SCHEMBL2641574

SCHEMBL2641574

CS(=O)(=O)c1ccc(Nc2nc3cccc(-c4ccc(S(C)(=O)=O)cc4)n3n2)cc1.CS(=O)(=O)c1ccc(Nc2nc3cccc(-c4ccc(S(C)(=O)=O)cc4)n3n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 20/20 1.00
JAK3 P52333 19/20 1.00
PTK2 Q05397 18/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2640560 1.00 JAK2 (1.00) JAK2JAK3PTK2
SCHEMBL2640652 0.95 JAK2 (0.91) JAK2JAK3PTK2
SCHEMBL3202575 0.92 JAK2 (0.85) JAK2JAK3PTK2
SCHEMBL2640637 0.92 JAK2 (1.00) JAK2JAK3PTK2
SCHEMBL3216706 0.91 JAK2 (0.83) JAK2JAK3PTK2
SCHEMBL2635085 0.91 JAK2 (1.00) JAK2JAK3PTK2
SCHEMBL3208718 0.90 JAK2 (0.82) JAK2JAK3PTK2
SCHEMBL3200475 0.89 JAK2 (0.80) JAK2JAK3PTK2
SCHEMBL22512323 0.89 JAK2 (0.78) JAK2JAK3PTK2
SCHEMBL2634700 0.88 JAK2 (1.00) JAK2JAK3PTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438066-A2 PREPARATION AND USES OF 1,2,4-TRIAZOLO [1,5a]PYRIDINE DERIVATIVES Cephalon, Inc. (US) 2012-04-11 EP disclosed
WO-2010141796-A2 PREPARATION AND USES OF 1,2,4-TRIAZOLO [1,5a] PYRIDINE DERIVATIVES CEPHALON, INC. (US) 2010-12-09 WO disclosed