SCHEMBL2596686

SCHEMBL2596686

CCCc1cc2cc(-n3c(S)nnc3-c3cc(C(C)C)c(O)cc3O)ccc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 20/20 0.44
HSP90AB1 P08238 20/20 0.44
HSP90B1 P14625 1/20 0.40
TRAP1 Q12931 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3915279 0.92 HSP90AA1 (0.45) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL15940182 0.86 HSP90AA1 (0.48) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL421210 0.80 HSP90AA1 (0.48) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL8931378 0.78 HSP90AB1 (0.46) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL421114 0.76 HSP90AA1 (0.58) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL789420 0.76 HSP90AA1 (0.49) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL421216 0.76 HSP90AA1 (0.57) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL3094973 0.75 HSP90AA1 (0.45) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL2596684 0.75 HSP90AA1 (0.45) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL4740722 0.74 HSP90AA1 (0.56) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011146801-A1 FORMULATION AND DOSING OF HSP90 INHIBITORY COMPOUNDS SYNTA PHARMACEUTICALS CORP. (US) 2011-11-24 WO claimed