SCHEMBL25738522

SCHEMBL25738522

O=c1cc(F)c2ccc(Br)cc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.47
TNKS2 Q9H2K2 3/20 0.42
TNKS O95271 1/20 0.42
CDK5 Q00535 3/20 0.41
CDK9 P50750 2/20 0.41
CAMK2A Q9UQM7 2/20 0.41
CCNB2 O95067 2/20 0.41
CDK1 P06493 2/20 0.41
CCNB1 P14635 2/20 0.41
CDK5R1 Q15078 2/20 0.41
CCNB3 Q8WWL7 2/20 0.41
CCNT1 O60563 1/20 0.41
CCNE2 O96020 1/20 0.41
CDK4 P11802 1/20 0.41
EIF2AK2 P19525 1/20 0.41
CCNA2 P20248 1/20 0.41
CCND1 P24385 1/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
CAMK2B Q13554 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL706591 0.85 PDE3B (0.43) METAP2TNKS2TNKSCDK5CDK9
SCHEMBL2798886 0.79 KDM4E (0.62) METAP2TNKS2TNKSHPGDTP53
SCHEMBL29892996 0.79 KDM4E (0.62) METAP2TNKS2TNKSHPGDTP53
SCHEMBL29171685 0.78 TP53 (0.47) METAP2TNKS2CDK5CDK9CAMK2A
SCHEMBL29831055 0.78 KDM4E (0.59) METAP2CDK5CDK9CAMK2ACCNB2
SCHEMBL30759515 0.78 TP53 (0.47) METAP2TNKS2CDK5CDK9CAMK2A
SCHEMBL14796728 0.78 KDM4E (0.59) METAP2CDK5CDK9CAMK2ACCNB2
SCHEMBL9393238 0.75 KDM4E (0.47) METAP2CDK5CDK9CAMK2ACCNB2
SCHEMBL6827495 0.75 CYP1A2 (0.62) TNKS2TNKSHPGDSMN1; SMN2KDM4E
SCHEMBL5469793 0.74 HPGD (0.67) METAP2TNKS2TNKSCDK5CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023109521-A1 PARP INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE THEREOF 凯复(苏州)生物医药有限公司 2023-06-22 WO disclosed