SCHEMBL2565231

SCHEMBL2565231

NC(=O)Oc1oc2c(Cl)cncc2c1Nc1ccc(I)cc1F

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 17/20 0.50
MAP2K2 P36507 3/20 0.43
IDO1 P14902 1/20 0.39
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2569333 0.85 MAP2K1 (0.57) MAP2K1MAP2K2IDO1
SCHEMBL2565784 0.83 MAP2K1 (0.58) MAP2K1MAP2K2
SCHEMBL2562768 0.82 MAP2K1 (0.55) MAP2K1MAP2K2IDO1CYP2C9CYP2C19
SCHEMBL2563462 0.81 MAP2K1 (0.54) MAP2K1MAP2K2IDO1CYP2C9CYP2C19
SCHEMBL2563469 0.81 MAP2K1 (0.54) MAP2K1MAP2K2IDO1CYP2C9CYP2C19
SCHEMBL2563464 0.80 MAP2K1 (0.54) MAP2K1MAP2K2IDO1
SCHEMBL2565295 0.79 MAP2K1 (0.57) MAP2K1MAP2K2IDO1
SCHEMBL12164526 0.78 MAP2K1 (0.72) MAP2K1MAP2K2CYP2C9CYP2C19KCNH2
SCHEMBL2568269 0.77 MAP2K1 (0.59) MAP2K1MAP2K2CYP2C9CYP2C19KCNH2
SCHEMBL2565371 0.75 MAP2K1 (0.74) MAP2K1MAP2K2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069354-B1 Aza-benzofuranyl compounds and methods of use GENENTECH INC (US) 2011-11-02 EP claimed