Piketoprofen

Piketoprofen

SCHEMBL26199

Cc1ccnc(NC(=O)C(C)c2cccc(C(=O)c3ccccc3)c2)c1

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.65
HTT P42858 3/20 0.65
ALDH1A1 P00352 3/20 0.65
LMNA P02545 3/20 0.65
MEN1 O00255 1/20 0.65
KMT2A Q03164 1/20 0.65
NPSR1 Q6W5P4 1/20 0.64
NPC1 O15118 1/20 0.62
RAB9A P51151 1/20 0.62
CYP3A4 P08684 2/20 0.62
CYP1A2 P05177 1/20 0.62
CYP2D6 P10635 1/20 0.62
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
SMN1; SMN2 Q16637 3/20 0.57
RIOK2 Q9BVS4 3/20 0.56
GSK3A P49840 2/20 0.56
MAPK10 P53779 2/20 0.56
PTGS1 P23219 3/20 0.54
PTGS2 P35354 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Piketoprofen SCHEMBL3156214 1.00 MAPT (0.65) MAPTHTTALDH1A1LMNAMEN1
Piketoprofen SCHEMBL3261211 1.00 MAPT (0.65) MAPTHTTALDH1A1LMNAMEN1
Piketoprofen SCHEMBL29706600 1.00 MAPT (0.65) MAPTHTTALDH1A1LMNAMEN1
Piketoprofen SCHEMBL19813145 0.99 MAPT (0.64) MAPTHTTALDH1A1LMNAMEN1
SCHEMBL3155175 0.87 POLB (0.73) MAPTHTTALDH1A1LMNAMEN1
Hydrochloric Acid SCHEMBL3258168 0.86 POLB (0.71) MAPTHTTALDH1A1LMNAMEN1
SCHEMBL27586219 0.84 RIOK2 (0.57) MAPTHTTALDH1A1LMNAMEN1
SCHEMBL31544567 0.79 HTT (0.69) MAPTHTTALDH1A1LMNAMEN1
SCHEMBL1820700 0.79 MAPT (0.85) MAPTHTTALDH1A1LMNAMEN1
SCHEMBL2183992 0.77 PSEN1 (0.82) MAPTHTTALDH1A1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2225 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023031749-A1 PALMITOYLETHANOLAMIDE SPRAY COMPOSITIONS SHILPA MEDICARE LIMITED (IN) 2023-03-09 WO claimed
EP-4034087-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS Research Inc. (CA) 2022-08-03 EP claimed
US-20220218611-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS RESEARCH INC. (CA) 2022-07-14 US claimed
WO-2021056106-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS RESEARCH INC. (CA) 2021-04-01 WO claimed
CN-107854469-A Topical ophthalmic or the husky star medicine of ear or nose use or external preparation for skin and combinations thereof 刘力 2018-03-30 CN claimed
US-20170225958-A1 FUNCTIONAL PARTICLES, PRODUCTION PROCESS AND USES SMART INOVATION, LDA (PT) 2017-08-10 US claimed
EP-3175865-A1 FUNCTIONAL PARTICLES, PRODUCTION PROCESS AND USES Smart Inovation Lda (PT) 2017-06-07 EP claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
EP-2560634-A1 NITRIC OXIDE RELEASING PRODRUGS OF THERAPEUTIC AGENTS Piramal Enterprises Limited (IN) 2013-02-27 EP claimed
US-20120183600-A1 NOVEL COMPOSITION FOR TREATING METABOLIC SYNDROME AND OTHER CONDITIONS CHEN CHIEN-HUNG (US) 2012-07-19 US claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
EP-0786999-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1999-01-20 EP claimed
EP-0792371-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1998-12-30 EP claimed
EP-0792371-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-09-03 EP claimed
EP-0786999-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-08-06 EP claimed
US-5543417-A 5 Alpha-reductase inhibitor and at least one of an antibacterial agent, a keratolytic agent or an anti-inflammatory agent MERCK & CO., INC. (US) 1996-08-06 US claimed
WO-1996012487-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1996012817-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed