Formestane

Formestane

SCHEMBL25717

C[C@]12CCC(=O)C(O)=C1CC[C@@H]1[C@@H]2CC[C@]2(C)C(=O)CC[C@@H]12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 1.00
TSHR P16473 1/20 1.00
THPO P40225 1/20 1.00
HIF1A Q16665 1/20 1.00
TDP1 Q9NUW8 1/20 1.00
CYP19A1 P11511 17/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formestane SCHEMBL3230067 1.00 CYP3A4 (1.00) CYP3A4TSHRTHPOHIF1ATDP1
Formestane SCHEMBL14291425 1.00 CYP3A4 (1.00) CYP3A4TSHRTHPOHIF1ATDP1
Formestane SCHEMBL22891821 1.00 CYP3A4 (1.00) CYP3A4TSHRTHPOHIF1ATDP1
Formestane SCHEMBL13838287 1.00 CYP3A4 (1.00) CYP3A4TSHRTHPOHIF1ATDP1
Formestane SCHEMBL13795108 1.00 CYP3A4 (1.00) CYP3A4TSHRTHPOHIF1ATDP1
Formestane SCHEMBL947479 1.00 CYP3A4 (1.00) CYP3A4TSHRTHPOHIF1ATDP1
SCHEMBL10942772 0.90 CYP3A4 (0.81) CYP3A4TSHRTHPOHIF1ATDP1
SCHEMBL10942767 0.90 CYP3A4 (0.81) CYP3A4TSHRTHPOHIF1ATDP1
Formestane SCHEMBL27563770 0.88 CYP19A1 (0.77) CYP3A4TSHRTHPOHIF1ATDP1
SCHEMBL7739598 0.87 CYP3A4 (0.77) CYP3A4TSHRTHPOHIF1ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 31956 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
EP-3645742-B1 ANTI-ROR1 ANTIBODIES AND METHODS OF MAKING AND USING THEREOF SYSTIMMUNE INC (US) 2026-04-29 EP claimed
US-20260103461-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF OLEMA PHARMACEUTICALS INC (US) 2026-04-16 US claimed
EP-4712980-A1 TREATMENT OF BREAST TISSUE Havah Therapeutics Pty Ltd (AU) 2026-03-25 EP claimed
EP-4680251-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER Thomas Jefferson University (US) 2026-01-21 EP claimed
EP-4680284-A2 BIODEGRADABLE DENDRITIC PARTICLES FOR SUSTAINED DRUG RELEASE THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2026-01-21 EP claimed
EP-4680226-A2 ACYLSULFONAMIDE KAT6A INHIBITORS Olema Pharmaceuticals, Inc. (US) 2026-01-21 EP claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
EP-4674894-A2 COPOLYMERS OF N-VINYLPYRROLIDONE WITH FUNCTIONALIZED MALEIC ACID MOIETIES Hemoteq AG (DE) 2026-01-07 EP claimed
EP-4663688-A2 CROSSLINKERS Hemoteq AG (DE) 2025-12-17 EP claimed
US-5002940-A Steroids, Phospholipids, Polyoxyethylene Glycol CIBA-GEIGY CORPORATION (US) 1991-03-26 US claimed
WO-1991000731-A1 COMBINATION THERAPY FOR PROPHYLAXIS AND/OR TREATMENT OF BENIGN PROSTATIC HYPERPLASIA ENDORECHERCHE INC. (CA) 1991-01-24 WO claimed
WO-1990010462-A1 COMBINATION THERAPY FOR TREATMENT OF ESTROGEN SENSITIVE DISEASES ENDORECHERCHE INC. (CA) 1990-09-20 WO claimed
EP-0181287-B1 DRY SUBSTANCES AND STABLE SUSPENSIONS CIBA-GEIGY AG (CH) 1990-03-21 EP claimed
US-4895715-A Method of treating gynecomastia SCHERING CORPORATION (US) 1990-01-23 US claimed
US-4749567-A WITH 6-HYDROXYANDROST-4-ENE-3, 17-DIONE, LINKED THROUGH THE HYDROXY THE DIRECTOR GENERAL OF THE MINISTRY OF AGRICULTURE AND FISHERIES (NZ) 1988-06-07 US claimed
US-4598072-A Combinations of an aromatase-inhibitor and an antiandrogen for prophylaxis and/or treatment of benign prostatic hyperplasia SCHERING AKTIENGESELLSCHAFT (DE) 1986-07-01 US claimed
US-4596797-A Urogenital disorders SCHERING AKTIENGESELLSCHAFT (DE) 1986-06-24 US claimed
EP-0181287-A2 Dry substances and stable suspensions CIBA-GEIGY AG (CH) 1986-05-14 EP claimed
US-4500523-A Suppression of premature labor by use of aromatase inhibitors CORNELL RESEARCH FOUNDATION, INC. (US) 1985-02-19 US claimed