SCHEMBL2566165

SCHEMBL2566165

CCCS(=O)(=O)CCCSc1nc2cc[nH]c2c(=O)n1-c1ccc(OCC2CC2)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.38
TP53 P04637 6/20 0.35
KMT2A Q03164 3/20 0.35
LMNA P02545 3/20 0.34
GAA P10253 1/20 0.34
MEN1 O00255 2/20 0.34
BRD4 O60885 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 1/20 0.33
APLNR P35414 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
PDE2A O00408 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE11A Q9HCR9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2570283 0.92 TSHR (0.34) TSHRTP53KMT2ALMNAGAA
SCHEMBL2567318 0.91 TSHR (0.36) TSHRTP53KMT2ALMNAGAA
SCHEMBL2566162 0.89 TSHR (0.35) TSHRTP53KMT2ALMNAGAA
SCHEMBL2997987 0.86 TSHR (0.40) TSHRTP53KMT2ALMNAGAA
SCHEMBL2564410 0.85 TSHR (0.41) TSHRTP53KMT2ALMNAGAA
SCHEMBL2568131 0.85 TSHR (0.46) TSHRTP53KMT2ALMNAGAA
SCHEMBL2990546 0.84 TSHR (0.40) TSHRTP53KMT2ALMNAGAA
SCHEMBL2566036 0.83 TP53 (0.38) TSHRTP53KMT2ALMNAGAA
SCHEMBL2990464 0.83 TSHR (0.35) TSHRTP53KMT2ALMNAGAA
SCHEMBL2569802 0.83 TSHR (0.35) TSHRTP53KMT2ALMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2382218-A1 DELTA-5-DESATURASE INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2011-11-02 EP disclosed
WO-2010087467-A1 DELTA-5-DESATURASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-05 WO disclosed