SCHEMBL2651047

SCHEMBL2651047

CCOC(=O)C=Cc1ccc(C2OCCO2)c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
L3MBTL1 Q9Y468 3/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
CYP3A4 P08684 2/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
ESR1 P03372 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2664362 1.00 NPC1 (0.42) NPC1RAB9ACASP3SENP8SENP7
SCHEMBL6853096 0.83 CA12 (0.54) NPC1RAB9ACASP3SENP8SENP7
SCHEMBL11218812 0.83 CA12 (0.54) NPC1RAB9ACASP3SENP8SENP7
SCHEMBL6853099 0.78 HCAR2 (0.51) NPC1RAB9ACASP3SENP8SENP7
SCHEMBL14290541 0.77 TTR (0.55) NPC1RAB9ACASP3SENP8SENP7
SCHEMBL21449475 0.76 CA12 (0.47) NPC1RAB9ACASP3SENP8SENP7
SCHEMBL2690695 0.75 HDAC8 (0.55) MAPTKDM4EMEN1KMT2AATM
SCHEMBL2690696 0.75 HDAC8 (0.55) MAPTKDM4EMEN1KMT2AATM
SCHEMBL2689193 0.75 CAPN1 (0.59) MAPTKDM4EMEN1KMT2ACYP3A4
SCHEMBL12035855 0.75 CAPN1 (0.59) MAPTKDM4EMEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6613942-B1 Nonpeptide; 4-hydroxy benzoic acid hydrazides NOVO NORDISK A/S (DK) 2003-09-02 US disclosed
EP-0994848-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2000-04-26 EP disclosed
WO-1999001423-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 1999-01-14 WO disclosed