SCHEMBL25692152

SCHEMBL25692152

CSN(C)c1ccccc1Nc1nc(Nc2ccc(C(=O)O)c(F)c2)ncc1C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.52
ROCK2 O75116 1/20 0.52
MAP4K4 O95819 1/20 0.52
PIM1 P11309 1/20 0.52
PRKACA P17612 1/20 0.52
CDK7 P50613 1/20 0.52
CDK9 P50750 1/20 0.52
HIPK2 Q9H2X6 1/20 0.52
IRAK4 Q9NWZ3 1/20 0.52
GSK3A P49840 1/20 0.51
GSK3B P49841 1/20 0.51
PTK2 Q05397 9/20 0.51
KDR P35968 2/20 0.49
JAK2 O60674 1/20 0.49
NTRK1 P04629 1/20 0.49
TYK2 P29597 1/20 0.49
JAK3 P52333 1/20 0.49
PTK2B Q14289 1/20 0.49
NTRK3 Q16288 1/20 0.49
NTRK2 Q16620 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25692158 0.88 PTK2 (0.63) CDC7ROCK2MAP4K4PIM1PRKACA
SCHEMBL25692191 0.87 GSK3A (0.69) CDC7ROCK2MAP4K4PIM1PRKACA
SCHEMBL25692320 0.83 AURKA (0.44) CDC7MAP4K4PIM1HIPK2IRAK4
SCHEMBL24752270 0.82 PTK2 (0.58) CDC7ROCK2MAP4K4PIM1PRKACA
SCHEMBL30001799 0.82 PTK2 (0.58) CDC7ROCK2MAP4K4PIM1PRKACA
SCHEMBL25692540 0.81 MAPK8 (0.64) CDC7ROCK2MAP4K4PIM1PRKACA
SCHEMBL25692215 0.78 PTK2 (0.58) PTK2KDRJAK2NTRK1TYK2
SCHEMBL25692119 0.78 PTK2 (0.54) CDC7ROCK2MAP4K4PIM1PRKACA
SCHEMBL25692237 0.77 MAPK3 (0.47) CDC7ROCK2MAP4K4PIM1PRKACA
SCHEMBL25692657 0.77 AURKA (0.54) CDC7ROCK2MAP4K4PIM1PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023121251-A1 EGFR AND HDAC DUAL INHIBITOR COMPOUNDS AND MEDICAL USE THEREOF 한국원자력의학원 2023-06-29 WO disclosed