SCHEMBL2640346

SCHEMBL2640346

Nc1ncc(O[C@H]2CCC(O)C2)nc1-c1nc2ccccc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ATR Q13535 16/20 0.51
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
EGFR P00533 1/20 0.44
PRKDC P78527 1/20 0.44
ATM Q13315 1/20 0.44
DGAT1 O75907 1/20 0.43
CHEK2 O96017 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL561078 1.00 ATR (0.51) ATRALDH1A1HPGDSMN1; SMN2NPSR1
SCHEMBL560943 1.00 ATR (0.51) ATRALDH1A1HPGDSMN1; SMN2NPSR1
SCHEMBL10135179 1.00 ATR (0.51) ATRALDH1A1HPGDSMN1; SMN2NPSR1
SCHEMBL560941 1.00 ATR (0.51) ATRALDH1A1HPGDSMN1; SMN2NPSR1
SCHEMBL560942 1.00 ATR (0.51) ATRALDH1A1HPGDSMN1; SMN2NPSR1
SCHEMBL10135180 1.00 ATR (0.51) ATRALDH1A1HPGDSMN1; SMN2NPSR1
SCHEMBL561077 1.00 ATR (0.51) ATRALDH1A1HPGDSMN1; SMN2NPSR1
SCHEMBL560077 0.75 ATR (0.61) ATRALDH1A1HPGDSMN1; SMN2NPSR1
SCHEMBL559766 0.75 ATR (0.63) ATRALDH1A1HPGDSMN1; SMN2NPSR1
SCHEMBL5638605 0.74 CHEK2 (0.66) ALDH1A1HPGDSMN1; SMN2CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569289-A1 PYRAZINES USEFUL AS INHIBITORS OF ATR KINASE Vertex Pharmaceuticals Incorporated (US) 2013-03-20 EP disclosed
WO-2011143419-A1 PYRAZINES USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-11-17 WO disclosed