SCHEMBL257597

SCHEMBL257597

CC(C)(C)OC(=O)Nc1ccc2c(c1)CCCN2

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.50
GAA P10253 1/20 0.48
KDM4E B2RXH2 1/20 0.48
MAPT P10636 1/20 0.48
TRPV1 Q8NER1 1/20 0.46
PIR O00625 1/20 0.44
GSK3B P49841 1/20 0.44
HSF1 Q00613 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
NR1I3 Q14994 5/20 0.42
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA9 Q16790 2/20 0.42
CA2 P00918 1/20 0.41
CYP17A1 P05093 2/20 0.41
EPHX2 P34913 1/20 0.41
DRD2 P14416 1/20 0.39
LIPE Q05469 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22160852 0.92 CA12 (0.43) PLAUNR1I3CA12CA1CA9
SCHEMBL17813292 0.84 BAZ2B (0.45) TRPV1GSK3BNPC1RAB9ANR1I3
SCHEMBL2229710 0.82 MEN1 (0.49) TRPV1NPC1RAB9ANR1I3CA12
SCHEMBL5053574 0.81 PLAU (0.56) PLAUGAAKDM4EMAPTTRPV1
SCHEMBL30464664 0.81 PLAU (0.56) PLAUGAAKDM4EMAPTTRPV1
SCHEMBL13783463 0.81 NPC1 (0.60) GAAMAPTNPC1RAB9A
SCHEMBL31169451 0.81 NPC1 (0.57) GAAMAPTTRPV1NPC1RAB9A
SCHEMBL3545975 0.80 PLAU (0.50) PLAUGAAKDM4EMAPTTRPV1
SCHEMBL691153 0.79 MAPT (0.60) PLAUGAAKDM4EMAPTTRPV1
SCHEMBL23520112 0.79 PPID (0.50) GAAKDM4EMAPTEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012029763-A1 DIAMINE, POLYIMIDE PRECURSOR, POLYIMIDE, LIQUID-CRYSTAL ALIGNMENT MATERIAL, LIQUID-CRYSTAL ALIGNMENT FILM, AND LIQUID-CRYSTAL DISPLAY ELEMENT 日産化学工業株式会社 (JP) 2012-03-08 WO disclosed
US-6930104-B2 Heterocyclic derivatives TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-16 US disclosed
US-20040157850-A1 Novel heterocyclic derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-08-12 US disclosed
EP-1382598-A1 NOVEL HETEROCYCLIC DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2004-01-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040157850-A1 Novel heterocyclic derivatives APP, BACE1, PSEN1 PLAU 2069/4885GAA 1685/4885KDM4E 4527/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.