SCHEMBL2648904

SCHEMBL2648904

C1=CN[C](NCc2ccccc2)C=C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.43
KCNH3 Q9ULD8 1/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
HSD17B10 Q99714 1/20 0.39
FABP1 P07148 1/20 0.38
FABP6 P51161 1/20 0.38
METAP2 P50579 1/20 0.38
IDO1 P14902 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 2/20 0.38
THRB P10828 1/20 0.38
MEN1 O00255 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
POLB P06746 1/20 0.37
RAD52 P43351 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28026789 0.73 HTT (0.42) HTTKCNH3CA1CA2HSD17B10
SCHEMBL12478183 0.72 HSD17B10 (0.46) HTTHSD17B10ALDH1A1KMT2ATHRB
SCHEMBL9294542 0.72 HTT (0.35) HTTKCNH3CA1CA2HSD17B10
N-Benzylaniline SCHEMBL7840 0.68 HTT (0.71) HTTKCNH3CA1CA2ALDH1A1
SCHEMBL22628164 0.68 HTT (0.71) HTTKCNH3CA1CA2ALDH1A1
SCHEMBL1924100 0.68 HTT (0.78) HTTCA1CA2ALDH1A1KMT2A
SCHEMBL4072346 0.68 IDO1 (0.39) HTTCA1CA2HSD17B10FABP1
SCHEMBL2066721 0.67 RECQL (0.31)
N-Benzylaniline SCHEMBL3602124 0.66 HTT (0.68) HTTKCNH3CA1CA2ALDH1A1
SCHEMBL20804371 0.66 HTT (0.61) HTTKCNH3CA1CA2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776954-A GLUCAGON ANTAGONISTS MERCK & CO., INC. (US) 1998-07-07 US claimed
EP-0859771-A4 SUBSTITUTED PYRIDYL PYRROLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO INC (US) 2000-03-15 EP disclosed
EP-0859771-A1 SUBSTITUTED PYRIDYL PYRROLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE Merck & Co., Inc. (US) 1998-08-26 EP disclosed
US-5776954-A GLUCAGON ANTAGONISTS MERCK & CO., INC. (US) 1998-07-07 US disclosed
WO-1997016442-A1 SUBSTITUTED PYRIDYL PYRROLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO., INC. (US) 1997-05-09 WO disclosed