SCHEMBL26037786

SCHEMBL26037786

COc1ccc(C(C)C)c2c1c(C)c(C(=O)O)n2C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.38
NQO2 P16083 1/20 0.38
ATM Q13315 2/20 0.38
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA7 P43166 2/20 0.37
CA9 Q16790 2/20 0.37
GPR35 Q9HC97 1/20 0.37
EDNRA P25101 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
MAPT P10636 5/20 0.34
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 3/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
MYC P01106 1/20 0.34
HPGD P15428 4/20 0.34
POLB P06746 3/20 0.34
HSD17B10 Q99714 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23809472 0.88 CYP19A1 (0.38) CYP19A1NQO2ATMCA1CA2
SCHEMBL26581499 0.83 CYP19A1 (0.45) CYP19A1NQO2ATMCA1CA2
SCHEMBL23809174 0.71 MCL1 (0.45) ATMCA1CA2GPR35KDM4E
SCHEMBL26581394 0.70 CYP19A1 (0.44) CYP19A1NQO2ATMNPSR1MAPT
SCHEMBL19332237 0.69 MAPT (0.39) CYP19A1NQO2ATMCA1CA2
SCHEMBL23809515 0.69 ATM (0.39) ATMMAPTALDH1A1HPGD
SCHEMBL23809479 0.66 KMT2A (0.44) ATMCA1CA2CA7CA9
SCHEMBL26048303 0.65 CYP19A1 (0.41) CYP19A1NQO2ATMNPSR1MAPT
SCHEMBL23809532 0.64 KMT2A (0.43) ATMMAPTALDH1A1KDM4EHPGD
SCHEMBL23809471 0.64 MAPT (0.36) CYP19A1NQO2CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3423435-B1 SUBSTITUTED INDOLE MCL-1 INHIBITORS UNIV VANDERBILT (US) 2023-08-23 EP disclosed