SCHEMBL25901263

SCHEMBL25901263

CCC[C@H](C(N)=O)[C@@H](CCC(F)(F)F)C(=O)N[C@H]1N=C(c2ccccc2)c2ccccc2N(C)C1=O

nearest known ligand 0.88

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOTCH1 P46531 19/20 0.88
NOTCH3 Q9UM47 17/20 0.88
NOTCH2 Q04721 1/20 0.79
NOTCH4 Q99466 1/20 0.79
RBPJ Q06330 2/20 0.79
PSEN1 P49768 1/20 0.79
PSEN2 P49810 1/20 0.79
APH1B Q8WW43 1/20 0.79
NCSTN Q92542 1/20 0.79
APH1A Q96BI3 1/20 0.79
PSENEN Q9NZ42 1/20 0.79
CCKBR P32239 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Osugacestat SCHEMBL12543868 0.97 NOTCH1 (0.84) NOTCH1NOTCH3NOTCH2NOTCH4RBPJ
Osugacestat SCHEMBL21577519 0.97 NOTCH1 (0.84) NOTCH1NOTCH3NOTCH2NOTCH4RBPJ
Osugacestat SCHEMBL18288911 0.97 NOTCH1 (0.84) NOTCH1NOTCH3NOTCH2NOTCH4RBPJ
Osugacestat SCHEMBL17420836 0.97 NOTCH1 (0.84) NOTCH1NOTCH3NOTCH2NOTCH4RBPJ
Osugacestat SCHEMBL15622455 0.97 NOTCH1 (0.84) NOTCH1NOTCH3NOTCH2NOTCH4RBPJ
Osugacestat SCHEMBL12543867 0.97 NOTCH1 (0.84) NOTCH1NOTCH3NOTCH2NOTCH4RBPJ
Osugacestat SCHEMBL29412689 0.97 NOTCH1 (0.84) NOTCH1NOTCH3NOTCH2NOTCH4RBPJ
SCHEMBL12690166 0.94 NOTCH1 (0.83) NOTCH1NOTCH3NOTCH2NOTCH4RBPJ
SCHEMBL22970147 0.94 NOTCH1 (0.80) NOTCH1NOTCH3NOTCH2NOTCH4RBPJ
SCHEMBL22660068 0.92 NOTCH1 (0.83) NOTCH1NOTCH3NOTCH2NOTCH4RBPJ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11697798-B2 Enhanced differentiation and maturation of pluripotent stem cell-derived myogenic cells REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2023-07-11 US disclosed