SCHEMBL2599462

SCHEMBL2599462

O=c1c2c(Cl)cccc2cc(CCNc2ncnc3c2ncn3[C@@H]2CCCCO2)n1-c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
CYP1A2 P05177 2/20 0.49
HPGD P15428 1/20 0.49
TSHR P16473 2/20 0.42
YTHDC1 Q96MU7 1/20 0.40
CYP2C19 P33261 1/20 0.39
PIK3CD O00329 3/20 0.37
PIK3CG P48736 2/20 0.37
ABCB11 O95342 1/20 0.37
TBXA2R P21731 1/20 0.37
PIK3R1 P27986 1/20 0.37
HTR2A P28223 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PDE3A Q14432 1/20 0.37
NFKB1 P19838 2/20 0.36
TP53 P04637 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16670934 0.87 NPC1 (0.53) NPC1RAB9ASMN1; SMN2CYP1A2HPGD
SCHEMBL16670935 0.87 NPC1 (0.53) NPC1RAB9ASMN1; SMN2CYP1A2HPGD
SCHEMBL2599461 0.86 NPC1 (0.48) NPC1RAB9ASMN1; SMN2CYP1A2HPGD
SCHEMBL936036 0.84 NPC1 (0.52) NPC1RAB9ASMN1; SMN2CYP1A2HPGD
SCHEMBL153714 0.83 PIK3CD (0.54) NPC1RAB9ASMN1; SMN2CYP1A2HPGD
SCHEMBL19656225 0.83 PIK3CD (0.54) NPC1RAB9ASMN1; SMN2CYP1A2HPGD
SCHEMBL153713 0.83 PIK3CD (0.54) NPC1RAB9ASMN1; SMN2CYP1A2HPGD
SCHEMBL31628325 0.83 PIK3CD (0.54) NPC1RAB9ASMN1; SMN2CYP1A2HPGD
SCHEMBL936140 0.80 NPC1 (0.51) NPC1RAB9ASMN1; SMN2CYP1A2HPGD
SCHEMBL179634 0.78 PIK3CD (0.55) NPC1RAB9ASMN1; SMN2CYP1A2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571357-A1 CHEMICAL COMPOUNDS, COMPOSITIONS AND METHODS FOR KINASE MODULATION Intellikine, Inc. (US) 2013-03-27 EP disclosed
WO-2011146882-A1 CHEMICAL COMPOUNDS, COMPOSITIONS AND METHODS FOR KINASE MODULATION INTELLIKINE, INC. (US) 2011-11-24 WO disclosed