclosed
US-6713566-B1 CATALYTIC HYDROBORATION OF OLEFINIC OR ACETYLENIC FUNCTIONA-LIZED MATERIAL UNDER MILD CONDITIONS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2004-03-30 US disclosed
EP-1071684-B1 IMIDAZO 1,2-a]PYRIDINES AS PERIPHERAL BENZODIAZEPINE RECEPTOR BINDING AGENTS AUSTRALIAN NUCLEAR SCIENCE TEC (AU) 2004-03-17 EP disclosed
US-20040048852-A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor PHARMACIA CORPORATION 2004-03-11 US disclosed
WO-2003097657-A9 AN ANTIMICROBIAL AGENT UNIV GRIFFITH (AU) 2004-03-11 WO disclosed
WO-2004019986-A1 METHODS OF TREATING ACUTE RESPIRATORY DISTRESS SYNDROME SCHERING AKTIENGESELLSCHAFT (DE) 2004-03-11 WO disclosed
WO-2004018487-A1 CHIRAL ORGANOSILICON HYDRIDES CHIROGEN PTY LIMITED (AU) 2004-03-04 WO disclosed
EP-1390337-A1 PRECURSORS FOR KETONES AND ALDEHYDES Givaudan SA (CH) 2004-02-25 EP disclosed
US-6696611-B2 Chemical methods CHIROGEN PTY. LIMITED (AU) 2004-02-24 US disclosed
US-6696449-B2 CONTROL DEGRADATION OF CONENCTING TISSUE; CARDIOVASCULAR DISORDERS PHARMACIA CORPORATION 2004-02-24 US disclosed
US-20040033995-A1 Compounds and inhibitors of phospholipases QUEENSLAND, THE UNIVERSITY OF (AU) 2004-02-19 US disclosed
US-20040034071-A1 Thioaryl sulfonamide hydroxamic acid compounds PHARMACIA CORPORATION 2004-02-19 US disclosed
US-6689794-B2 SUPPRESSING MATRIX METALLOPROTEINASE AND/OR AGGRECANASE ACTIVITY PHARMACIA CORPORATION 2004-02-10 US disclosed
US-20040024024-A1 Aromatic sulfone hydroxamates and their use as protease inhibitors PHARMACIA CORPORATION 2004-02-05 US disclosed
WO-2004011460-A2 PYRAZOLYLBENZOTHIAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS QLT, INC. (CA) 2004-02-05 WO disclosed
WO-2004011473-A1 ORGANOGERMANIUM COMPOUNDS AND METHODS FOR THEIR USE CHIROGEN PTY LIMITED (AU) 2004-02-05 WO disclosed
EP-1385836-A2 AROMATIC SULFONE HYDROXAMATES AND THEIR USE AS PROTEASE INHIBITORS Pharmacia Corporation (US) 2004-02-04 EP disclosed
EP-0813525-B9 BENZAMIDINE DERIVATIVES THEIR PREPARATION AND THEIR USE AS ANTI-COAGULANTS BERLEX LAB (US) 2004-02-04 EP disclosed
US-6686364-B2 4-HYDROXY-3-((3,5-DIFLUORO-6-(3 -DIMETHYLAMINOCARBONYLPHENOXY)-4-(2-METHOXY-4-CARBOXYPHENOXY) PYRIDIN-2-YL)OXY)BENZAMIDINE, FOR EXAMPLE; FACTOR XA INHIBITORS BERLEX LABORATORIES, INC. 2004-02-03 US disclosed
US-6683093-B2 ENZYME INHIBITORS; CARDIOVASCULAR DISORDERS; ANTIINFLAMMATORY AGENTS; AUTOIMMUNE DISEASE PHARMACIA CORPORATION 2004-01-27 US disclosed
US-6683078-B2 REDUCING DEGRADATION OF CONNECTIVE TISSUE DUE TO CANCER OR INFLAMMATION PHARMACIA CORPORATION 2004-01-27 US disclosed
WO-2004007461-A1 8-HYDROXY QUINOLINE DERIVATIVES PRANA BIOTECHNOLOGY LIMITED (AU) 2004-01-22 WO disclosed
US-6680401-B1 BORON COMPOUNDS SUCH AS 4-(METHOXYMETHYL)-1,3,2-DIOXABOROLANE, USED AS COUPLERS OR CHEMICAL INTERMEDIATES FOR DRUGS, PESTICIDES OR IN COMBINATORIAL CHEMISTRY COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2004-01-20 US disclosed
WO-2004004834-A1 COMPOUNDS AND METHODS FOR TREATING CANCER AND INFLAMMATION QLT INC. (CA) 2004-01-15 WO disclosed
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors PHARMACIA ITALIA S.P.A. 2004-01-15 US disclosed
US-20040010140-A1 Process for preparation of bicyclic and polycyclic molecules MONASH UNIVERSITY (AU) 2004-01-15 US disclosed
US-20040010019-A1 Aromatic sulfone hydroxamates and their use as protease inhibitors PHARMACIA CORPORATION 2004-01-15 US disclosed
WO-2004004713-A1 FREDERICAMYCIN DERIVATIVES AS MEDICAMENTS FOR TREATING TUMOURS BIOFRONTERA DISCOVERY GMBH (DE) 2004-01-15 WO disclosed
EP-1379508-A2 N-(ARYL)-2-ARYLETHENESULFONAMIDES AND THERAPEUTIC USES THEREOF Temple University of the Commonwealth System of Higher Education (US) 2004-01-14 EP disclosed
US-6676926-B2 FOR ADMINISTERING TO A HUMAN IN NEED OF SUCH DIAGNOSIS AND MEASURING THE RADIOACTIVITY ARISING FROM THE ADMINISTRATION OF THE COMPOUND TO THE HUMAN EITHER BY USING A GAMMA CAMERA OR BY POSITRON EMISSION TOMOGRAPHY SCHERING AKTIENGESELLSCHAFT (DE) 2004-01-13 US disclosed
US-20040002424-A1 2-Amino-4-bicyclylamino-6H-1,3,5-triazines, processes for their preparation and their use as herbicides and plant growth regulators BAYER INTELLECTUAL PROPERTY GMBH (DE) 2004-01-01 US disclosed
WO-2004000314-A1 METHODS OF USING BENZOTHIOPHENONE DERIVATIVES TO TREAT CANCER OR INFLAMMATION QLT INC. (CA) 2003-12-31 WO disclosed
WO-2004000811-A1 ARYLSULFONYLHYDROXAMIC ACID AND AMIDE DERIVATIVES AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2003-12-31 WO disclosed
CN-1132836-C Synthesis of various lamellarin compounds and analogs and intermediates THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2003-12-31 CN disclosed
US-6670473-B2 Inhibitors of nitric oxide synthase (nos) BERLEX LABORATORIES, INC. 2003-12-30 US disclosed
WO-2003106404-A1 USE OF ALKYLAMIDOMANDELATES AS FLAVOURINGS SYMRISE GMBH & CO. KG (DE) 2003-12-24 WO disclosed
WO-2003105843-A1 METHODS OF USING ISOTHIAZOLE DERIVATIVES TO TREAT CANCER OR INFLAMMATION KINETEK PHARMACEUTICALS, INC. (CA) 2003-12-24 WO disclosed
WO-2003103675-A2 COMBINATION TREATMENTS FOR PURINOCEPTOR-RELATED DISORDERS ENDACEA, INC. (US) 2003-12-18 WO disclosed
US-20030232873-A1 Tetrahydrocarbazol derivatives as ligands for G-protein-coupled receptors (GPCR) ZENTARIS AG (DE) 2003-12-18 US disclosed
WO-2003104223-A1 PYRAZOLE-DERIVATIVES AS P38 KINASE INHIBITORS PHARMACIA CORPORATION (US) 2003-12-18 WO disclosed
US-20030232766-A1 Combinatorial libraries of monosaccharides VAST BIOSCIENCE PTY LIMITED (AU) 2003-12-18 US disclosed
EP-1206467-B1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LAB (US) 2003-12-17 EP disclosed
WO-2003101373-A2 THIAZOLIDINEDIONE DERIVATIVES IN THERAPEUTIC AND PROPHYLACTIC METHODS QLT INC. (CA) 2003-12-11 WO disclosed
US-20030224942-A1 Alkylamino-1,3,5-triazines, processes for their preparation and their use as herbicides and plant growth regulators AHRENS HARTMUT (DE) 2003-12-04 US disclosed
US-20030225108-A1 Process for making substituted pyrazoles PHARMACIA CORPORATION 2003-12-04 US disclosed
US-20030224032-A1 Antimicrobial coatings UNISEARCH LIMITED (AU) 2003-12-04 US disclosed
EP-1366015-A1 BENZENE-1 2-DIOL MANNICH BASES LIGANDS POLYMERS AND METHOD OF SELECTIVE METAL IONS REMOVAL TECHNOLOGICAL RESOURCES PTY. LTD. (AU) 2003-12-03 EP disclosed
US-6656954-B2 Such as N-hydroxy-2-(((4-phenoxyphenyl)-sulfonyl)methyl) benzamide which inhibits matrix metalloprotease activity PHARMACIA CORPORATION 2003-12-02 US disclosed
WO-2003097657-A1 AN ANTIMICROBIAL AGENT GRIFFITH UNIVERSITY (AU) 2003-11-27 WO disclosed
WO-2003097621-A1 METHODS OF USING THIAZOLIDINEDITHIONE DERIVATIVES QLT INC. (CA) 2003-11-27 WO disclosed
WO-2003096979-A2 DRUG THERAPY FOR CELIAC SPRUE THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2003-11-27 WO disclosed
US-20030220520-A1 Process for preparing organic boronic acid derivatives using diboronic acid COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2003-11-27 US disclosed
EP-1363880-A1 SYNTHESIS FOR THE PREPARATION OF COMPOUNDS FOR SCREENING AS POTENTIAL TUBULIN BINDING AGENTS THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2003-11-26 EP disclosed
WO-2003095494-A1 GENERATION OF SURFACE COATING DIVERSITY BIO-LAYER PTY LIMITED (AU) 2003-11-20 WO disclosed
WO-2003094916-A1 METHODS OF USING THIAZOLIDINE DERIVATIVES TO TREAT CANCER OR INFLAMMATION QLT INC. (CA) 2003-11-20 WO disclosed
EP-0973392-B1 SULFONYL DIVALENT ARYL OR HETEROARYL HYDROXAMIC ACID COMPOUNDS MONSANTO CO (US) 2003-11-19 EP disclosed
US-6646009-B2 Use against proliferative disorders including cancer, and as a radioprotective compound for normal cells from ionizing radiation Temple University — Of Commonwealth System of Higher Education 2003-11-11 US disclosed
WO-2003091247-A2 PIPERIDINYL-AND PIPERAZINYL-SULFONYLMETHYL HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2003-11-06 WO disclosed
EP-1358155-A1 AROMATIC SULFONYL ALPHA-CYCLOAMINO HYDROXAMATES AND THEIR USE AS MMP INHIBITORS Pharmacia Corporation (US) 2003-11-05 EP disclosed
WO-2003087060-A1 FREDERICAMYCIN DERIVATIVES BIOFRONTERA DISCOVERY GMBH (DE) 2003-10-23 WO disclosed
US-20030198692-A1 Microbial inhibitory compositions UNISEARCH LIMITED (AU) 2003-10-23 US disclosed
EP-1353911-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2003-10-22 EP disclosed
EP-1149075-A4 SYNTHESIS OF DITHIOESTER CHAIN TRANSFER AGENTS AND USE OF BIS(THIOACYL) DISULFIDES OR DITHIOESTERS AS CHAIN TRANSFER AGENTS DU PONT (US) 2003-10-22 EP disclosed
CN-1449379-A Sulfonium salt compound WAKO PURE CHEM IND LTD (JP) 2003-10-15 CN disclosed
US-20030191144-A1 Compounds, compositions and methods for modulating beta-amyloid production ACTIVE PASS PHARMACEUTICALS, INC. (CA) 2003-10-09 US disclosed
US-20030191317-A1 Sulfonyl aryl or heteroaryl hydroxamic acid compounds G. D. SEARLE & CO., (US) 2003-10-09 US disclosed
WO-2003080631-A2 PLASMA CARBOXYPEPTIDASE B INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 2003-10-02 WO disclosed
US-20030187035-A1 Substituted hydrazones as inhibitors of cyclooxygenase-2 TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2003-10-02 US disclosed
US-20030187256-A1 Benoxazinones/benzothiazinones as serine protease inhibitors BERRYMAN KENT ALAN (US) 2003-10-02 US disclosed
EP-0813525-B1 BENZAMIDINE DERIVATIVES THEIR PREPARATION AND THEIR USE AS ANTI-COAGULANTS BERLEX LAB (US) 2003-10-01 EP disclosed
EP-0920430-B1 PURINE DERIVATIVES AND THEIR USE AS ANTI-COAGULANTS SCHERING AG (DE) 2003-09-24 EP disclosed
EP-0984959-B1 AROMATIC SULFONYL ALPHA-HYDROXY HYDROXAMIC ACID COMPOUNDS PHARMACIA CORP (US) 2003-09-24 EP disclosed
US-20030176363-A1 Novel compounds and methods PHARMAXIS PTY LTD. (AU) 2003-09-18 US disclosed
US-20030171404-A1 Use of sulfonyl aryl or heteroaryl hydroxamic acids and derivatives thereof as aggrecanase inhibitors PHARMACIA CORPORATION 2003-09-11 US disclosed
EP-0896533-B1 PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS TULARIK INC (US) 2003-09-10 EP disclosed
EP-1000070-B1 SILICON-CONTAINING CHAIN EXTENDERS AORTECH BIOMATERIALS PTY LTD (AU) 2003-09-10 EP disclosed
EP-0939627-B1 PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS TULARIK INC (US) 2003-09-10 EP disclosed
US-20030166816-A1 Prepolymeric (meth) acrylates with polycyclic or aromatic segments 3M INNOVATIVE PROPERTIES COMPANY 2003-09-04 US disclosed
WO-2003072063-A2 AMINO-SUBSTITUTED SULFONANILIDES AND DERIVATIVES THEREOF FOR TREATING PROLIFERATIVE DISORDERS TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2003-09-04 WO disclosed
WO-2003072062-A2 AMINO-SUBSTITUTED (E)-2,6-DIALKOXYSTYRYL 4-SUBSTITUTED BENZYLSULFONES FOR TREATING PROLIFERATIVE DISORDERS TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2003-09-04 WO disclosed
US-20030166979-A1 Catalytic reduction using hydrogen DAKTERNIEKS DAINIS (AU) 2003-09-04 US disclosed
WO-2003070715-A1 AN ANTIMICROBIAL AGENT GRIFFITH UNIVERSITY (AU) 2003-08-28 WO disclosed
US-20030162817-A1 Pentafluorobenzenesulfonamides and analogs TULARIK INC. 2003-08-28 US disclosed
US-20030158205-A1 Piperazine derivatives and their use as anti-inflammatory agents SCHERING AKTIENGESELLSCHAFT (DE) 2003-08-21 US disclosed
WO-2003066873-A1 ESTERASES WITH LIPASE ACTIVITY COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2003-08-14 WO disclosed
EP-1334092-A1 PROCESS FOR PREPARATION OF BICYCLIC AND POLYCYCLIC MOLECULES Monash University (AU) 2003-08-13 EP disclosed
EP-1334719-A2 Pentafluorobenzenesulfonamides and analogs TULARIK, INC. (US) 2003-08-13 EP disclosed
US-20030148062-A1 POLYMERIC MEMBRANE COMPONENTS RESIDE WITHIN THE INTERSTITIAL GAPS OF THE SUBSTRATE; ULTRA-THIN; POLYMERIZATION AND CROSSLINKING OF POLYACRYLAMIDE GEL SOLOMON DAVID HENRY (AU) 2003-08-07 US disclosed
EP-1332138-A1 RADIOPHARMACEUTICALS FOR DIAGNOSING ALZHEIMER'S DISEASE SCHERING AKTIENGESELLSCHAFT (DE) 2003-08-06 EP disclosed
US-6603004-B2 Reacting diboron tetrahydroxide with boronic acid derivatives in presence of group 8-11 metal catalyst; one pot; no need for hydrolysis or hydrogenolysis COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2003-08-05 US disclosed
US-20030144302-A1 Process for making substituted pyrazoles PHARMACIA CORPORATION 2003-07-31 US disclosed
US-20030139376-A1 Lipoxin A4 analogs SCHERING AKTIENGESELLSCHAFT (DE) 2003-07-24 US disclosed
US-20030139425-A1 Piperazine derivatives and their use as anti-inflammatory agents SCHERING AKTIENGESELLSCHAFT (DE) 2003-07-24 US disclosed
US-20030139470-A1 3,4-dihydroxybenzyl-substituted carbonic acid derivatives and the use thereof as antioxidants HAARMANN & REIMER GMBH (DE) 2003-07-24 US disclosed
WO-2003055919-A1 AQUEOUS DISPERSIONS OF POLYMER PARTICLES UNIVERSITY OF SYDNEY (AU) 2003-07-10 WO disclosed
US-20030125381-A1 Inhibition of two-component signal transduction systems UNISEARCH LIMITED (AU) 2003-07-03 US disclosed
US-6585873-B1 Polymer gels and methods for their preparation UNIVERSITY OF MELBOURNE (AU) 2003-07-01 US disclosed
WO-2003051837-A2 TETRAHYDROCARBOZOLE DERIVATIVES AS LIGANDS FOR G-PROTEIN COUPLED RECEPTORS (GPCR) ZENTARIS GMBH (DE) 2003-06-26 WO disclosed
US-6583299-B1 Matrix metalloprotease inhibitors; nonsuppression of tumor necrosis factor production G.D. SEARLE & CO. 2003-06-24 US disclosed
WO-2003049698-A2 SUBSTITUTED HYDRAZONES AS INHIBITORS OF CYCLOOXYGENASE-2 TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2003-06-19 WO disclosed
US-20030114638-A1 Alkene borates and a process for covalently coupling organic compounds COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2003-06-19 US disclosed
US-20030104945-A1 2,4-Diamino-1,3,5-triazines, their preparation, and their use as herbicides and plant growth regulators AVENTIS CROPSCIENCE GMBH (DE) 2003-06-05 US disclosed
WO-2003045944-A1 AROMATIC SULFONE HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2003-06-05 WO disclosed
WO-2003045379-A1 HYDRAZONOPYRAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTICS KINETEK PHARMACEUTICALS, INC. (CA) 2003-06-05 WO disclosed
US-20030105375-A1 Purification of 4,4'(5')- di-t-butylcyclohexano-18-crown-6 PG RESEARCH FOUNDATION 2003-06-05 US disclosed
US-6573266-B1 Compounds used for treating multitiple sclerosis and encephalomyelitis SCHERING AKTIENGESELLSCHAFT (DE) 2003-06-03 US disclosed
WO-2003043960-A2 IMPROVED PURIFICATION OF 4, 4'(5')-DI-t-BUTYLCYCLOHEXANO-18-CROWN-6 PG RESEARCH FOUNDATION (US) 2003-05-30 WO disclosed
US-6566413-B1 For dental and dental engineering applications 3M ESPE AG (DE) 2003-05-20 US disclosed
US-20030092678-A1 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2003-05-15 US disclosed
WO-2003040080-A2 LIPOXIN A4 ANALOGS SCHERING AKTIENGESELLSCHAFT (DE) 2003-05-15 WO disclosed
US-20030092864-A1 Silicon-based polycarbonates AORTECH BIOMATERIALS PTY LTD. 2003-05-15 US disclosed
US-20030087761-A1 Synergistic active compound combinations for controlling harmful plants AVENTIS CROPSCIENCE GMBH (DE) 2003-05-08 US disclosed
US-20030087942-A1 Method for the treatment and prevention of cachexia WASHINGTON UNIVERSITY 2003-05-08 US disclosed
US-6559310-B2 Reacting a halogen aromatic derivative at a coupling position with a diboron derivative in the presence of a Group VIII metal catalyst and a suitable base for covalently coupling organic compounds COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2003-05-06 US disclosed
US-20030083332-A1 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2003-05-01 US disclosed
US-6555537-B2 Inhibit activity of chemokines, macrophage inflammatory protein-1 (MIP-1 alpha) and RANTES; 1-((4-chlorophenoxy)methyl)-carbonyl-2-methyl-4-(4-fluorobenzyl)piperazine for example SCHERING AKTIENGESELLSCHAFT (DE) 2003-04-29 US disclosed
US-20030078265-A1 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2003-04-24 US disclosed
EP-1139973-B1 POLYMERISABLE MATERIALS WHICH ARE BASED ON HARDENABLE SILOXANE COMPOUNDS 3M ESPE AG (DE) 2003-04-23 EP disclosed
US-6551684-B1 Substrate with interstitial gaps having polymeric membrane within the gaps that are thinner than the cross-sectional thickness of the substrate GRADIPORE LIMITED (AU) 2003-04-22 US disclosed
US-20030073718-A1 Aromatic sulfone hydroxamic acids and their use as protease inhibitors PHARMACIA CORPORATION 2003-04-17 US disclosed
US-20030073669-A1 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2003-04-17 US disclosed
US-20030073845-A1 Sulfonyl aryl hydroxamates and their use as matrix metalloprotease inhibitors PHARMACIA CORPORATION 2003-04-17 US disclosed
EP-0922045-B1 BICYCLIC PYRIMIDINE DERIVATIVES AND THEIR USE AS ANTI-COAGULANTS SCHERING AG (DE) 2003-04-16 EP disclosed
EP-1301522-A1 NOVEL COMPOUNDS AND METHODS Pharmaxis Pty Ltd (AU) 2003-04-16 EP disclosed
US-6548505-B1 Protecting biological materials from damage caused by radiation; side effect reduction during radiotherapy or chemotherapy; indole, benzimidazole, benzoxazole or benzothiazole compounds substituted with 4-alkylpiperazino PETER MACCALLUM CANCER INSTITUTE (AU) 2003-04-15 US disclosed
US-20030069210-A1 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2003-04-10 US disclosed
US-20030069307-A1 2-(3,4-Dihydroxyphenyl)ethyl-substituted carbonic acid derivatives and their use HAARMANN & REIMER GMBH (DE) 2003-04-10 US disclosed
CN-1105114-C Sulfonyl divalent aryl alpha-hydroxamic acid compounds MANSANTO CO (US) 2003-04-09 CN disclosed
WO-2003026663-A1 PROCESS FOR MAKING SUBSTITUTED PYRAZOLES PHARMACIA CORPORATION (US) 2003-04-03 WO disclosed
EP-1296941-A2 3,4-DIHYDROXYBENZYL-SUBSTITUTED CARBONIC ACID DERIVATIVES AND THE USE THEREOF AS ANTIOXIDANTS HAARMANN & REIMER GMBH (DE) 2003-04-02 EP disclosed
EP-1296673-A1 ANTIMICROBIAL COATINGS UNISEARCH LIMITED (AU) 2003-04-02 EP disclosed
US-6541489-B1 Excellent inhibitory activity of one or more matrix metalloprotease (MMP) enzymes, such as MMP-2, MMP-9, and MMP-13, while exhibiting substantially less inhibition at least of MMP- 1 G. D. SEARLE & COMPANY 2003-04-01 US disclosed
US-6541476-B1 Treating multiple sclerosis or encephalomyelitis in a human SCHERING AKTIENGESELLSCHAFT (DE) 2003-04-01 US disclosed
US-20030060452-A1 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2003-03-27 US disclosed
US-20030060474-A1 Platelet adenosine diphosphate receptor antagonists SCHERING AKTIENGESELLSCHAFT (DE) 2003-03-27 US disclosed
EP-1294705-A1 SYNTHESIS OF CYCLIC COMPOUNDS UNISEARCH LIMITED (AU) 2003-03-26 EP disclosed
US-6534509-B1 Derivatives are useful as anti-inflammatory agents. This invention is also directed to pharmacetutical compostions for inflammation SCHERING AKTIENGESELLSCHAFT (DE) 2003-03-18 US disclosed
WO-2003020268-A1 METHOD FOR THE TREATMENT AND PREVENTION OF CACHEXIA WASHINGTON UNIVERSITY (US) 2003-03-13 WO disclosed
EP-0939628-B1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 2003-03-05 EP disclosed
EP-1284979-A1 PREPOLYMERIC (METH)ACRYLATES WITH POLYCYCLIC OR AROMATIC SEGMENTS 3M Espe AG (DE) 2003-02-26 EP disclosed
EP-1285912-A2 Process for the selective reduction of alkynic compounds BASF AKTIENGESELLSCHAFT (DE) 2003-02-26 EP disclosed
WO-2003014122-A1 DERIVATIVES OF MORPHINE-LIKE OPIOID COMPOUNDS POLYCHIP PHARMACEUTICALS PTY LTD (AU) 2003-02-20 WO disclosed
EP-1284145-A1 2-(3,4-Dihydroxyphenyl)ethyl substituted carbonic acid derivatives and their use HAARMANN & REIMER GMBH (DE) 2003-02-19 EP disclosed
EP-0988292-B1 PIPERAZINE DERIVATIVES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS SCHERING AG (DE) 2003-02-12 EP disclosed
US-20030027794-A1 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2003-02-06 US disclosed
US-6515160-B2 Boronic compounds COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2003-02-04 US disclosed
WO-2003007954-A2 SULFONYL ARYL HYDROXAMATES AND THEIR USE AS MATRIX METALLOPROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2003-01-30 WO disclosed
WO-2003007930-A2 USE OF SULFONYL ARYL OR HETEROARYL HYDROXAMIC ACIDS AND DERIVATIVES THEREOF AS AGGRECANASE INHIBITORS PHARMACIA CORPORATION (US) 2003-01-30 WO disclosed
US-6512081-B1 Synthesis of dithioester chain transfer agents and use of bis(thioacyl) disulfides or dithioesters as chain transfer agents E.I. DUPONT NEMOURS AND COMPANY 2003-01-28 US disclosed
EP-1056751-A4 BORONIC COMPOUNDS COMMW SCIENT IND RES ORG (AU) 2003-01-22 EP disclosed
US-6509335-B1 This invention discloses benzoxazinone and benzothiazinone compounds which display inhibitory effects on serine proteases such as factor Xa, thrombin, and/or factor VIIa. The invention also discloses pharmaceutically acceptable salts of WARNER-LAMBERT COMPANY 2003-01-21 US disclosed
EP-1274420-A1 MICROBIAL INHIBITORY COMPOSITIONS Unisearch Limited (AU) 2003-01-15 EP disclosed
US-6506925-B2 Synthesis from haloalkenes or pseudo-haloalkenes COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2003-01-14 US disclosed
US-20030004137-A1 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. (US) 2003-01-02 US disclosed
US-20030004064-A1 Synergistic active compound combinations for controlling harmful plants AVENTIS CROPSCIENCE GMBH (DE) 2003-01-02 US disclosed
EP-1090008-A4 SYNTHESES OF A VARIETY OF LAMELLARIN COMPOUNDS AND ANALOGUES UNIV AUSTRALIAN (AU) 2003-01-02 EP disclosed
WO-2002102370-A1 BIOFILM DEGRADING OR SLOUGHING COMPOSITIONS AND METHODS UNISEARCH LIMITED (AU) 2002-12-27 WO disclosed
WO-2002102560-A1 BORON-BASED WOOD PRESERVATIVES AND TREATMENT OF WOOD WITH BORON-BASED PRESERVATIVES THE UNIVERSITY OF MELBOURNE (AU) 2002-12-27 WO disclosed
CN-1387514-A Aromatic sulfone hydroxamic acid metalloprotease inhibitor SEARLE & CO (US) 2002-12-25 CN disclosed
US-20020193604-A1 Aryl borates COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2002-12-19 US disclosed
US-6492367-B1 Sulfamato hydroxamic acid metalloprotease inhibitor G. D. SEARLE & COMPANY 2002-12-10 US disclosed
US-20020183323-A1 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. 2002-12-05 US disclosed
WO-2002096850-A1 PRECURSORS FOR KETONES AND ALDEHYDES GIVAUDAN SA (CH) 2002-12-05 WO disclosed
US-20020177598-A1 Piperazine derivatives and their use as anti-inflammatory agents SCHERING AKTIENGSCHELLSCHAFT 2002-11-28 US disclosed
US-20020177588-A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor PHARMACIA CORPORATION 2002-11-28 US disclosed
WO-2002092588-A2 AROMATIC SULFONE HYDROXAMATES AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2002-11-21 WO disclosed
US-20020173508-A1 Aromatic sulfonyl alpha-hydroxy hydroxamic acid compounds PHARMACIA CORPORATION 2002-11-21 US disclosed
US-6482860-B1 such as batabulin (2-Fluoro-1-methoxy-4-pentafluorophenylsulfonamidobenzene), use as antiproliferative agents to treat cancer TULARIK INC. 2002-11-19 US disclosed
US-6479485-B2 4-HYDROXY-3-((3,4-DIFLUORO-6-(3 -DIMETHYLAMINOCARBONYLPHENOXY)-4-(2-METHOXY-4-CARBOXYPHENOXY) PYRIDIN-2-YL)OXY)BENZAMIDINE, FOR EXAMPLE; INHIBITION OF BLOOD COAGGULATION FACTOR XA BERLEX LABORATORIES, INC. 2002-11-12 US disclosed
US-20020165203-A1 N-heterocyclic derivatives as NOS inhibitors BERLEX LABORATORIES, INC. 2002-11-07 US disclosed
US-20020165412-A1 N-(aryl)-2-arylethenesulfonamides and therapeutic uses thereof ONCONOVA THERAPEUTICS, INC. 2002-11-07 US disclosed
EP-1254899-A2 Piperazine derivatives and their use as anti-inflammatory agents Schering Aktiengesellschaft (DE) 2002-11-06 EP disclosed
US-6476027-B1 N-hydroxy 4-sulfonyl butanamide compounds MONSANTO COMPANY 2002-11-05 US disclosed
US-20020161114-A1 Shape memory polyurethane or polyurethane-urea polymers AORTECH BIOMATERIALS PTY LTD. (AU) 2002-10-31 US disclosed
WO-2002085459-A2 ANTIANGIOGENIC COMBINATION THERAPY FOR THE TREATMENT OF CANCER PHARMACIA CORPORATION (US) 2002-10-31 WO disclosed
EP-1203038-A4 SHAPE MEMORY POLYURETHANE OR POLYURETHANE-UREA POLYMERS AORTECH BIOMATERIALS PTY LTD (AU) 2002-10-30 EP disclosed
EP-1187827-A4 ANTIVIRAL AGENTS BIOTA SCIENT MANAGEMENT (AU) 2002-10-24 EP disclosed
US-6469171-B1 NON-TOXIC MODULATORS OF THE MULTIDRUG RESISTANT PHENOTYPE THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2002-10-22 US disclosed
US-20020151743-A1 Process for preparing organic boronic avid derivatives using diboronic acid COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2002-10-17 US disclosed
US-6465459-B2 INHIBIT THE ENZYME, FACTOR XA BERLEX LABORATORIES, INC. 2002-10-15 US disclosed
CN-1373751-A 'Alpha'-amino-'beta'-sulfonyl hydroxamic acid compounds SEARLE & CO (US) 2002-10-09 CN disclosed
US-20020143036-A1 Pentafluorobenzenesulfonamides and analogs TULARIK INC. 2002-10-03 US disclosed
EP-0877730-B1 ARYL ACRYLICS FOR USE AS FUNGICIDE MONSANTO TECHNOLOGY LLC (US) 2002-10-02 EP disclosed
US-20020131932-A1 Radiopharmaceuticals for diagnosing alzheimer's disease SCHERING AG (DE) 2002-09-19 US disclosed
US-20020133039-A1 Chemical methods DEAKIN UNIVERSITY (AU) 2002-09-19 US disclosed
EP-0984997-B1 SILICON-BASED POLYCARBONATES AORTECH BIOMATERIALS PTY LTD (AU) 2002-09-18 EP disclosed
CN-1370144-A Aromatic sulfone hydroxamic acid metalloprotease inhibitor SEARLE & CO (US) 2002-09-18 CN disclosed
CN-1370048-A Azabicyclo and azacyclo oxime and amine compounds as pesticides AVENTIS CROPSCIONCE GMBH (DE) 2002-09-18 CN disclosed
US-6451791-B1 Amidoaromatic ring sulfonamide hydroxamic acid compounds MONSANTO COMPANY 2002-09-17 US disclosed
WO-2002070456-A1 BENZENE-1 2-DIOL MANNICH BASES LIGANDS POLYMERS AND METHOD OF SELECTIVE METAL IONS REMOVAL TECHNOLOGICAL RESOURCES PTY LIMITED (AU) 2002-09-12 WO disclosed
US-6448250-B1 INHIBITS THE ACTIVITY OF ONE OR MORE OF THE FOLLOWING MATRIX METALLOPROTEINASES: MMP-2, MMP-9, AND MMP-13, WHILE EXHIBITING SUBSTANTIALLY LESS INHIBITORY ACTIVITY AGAINST MMP-1 G. D. SEARLE & COMPANY 2002-09-10 US disclosed
WO-2002067865-A2 N-(ARYL)-2-ARYLETHENESULFONAMIDES AND THERAPEUTIC USES THEREOF TEMPLE UNIVERSITY OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2002-09-06 WO disclosed
EP-1236727-A1 Azabicyclo compounds as pesticides Bayer CropScience GmbH (DE) 2002-09-04 EP disclosed
US-6437073-B1 Non-elastomeric polyurethane compositions AORTECH BIOMATERIALS PTY LTD. (AU) 2002-08-20 US disclosed
WO-2002062756-A1 AROMATIC SULFONYL ALPHA-CYCLOAMINO HYDROXAMATES AND THEIR USE AS MMP INHIBITORS PHARMACIA CORPORATION (US) 2002-08-15 WO disclosed
EP-0986541-A4 PROCESS FOR COVALENTLY COUPLING ORGANIC COMPOUNDS UTILIZING DIBORON DERIVATIVES COMMW SCIENT IND RES ORG (AU) 2002-08-14 EP disclosed
US-6432947-B1 NERVOUS SYSTEM DISORDERS; MUSCLE RELAXANTS; ANTIDIABETIC AGENTS BERLEX LABORATORIES, INC. 2002-08-13 US disclosed
US-6432963-B1 ANTIINFLAMMATORY AGENTS; TYROSINE KINASE INHIBITOR YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2002-08-13 US disclosed
WO-2002060872-A1 SYNTHESIS FOR THE PREPARATION OF COMPOUNDS FOR SCREENING AS POTENTIAL TUBULIN BINDING AGENTS THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2002-08-08 WO disclosed
US-20020103141-A1 Antiangiogenic combination therapy for the treatment of cancer PHARMACIA CORPORATION 2002-08-01 US disclosed
US-20020103239-A1 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds BEDELL LOUIS J (US) 2002-08-01 US disclosed
EP-1224190-A1 SUBSTITUTED DIBORON COMPOUNDS Commonwealth Scientific and Research Organisation (AU) 2002-07-24 EP disclosed
CN-1360577-A Hydroxamic acid derivs. as matrix metalloprotease inhibitors SEARLE & CO (US) 2002-07-24 CN disclosed
US-6420452-B1 POLYURETHANES WITH EXTENDERS AORTECH BIOMATERIALS PTY LTD (AU) 2002-07-16 US disclosed
WO-2002053572-A1 DELIVERY SYSTEMS ALCHEMIA PTY LTD (AU) 2002-07-11 WO disclosed
US-20020086866-A1 Quinoxalinones as serine protease inhibitors DUDLEY DANETTE ANDREA (US) 2002-07-04 US disclosed
WO-2002050045-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2002-06-27 WO disclosed
US-6410536-B1 ANTICOAGULANTS WARNER-LAMBERT COMPANY 2002-06-25 US disclosed
WO-2002047681-A1 REGULATION OF BACTERIAL VIRULENCE UNISEARCH LIMITED (AU) 2002-06-20 WO disclosed
EP-1214317-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2002-06-19 EP disclosed
EP-1019414-A4 PROCESS FOR PREPARING ORGANIC BORONIC ACID DERIVATIVES USING DIBORONIC ACID COMMW SCIENT IND RES ORG (AU) 2002-05-29 EP disclosed
US-6388131-B2 Benzenesulfonamide compounds, which encompasses the compound batabulin (2-Fluoro-1-methoxy-4-pentafluorophenylsulfonamidobenzene) TULARIK, INC. 2002-05-14 US disclosed
WO-2002036581-A1 RADIOPHARMACEUTICALS FOR DIAGNOSING ALZHEIMER'S DISEASE SCHERING AKTIENGESELLSCHAFT (DE) 2002-05-10 WO disclosed
EP-1203038-A1 SHAPE MEMORY POLYURETHANE OR POLYURETHANE-UREA POLYMERS AorTech Biomaterials Pty Ltd (AU) 2002-05-08 EP disclosed
WO-2002034736-A1 PROCESS FOR PREPARATION OF BICYCLIC AND POLYCYCLIC MOLECULES MONASH UNIVERSITY (AU) 2002-05-02 WO disclosed
US-6380258-B2 METALLOPROTEASE INHIBITOR G. D. SEARLE, L.L.C. 2002-04-30 US disclosed
US-6379649-B1 USEFUL FOR DIAGNOSIS AND TREATMENT, INCLUDING RADIOTHERAPY, OF DISORDERS THAT ARE CHARACTERIZED BY AN ABNORMAL DENSITY OF PERIPHERAL BENZODIAZEPINE RECEPTORS; NERVE SYSTEM DISPORDERS AUSTRALIAN NUCLEAR SCIENCE & TECHNOLOGY ORGANISATION (AU) 2002-04-30 US disclosed
WO-2002032963-A1 IMMUNOADJUVANT SYSTEMS ALCHEMIA PTY LTD (AU) 2002-04-25 WO disclosed
US-20020045654-A1 Sulfonylbenzene compounds as anti-inflammatory/analgesic agents ANDO KAZUO (JP) 2002-04-18 US disclosed
WO-2002028345-A2 ALDEHYDE-RELEASING COMPOUNDS LA TROBE UNIVERSITY (AU) 2002-04-11 WO disclosed
US-6362183-B1 PROTEASE INHIBITORS; RHEUMATIC DISEASES; ANTITUMOR AGENTS G. D. SEARLE & COMPANY 2002-03-26 US disclosed
US-20020035109-A1 Benzamidine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. 2002-03-21 US disclosed
EP-1187859-A1 POLYMER GELS, METHODS FOR THEIR PREPARATION AND THEIR USE IN ELECTROPHORETIC APPLICATIONS THE UNIVERSITY OF MELBOURNE (AU) 2002-03-20 EP disclosed
EP-1187827-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 2002-03-20 EP disclosed
US-20020032339-A1 ARYL BORATES BORON MOLECULAR LIMITED (AU) 2002-03-14 US disclosed
US-20020032223-A1 Benzamidine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. 2002-03-14 US disclosed
US-20020028820-A1 Benzamidine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. 2002-03-07 US disclosed
US-20020028901-A1 Siloxane-containing polyurethane-urea compositions ELASTOMEDIC PTY LIMITED 2002-03-07 US disclosed
EP-1121365-A4 ORGANOBORON DERIVATIVES AND PROCESS FOR COUPLING ORGANIC COMPOUNDS COMMW SCIENT IND RES ORG (AU) 2002-03-06 EP disclosed
EP-1183239-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE &amp; CO. (US) 2002-03-06 EP disclosed
US-6350746-B1 FACTOR XA ENZYME INHIBITORS BERLEX LABORATORIES, INC. 2002-02-26 US disclosed
US-6348474-B1 COMPOUNDS AS ANTIDIABETIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed
US-6346639-B1 Boronic compounds THE COMMONWEALTH OF AUSTRALIA COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANIZATION (AU) 2002-02-12 US disclosed
US-20020016489-A1 Alkene borates and a process for covalently coupling organic compounds COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION 2002-02-07 US disclosed
EP-1177173-A1 HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS G.D. SEARLE & CO. (US) 2002-02-06 EP disclosed
US-20020013496-A1 Benzene compounds as antiproliferative and cholesterol lowering agents AMGEN INC. 2002-01-31 US disclosed
CN-1333777-A Organoboron derivatives and methods of coupling organic compounds COMMW SCIENT IND RES ORG (AU) 2002-01-30 CN disclosed
WO-2002004472-A1 NOVEL COMPOUNDS AND METHODS PHARMAXIS PTY LTD (AU) 2002-01-17 WO disclosed
EP-1044194-A4 RECEPTOR WITH AN AFFINITY FOR COMPOUNDS OF THE OXAZOLINE CLASS UNIV MELBOURNE (AU) 2002-01-09 EP disclosed
WO-2002000639-A1 SYNTHESIS OF CYCLIC COMPOUNDS UNISEARCH LIMITED (AU) 2002-01-03 WO disclosed
WO-2001098235-A2 3,4-DIHYDROXYBENZYL-SUBSTITUTED CARBONIC ACID DERIVATIVES AND THE USE THEREOF AS ANTIOXIDANTS HAARMANN & REIMER GMBH (DE) 2001-12-27 WO disclosed
US-6333391-B1 FROM AMINES AND CARBOXYLIC ACIDS OR ANHYDRIDES, IN WATER; COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2001-12-25 US disclosed
WO-2001094348-A1 ANTIVIRAL AGENTS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2001-12-13 WO disclosed
WO-2001092271-A1 PREPOLYMERIC (METH)ACRYLATES WITH POLYCYCLIC OR AROMATIC SEGMENTS 3M ESPE AG (DE) 2001-12-06 WO disclosed
US-20010049449-A1 Aromatic sulfonyl alpha-cycloamino hydroxamates and their use as MMP inhibitors PHARMACIA CORPORATION 2001-12-06 US disclosed
WO-2001085680-A2 SULFONYL ARYL OR HETEROARYL HYDROXAMIC ACID COMPOUNDS PHARMACIA CORPORATION (US) 2001-11-15 WO disclosed
US-6316484-B1 FOR THERAPY OR PROPHYLAXIS OF ATHEROSCLEROSIS AND HYPERCHOLESTEROLEMIA TULARIK INC. 2001-11-13 US disclosed
US-20010039287-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR PHARMACIA CORPORATION 2001-11-08 US disclosed
EP-0764165-B1 PREPARATION OF STEREOCHEMICALLY PURE OXIMES WITH MUSCARINIC ACTIVITY WARNER LAMBERT CO (US) 2001-11-07 EP disclosed
EP-1149075-A1 SYNTHESIS OF DITHIOESTER CHAIN TRANSFER AGENTS AND USE OF BIS(THIOACYL) DISULFIDES OR DITHIOESTERS AS CHAIN TRANSFER AGENTS E.I. DU PONT DE NEMOURS AND COMPANY (US) 2001-10-31 EP disclosed
US-6306884-B1 ANTICOAGULANTS AND BLOOD COAGULATION FACTOR BERLEX LABORATORIES, INC. 2001-10-23 US disclosed
WO-2001076594-A1 ANTIMICROBIAL COATINGS UNISEARCH LIMITED (AU) 2001-10-18 WO disclosed
EP-1071684-A4 IMIDAZO 1,2-a]PYRIDINES AS PERIPHERAL BENZODIAZEPINE RECEPTOR BINDING AGENTS AUSTRALIAN NUCLEAR SCIENCE TEC (AU) 2001-10-04 EP disclosed
WO-2001068090-A1 MICROBIAL INHIBITORY COMPOSITIONS UNISEARCH LIMITED (AU) 2001-09-20 WO disclosed
US-20010020021-A1 SULFONYL DIVALENT ARYL OR HETEROARYL HYDROXAMIC ACID COMPOUNDS G.D. SEARLE & CO. 2001-09-06 US disclosed
US-20010020079-A1 Electrophoresis gels and cross-linking agents for their preparation THE UNIVERSITY OF MELBOURNE 2001-09-06 US disclosed
US-6284923-B1 BENZENESULFONIMIDES FOR TREATMENT OF CANCER AND ANTICHOLESTEROL AGENTS TULARIK INC 2001-09-04 US disclosed
US-20010014688-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR BARTA THOMAS E (US) 2001-08-16 US disclosed
EP-1121365-A1 ORGANOBORON DERIVATIVES AND PROCESS FOR COUPLING ORGANIC COMPOUNDS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2001-08-08 EP disclosed
CN-1307580-A Synthesis of various lamellarin compounds and analogs UNIV AUSTRALIAN (AU) 2001-08-08 CN disclosed
EP-0920405-B1 FLUOROVINYL DERIVATIVE COMPOUND, LIQUID CRYSTAL COMPOSITION, AND LIQUID CRYSTAL DISPLAY DEVICE CHISSO CORP (JP) 2001-07-11 EP disclosed
US-6258806-B1 PEPTIDES WITH CYCLIC DIAZAALKANES FOR PREVENTION OF PREMATURE METABOLISM METHOD FOR INHIBITING AN HIV PROTEASE IN A MAMMAL IN NEED OF SUCH PROTEASE INHIBITION, COMPRISING ADMINISTERING TO SAID MAMMAL AN EFFECTIVE DOSAGE NARHEX LIMITED (HK) 2001-07-10 US disclosed
EP-1078010-A4 NON-ELASTOMERIC POLYURETHANE COMPOSITIONS ELASTOMEDIC PTY LTD (AU) 2001-07-04 EP disclosed
EP-1112250-A1 THERAPEUTIC COMPOUNDS AND METHODS Institute of Molecular and Cell Biology (SG) 2001-07-04 EP disclosed
US-6242454-B1 Benzamidine derivatives substituted by amino acid and hydroxy acid derivatives and their use as anti-coagulants BERLEX LABORATORIES INC. 2001-06-05 US disclosed
EP-0983257-A4 AROMATIC SULFONYL ALPHA-CYCLOAMINO HYDROXAMIC ACID COMPOUNDS MONSANTO CO (US) 2001-05-02 EP disclosed
EP-0984959-A4 AROMATIC SULFONYL ALPHA-HYDROXY HYDROXAMIC ACID COMPOUNDS MONSANTO CO (US) 2001-05-02 EP disclosed
EP-0973392-A4 SULFONYL DIVALENT ARYL OR HETEROARYL HYDROXAMIC ACID COMPOUNDS MONSANTO CO (US) 2001-05-02 EP disclosed
WO-2001029051-A1 SUBSTITUTED DIBORON COMPOUNDS COMMONWEALTH SCIENTIFIC AND RESEARCH ORGANISATION (AU) 2001-04-26 WO disclosed
US-6221886-B1 Thio acid derived monocyclic N-heterocyclics as anticoagulants BERLEX LABORATORIES, INC. 2001-04-24 US disclosed
EP-1091955-A1 QUINOLONES AS SERINE PROTEASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2001-04-18 EP disclosed
EP-1090008-A1 SYNTHESES OF A VARIETY OF LAMELLARIN COMPOUNDS AND ANALOGUES THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2001-04-11 EP disclosed
US-6215016-B1 HEMATOPOIETIC AGENTS; PREVENTING CYTOPENIA TORAY INDUSTRIES, INC. (JP) 2001-04-10 US disclosed
US-6207665-B1 TO TREAT INFLAMMATORY DISORDERS IN HUMANS SCHERING AKTIENGESELLSCHAFT (DE) 2001-03-27 US disclosed
US-6207076-B1 HIGH ELASTIC CONSTANT RATIO, LOW VISCOSITY, WIDE NEMATIC PHASE TEMPERATURE RANGE, CHEMICAL STABILITY CHISSO CORPORATION (JP) 2001-03-27 US disclosed
WO-2001019822-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2001-03-22 WO disclosed
US-6197906-B1 ASSYMETRIC AGENTS SUCH AS (2-METHACRYLOYLOXYETHYL)ACRYLAMIDE, (2-ACRYLOYLOXYETHYL)METHACRYLAMIDE, AND (N-METHYL-N-ACRYLOYLAMINO)ETHYL METHACRYLATE THE UNIVERSITY OF MELBOURNE (AU) 2001-03-06 US disclosed
EP-1078010-A1 NON-ELASTOMERIC POLYURETHANE COMPOSITIONS Elastomedic Pty Limited (AU) 2001-02-28 EP disclosed
US-6194414-B1 CANCER THERAPY; PREVENT RADIATION DAMAGE THE INNER AND EASTERN HEALTH CARE NETWORK (AU) 2001-02-27 US disclosed
US-6184245-B1 Cyclic ketone derivatives and their medical applications TORAY INDUSTRIES INC. (JP) 2001-02-06 US disclosed
WO-2001007499-A1 SHAPE MEMORY POLYURETHANE OR POLYURETHANE-UREA POLYMERS AORTECH BIOMATERIALS PTY LTD. (AU) 2001-02-01 WO disclosed
EP-1071684-A1 IMIDAZO 1,2-a]PYRIDINES AS PERIPHERAL BENZODIAZEPINE RECEPTOR BINDING AGENTS AUSTRALIAN NUCLEAR SCIENCE &amp; TECHNOLOGY ORGANISATION (AU) 2001-01-31 EP disclosed
EP-0981517-A4 PREPARATION OF FUSED POLYCYCLIC ALKALOIDS BY RING CLOSURE OF AZOMETHINE YLIDES, NOVEL COMPOUNDS THEREOF AND THEIR USE AS CHEMOTHERAPEUTIC AGENTS UNIV AUSTRALIAN (AU) 2001-01-24 EP disclosed
EP-1068190-A1 QUINOXALINONES AS SERINE PROTEASE INHIBITORS SUCH AS FACTOR XA AND THROMBIN WARNER-LAMBERT COMPANY LLC (US) 2001-01-17 EP disclosed
EP-1068191-A1 BENZOXAZINONES/BENZOTHIAZINONES AS SERINE PROTEASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2001-01-17 EP disclosed
CN-1279669-A Aromatic sulfone hydroxamic acid metalloprotease inhibitors SEARLE & CO (US) 2001-01-10 CN disclosed
WO-2000078746-A1 ANTIVIRAL AGENTS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2000-12-28 WO disclosed
US-6166014-A Thio acid derived monocyclic N-heterocyclics as anticoagulants BERLEX LABORATORIES, INC. (US) 2000-12-26 US disclosed
US-6166088-A CONTROLLING THROMBOSIS BERLEX LABORATORIES, INC. (US) 2000-12-26 US disclosed
US-6162807-A Thio acid derived monocyclic N-heterocyclics as anticoagulants BERLEX LABORATORIES, INC. (US) 2000-12-19 US disclosed
EP-1056751-A1 BORONIC COMPOUNDS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2000-12-06 EP disclosed
CN-1275984-A Process for preparing organic boronic acid derivatives using diboronic acid COMMW SCIENT IND RES ORG (AU) 2000-12-06 CN disclosed
WO-2000069821-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE & CO. (US) 2000-11-23 WO disclosed
WO-2000069819-A1 HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS G.D. SEARLE & CO. (US) 2000-11-23 WO disclosed
EP-1054004-A1 NOVEL PYRIMIDINE-5-CARBOXAMIDE DERIVATIVES YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2000-11-22 EP disclosed
US-6150382-A ENZYME INHIBITORS OF BLOOD COAGULATION FACTOR XA, A SERINE PROTEASE CLASS OF ENZYMES; E.G., 4-HYDROXY-3-((4-(2-CARBOXY-METHYL)THIO-6-(3-(1-METHYL)-6-(3-(1 -METHYL)IMIDAZOLIN-2-YL)-PHENOXY-3,5-DIFLUOROPYRIDINE AND DERIVATIVES BERLEX LABORATORIES, INC. (US) 2000-11-21 US disclosed
EP-1044194-A1 RECEPTOR WITH AN AFFINITY FOR COMPOUNDS OF THE OXAZOLINE CLASS THE UNIVERSITY OF MELBOURNE (AU) 2000-10-18 EP disclosed
EP-1042290-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE &amp; CO. (US) 2000-10-11 EP disclosed
CN-1268940-A Preparation of thiochloroformates BASF AG (DE) 2000-10-04 CN disclosed
WO-2000056792-A1 POLYMER GELS, METHODS FOR THEIR PREPARATION AND THEIR USE IN ELECTROPHORETIC APPLICATIONS THE UNIVERSITY OF MELBOURNE (AU) 2000-09-28 WO disclosed
US-6121304-A SUCH AS 1-(PENTAFLUOROPHENYLSULFONYL)INDOLE; USEFUL IN TREATING ATHEROSCLEROSIS AND HYPERCHOLESTEROLERNIA TULARIK INC (US) 2000-09-19 US disclosed
CN-1264386-A Alkene borates and process for covalently coupling organic compounds COMMW SCIENT IND RES ORG (AU) 2000-08-23 CN disclosed
CN-1262677-A Preparation of fused polycyclic alkaloids by ring closure of azomethine ylides, novel compounds thereof and their use as chemotherapeutic agents UNIV AUSTRALIAN (AU) 2000-08-09 CN disclosed
US-6100292-A Ketone derivatives and their medical applications TORAY INDUSTRIES, INC. (JP) 2000-08-08 US disclosed
EP-0920412-A4 ELECTROPHORESIS GELS AND CROSS-LINKING AGENTS FOR THEIR PREPARATION UNIV MELBOURNE (AU) 2000-08-02 EP disclosed
EP-1019414-A1 PROCESS FOR PREPARING ORGANIC BORONIC ACID DERIVATIVES USING DIBORONIC ACID COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2000-07-19 EP disclosed
US-6087359-A A MATRIX METALLOPROTEASE ENZYME INHIBITOR PHARMACIA CORPORATION 2000-07-11 US disclosed
EP-1005453-A1 SUBSTITUTED BENZENE COMPOUNDS AS ANTIPROLIFERATIVE AND CHOLESTEROL LOWERING AGENTS TULARIK, INC. (US) 2000-06-07 EP disclosed
US-6071895-A RETROVIRAL PROTEASES INHIBITOR; USEFUL FOR TREATMENT OF HUMAN IMMUNODEFICIENCY VIRUS VIRAL INFECTIONS SUCH AS ACQUIRED IMMUNODEFICIENCY SYNDROME(AIDS); COMPOUND CONTAINING A CYCLIC DIAZAALKANE GROUP NARHEX LIMITED (HK) 2000-06-06 US disclosed
US-6071912-A INHIBIT HUMAN FACTOR XA AND ARE THEREFORE USEFUL AS PHARMACOLOGICAL AGENTS FOR THE TREATMENT OF DISEASE-STATES CHARACTERIZED BY THROMBOTIC ACTIVITY; AMINO-, OXY- AND THIA-SUBSTITUTED TRIAZINES BERLEX LABORATORIES, INC. (US) 2000-06-06 US disclosed
CN-1255123-A Method for Covalently Coupling Organic Compounds Using Diboron Derivatives COMMW SCIENT IND RES ORG (AU) 2000-05-31 CN disclosed
CN-1254337-A N-hydroxy 4-sulfonylbutyramide compounds MONSANTO CO (US) 2000-05-24 CN disclosed
CN-1253559-A Sulfonyl divalent aryl alpha-hydroxamic acid compounds MONSANTO CO (US) 2000-05-17 CN disclosed
CN-1253474-A Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds MONSANTO CO (US) 2000-05-17 CN disclosed
WO-2000021966-A1 ORGANOBORON DERIVATIVES AND PROCESS FOR COUPLING ORGANIC COMPOUNDS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2000-04-20 WO disclosed
EP-0986541-A1 PROCESS FOR COVALENTLY COUPLING ORGANIC COMPOUNDS UTILIZING DIBORON DERIVATIVES COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2000-03-22 EP disclosed
WO-2000014063-A1 THERAPEUTIC COMPOUNDS AND METHODS INSTITUTE OF MOLECULAR & CELL BIOLOGY (SG) 2000-03-16 WO disclosed
EP-0888271-A4 BENZAMIDINE DERIVATIVES SUBSTITUTED BY AMINO ACID AND HYDROXY ACID DERIVATIVES AND THEIR USE AS ANTI-COAGULANTS BERLEX LAB (US) 2000-03-15 EP disclosed
EP-0984959-A1 AROMATIC SULFONYL ALPHA-HYDROXY HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 2000-03-15 EP disclosed
EP-0983257-A1 AROMATIC SULFONYL ALPHA-CYCLOAMINO HYDROXAMIC ACID COMPOUNDS Monsanto Company (US) 2000-03-08 EP disclosed
EP-0983267-A1 AMIDOAROMATIC RING SULFONAMIDE HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 2000-03-08 EP disclosed
US-6034084-A CARDIOVASCULAR DISORDERS BERLEX LABORATORIES, INC. (US) 2000-03-07 US disclosed
US-6034103-A THROMBOSIS THERAPY BERLEX LABORATORIES, INC. (US) 2000-03-07 US disclosed
EP-0981517-A1 PREPARATION OF FUSED POLYCYCLIC ALKALOIDS BY RING CLOSURE OF AZOMETHINE YLIDES, NOVEL COMPOUNDS THEREOF AND THEIR USE AS CHEMOTHERAPEUTIC AGENTS THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 2000-03-01 EP disclosed
EP-0980867-A1 KETONE DERIVATIVES AND MEDICINAL USE THEREOF TORAY INDUSTRIES, INC. (JP) 2000-02-23 EP disclosed
EP-0977745-A1 THIOARYL SULFONAMIDE HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 2000-02-09 EP disclosed
WO-1998050365-A9 PREPARATION OF FUSED POLYCYCLIC ALKALOIDS BY RING CLOSURE OF AZOMETHINE YLIDES, NOVEL COMPOUNDS THEREOF AND THEIR USE AS CHEMOTHERAPEUTIC AGENTS UNIV AUSTRALIAN (AU) 2000-02-03 WO disclosed
EP-0973392-A1 SULFONYL DIVALENT ARYL OR HETEROARYL HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 2000-01-26 EP disclosed
CN-1242770-A Cyclic ketone derivative and pharmaceutical use thereof TORAY INDUSTRIES (JP) 2000-01-26 CN disclosed
US-6013649-A BOND DISORDERS; AUTOIMMUNE DISEASES; ANTITUMOR AGENTS MONSANTO COMPANY (US) 2000-01-11 US disclosed
US-6013836-A PARTICULARLY ACTIVE AGAINST MOTHS AND BEETLES AND THEIR INSECT GROWTH REGULATING ACTIVITY WITHOUT ADVERSE IMPACT ON BENEFICIAL INSECTS; CROPS; FORESTRY ROHM AND HAAS COMPANY (US) 2000-01-11 US disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1999067250-A1 SYNTHESES OF A VARIETY OF LAMELLARIN COMPOUNDS AND ANALOGUES THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 1999-12-29 WO disclosed
US-6004981-A HUMAN FACTOR XA INHIBITORS BERLEX LABORATORIES, INC. 1999-12-21 US disclosed
US-6004985-A BLOOD-COAGULATION FACTOR XA INHIBITORS BERLEX LABORATORIES, INC. (US) 1999-12-21 US disclosed
CN-1238688-A Thiol sulfonamide metalloprotease inhibitors MONSANTO CO (US) 1999-12-15 CN disclosed
EP-0962456-A1 CYCLIC KETONE DERIVATIVE AND PHARMACEUTICAL USE THEREOF TORAY INDUSTRIES, INC. (JP) 1999-12-08 EP disclosed
US-5994375-A ANTICOAGULANTS BERLEX LABORATORIES, INC. (US) 1999-11-30 US disclosed
CN-1235172-A Process for producing cycloolefin copolymer, cycloolefin copolymer produced by the process, and use of the copolymer HOECHST AG (DE) 1999-11-17 CN disclosed
WO-1999051594-A1 IMIDAZO[1,2-a]PYRIDINES AS PERIPHERAL BENZODIAZEPINE RECEPTOR BINDING AGENTS AUSTRALIAN NUCLEAR SCIENCE & TECHNOLOGY ORGANISATION (AU) 1999-10-14 WO disclosed
WO-1999050257-A1 BENZOXAZINONES/BENZOTHIAZINONES AS SERINE PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1999-10-07 WO disclosed
WO-1999050263-A1 QUINOLONES AS SERINE PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1999-10-07 WO disclosed
WO-1999050254-A1 QUINOXALINONES AS SERINE PROTEASE INHIBITORS SUCH AS FACTOR XA AND THROMBIN WARNER-LAMBERT COMPANY (US) 1999-10-07 WO disclosed
WO-1999050327-A1 NON-ELASTOMERIC POLYURETHANE COMPOSITIONS CARDIAC CRC NOMINEES PTY. LTD. (AU) 1999-10-07 WO disclosed
CN-1230884-A Thiol sulfone metalloprotease inhibitors MONSANTO CO (US) 1999-10-06 CN disclosed
US-5942504-A INHIBITORS OF RETROVIRAL PROTEASES; TREATMENT OF AIDS AND HIV NARHEX LIMITED (HK) 1999-08-24 US disclosed
EP-0934310-A1 THIO ACID DERIVED MONOCYCLIC $i(N)-HETEROCYCLICS AS ANTICOAGULANTS SCHERING AKTIENGESELLSCHAFT (DE) 1999-08-11 EP disclosed
CN-1225009-A Pentafluorobenzenesulfonamides and analogs thereof TULARIK INC (US) 1999-08-04 CN disclosed
WO-1999033845-A1 BORONIC COMPOUNDS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 1999-07-08 WO disclosed
EP-0920412-A1 ELECTROPHORESIS GELS AND CROSS-LINKING AGENTS FOR THEIR PREPARATION THE UNIVERSITY OF MELBOURNE (AU) 1999-06-09 EP disclosed
WO-1999025687-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE & CO. (US) 1999-05-27 WO disclosed
WO-1999024411-A1 RECEPTOR WITH AN AFFINITY FOR COMPOUNDS OF THE OXAZOLINE CLASS THE UNIVERSITY OF MELBOURNE (AU) 1999-05-20 WO disclosed
EP-0896533-A4 PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS TULARIK INC (US) 1999-04-28 EP disclosed
US-5889005-A Benzamidine derivatives and their use for treating thrombotic diseases BERLEX LABORATORIES, INC. (US) 1999-03-30 US disclosed
US-5888992-A PROTEASE INHIBITOR; VIRICIDE NARHEX LIMITED (HK) 1999-03-30 US disclosed
WO-1999012940-A1 PROCESS FOR PREPARING ORGANIC BORONIC ACID DERIVATIVES USING DIBORONIC ACID COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 1999-03-18 WO disclosed
US-5883100-A Benzamidine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. (US) 1999-03-16 US disclosed
US-5880151-A TREATING OR PREVENTING DISEASE CHARACTERIZED BY HIGH LEVELS OF LOW DENSITY LIPOPROTEIN PARTICLES OR CHOLESTEROL IN BLOOD TULARIK INC. (US) 1999-03-09 US disclosed
US-5879585-A EXHIBIT GOOD MISCIBILITY WITH OTHER LIQUID CRYSTALLINE COMPOUNDS; USEFUL FOR DISPLAY OF WATCHES, COMPUTER TERMINALS, AND TELEVISIONS CHISSO CORPORATION (JP) 1999-03-09 US disclosed
WO-1999010320-A1 SUBSTITUTED BENZENE COMPOUNDS AS ANTIPROLIFERATIVE AND CHOLESTEROL LOWERING AGENTS TULARIK INC. (US) 1999-03-04 WO disclosed
US-5877181-A Benzamidine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. (US) 1999-03-02 US disclosed
US-5877119-A HERBICIDE ROHM AND HAAS COMPANY (US) 1999-03-02 US disclosed
EP-0896533-A2 PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS TULARIK, INC. (US) 1999-02-17 EP disclosed
US-5872111-A TOILET BAR SOAP, FACIAL BODY CLEANSER, SHAMPOO, CONDITIONER, COSMETIC,SHAVING CREAM OR LOTION, SHOWER GEL, FABRIC SOFTENING CONDITIONER, AND UNDERARM DEODORANT/ANTI-PERSPIRANT LEVER BROTHERS COMPANY, DIVISION OF CONOPCO, INC. (US) 1999-02-16 US disclosed
WO-1999005099-A1 SYNTHESIS OF DITHIOESTER CHAIN TRANSFER AGENTS AND USE OF BIS(THIOACYL) DISULFIDES OR DITHIOESTERS AS CHAIN TRANSFER AGENTS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 1999-02-04 WO disclosed
EP-0888271-A1 BENZAMIDINE DERIVATIVES SUBSTITUTED BY AMINO ACID AND HYDROXY ACID DERIVATIVES AND THEIR USE AS ANTI-COAGULANTS BERLEX LABORATORIES, INC. (US) 1999-01-07 EP disclosed
US-5846972-A Bicyclic pyrimidine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. (US) 1998-12-08 US disclosed
US-5846970-A Bicyclic pyrimidine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. (US) 1998-12-08 US disclosed
US-5843867-A Substituted pyridine compounds ROHM AND HAAS COMPANY (US) 1998-12-01 US disclosed
EP-0813556-B1 LIQUID PHASE POWDER BED SYNDIOTACTIC VINYLAROMATIC POLYMERIZATION DOW CHEMICAL CO (US) 1998-11-25 EP disclosed
WO-1998050365-A1 PREPARATION OF FUSED POLYCYCLIC ALKALOIDS BY RING CLOSURE OF AZOMETHINE YLIDES, NOVEL COMPOUNDS THEREOF AND THEIR USE AS CHEMOTHERAPEUTIC AGENTS THE AUSTRALIAN NATIONAL UNIVERSITY (AU) 1998-11-12 WO disclosed
US-5824625-A HERBICIDES, HETEROCYCLIC GROUP(S) ATTACHED TO PYRIDINE RING ROHM AND HAAS COMPANY 1998-10-20 US disclosed
WO-1998045265-A1 PROCESS FOR COVALENTLY COUPLING ORGANIC COMPOUNDS UTILIZING DIBORON DERIVATIVES COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 1998-10-15 WO disclosed
CN-1194580-A Ketone derivatives and medical use thereof TORAY INDUSTRIES (JP) 1998-09-30 CN disclosed
WO-1998039313-A1 THIOARYL SULFONAMIDE HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 1998-09-11 WO disclosed
WO-1998039315-A1 AROMATIC SULFONYL ALPHA-CYCLOAMINO HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 1998-09-11 WO disclosed
WO-1998039326-A1 AROMATIC SULFONYL ALPHA-HYDROXY HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 1998-09-11 WO disclosed
WO-1998038859-A1 SULFONYL DIVALENT ARYL OR HETEROARYL HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 1998-09-11 WO disclosed
WO-1998039329-A1 AMIDOAROMATIC RING SULFONAMIDE HYDROXAMIC ACID COMPOUNDS MONSANTO COMPANY (US) 1998-09-11 WO disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed
EP-0857067-A1 RADIOPROTECTORS The Inner and Eastern Health Care Network (AU) 1998-08-12 EP disclosed
US-5753635-A Purine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. (US) 1998-05-19 US disclosed
EP-0841063-A1 KETONE DERIVATIVES AND MEDICINAL USE THEREOF TORAY INDUSTRIES, INC. (JP) 1998-05-13 EP disclosed
EP-0837045-A1 Liquid crystalline compound having alkynyl group, and liquid crystal composition and liquid crystal display device therefrom Chisso Corporation (JP) 1998-04-22 EP disclosed
WO-1998015547-A1 THIO ACID DERIVED MONOCYCLIC N-HETEROCYCLICS AS ANTICOAGULANTS SCHERING AKTIENGESELLSCHAFT (DE) 1998-04-16 WO disclosed
US-5739140-A AGRICULTURAL FUNGICIDES MONSANTO COMPANY (US) 1998-04-14 US disclosed
WO-1998001419-A1 ELECTROPHORESIS GELS AND CROSS-LINKING AGENTS FOR THEIR PREPARATION THE UNIVERSITY OF MELBOURNE (AU) 1998-01-15 WO disclosed
EP-0813525-A1 BENZAMIDINE DERIVATIVES THEIR PREPARATION AND THEIR USE AS ANTI-COAGULANTS BERLEX LABORATORIES, INC. (US) 1997-12-29 EP disclosed
US-5693641-A ENZYME INHIBITOR TREATING BLOOD DISORDER BERLEX LABORATORIES INC. (US) 1997-12-02 US disclosed
US-5691364-A Benzamidine derivatives and their use as anti-coagulants BERLEX LABORATORIES, INC. (US) 1997-11-25 US disclosed
US-5679688-A RETROVIRAL PROTEASE INHIBITORS; AIDS THERAPY NARHEX LIMITED (HK) 1997-10-21 US disclosed
WO-1997030677-A2 PENTAFLUOROBENZENESULFONAMIDES AND ANALOGS TULARIK, INC. (US) 1997-08-28 WO disclosed
WO-1997029067-A1 BENZAMIDINE DERIVATIVES SUBSTITUTED BY AMINO ACID AND HYDROXY ACID DERIVATIVES AND THEIR USE AS ANTI-COAGULANTS BERLEX LABORATORIES, INC. (DE) 1997-08-14 WO disclosed
US-5648349-A PHOSPHOLIPASE INHIBITORS MONSANTO COMPANY (US) 1997-07-15 US disclosed
US-5643854-A HERBICIDES ROHM AND HAAS COMPANY (US) 1997-07-01 US disclosed
EP-0586556-B1 SUBSTITUTED 2,6-SUBSTITUTED PYRIDINE HERBICIDES ROHM & HAAS (US) 1997-04-16 EP disclosed
WO-1997004776-A1 RADIOPROTECTORS THE INNER AND EASTERN HEALTH CARE NETWORK (AU) 1997-02-13 WO disclosed
CN-1135212-A polar substituted hydrocarbons NARHEX AUSTRALIA PTY LTD (AU) 1996-11-06 CN disclosed
WO-1996028427-A1 BENZAMIDINE DERIVATIVES THEIR PREPARATION AND THEIR USE AS ANTI-COAGULANTS BERLEX LABORATORIES, INC. (US) 1996-09-19 WO disclosed
EP-0717736-A4 POLAR-SUBSTITUTED HYDROCARBONS NARHEX LTD (HK) 1996-08-28 EP disclosed
EP-0717736-A1 POLAR-SUBSTITUTED HYDROCARBONS NARHEX LIMITED (HK) 1996-06-26 EP disclosed
WO-1996016094-A1 PREPARATION OF SYNDIOTACTIC POLYOLEFINS FROM PROCHIRAL OLEFINS THE DOW CHEMICAL COMPANY (US) 1996-05-30 WO disclosed
US-5514812-A Preparation of stereochemically pure oximes with muscarinic activity WARNER-LAMBERT COMPANY (US) 1996-05-07 US disclosed
US-5512536-A HERBICIDE ROHN AND HAAS COMPANY (US) 1996-04-30 US disclosed
US-5504255-A Optically active compounds and a method for producing them CHISSO CORPORATION (JP) 1996-04-02 US disclosed
US-5504237-A PLA2 inhibitors MONSANTO COMPANY (US) 1996-04-02 US disclosed
EP-0445731-B1 Azabicyclo and azacyclo oxime and amine cholinergic agents and pharmaceutically acceptable salts thereof WARNER LAMBERT CO (US) 1996-01-10 EP disclosed
US-5482938-A Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment WARNER-LAMBERT COMPANY (US) 1996-01-09 US disclosed
CN-1112564-A Metallocenes and their use as catalysts HOECHST AG (DE) 1995-11-29 CN disclosed
WO-1995031202-A1 CAGE COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS ANTIVIRAL AGENTS COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 1995-11-23 WO disclosed
US-5464842-A Azabicyclo oxime and amine cholinergic agents and methods of treatment WARNER-LAMBERT COMPANY (US) 1995-11-07 US disclosed
CN-1108666-A Process for preparing polyolefins HOECHST AG (DE) 1995-09-20 CN disclosed
US-5446175-A Optically active compounds and a method for producing them CHISSO CORPORATION (JP) 1995-08-29 US disclosed
US-5434288-A Phospholipase A2 inhibitor MONSANTO COMPANY (US) 1995-07-18 US disclosed
US-5424333-A Anthelmintic N'-substituted-N,N'-disubstitutedhydrazines ROHM AND HAAS COMPANY (US) 1995-06-13 US disclosed
EP-0382463-B1 Maleimide compounds and fungicides containing them SUNTORY LTD (JP) 1995-04-26 EP disclosed
WO-1995007269-A1 POLAR-SUBSTITUTED HYDROCARBONS NARHEX LIMITED (HK) 1995-03-16 WO disclosed
EP-0641337-A1 CYCLIC ALKYLIDENE SUBSTITUTED PYRIDINE HERBICIDES ROHM AND HAAS COMPANY (US) 1995-03-08 EP disclosed
US-5391540-A Herbicides ROHM AND HAAS COMPANY (US) 1995-02-21 US disclosed
EP-0292990-B1 4-Halopyridine-3-carboxamide compounds and herbicidal composition thereof DAICEL CHEM (JP) 1995-02-01 EP disclosed
US-5380812-A Storage stability DOW CORNING CORPORATION (US) 1995-01-10 US disclosed
US-5364922-A Storage stable polymers DOW CORNING CORPORATION (US) 1994-11-15 US disclosed
US-5354762-A Insecticides ROHM AND HAAS COMPANY (US) 1994-10-11 US disclosed
EP-0371264-B1 Phosphonate reagent compositions and methods of making same UNIV LOYOLA CHICAGO (US) 1994-09-14 EP disclosed
US-5346911-A Analgesics, cognition activators, treatment of alzheimer*s s disease WARNER-LAMBERT COMPANY (US) 1994-09-13 US disclosed
US-5318978-A Azabicyclo oxime and amine cholinergic agents and methods of treatment WARNER-LAMBERT COMPANY (US) 1994-06-07 US disclosed
US-5306718-A Analgesics, cognition activators WARNER-LAMBERT COMPANY (US) 1994-04-26 US disclosed
US-5306638-A Stereoselective EASTMAN KODAK COMPANY (US) 1994-04-26 US disclosed
EP-0586556-A1 SUBSTITUTED 2,6-SUBSTITUTED PYRIDINE HERBICIDES. MONSANTO CO (US) 1994-03-16 EP disclosed
EP-0581095-A2 Substituted acrylic acid esters and plant-protecting agents containing them BASF Aktiengesellschaft (DE) 1994-02-02 EP disclosed
EP-0573575-A1 SUBSTITUTED PYRIDINE COMPOUNDS ROHM AND HAAS COMPANY (US) 1993-12-15 EP disclosed
EP-0361645-B1 ORGANIC HYDRAZINE DERIVATIVES FOR PHARMACEUTICAL USE ROHM AND HAAS COMPANY (US) 1993-09-29 EP disclosed
EP-0347216-B1 INSECTICIDAL N'-SUBSTITUTED-N-ALKYLCARBONYL-N'-ACYLHYDRAZINES AND N'-SUBSTITUTED -N-ACYL-N'-ALKYLCARBONYL HYDRAZINES ROHM AND HAAS COMPANY (US) 1993-09-01 EP disclosed
EP-0312019-B1 CONDENSED HETEROCYCLIC COMPOUNDS, A PROCESS FOR PREPARING THE SAME AND A HERBICIDAL COMPOSITION THEREOF DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1993-08-04 EP disclosed
US-5228897-A Herbicides MONSANTO COMPANY (US) 1993-07-20 US disclosed
US-5225443-A Lepidotera and Coleoptera insecticides to protect plants ROHM AND HAAS COMPANY (US) 1993-07-06 US disclosed
EP-0339854-B1 SYNTHESIS OF N-T-ALKYL-1,2-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1993-05-26 EP disclosed
WO-1993008191-A1 AZABICYCLO OXIME AND AMINE CHOLINERGIC AGENTS AND METHODS OF TREATMENT WARNER-LAMBERT COMPANY (US) 1993-04-29 WO disclosed
EP-0173848-B1 BENZOPYRAN COMPOUNDS FOR USE IN THE CARDIOVASCULAR SYSTEM BEECHAM GROUP PLC (GB) 1992-12-23 EP disclosed
EP-0261755-B1 FIVE-MEMBERED HETEROCYCLIC DERIVATIVES OF N'-SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1992-12-16 EP disclosed
WO-1992021674-A1 CYCLIC ALKYLIDENE SUBSTITUTED PYRIDINE HERBICIDES MONSANTO COMPANY (US) 1992-12-10 WO disclosed
US-5169432-A 2-and/or 6-fluoroalkyl substituted and a carbonyl oxy(thio) ester or a heterocyclo-carbonyl at the 3 or 5 position MONSANTO COMPANY (US) 1992-12-08 US disclosed
WO-1992020659-A1 SUBSTITUTED 2,6-SUBSTITUTED PYRIDINE HERBICIDES MONSANTO COMPANY (US) 1992-11-26 WO disclosed
CN-1066060-A Medicinal compound LILLY CO ELI (US) 1992-11-11 CN disclosed
EP-0510947-A1 N-Hydroxy (thio)ureas as 5-lipoxygenase inhibitors ELI LILLY AND COMPANY (US) 1992-10-28 EP disclosed
US-5156670-A Low soil mobility MONSANTO COMPANY (US) 1992-10-20 US disclosed
WO-1992014711-A1 SUBSTITUTED PYRIDINE COMPOUNDS MONSANTO COMPANY (US) 1992-09-03 WO disclosed
US-5130485-A For treatment of asthma, arthritis, allergy, inflammatory bowel disease, psoriasis, respiratory system disorders and antiischemic agents ELI LILLY AND COMPANY (US) 1992-07-14 US disclosed
US-5125956-A Preemergence herbicides MONSANTO COMPANY (US) 1992-06-30 US disclosed
EP-0245950-B1 INSECTICIDAL N-SUBSTITUTED-N' - SUBSTITUTED-N, N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1992-06-17 EP disclosed
US-5117057-A Insecticidal N' substituted-N-N'-disubstituted-hydrazines ROHM AND HAAS COMPANY (US) 1992-05-26 US disclosed
US-5110986-A Reaction of a 1,3,4-oxadiazole with a tert-alkyl cation precursor in presence of strong acid catalyst ROHM AND HAAS COMPANY (US) 1992-05-05 US disclosed
EP-0176689-B1 BENZOPYRAN COMPOUNDS FOR THE TREATMENT OF SMOOTH MUSCLES CONTRACTION BEECHAM GROUP PLC (GB) 1992-04-01 EP disclosed
EP-0204285-B1 IMIDAZOHETEROCYCLIC COMPOUNDS PROCESSES FOR PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-01-15 EP disclosed
EP-0253468-B1 SIX-MEMBERED HETEROCYCLIC DERIVATIVES OF N'SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-11-06 EP disclosed
EP-0207614-B1 BENZOPYRAN COMPOUNDS IN THE TREATMENT OF INCONTINENCE BEECHAM GROUP PLC (GB) 1991-09-25 EP disclosed
CN-1054601-A Azabicyclo and azepine cyclic oximes and amine cholinergic agents thing and methods of treatment thereof WARNER LAMBERT CO (US) 1991-09-18 CN disclosed
EP-0445731-A1 Azabicyclo and azacyclo oxime and amine cholinergic agents and pharmaceutically acceptable salts thereof WARNER-LAMBERT COMPANY (US) 1991-09-11 EP disclosed
US-5039696-A Maleimide derivatives and fungicides for agriculture and horticulture containing the same SUNTORY LIMITED (JP) 1991-08-13 US disclosed
US-5032596-A Hypotensive BEECHAM GROUP P.L.C. (GB) 1991-07-16 US disclosed
EP-0234944-B1 INSECTICIDAL N'-SUBSTITUTED-N-ACYL-N'-ALKYLCARBONYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-04-10 EP disclosed
EP-0232075-B1 INSECTICIDAL N'-SUBSTITUTED-N-ALKYLCARBONYL-N'-ACYL HYDRAZINES ROHM AND HAAS COMPANY (US) 1991-03-13 EP disclosed
EP-0286746-B1 INSECTICIDAL N-(OPTIONALLY SUBSTITUTED) - N'-SUBSTITUTED-N,N'-DISUBSTITUTED- HYDRAZINES ROHM AND HAAS COMPANY (US) 1991-02-27 EP disclosed
US-4985461-A Insecticidal N'-substituted-N,N'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1991-01-15 US disclosed
US-4978385-A 4-halopyridine-3-carboxamide compounds and herbicidal compositions thereof DAICEL CHEMICAL INDUSTRIES LTD. (JP) 1990-12-18 US disclosed
EP-0193853-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1990-09-12 EP disclosed
EP-0382463-A1 Maleimide compounds and fungicides containing them SUNTORY LIMITED (JP) 1990-08-16 EP disclosed
US-4943314-A Pyridine-3-carboxamide derivatives having plant growth inhibiting activity DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1990-07-24 US disclosed
US-4936121-A Condensed heterocyclic compounds, a process for preparing the same and a herbicidal composition thereof DAICEL CHEMICAL INDUSTRIES LTD. (JP) 1990-06-26 US disclosed
EP-0361645-A2 Organic hydrazine derivatives for pharmaceutical use ROHM AND HAAS COMPANY (US) 1990-04-04 EP disclosed
EP-0347216-A2 Insecticidal N'-substituted-N-alkylcarbonyl-N'-acylhydrazines and N'-substituted -N-acyl-N'-alkylcarbonyl hydrazines ROHM AND HAAS COMPANY (US) 1989-12-20 EP disclosed
US-4886546-A Pyrone-3-carboxamide compounds and herbicidal composition thereof DAICEL CHEMICAL INDUSTRIES LTD. (JP) 1989-12-12 US disclosed
EP-0339071-A1 IMIDAZO(1,2-a)(PYRIDAZINES OR PYRAZINES) FOR TREATMENT OF DISEASES RELATED TO BONE LOSS Aktiebolaget Hässle (SE) 1989-11-02 EP disclosed
EP-0339854-A2 Synthesis of N-t-alkyl-1,2-diacylhydrazines ROHM AND HAAS COMPANY (US) 1989-11-02 EP disclosed
EP-0149760-B1 SUBSTITUTED O-ACYL GLYCOSYLAMIDES, METHODS FOR THEIR PREPARATION AND THEIR USE BAYER AG (DE) 1989-08-23 EP disclosed
EP-0193887-B1 SUBSTITUTED O-SULFONYL-GLYCOSYL AMIDES, METHOD FOR THEIR PREPARATION AND THEIR USE AS MEDIACMENTS BAYER AG (DE) 1989-07-26 EP disclosed
US-4844732-A PLANT GROWTH REGULATORS DAICEL CHEMICAL INDUSTRIES LTD. (JP) 1989-07-04 US disclosed
EP-0149093-B1 N-GLYCOSYLATED UREAS, CARBAMATES AND THIOCARBAMATES, THEIR PREPARATION METHOD AND THEIR USE BAYER AG (DE) 1989-05-31 EP disclosed
WO-1989003833-A1 IMIDAZO(1,2-a)(PYRIDAZINES OR PYRAZINES) FOR TREATMENT OF DISEASES RELATED TO BONE LOSS Aktiebolaget Hässle (SE) 1989-05-05 WO disclosed
EP-0312019-A2 Condensed heterocyclic compounds, a process for preparing the same and a herbicidal composition thereof DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1989-04-19 EP disclosed
EP-0140321-B1 USE OF DERIVATIVES OF AMIDES OF CARBOXYLIC ACIDS IN WHICH THE N ATOM IS SUBSTITUTED BY A GLYCOSYL RADICAL AS GROWTH PROMOTOR IN ANIMAL NUTRITION BAYER AG (DE) 1989-04-12 EP disclosed
EP-0143385-B1 PHOSPHORYLISED GLYCOSIL AMIDES, UREAS, CARBAMATES AND THIOCARBAMATES, METHOD FOR THEIR PREPARATION AND THEIR USE BAYER AG (DE) 1989-03-15 EP disclosed
EP-0301713-A2 Chroman derivatives for treatment of pulmonary hypertension BEECHAM GROUP PLC (GB) 1989-02-01 EP disclosed
EP-0292990-A1 4-Halopyridine-3-carboxamide compounds and herbicidal composition thereof DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1988-11-30 EP disclosed
US-4786639-A ADMINISTERING BENZOPYRAN DERIVATIVES BEECHAM GROUP P.L.C. (GB) 1988-11-22 US disclosed
EP-0286746-A1 Insecticidal N-(optionally substituted) - N'-substituted-N,N'-disubstituted- hydrazines ROHM AND HAAS COMPANY (US) 1988-10-19 EP disclosed
US-4777256-A PLANT GROWTH REGULATORS, ANTIINFLAMMATORY AGENTS DAICEL CHEMICAL INDUSTRIES LTD. (JP) 1988-10-11 US disclosed
US-4772603-A CHROMENE COMPOUNDS BEECHAM GROUP P.L.C. (GB) 1988-09-20 US disclosed
US-4755598-A 1'-(substituted)ethyl-7β-[2-(2-aminothiazol-4-yl)acetamido]-3-[[[1-(2-dimethylaminoethyl)-1H-tetrazol-5-yl]thio]methyl]ceph-3-em-4-carboxylate derivatives having antibacterial utility TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-07-05 US disclosed
US-4744819-A 4-oxo pyridinecarboxamide derivatives as plant growth regulators DAICEL CHEMICAL INDUSTRIES LTD. (JP) 1988-05-17 US disclosed
US-4739083-A REACTING 1,3-DIOXAN-4-ONE WITH (AMINE OR IMINE) SUBSTITUTED AMIDE DAICEL CHEMICAL INDUSTRIES LTD. (JP) 1988-04-19 US disclosed
US-4738963-A NITROGEN SUBSTITUTED BENZO(B)PYRAN BEECHAM GROUP P.L.C. (GB) 1988-04-19 US disclosed
US-4737488-A Immune system-stimulating N-glycosylated ureas and carbamates BAYER AKTIENGESELLSCHAFT (DE) 1988-04-12 US disclosed
EP-0261755-A2 Five-membered heterocyclic derivatives of N'-substituted-N,N'-Diacylhydrazines ROHM AND HAAS COMPANY (US) 1988-03-30 EP disclosed
US-4725306-A Pyridinecarboxamide plant growth inhibitors DAICEL CHEMICAL INDUSTRIES LTD. (JP) 1988-02-16 US disclosed
US-4725601-A Certain imidazo[1,2-a]pyridines useful in the treatment of ulcers FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-02-16 US disclosed
EP-0253468-A2 Six-membered heterocyclic derivatives of N'substituted-N,N'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1988-01-20 EP disclosed
US-4716152-A IMMUNOSTIMULANTS BAYER AKTIENGESELLSCHAFT (DE) 1987-12-29 US disclosed
US-4710491-A N-glycosylated carboxylic acid derivatives as agents for combating rheumatic diseases TROPONWERKE GMBH & CO., KG (DE) 1987-12-01 US disclosed
EP-0245950-A2 Insecticidal n-substituted-n' - substituted-n, n'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1987-11-19 EP disclosed
US-4699899-A IMMUNE STIMULANTS BAYER AKTIENGESELLSCHAFT (DE) 1987-10-13 US disclosed
EP-0234944-A1 Insecticidal N'-substituted-N-acyl-N'-alkylcarbonylhydrazines ROHM AND HAAS COMPANY (US) 1987-09-02 EP disclosed
EP-0232075-A1 Insecticidal N'-substituted-N-alkylcarbonyl-N'-acyl hydrazines ROHM AND HAAS COMPANY (US) 1987-08-12 EP disclosed
US-4686208-A Phosphorylated glycosyl-amides, -ureas, -carbamates and -thiocarbamates and method of use BAYER AKTIENGESELLSCHAFT (DE) 1987-08-11 US disclosed
US-4683222-A STIMULANTS FOR IMMUNE SYSTEM BAYER AKTIENGESELLSCHAFT (DE) 1987-07-28 US disclosed
US-4680287-A N-glycosylated carboxamide derivatives as growth-promoters in livestock feeding BAYER AKTIENGESELLSCHAFT (DE) 1987-07-14 US disclosed
CN-86104313-A The preparation method of Imidazoheterocyclic compounds 1987-03-04 CN disclosed
EP-0091645-B1 DERIVATIVES OF AMIDES OF CARBOXYLIC ACIDS IN WHICH THE N ATOM IS SUBSTITUTED BY A GLYCOSYL RADICAL, METHOD FOR THEIR PREPARATION AND THEIR USE TO INFLUENCE THE IMMUNOGENIC SYSTEM BAYER AG (DE) 1987-02-25 EP disclosed
EP-0207614-A2 Benzopyran compounds in the treatment of incontinence BEECHAM GROUP PLC (GB) 1987-01-07 EP disclosed
US-4631272-A N-acylated 1-alkylamino-1-deoxy-ketose derivatives, a process for their preparation and their use BAYER AKTIENGESELLSCHAFT (DE) 1986-12-23 US disclosed
US-4629734-A HYPOTENSIVE AGENTS BEECHAM GROUP P.L.C. (GB) 1986-12-16 US disclosed
EP-0204285-A1 Imidazoheterocyclic compounds processes for preparation thereof and pharmaceutical compositions comprising them FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1986-12-10 EP disclosed
EP-0193887-A2 Substituted O-sulfonyl-glycosyl amides, method for their preparation and their use as mediacments BAYER AG (DE) 1986-09-10 EP disclosed
EP-0189596-A1 Benzofuran and benzothiophene derivatives SHIONOGI & CO., LTD. (JP) 1986-08-06 EP disclosed
EP-0176689-A2 Benzopyran compounds for the treatment of smooth muscles contraction BEECHAM GROUP PLC (GB) 1986-04-09 EP disclosed
EP-0173848-A2 Benzopyran compounds for use in the cardiovascular system BEECHAM GROUP PLC (GB) 1986-03-12 EP disclosed
US-4574122-A ANTIBODIES, IMMUNOLOGY BAYER AKTIENGESELLSCHAFT (DE) 1986-03-04 US disclosed
US-4556415-A POST-EMERGENCE MONSANTO COMPANY (US) 1985-12-03 US disclosed
EP-0155625-A2 Glycolipid-like substances in liposome form BAYER AG (DE) 1985-09-25 EP disclosed
EP-0152856-A2 N-acylated 1-alkylamimo-1-desoxy ketose derivatives, method for their preparation and use BAYER AG (DE) 1985-08-28 EP disclosed
EP-0152630-A2 Organosiloxane polymers and compositions containing same curable upon exposure to gaseous oxygen UNION CARBIDE CORPORATION (US) 1985-08-28 EP disclosed
EP-0149760-A2 Substituted O-acyl glycosylamides, methods for their preparation and their use BAYER AG (DE) 1985-07-31 EP disclosed
EP-0149093-A2 N-glycosylated ureas, carbamates and thiocarbamates, their preparation method and their use BAYER AG (DE) 1985-07-24 EP disclosed
EP-0147777-A2 Derivatives of M-glycosylated amides of carboxylic acids as a product for combating diseases of the rheumatism type Troponwerke GmbH &amp; Co. KG (DE) 1985-07-10 EP disclosed
US-4526954-A Contains olefinically polyunsaturated radical containing 1,3- or 1,4-pentadienylene group bonded to silicon UNION CARBIDE CORPORATION (US) 1985-07-02 US disclosed
EP-0144894-A2 Therapeutic application of substituted O-acyl-glycosides BAYER AG (DE) 1985-06-19 EP disclosed
EP-0143385-A2 Phosphorylised glycosil amides, ureas, carbamates and thiocarbamates, method for their preparation and their use BAYER AG (DE) 1985-06-05 EP disclosed
EP-0140321-A2 Use of derivatives of amides of carboxylic acids in which the N atom is substituted by a glycosyl radical as growth promotor in animal nutrition BAYER AG (DE) 1985-05-08 EP disclosed
EP-0128028-A2 Cephalosporin derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1984-12-12 EP disclosed
EP-0091645-A1 Derivatives of amides of carboxylic acids in which the N atom is substituted by a glycosyl radical, method for their preparation and their use to influence the immunogenic system BAYER AG (DE) 1983-10-19 EP disclosed
US-4349552-A TREATMENT OF CANCER FUJISAWA PHARMACEUTICAL COMPANY, LTD. (JP) 1982-09-14 US disclosed
EP-0002938-B1 NOVEL HETEROCYCLIC CARBOTHIOAMIDES, COMPOSITIONS CONTAINING THEM, THEIR PREPARATION AND USE ELI LILLY AND COMPANY (US) 1982-05-12 EP disclosed
EP-0002939-B1 NOVEL CARBOTHIOAMIDES, COMPOSITIONS CONTAINING THEM AND THEIR PREPARATION ELI LILLY AND COMPANY (US) 1982-04-21 EP disclosed
EP-0003081-B1 THIAZOLIDINECARBOTHIOAMIDES, THEIR PREPARATION, COMPOSITIONS AND USE AS INSECTICIDES ELI LILLY AND COMPANY (US) 1981-12-30 EP disclosed
US-4289766-A Heterocyclic carbothioamides ELI LILLY AND COMPANY (US) 1981-09-15 US disclosed
US-4289778-A SYSTEMIC INSECTICIDES ELI LILLY AND COMPANY (US) 1981-09-15 US disclosed
EP-0010941-A1 5-Fluorouracil derivatives, preparation thereof and their pharmaceutical compositions FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1980-05-14 EP disclosed
US-4195092-A INSECTICIDES FOR TREATING MEXICAN BEAN BEETLE ELI LILLY AND COMPANY (US) 1980-03-25 US disclosed
US-4166908-A SELECTIVE PREEMERGENT ACTIVITY AMERICAN CYANAMID COMPANY (US) 1979-09-04 US disclosed
EP-0003081-A2 Thiazolidinecarbothioamides, their preparation, compositions and use as insecticides ELI LILLY AND COMPANY (US) 1979-07-25 EP disclosed
EP-0002939-A2 Novel carbothioamides, compositions containing them and their preparation ELI LILLY AND COMPANY (US) 1979-07-11 EP disclosed
EP-0002938-A2 Novel heterocyclic carbothioamides, compositions containing them, their preparation and use ELI LILLY AND COMPANY (US) 1979-07-11 EP disclosed
US-3971825-A (5,6) (10,11) BIS-METHYLENE, BRONCHODILATORS SANKYO COMPANY LIMITED (JA) 1976-07-27 US disclosed
US-3943153-A BACTERICIDES MERCK & CO., INC. (US) 1976-03-09 US disclosed
US-3943153-A BACTERICIDES MERCK & CO., INC. (US) 1976-03-09 US disclosed