SCHEMBL2644444

SCHEMBL2644444

COc1ccc(Oc2cc(Sc3nccn3C)c3nc(-c4ccccn4)[nH]c3c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
RUNX1 Q01196 2/20 0.49
CBFB Q13951 14/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
ALDH1A1 P00352 2/20 0.43
TP53 P04637 2/20 0.43
HPGD P15428 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
ALOX15 P16050 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GCK P35557 2/20 0.40
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
LMNA P02545 1/20 0.37
PKM P14618 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2646299 0.87 GCK (0.39) NPC1RAB9ARUNX1CBFBSMN1; SMN2
SCHEMBL2645178 0.85 NPC1 (0.55) NPC1RAB9ARUNX1CBFBSMN1; SMN2
SCHEMBL2645879 0.75 GCK (0.39) NPC1CBFBHPGDCYP3A4CYP2C19
SCHEMBL2647458 0.71 GCK (0.42) NPC1RAB9ARUNX1CBFBSMN1; SMN2
SCHEMBL2645683 0.71 CBFB (0.43) NPC1RAB9ARUNX1CBFBGCK
SCHEMBL2647096 0.70 GCK (0.44) NPC1RAB9ARUNX1CBFBSMN1; SMN2
SCHEMBL2645245 0.68 CBFB (0.63) NPC1RAB9ARUNX1CBFBSMN1; SMN2
SCHEMBL10351275 0.67 NPC1 (1.00) NPC1RAB9ARUNX1CBFBSMN1; SMN2
SCHEMBL2645214 0.67 CBFB (0.54) NPC1RAB9ARUNX1CBFBSMN1; SMN2
SCHEMBL2644975 0.66 CBFB (0.46) NPC1RAB9ARUNX1CBFBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1702919-B1 NOVEL 2-HETEROARYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVE MSD KK (JP) 2012-05-30 EP disclosed
EP-1702919-A1 NOVEL 2-HETEROARYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2006-09-20 EP disclosed