SCHEMBL25809239

SCHEMBL25809239

CC(C)(C)OC(=O)NC[C@H](S)CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 1/20 0.39
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.36
PCSK9 Q8NBP7 1/20 0.36
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
SYK P43405 1/20 0.34
CYP3A4 P08684 2/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25809213 1.00 SERPINE1 (0.39) SERPINE1MEN1GAAKMT2ATDP1
SCHEMBL20297742 1.00 SERPINE1 (0.39) SERPINE1MEN1GAAKMT2ATDP1
SCHEMBL25400155 0.84 SERPINE1 (0.40) SERPINE1MEN1GAAKMT2ATDP1
SCHEMBL30015389 0.84 SERPINE1 (0.40) SERPINE1MEN1GAAKMT2ATDP1
SCHEMBL6854629 0.84 SERPINE1 (0.40) SERPINE1MEN1GAAKMT2ATDP1
SCHEMBL18340909 0.83 CYP2D6 (0.37)
SCHEMBL26314494 0.82 SERPINE1 (0.39) SERPINE1MEN1GAAKMT2ATDP1
SCHEMBL18990457 0.81 SERPINE1 (0.43) SERPINE1MEN1GAAKMT2ATDP1
SCHEMBL20298107 0.81 SERPINE1 (0.43) SERPINE1MEN1GAAKMT2ATDP1
SCHEMBL17860151 0.81 TDP1 (0.39) SERPINE1MEN1GAAKMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3313828-B1 METALLO-BETA-LACTAMASE INHIBITORS MERCK SHARP & DOHME LLC (US) 2023-07-12 EP disclosed
EP-3313828-B1 METALLO-BETA-LACTAMASE INHIBITORS MERCK SHARP & DOHME LLC (US) 2023-07-12 EP disclosed