SCHEMBL2641778

SCHEMBL2641778

COc1ccc(/C=C/c2cccc(Br)n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.56
TRPA1 O75762 1/20 0.53
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
RELA Q04206 5/20 0.51
CYP1A2 P05177 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
KDM4E B2RXH2 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
HPGD P15428 1/20 0.50
CYP2C19 P33261 1/20 0.50
DHFR P00374 1/20 0.48
APP P05067 4/20 0.47
NFE2L2 Q16236 2/20 0.47
ESR1 P03372 2/20 0.47
ABL1 P00519 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2641784 1.00 MAPT (0.56) MAPTTRPA1NPC1RAB9AMEN1
SCHEMBL4536873 0.84 MEN1 (0.58) NPC1MEN1KMT2ARELACYP1A2
SCHEMBL4536867 0.84 MEN1 (0.58) NPC1MEN1KMT2ARELACYP1A2
SCHEMBL5864850 0.81 GRM4 (0.65) MAPTTRPA1NPC1RAB9ARELA
SCHEMBL5864846 0.81 GRM4 (0.65) MAPTTRPA1NPC1RAB9ARELA
Hydrochloric Acid SCHEMBL5865178 0.79 GRM4 (0.63) MAPTTRPA1NPC1RAB9ARELA
Hydrochloric Acid SCHEMBL5865175 0.79 GRM4 (0.63) MAPTTRPA1NPC1RAB9ARELA
SCHEMBL4542155 0.79 GRM4 (0.61) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL4542158 0.79 GRM4 (0.61) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL5864866 0.78 MAPT (0.53) MAPTTRPA1NPC1RAB9ARELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011141515-A1 DIAGNOSTIC AGENTS FOR AMYLOID BETA IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-11-17 WO claimed
WO-2011141515-A1 DIAGNOSTIC AGENTS FOR AMYLOID BETA IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-11-17 WO disclosed