SCHEMBL2564516

SCHEMBL2564516

CC(=O)N(Cl)C12CC3CC(C)(CC(C)(C3)C1)C2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 5/20 0.53
GRIN2A Q12879 5/20 0.53
GRIN2D O15399 4/20 0.53
GRIN3B O60391 4/20 0.53
GRIN2B Q13224 4/20 0.53
GRIN2C Q14957 4/20 0.53
GRIN3A Q8TCU5 4/20 0.53
EPHX2 P34913 4/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 2/20 0.38
SLC22A1 O15245 1/20 0.38
ESR1 P03372 1/20 0.38
ADRB3 P13945 1/20 0.38
ACHE P22303 1/20 0.38
OPRK1 P41145 1/20 0.38
MTOR P42345 1/20 0.38
HTT P42858 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28011393 0.81 GRIN1 (0.57) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
SCHEMBL15562785 0.79 GRIN1 (0.53) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
SCHEMBL659842 0.70 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
Hydrochloric Acid SCHEMBL11656331 0.69 GRIN1 (0.95) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
SCHEMBL28098360 0.68 GRIN1 (0.41) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
SCHEMBL812216 0.68 GRIN1 (0.68) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
SCHEMBL28833937 0.67 GRIN2D (0.41) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
SCHEMBL7453250 0.67 MEN1 (0.58) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
SCHEMBL733617 0.67 EPHX2 (0.62) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
Ammonia Solution, Strong SCHEMBL14695768 0.66 GRIN1 (0.65) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097372-B1 PROCESS FOR THE PREPARATION OF MEMANTINE AND ITS HYDROCHLORIC ACID SALT FORM KRKA D D NOVO MESTO (SI) 2017-05-31 EP claimed
EP-2097372-A1 PROCESS FOR THE PREPARATION OF MEMANTINE AND ITS HYDROCHLORIC ACID SALT FORM KRKA, D.D., Novo Mesto (SI) 2009-09-09 EP claimed
WO-2008040560-A1 PROCESS FOR THE PREPARATION OF MEMANTINE AND ITS HYDROCHLORIC ACID SALT FORM KRKA, D.D., NOVO MESTO (SI) 2008-04-10 WO claimed
EP-1908748-A1 Process for the preparation of memantine and its hydrochloric acid salt form KRKA (SI) 2008-04-09 EP claimed
EP-2097372-B1 PROCESS FOR THE PREPARATION OF MEMANTINE AND ITS HYDROCHLORIC ACID SALT FORM KRKA D D NOVO MESTO (SI) 2017-05-31 EP disclosed
EP-2555616-A1 PROCESS FOR THE PREPARATION OF MEMANTINE HYDROCHLORIDE Hetero Research Foundation (IN) 2013-02-13 EP disclosed
WO-2011125062-A1 PROCESS FOR THE PREPARATION OF MEMANTINE HYDROCHLORIDE HETERO RESEARCH FOUNDATION (IN) 2011-10-13 WO disclosed
EP-2097372-A1 PROCESS FOR THE PREPARATION OF MEMANTINE AND ITS HYDROCHLORIC ACID SALT FORM KRKA, D.D., Novo Mesto (SI) 2009-09-09 EP disclosed
EP-2097372-A1 PROCESS FOR THE PREPARATION OF MEMANTINE AND ITS HYDROCHLORIC ACID SALT FORM KRKA, D.D., Novo Mesto (SI) 2009-09-09 EP disclosed
WO-2008040560-A1 PROCESS FOR THE PREPARATION OF MEMANTINE AND ITS HYDROCHLORIC ACID SALT FORM KRKA, D.D., NOVO MESTO (SI) 2008-04-10 WO disclosed
WO-2008040560-A1 PROCESS FOR THE PREPARATION OF MEMANTINE AND ITS HYDROCHLORIC ACID SALT FORM KRKA, D.D., NOVO MESTO (SI) 2008-04-10 WO disclosed
EP-1908748-A1 Process for the preparation of memantine and its hydrochloric acid salt form KRKA (SI) 2008-04-09 EP disclosed
EP-1908748-A1 Process for the preparation of memantine and its hydrochloric acid salt form KRKA (SI) 2008-04-09 EP disclosed