SCHEMBL26029263

SCHEMBL26029263

c1ncc(-c2cc3nccn3c(Nc3cc[nH]n3)n2)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 5/20 0.42
MAP4K2 Q12851 6/20 0.39
MAP4K4 O95819 2/20 0.39
PKN2 Q16513 2/20 0.39
AURKB Q96GD4 2/20 0.39
SLK Q9H2G2 2/20 0.39
AURKA O14965 1/20 0.39
JAK2 O60674 1/20 0.39
INSR P06213 1/20 0.39
LCK P06239 1/20 0.39
LYN P07948 1/20 0.39
RET P07949 1/20 0.39
ROS1 P08922 1/20 0.39
SRC P12931 1/20 0.39
FER P16591 1/20 0.39
KDR P35968 1/20 0.39
BLK P51451 1/20 0.39
RPS6KA3 P51812 1/20 0.39
PRKCD Q05655 1/20 0.39
BTK Q06187 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26007557 0.84 SYK (0.40) SYKMAP4K2MAP4K4PKN2AURKB
SCHEMBL26011193 0.83 SYK (0.42) SYKMAP4K2MAP4K4PKN2AURKB
SCHEMBL26005518 0.80 SYK (0.41) SYKMAP4K2MAP4K4PKN2AURKB
SCHEMBL3044547 0.78 SYK (0.33) SYKMAP4K2MAP4K4PKN2AURKB
SCHEMBL26022798 0.78 MAPK1 (0.42) SYKMAP4K2MAP4K4PKN2AURKB
SCHEMBL13221039 0.78 PAK1 (0.42) SYK
SCHEMBL26007684 0.75 PDE2A (0.33) SYKMAP4K2MAP4K4PKN2AURKB
SCHEMBL26035235 0.75 SYK (0.32) SYKMAP4K2MAP4K4PKN2AURKB
SCHEMBL13220904 0.72 ALK (0.49) SYKMAP4K2MAP4K4PKN2AURKB
SCHEMBL26009808 0.71 ATR (0.40) SYKJAK2FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154426-A1 CDK INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2023-08-17 WO disclosed