SCHEMBL25796181

SCHEMBL25796181

CS(=O)(=O)Nc1cc(N2CCc3cc(N4CCOCC4)ccc3C2=O)ccc1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.38
KIF11 P52732 1/20 0.38
CDK1 P06493 1/20 0.38
CDK2 P24941 1/20 0.38
ADRB3 P13945 5/20 0.38
ADRB1 P08588 4/20 0.38
ADRB2 P07550 3/20 0.37
BTK Q06187 2/20 0.37
ACLY P53396 1/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37
MAPK14 Q16539 1/20 0.37
EPHX2 P34913 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
MCL1 Q07820 1/20 0.36
MAPT P10636 2/20 0.35
PKM P14618 1/20 0.35
PSMD14 O00487 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25796194 0.85 BTK (0.42) ADRB3ADRB1ADRB2BTKPIK3CA
SCHEMBL25795912 0.84 BTK (0.38) PRKDCBTKMCL1MAPTEGFR
SCHEMBL30549624 0.84 BTK (0.38) PRKDCBTKMCL1MAPTEGFR
SCHEMBL30549742 0.83 TRPV1 (0.41) MAPT
SCHEMBL25795808 0.83 KCNH2 (0.44) BTKMAPK14MAPT
SCHEMBL25796278 0.82 BTK (0.38) ADRB3ADRB1ADRB2BTKLRRK2
SCHEMBL25795650 0.81 HRH3 (0.41) ADRB3ACLYMCL1
SCHEMBL25797450 0.81 AOC3 (0.43) ADRB3MCL1PKM
SCHEMBL30550018 0.81 HRH3 (0.41) ADRB3ACLYMCL1
SCHEMBL30549782 0.81 BACE1 (0.38) ADRB3PIK3CDPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023109912-A1 3, 4-DIHYDROISOQUINOLIN-1 (2H) -ONES DERIVATIVES AS STING ANTAGONISTS AND THE USE THEREOF BEIGENE, LTD. (KY) 2023-06-22 WO disclosed