SCHEMBL2649158

SCHEMBL2649158

Cc1[nH]cc2c(=O)n(-c3ccc(Cl)cc3)nc-2c1-c1cccc(-c2ncc[nH]2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 7/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
LMNA P02545 2/20 0.35
CHEK1 O14757 1/20 0.35
EGFR P00533 1/20 0.35
KDR P35968 1/20 0.35
BRD4 O60885 1/20 0.35
PSD A5PKW4 2/20 0.35
NPSR1 Q6W5P4 2/20 0.34
AURKA O14965 1/20 0.34
SYK P43405 1/20 0.34
MAPT P10636 4/20 0.33
HTT P42858 3/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
NOD2 Q9HC29 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2649146 0.90 NISCH (0.39) GAASMN1; SMN2NPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL7443190 0.89 NISCH (0.38) GAASMN1; SMN2NPC1RAB9AMEN1
SCHEMBL2649481 0.84 PSD (0.50) GAASMN1; SMN2NPC1RAB9APSD
SCHEMBL2649751 0.83 KIT (0.40) GAASMN1; SMN2NPC1RAB9AMEN1
SCHEMBL2648853 0.83 GAA (0.39) GAASMN1; SMN2NPC1RAB9AMEN1
SCHEMBL2650770 0.83 GAA (0.47) GAASMN1; SMN2NPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL2662150 0.82 GAA (0.46) GAASMN1; SMN2NPC1RAB9AMEN1
SCHEMBL2649984 0.82 SMN1; SMN2 (0.43) GAASMN1; SMN2NPC1RAB9AMEN1
SCHEMBL2649448 0.82 DHODH (0.40) GAASMN1; SMN2NPC1RAB9AMEN1
SCHEMBL2649310 0.82 CSNK2A1 (0.42) GAASMN1; SMN2MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1064283-A1 PYRAZOLO-PYRIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2001-01-03 EP claimed
WO-1999048892-A1 PYRAZOLO-PYRIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 1999-09-30 WO claimed
EP-1064283-A1 PYRAZOLO-PYRIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2001-01-03 EP disclosed
WO-1999048892-A1 PYRAZOLO-PYRIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 1999-09-30 WO disclosed