SCHEMBL25925335

SCHEMBL25925335

COc1ccc(C(C)NN=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.54
CA2 P00918 2/20 0.54
ACHE P22303 1/20 0.54
ACP3 P15309 2/20 0.48
ACACB O00763 1/20 0.47
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
CA12 O43570 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
PKM P14618 1/20 0.42
KDM1A O60341 1/20 0.42
CNR2 P34972 5/20 0.41
CNR1 P21554 2/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
DRD4 P21917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28660520 0.81 CA1 (0.58) CA1CA2ACHEACP3ACACB
SCHEMBL12870269 0.78 CA1 (0.55) CA1CA2ACHEACP3ACACB
SCHEMBL13741075 0.78 CA1 (0.55) CA1CA2ACHEACP3ACACB
SCHEMBL278257 0.78 CA1 (0.55) CA1CA2ACHEACP3ACACB
SCHEMBL24105692 0.75 CA1 (0.56) CA1CA2ACHEACP3ACACB
SCHEMBL8239398 0.75 CA1 (0.56) CA1CA2ACHEACP3ACACB
SCHEMBL13462356 0.75 CA1 (0.56) CA1CA2ACHEACP3ACACB
SCHEMBL327954 0.75 CA1 (0.56) CA1CA2ACHEACP3ACACB
SCHEMBL11846483 0.75 ACP3 (0.47) ACP3ALDH1A1MEN1KMT2ADRD3
SCHEMBL19286211 0.75 CA1 (0.56) CA1CA2ACHEACP3ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4219502-A1 IMIDAZO[1,5-A]PYRAZINE DERIVATIVES AS PI3KDELTA INHIBITORS BeiGene, Ltd. (KY) 2023-08-02 EP disclosed