SCHEMBL25698477

SCHEMBL25698477

CC(C)(C)OC(=O)NC[C@]1(CO)C[C@@H](N(Cc2ccccc2)Cc2ccccc2)C1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.45
CTSS P25774 4/20 0.43
CTSL P07711 3/20 0.43
CTSB P07858 3/20 0.43
IDO1 P14902 1/20 0.42
SYK P43405 1/20 0.41
NPFFR1 Q9GZQ6 1/20 0.40
NPFFR2 Q9Y5X5 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
SIGMAR1 Q99720 3/20 0.39
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
CTSK P43235 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25698474 1.00 AKT1 (0.45) AKT1CTSSCTSLCTSBIDO1
SCHEMBL25572358 0.83 AKT1 (0.44) AKT1CTSSCTSLCTSBIDO1
SCHEMBL25698468 0.83 AKT1 (0.44) AKT1CTSSCTSLCTSBIDO1
SCHEMBL25572361 0.83 AKT1 (0.44) AKT1CTSSCTSLCTSBIDO1
SCHEMBL13664871 0.78 AKT1 (0.52) AKT1CTSSCTSLCTSBIDO1
SCHEMBL6185852 0.74 NAMPT (0.44) IDO1SYKNPFFR1NPFFR2
SCHEMBL25568275 0.74 KDM4E (0.39) ALDH1A1KMT2A
SCHEMBL25568276 0.74 KDM4E (0.39) ALDH1A1KMT2A
SCHEMBL6863653 0.73 KDM1A (0.57) AKT1CTSSCTSLCTSBALDH1A1
SCHEMBL21071384 0.73 KDM1A (0.57) AKT1CTSSCTSLCTSBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091438-A1 CHROMANE AMIDINE MONOBACTAM ANTIBIOTICS MERCK SHARP & DOHME LLC (US) 2023-05-25 WO disclosed