SCHEMBL257050

SCHEMBL257050

Cn1cc(-c2cc(C(=O)Nc3cccc(F)c3)c(OCc3ccccc3)cc2C(=O)N2CCOCC2)cn1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 9/20 0.51
MET P08581 3/20 0.50
CYP3A4 P08684 1/20 0.45
SLCO1B1 Q9Y6L6 1/20 0.45
SGMS2 Q8NHU3 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
AURKB Q96GD4 1/20 0.42
PTGER1 P34995 1/20 0.42
NMT2 O60551 1/20 0.41
NMT1 P30419 1/20 0.41
FSCN1 Q16658 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15204962 0.95 LRRK2 (0.55) LRRK2METSGMS2HTR2AHTR2C
SCHEMBL165714 0.89 LRRK2 (0.53) LRRK2METCYP3A4AURKB
SCHEMBL256246 0.89 LRRK2 (0.67) LRRK2METCYP3A4SLCO1B1SGMS2
SCHEMBL257185 0.87 LRRK2 (0.61) LRRK2CYP3A4SLCO1B1
SCHEMBL176196 0.87 LRRK2 (0.68) LRRK2METSGMS2
SCHEMBL165664 0.86 HSD17B10 (0.49) LRRK2CYP3A4SLCO1B1HSD17B10NMT2
SCHEMBL256499 0.85 CNR1 (0.47) LRRK2METCYP3A4AURKB
SCHEMBL176062 0.84 LRRK2 (0.54) LRRK2CYP3A4SLCO1B1
SCHEMBL175796 0.84 LRRK2 (0.68) LRRK2METSGMS2
SCHEMBL256260 0.84 LRRK2 (0.46) LRRK2CYP3A4SLCO1B1HSD17B10NMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028629-A1 2 - (BENZYLOXY) BENZAMIDES AS LRRK2 KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed