SCHEMBL25872018

SCHEMBL25872018

COC(=O)CCCN1Cc2cc(N)c(Br)cc2C1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
HDAC6 Q9UBN7 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
TNF P01375 2/20 0.39
KAT2B Q92831 3/20 0.38
AOC3 Q16853 2/20 0.36
PARP1 P09874 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
REN P00797 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2181132 0.81 KDM4E (0.48) KDM4EALDH1A1HPGDHDAC6HDAC3
SCHEMBL2178732 0.81 HDAC6 (0.46) KDM4EALDH1A1HPGDHDAC6HDAC3
SCHEMBL16850283 0.77 KDM4E (0.49) KDM4EALDH1A1HPGDHDAC6HDAC3
SCHEMBL16850273 0.74 KDM4E (0.54) KDM4EALDH1A1HPGDHDAC6HDAC3
SCHEMBL18766026 0.73 KDM4E (0.46) KDM4EALDH1A1HPGDHDAC6HDAC4
SCHEMBL1500259 0.73 AOC3 (0.47) KDM4EALDH1A1HPGDHDAC6AOC3
SCHEMBL25872020 0.72 IRAK4 (0.56)
SCHEMBL449230 0.70 HDAC6 (0.42) KDM4EALDH1A1HPGDHDAC6HDAC3
SCHEMBL8046017 0.69 AOC3 (0.47) KDM4EALDH1A1HPGDHDAC6KAT2B
SCHEMBL16850282 0.69 KDM4E (0.47) KDM4EALDH1A1HPGDTNFKAT2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023116920-A1 PENTA- FUSED HEXA-HETEROCYCLIC COMPOUND, PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE 杭州多域生物技术有限公司 2023-06-29 WO disclosed