SCHEMBL25756887

SCHEMBL25756887

COC(=O)CCCCCCCc1ccc(NC(=O)c2ccc(C)c(C#Cc3cnc4cc(C)cnn34)c2)cc1C(F)(F)F

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 18/20 0.59
RET P07949 3/20 0.59
ABL2 P42684 2/20 0.59
GAK O14976 1/20 0.59
MLNR O43193 1/20 0.59
RIPK2 O43353 1/20 0.59
JAK2 O60674 1/20 0.59
NR1I2 O75469 1/20 0.59
ABCB11 O95342 1/20 0.59
MAP4K4 O95819 1/20 0.59
EGFR P00533 1/20 0.59
NR3C1 P04150 1/20 0.59
ERBB2 P04626 1/20 0.59
NTRK1 P04629 1/20 0.59
LCK P06239 1/20 0.59
FYN P06241 1/20 0.59
PGR P06401 1/20 0.59
CSF1R P07333 1/20 0.59
YES1 P07947 1/20 0.59
LYN P07948 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25756898 0.91 ABL1 (0.72) ABL1RETABL2GAKMLNR
SCHEMBL25756905 0.85 ABL1 (0.72) ABL1RETABL2GAKMLNR
SCHEMBL25756904 0.84 ABL1 (0.71) ABL1RETABL2GAKMLNR
SCHEMBL25757199 0.84 ABL1 (0.54) ABL1RETABL2GAKMLNR
SCHEMBL25638630 0.83 ABL1 (0.83) ABL1RETABL2GAKMLNR
SCHEMBL25422487 0.83 ABL1 (0.70) ABL1RETABL2GAKMLNR
SCHEMBL25243927 0.83 ABL1 (0.70) ABL1RETABL2GAKMLNR
SCHEMBL18298082 0.78 ABL1 (0.80) ABL1RETABL2GAKMLNR
SCHEMBL31697365 0.78 ABL1 (0.80) ABL1RETABL2GAKMLNR
SCHEMBL20811900 0.77 ABL1 (0.82) ABL1RETABL2GAKMLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023119334-A1 ANTI-CANCER COMPOUND BY COMBINING PONATINIB MOLECULE WITH HDAC INHIBITOR MOLECULE USING A VARIABLE LENGTH LINKER AMRITA VISHWA VIDYAPEETHAM (IN) 2023-06-29 WO disclosed