SCHEMBL2586779

SCHEMBL2586779

CN(C(=O)C(O)c1ccc(-c2noc(-c3cnn(-c4ccccc4)c3C(F)(F)F)n2)cc1)C1CCCCC1

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.66
S1PR3 Q99500 9/20 0.39
S1PR4 O95977 2/20 0.39
S1PR5 Q9H228 2/20 0.39
CYP2C8 P10632 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2579544 0.84 S1PR1 (0.77) S1PR1S1PR3
SCHEMBL27921152 0.84 S1PR1 (0.77) S1PR1S1PR3
SCHEMBL2576403 0.83 S1PR1 (0.82) S1PR1
SCHEMBL12289131 0.81 S1PR1 (0.81) S1PR1
SCHEMBL12288618 0.80 S1PR1 (0.77) S1PR1S1PR3
SCHEMBL14696697 0.80 S1PR1 (0.75) S1PR1S1PR3S1PR4S1PR5
SCHEMBL14696699 0.80 S1PR1 (0.75) S1PR1S1PR3S1PR4S1PR5
SCHEMBL14696698 0.80 S1PR1 (0.75) S1PR1S1PR3S1PR4S1PR5
SCHEMBL2577490 0.80 S1PR1 (1.00) S1PR1
SCHEMBL14696212 0.80 S1PR1 (0.75) S1PR1S1PR3S1PR4S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2560969-A1 4 - (5 - ISOXAZOLYL OR 5 - PYRRAZOLYL -1,2,4- OXADIAZOL - 3 - YL) -MANDELIC ACID AMIDES AS SPHINGOSIN- 1 - PHOSPHATE 1 RRECEPTOR AGONISTS Bristol-Myers Squibb Company (US) 2013-02-27 EP disclosed
WO-2011133734-A1 4 - (5 - ISOXAZOLYL OR 5 - PYRRAZOLYL -1,2,4- OXADIAZOL - 3 - YL) -MANDELIC ACID AMIDES AS SPHINGOSIN- 1 - PHOSPHATE 1 RRECEPTOR AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-10-27 WO disclosed