SCHEMBL2582540

SCHEMBL2582540

Cc1ccc(C(=O)NC2(c3ncccn3)CC2)cc1-c1ccc2oc(-c3ccc(F)cc3)c(C(=O)N(C)F)c2c1

nearest known ligand 0.83

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.83
CYP3A4 P08684 5/20 0.83
KCNH2 Q12809 3/20 0.83
NR1I2 O75469 1/20 0.70
MAPK14 Q16539 1/20 0.37
ABL1 P00519 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2142804 0.91 CYP2C8 (1.00) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL2141750 0.84 CYP2C8 (0.88) CYP2C8CYP3A4KCNH2NR1I2ABL1
SCHEMBL2143177 0.84 CYP2C8 (0.87) CYP2C8CYP3A4KCNH2NR1I2ABL1
SCHEMBL2141388 0.83 CYP2C8 (0.86) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL2141972 0.82 CYP2C8 (1.00) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL2141169 0.81 CYP2C8 (0.83) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL2143486 0.81 CYP2C8 (0.83) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL12293914 0.81 CYP2C8 (0.70) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL9912760 0.81 CYP2C8 (0.82) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL12293750 0.81 CYP2C8 (0.85) CYP2C8CYP3A4KCNH2NR1I2ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048887-B2 Compounds for the treatment of hepatitis C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-11-01 US claimed