SCHEMBL26451247

SCHEMBL26451247

CN(C)c1nc2ccc(-c3nc(Nc4ccc(CN5CCN(S(C)(=O)=O)CC5)cn4)ncc3F)cc2s1

nearest known ligand 0.76

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DYRK2 Q92630 13/20 0.76
CDK6 Q00534 7/20 0.74
CCND1 P24385 3/20 0.53
CDK4 P11802 2/20 0.53
CCND3 P30281 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30569708 1.00 DYRK2 (0.76) DYRK2CDK6CCND1CDK4CCND3
SCHEMBL30569710 0.93 DYRK2 (0.74) DYRK2CDK6CCND1CDK4CCND3
SCHEMBL26451650 0.93 DYRK2 (0.74) DYRK2CDK6CCND1CDK4CCND3
SCHEMBL26447947 0.90 DYRK2 (0.81) DYRK2CDK6CCND1CDK4CCND3
SCHEMBL30679266 0.90 DYRK2 (0.81) DYRK2CDK6CCND1CDK4CCND3
SCHEMBL26680021 0.88 DYRK2 (0.66) DYRK2CDK6
SCHEMBL26447961 0.88 DYRK2 (0.81) DYRK2CDK6CCND1CDK4
SCHEMBL30569702 0.88 DYRK2 (0.81) DYRK2CDK6CCND1CDK4
SCHEMBL26447954 0.88 DYRK2 (0.80) DYRK2CDK6CCND1CDK4CCND3
Hydrochloric Acid SCHEMBL30679271 0.87 DYRK2 (0.81) DYRK2CDK6CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4282864-B1 CDK6/DYRK2 DUAL-TARGET INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF JIANGSU TASLY DIYI PHARMACEUTICAL CO LTD (CN) 2025-08-13 EP disclosed
EP-4282864-A1 CDK6/DYRK2 DUAL-TARGET INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF Jiangsu Tasly Diyi Pharmaceutical Co., Ltd. (CN) 2023-11-29 EP disclosed