SCHEMBL25878648

SCHEMBL25878648

C[C@H](CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C1CC2(C1)CN(C)C2

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 16/20 0.62
CRBN Q96SW2 16/20 0.62
IKZF3 Q9UKT9 2/20 0.51
TNF P01375 1/20 0.51
IL1B P01584 1/20 0.51
TBXA2R P21731 1/20 0.51
IKZF1 Q13422 1/20 0.51
STAT3 P40763 2/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC2 Q92769 1/20 0.49
ALDH1A1 P00352 1/20 0.47
CHRM2 P08172 1/20 0.47
OPRM1 P35372 1/20 0.47
CYP1A2 P05177 1/20 0.47
TSHR P16473 1/20 0.47
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22836351 0.91 DDB1 (0.64) DDB1CRBNIKZF3TNFIL1B
SCHEMBL22835996 0.91 DDB1 (0.64) DDB1CRBNIKZF3TNFIL1B
SCHEMBL22836002 0.91 DDB1 (0.64) DDB1CRBNIKZF3TNFIL1B
SCHEMBL25894759 0.89 CRBN (0.65) DDB1CRBNIKZF3TNFIL1B
SCHEMBL22836599 0.86 DDB1 (0.62) DDB1CRBNSTAT3HDAC1HDAC2
SCHEMBL22835405 0.86 DDB1 (0.62) DDB1CRBNSTAT3HDAC1HDAC2
SCHEMBL22835408 0.86 DDB1 (0.62) DDB1CRBNSTAT3HDAC1HDAC2
SCHEMBL29502275 0.86 DDB1 (0.62) DDB1CRBNSTAT3HDAC1HDAC2
SCHEMBL23568512 0.86 DDB1 (0.66) DDB1CRBNIKZF3TNFIL1B
SCHEMBL22849504 0.86 DDB1 (0.66) DDB1CRBNIKZF3TNFIL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11707457-B2 IRAK degraders and uses thereof KYMERA THERAPEUTICS, INC. (US) 2023-07-25 US disclosed
US-11707457-B2 IRAK degraders and uses thereof KYMERA THERAPEUTICS, INC. (US) 2023-07-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11707457-B2 IRAK degraders and uses thereof IRAK2, IRAK3, IRAK1 DDB1 1267/4885CRBN 187/4885IKZF3 135/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.