SCHEMBL2593701

SCHEMBL2593701

O=C(Nc1cccc(C23CC2COCC(=S)N3)c1)c1ncc(C(F)(F)F)cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.56
BACE2 Q9Y5Z0 6/20 0.44
ALDH1A1 P00352 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703053 0.87 BACE1 (0.56) BACE1BACE2
SCHEMBL2594835 0.81 BACE1 (0.51) BACE1
SCHEMBL7704675 0.81 BACE1 (0.51) BACE1
SCHEMBL7710580 0.80 BACE1 (0.46) BACE1BACE2
SCHEMBL2594187 0.80 BACE1 (0.46) BACE1BACE2
SCHEMBL2591429 0.80 BACE1 (0.70) BACE1BACE2
SCHEMBL2595074 0.80 BACE1 (0.70) BACE1BACE2
SCHEMBL15929894 0.73 HTT (0.58) BACE1ALDH1A1RAB9A
SCHEMBL362119 0.72 BACE1 (1.00) BACE1
SCHEMBL361903 0.71 BACE1 (1.00) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138293-A1 2,5,6,7-TETRAHYDRO-[1,4]OXAZEPIN-3-YLAMINE OR 2,3,6,7-TETRAHYDRO-[1,4]OXAZEPIN-5-YLAMINE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2011-11-10 WO disclosed