SCHEMBL26330423

SCHEMBL26330423

COc1cc2nc(N)n3nc(C)nc3c2cc1F

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.50
ADORA2B P29275 19/20 0.50
PDE10A Q9Y233 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29475899 0.79 ADORA2A (0.46) ADORA2AADORA2B
SCHEMBL27164673 0.78 ADORA2A (0.51) ADORA2AADORA2B
SCHEMBL27164710 0.77 ADORA2A (0.48) ADORA2AADORA2B
SCHEMBL27164696 0.77 ADORA2A (0.47) ADORA2AADORA2B
SCHEMBL25418823 0.76 ADORA2A (0.49) ADORA2AADORA2B
SCHEMBL25418821 0.76 ADORA2A (0.49) ADORA2AADORA2B
SCHEMBL25423986 0.76 ADORA2A (0.49) ADORA2AADORA2B
SCHEMBL30427984 0.76 ADORA2A (0.49) ADORA2AADORA2B
SCHEMBL26330309 0.76 PDE10A (0.47) ADORA2AADORA2BPDE10A
SCHEMBL21996552 0.74 ADORA2A (0.67) ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023158626-A1 ADENOSINE RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE THEREOF MERCK SHARP & DOHME LLC (US) 2023-08-24 WO disclosed