SCHEMBL25839035

SCHEMBL25839035

Cn1c(=O)[nH]c2ncc(I)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 10/20 0.47
PDE3A Q14432 10/20 0.47
PDE2A O00408 8/20 0.47
ADORA2A P29274 1/20 0.44
ADORA2B P29275 1/20 0.44
LMNA P02545 3/20 0.40
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
PABPC1 P11940 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
APAF1 O14727 1/20 0.38
CASP6 P55212 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11922289 0.81 PDE3B (0.54) PDE3BPDE3APDE2AADORA2AADORA2B
SCHEMBL15221682 0.79 PDE3B (0.47) PDE3BPDE3APDE2AADORA2AADORA2B
SCHEMBL1585845 0.79 HSD17B10 (0.53) PDE3BPDE3APDE2AADORA2AADORA2B
SCHEMBL29705394 0.79 HSD17B10 (0.53) PDE3BPDE3APDE2AADORA2AADORA2B
SCHEMBL17813540 0.77 PDE3B (0.45) PDE3BPDE3APDE2AADORA2AADORA2B
SCHEMBL28523335 0.76 PDE3B (0.44) PDE3BPDE3APDE2AADORA2AADORA2B
SCHEMBL2207001 0.74 GRIN1 (0.60) PDE3BPDE3APDE2AADORA2AADORA2B
SCHEMBL11238693 0.73 PDE3B (0.59) PDE3BPDE3APDE2A
SCHEMBL12830376 0.72 PDE3B (0.47) PDE3BPDE3APDE2AADORA2AADORA2B
SCHEMBL28522267 0.72 PDE3B (0.41) PDE3BPDE3APDE2AADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed