SCHEMBL2651653

SCHEMBL2651653

N#Cc1cccnc1-c1ccccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.48
LMNA P02545 3/20 0.48
CCR1 P32246 2/20 0.48
CCR5 P51681 2/20 0.48
CCR8 P51685 2/20 0.48
CYP1A2 P05177 1/20 0.48
POLB P06746 1/20 0.48
METAP1 P53582 1/20 0.48
BLM P54132 1/20 0.48
HIF1A Q16665 1/20 0.48
DOHH Q9BU89 1/20 0.48
P4HTM Q9NXG6 1/20 0.48
GRM5 P41594 3/20 0.45
TGFBR1 P36897 1/20 0.45
CNR2 P34972 1/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 3/20 0.42
MAPT P10636 2/20 0.42
MEN1 O00255 1/20 0.42
USP2 O75604 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29741178 1.00 KDM4E (0.48) KDM4ELMNACCR1CCR5CCR8
SCHEMBL9449076 0.98 KDM4E (0.46) KDM4ELMNACCR1CCR5CCR8
SCHEMBL2651055 0.86 CCR1 (0.40) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL27792926 0.84 KDM4E (0.64) KDM4ELMNACCR1CCR5CCR8
SCHEMBL31267979 0.83 CNR2 (0.49) KDM4ECYP1A2POLBBLMCNR2
SCHEMBL8936053 0.83 KDM4E (0.47) KDM4ELMNACCR1CCR5CCR8
SCHEMBL9715965 0.81 KDM4E (0.48) KDM4ELMNACCR1CCR5CCR8
SCHEMBL12470406 0.80 KDM4E (0.43) KDM4ELMNACCR1CCR5CCR8
SCHEMBL29761073 0.80 GRM5 (0.43) CYP1A2GRM5CNR2ALDH1A1HPGD
SCHEMBL18411456 0.80 KDM4E (0.52) KDM4ELMNACCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110105336-A Viologen derivative electrochromic material and preparation method thereof 华南理工大学 2019-08-09 CN claimed
WO-2023139085-A1 NEW BENZIMIDAZOLE PYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2023-07-27 WO disclosed
CN-109679129-B Method for modifying surface of polyolefin material 宿迁市南京工业大学新材料研究院 2021-06-29 CN disclosed
CN-104961677-A 11beta-HSD1 inhibitor of cyanobipyridine tert-alcohol structure and application of 11beta-HSD1 inhibitor FOSHAN SAIWEISI PHARMACEUTICAL TECHNOLOGY CO LTD 2015-10-07 CN disclosed
CN-104961677-A 11beta-HSD1 inhibitor of cyanobipyridine tert-alcohol structure and application of 11beta-HSD1 inhibitor FOSHAN SAIWEISI PHARMACEUTICAL TECHNOLOGY CO LTD 2015-10-07 CN disclosed
EP-1383768-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2004-01-28 EP disclosed
WO-2002076983-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2002-10-03 WO disclosed