SCHEMBL2646162

SCHEMBL2646162

CCS(=O)(=O)c1ccc(Oc2cc(Oc3cccnc3OC(F)F)c3nc(-c4ccccn4)[nH]c3c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GCK P35557 14/20 0.49
CBFB Q13951 5/20 0.43
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2644782 0.86 GCK (0.62) GCK
SCHEMBL2643943 0.84 GCK (0.51) GCKCBFBALDH1A1TP53CYP3A4
SCHEMBL2647193 0.83 CBFB (0.41) GCKCBFBALDH1A1TP53CYP3A4
SCHEMBL2644981 0.83 GCK (0.53) GCKCBFBALDH1A1TP53CYP3A4
SCHEMBL2645422 0.82 GCK (0.53) GCKCBFBALDH1A1TP53CYP3A4
SCHEMBL3549191 0.81 GCK (0.47) GCK
SCHEMBL2644037 0.79 CBFB (0.49) GCKCBFBALDH1A1TP53CYP3A4
SCHEMBL2645534 0.78 GCK (0.50) GCKCBFBALDH1A1TP53CYP3A4
SCHEMBL2645485 0.78 CBFB (0.50) GCKCBFBALDH1A1TP53CYP3A4
SCHEMBL2645829 0.78 GCK (0.52) GCKCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1702919-B1 NOVEL 2-HETEROARYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVE MSD KK (JP) 2012-05-30 EP disclosed
EP-1702919-A1 NOVEL 2-HETEROARYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2006-09-20 EP disclosed