SCHEMBL25699731

SCHEMBL25699731

CC1CN(c2ccc(C#N)c3ncccc23)CC(CN2CCN(c3ccnc(N4CCN(C)CC4)n3)CC2)O1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 13/20 0.46
TLR7 Q9NYK1 13/20 0.46
TLR8 Q9NR97 12/20 0.46
CCNT1 O60563 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CDK9 P50750 1/20 0.35
SORD Q00796 1/20 0.35
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
HRH1 P35367 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24120216 1.00 TLR9 (0.46) TLR9TLR7TLR8CCNT1CCNA2
SCHEMBL24120538 0.93 TLR9 (0.44) TLR9TLR7TLR8
SCHEMBL21815335 0.93 TLR9 (0.44) TLR9TLR7TLR8
SCHEMBL24120227 0.92 TLR9 (0.48) TLR9TLR7TLR8HRH1HRH3
SCHEMBL25700218 0.92 TLR9 (0.48) TLR9TLR7TLR8HRH1HRH3
SCHEMBL25417310 0.92 TLR9 (0.48) TLR9TLR7TLR8HRH1HRH3
SCHEMBL24120228 0.92 TLR9 (0.47) TLR9TLR7TLR8HRH1HRH3
SCHEMBL25699773 0.92 TLR9 (0.51) TLR9TLR7TLR8ALDH1A1HRH1
SCHEMBL24120542 0.92 TLR9 (0.51) TLR9TLR7TLR8ALDH1A1HRH1
SCHEMBL21815378 0.91 TLR9 (0.43) TLR9TLR7TLR8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3856737-B1 HETEROCYCLYL COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE HOFFMANN LA ROCHE (CH) 2023-05-17 EP disclosed