SCHEMBL25907310

SCHEMBL25907310

Cc1cc(C2(C=O)COC2)ncc1NC(=O)c1cccc(C#N)c1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.46
BRAF P15056 2/20 0.43
RORC P51449 10/20 0.42
CNR1 P21554 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TP53 P04637 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29631546 0.79 IDO1 (0.60) GRM5BRAFCNR1NPC1RAB9A
SCHEMBL20898564 0.79 IDO1 (0.60) GRM5BRAFCNR1NPC1RAB9A
SCHEMBL29631509 0.69 IDO1 (0.75) GRM5BRAFMEN1KMT2ANPC1
SCHEMBL20899512 0.69 IDO1 (0.75) GRM5BRAFMEN1KMT2ANPC1
SCHEMBL20898568 0.65 IDO1 (0.80) BRAFNPC1RAB9ASMN1; SMN2TP53
SCHEMBL19087022 0.64 GRM5 (0.67) GRM5BRAFMEN1KMT2A
SCHEMBL6541906 0.64 RXFP1 (0.56) GRM5MEN1KMT2ANPC1RAB9A
SCHEMBL9588685 0.64 GRM5 (0.69) GRM5BRAF
SCHEMBL30798963 0.64 F2 (0.55) GRM5BRAFMEN1KMT2ASMN1; SMN2
SCHEMBL27383419 0.64 NPC1 (0.63) GRM5BRAFCNR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3694506-B1 NOVEL SUBSTITUTED PHENYLOXETANE AND PHENYLTETRAHYDROFURAN COMPOUNDS AS INDOLEAMINE 2,3-DIOXYGENASE (IDO) INHIBITORS MERCK SHARP & DOHME LLC (US) 2023-08-02 EP disclosed