SCHEMBL2652533

SCHEMBL2652533

Fc1cccc(F)c1-c1cccnc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 9/20 0.58
ALDH1A1 P00352 3/20 0.58
CYP3A4 P08684 3/20 0.58
CYP1A2 P05177 2/20 0.58
KDM4E B2RXH2 1/20 0.50
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
MAPT P10636 1/20 0.50
HPGD P15428 1/20 0.50
ALOX15 P16050 1/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
HSD17B10 Q99714 1/20 0.50
TDO2 P48775 1/20 0.47
CYP2E1 P05181 2/20 0.47
CYP2B6 P20813 2/20 0.47
MEN1 O00255 1/20 0.47
PSIP1 O75475 1/20 0.47
AXL P30530 1/20 0.47
MKNK1 Q9BUB5 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8126224 0.87 CYP2A6 (0.48) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL21578105 0.82 CYP2A6 (0.64) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL18797731 0.81 DHODH (0.55) ALDH1A1KDM4ELMNAHTTSMN1; SMN2
SCHEMBL11965538 0.81 CYP2A6 (0.78) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL29706657 0.80 AXL (0.55) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL8504194 0.80 AXL (0.55) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL4147013 0.80 CYP2A6 (0.61) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL29257373 0.79 CYP2A6 (0.48) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL2665899 0.77 CYP2A6 (0.47) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E
SCHEMBL28603188 0.77 CYP2A6 (0.47) CYP2A6ALDH1A1CYP3A4CYP1A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107207529-A Bicyclic compounds as pest control agents 拜耳作物科学股份公司 2017-09-26 CN disclosed
EP-1381606-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2004-01-21 EP disclosed
WO-2002074773-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2002-09-26 WO disclosed
US-4797490-A Process for the preparation of 3-(2'-fluorophenyl)pyridine PFIZER INC. (US) 1989-01-10 US disclosed
US-4636506-A BACTERICIDES, STAPHYLOCOCCUS PFIZER, INC. (US) 1987-01-13 US disclosed