SCHEMBL2638306

SCHEMBL2638306

Cc1cc(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)cc(Oc2cc(Cl)cc(C#N)c2)c1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 8/20 0.48
CA2 P00918 8/20 0.48
CA12 O43570 7/20 0.48
CA9 Q16790 6/20 0.48
P2RX4 Q99571 6/20 0.45
CA5A P35218 3/20 0.43
CA7 P43166 3/20 0.43
CA5B Q9Y2D0 3/20 0.43
CA14 Q9ULX7 1/20 0.43
CYP2C8 P10632 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ADRA2B P18089 1/20 0.43
HTR2C P28335 1/20 0.43
P2RX3 P56373 1/20 0.43
SLC6A3 Q01959 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
P2RX7 Q99572 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
POLB P06746 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2638930 0.90 CA1 (0.45) CA1CA2CA12CA9P2RX4
SCHEMBL2638800 0.89 CA1 (0.53) CA1CA2CA12CA9CA5A
SCHEMBL2638407 0.87 CA1 (0.53) CA1CA2CA12CA9P2RX4
SCHEMBL2638824 0.87 CA1 (0.51) CA1CA2CA12CA9P2RX4
SCHEMBL4602268 0.86 CA1 (0.53) CA1CA2CA12CA9P2RX4
SCHEMBL2638397 0.86 CA1 (0.51) CA1CA2CA12CA9P2RX4
SCHEMBL2639938 0.86 CA1 (0.53) CA1CA2CA12CA9P2RX4
SCHEMBL2639061 0.86 CA1 (0.57) CA1CA2CA12CA9CA5A
SCHEMBL4604854 0.85 P2RX4 (0.47) CA1CA2CA12CA9P2RX4
SCHEMBL4604671 0.85 CA1 (0.53) CA1CA2CA12CA9P2RX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4810529-B2 2011-11-09 JP claimed
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP claimed
EP-1742908-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-01-17 EP claimed
WO-2005102989-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2005-11-03 WO claimed
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP disclosed