SCHEMBL25848970

SCHEMBL25848970

Cc1cc(C(F)(F)F)ccc1CNC(=O)c1ccc(S(C)(=O)=O)s1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 5/20 0.44
NR1H4 Q96RI1 3/20 0.44
DDR1 Q08345 4/20 0.43
ELANE P08246 2/20 0.43
HDAC1 Q13547 4/20 0.41
HDAC6 Q9UBN7 4/20 0.41
MCL1 Q07820 5/20 0.41
HDAC4 P56524 3/20 0.40
HDAC3 O15379 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25848857 0.92 EPHX2 (0.45) EPHX2NR1H4DDR1ELANEHDAC1
SCHEMBL25848961 0.90 TRPV1 (0.48) EPHX2NR1H4DDR1ELANEHDAC1
SCHEMBL24196659 0.89 MCL1 (0.42) EPHX2NR1H4DDR1ELANEHDAC1
SCHEMBL25848940 0.83 LSS (0.50) EPHX2NR1H4HDAC1HDAC6HDAC4
SCHEMBL30393777 0.83 ELANE (0.43) EPHX2ELANEHDAC1HDAC6HDAC4
SCHEMBL24196156 0.83 ELANE (0.43) EPHX2ELANEHDAC1HDAC6HDAC4
SCHEMBL25304798 0.83 NAMPT (0.41) EPHX2DDR1ELANEHDAC1HDAC6
SCHEMBL25848848 0.82 EPHX2 (0.48) EPHX2NR1H4DDR1HDAC1HDAC6
SCHEMBL25848869 0.82 ELANE (0.39) EPHX2ELANEHDAC1HDAC6HDAC4
SCHEMBL25848856 0.81 EPHX2 (0.43) EPHX2NR1H4DDR1HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230219921-A1 KCNT1 INHIBITORS AND METHODS OF USE PRAXIS PRECISION MEDICINES, INC. 2023-07-13 US disclosed
US-20230219921-A1 KCNT1 INHIBITORS AND METHODS OF USE PRAXIS PRECISION MEDICINES, INC. 2023-07-13 US disclosed
EP-4175624-A1 KCNT1 INHIBITORS AND METHODS OF USE Praxis Precision Medicines, Inc. (US) 2023-05-10 EP disclosed
CN-116075297-A KCNT1 inhibitors and methods of use 普拉西斯精密医药公司 2023-05-05 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230219921-A1 KCNT1 INHIBITORS AND METHODS OF USE KCNT1, KCNT2, KCNQ2 EPHX2 2590/4885NR1H4 3085/4885DDR1 3524/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.